nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
ACAT inhibitors derived from hetero-Diels-Alder cycloadducts of thioaldehydes
|
Wilde, Richard G. |
|
1996 |
4 |
9 |
p. 1493-1513 21 p. |
artikel |
2 |
20-Amino and 20,21-aziridinyl pregnene steroids: Development of potent inhibitors of 17α-hydroxylase/C17,20-lyase (P450 17)
|
Njar, Vincent C.O. |
|
1996 |
4 |
9 |
p. 1447-1453 7 p. |
artikel |
3 |
A new class of HIV-1 protease inhibitor: The crystallographic structure, inhibition and chemical synthesis of an aminimide peptide isostere
|
Rutenber, Earl E. |
|
1996 |
4 |
9 |
p. 1545-1558 14 p. |
artikel |
4 |
3-Carboxy-20-keto steroids are dual uncompetitive inhibitors of human steroid 5α-reductase types 1 and 2
|
Yamashita, Dennis S. |
|
1996 |
4 |
9 |
p. 1481-1485 5 p. |
artikel |
5 |
Design, synthesis, and in vitro inhibitory activity toward human leukocyte elastase, cathepsin G, and proteinase 3 of saccharin-derived sulfones and congeners
|
Groutas, William C. |
|
1996 |
4 |
9 |
p. 1393-1400 8 p. |
artikel |
6 |
Discovery and optimization of nonpeptide HIV-1 protease inhibitors
|
Tummino, Peter J. |
|
1996 |
4 |
9 |
p. 1401-1410 10 p. |
artikel |
7 |
Graphical abstracts
|
|
|
1996 |
4 |
9 |
p. vii-xi nvt p. |
artikel |
8 |
Inhibition of steroid C17(20) lyase with C-17-heteroaryl steroids
|
Burkhart, Joseph P. |
|
1996 |
4 |
9 |
p. 1411-1420 10 p. |
artikel |
9 |
Inhibitors of farnesyl:protein transferase—A possible cancer chemotherapeutic
|
Scholten, Jeffrey D. |
|
1996 |
4 |
9 |
p. 1537-1543 7 p. |
artikel |
10 |
Inhibitors of human nitric oxide synthase isoforms with the carbamidine moiety as a common structural element
|
Moore, William M. |
|
1996 |
4 |
9 |
p. 1559-1564 6 p. |
artikel |
11 |
Mechanism-based inactivation of γ-aminobutyric acid aminotransferase by 3-amino-4-fluorobutanoic acid
|
Silverman, Richard B. |
|
1996 |
4 |
9 |
p. 1521-1535 15 p. |
artikel |
12 |
Preface
|
Silverman, Richard B. |
|
1996 |
4 |
9 |
p. xiii- 1 p. |
artikel |
13 |
Properties of analogues of an intermediate in the process of mechanism-based inactivation of carboxypeptidase A
|
Ghosh, Soumitra S. |
|
1996 |
4 |
9 |
p. 1487-1492 6 p. |
artikel |
14 |
Quiescent affinity inactivators of protein tyrosine phosphatases
|
Taylor, William P. |
|
1996 |
4 |
9 |
p. 1515-1520 6 p. |
artikel |
15 |
Solution conformations of KNI-272, a tripeptide HIV protease inhibitor designed on the basis of substrate transition state: Determined by NMR spectroscopy and simulated annealing calculations
|
Ohno, Yasushi |
|
1996 |
4 |
9 |
p. 1565-1572 8 p. |
artikel |
16 |
Structure-based design of achiral, nonpeptidic hydroxybenzamide as a novel P2/P2′ replacement for the symmetry-based HIV protease inhibitors
|
Randad, Ramnarayan S. |
|
1996 |
4 |
9 |
p. 1471-1480 10 p. |
artikel |
17 |
Structure-based design of parasitic protease inhibitors
|
Li, Rongshi |
|
1996 |
4 |
9 |
p. 1421-1427 7 p. |
artikel |
18 |
Synthesis of complex δ-acetylenic amino acids as potential multisubstrate adduct inhibitors of methyltransferases
|
Burns, Mark R. |
|
1996 |
4 |
9 |
p. 1455-1470 16 p. |
artikel |
19 |
The rationale for E2020 as a potent acetylcholinesterase inhibitor
|
Kawakami, Yoshiyuki |
|
1996 |
4 |
9 |
p. 1429-1446 18 p. |
artikel |