| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Aminothiazolones as potent, selective and cell active inhibitors of the PIM kinase family
|
Quevedo, Camilo E.
|
|
|
28 |
22 |
p.
|
artikel
|
| 2 |
Analogs of nitrofuran antibiotics are potent GroEL/ES inhibitor pro-drugs
|
Stevens, Mckayla
|
|
|
28 |
22 |
p.
|
artikel
|
| 3 |
A new Pb2+-specific DNAzyme by revisiting the catalytic core of 10–23 DNAzyme
|
Li, Yang
|
|
|
28 |
22 |
p.
|
artikel
|
| 4 |
An expedient process for reducing the formation of process-related impurities during solid-phase synthesis of potential nucleic acid-based drugs
|
Grajkowski, Andrzej
|
|
|
28 |
22 |
p.
|
artikel
|
| 5 |
Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor
|
Ribeiro, Jean F.R.
|
|
|
28 |
22 |
p.
|
artikel
|
| 6 |
Design and synthesis of Coenzyme A analogues as Aurora kinase A inhibitors: An exploration of the roles of the pyrophosphate and pantetheine moieties
|
Bellany, Fiona
|
|
|
28 |
22 |
p.
|
artikel
|
| 7 |
Design and synthesis of novel methoxypyridine-derived gamma-secretase modulators
|
Rynearson, Kevin D.
|
|
|
28 |
22 |
p.
|
artikel
|
| 8 |
Design, synthesis, and multitargeted profiling of N-benzylpyrrolidine derivatives for the treatment of Alzheimer’s disease
|
Choubey, Priyanka Kumari
|
|
|
28 |
22 |
p.
|
artikel
|
| 9 |
Discovery and structure activity relationships of 7-benzyl triazolopyridines as stable, selective, and reversible inhibitors of myeloperoxidase
|
Shaw, Scott A.
|
|
|
28 |
22 |
p.
|
artikel
|
| 10 |
Druggable targets from coronaviruses for designing new antiviral drugs
|
Silva, Leandro Rocha
|
|
|
28 |
22 |
p.
|
artikel
|
| 11 |
Editorial Board
|
|
|
|
28 |
22 |
p.
|
artikel
|
| 12 |
Evaluation of 1,1-cyclopropylidene as a thioether isostere in the 4-thio-thienopyrimidine (TTP) series of antimalarials
|
Barrows, Robert D.
|
|
|
28 |
22 |
p.
|
artikel
|
| 13 |
Fluorinated 2-Arylcyclopropan-1-amines – A new class of sigma receptor ligands
|
Schinor, Benjamin
|
|
|
28 |
22 |
p.
|
artikel
|
| 14 |
Fragment based drug design and diversity-oriented synthesis of carboxylic acid isosteres
|
Ferri, Martina
|
|
|
28 |
22 |
p.
|
artikel
|
| 15 |
Graphical Abstract Contents Continued
|
|
|
|
28 |
22 |
p.
|
artikel
|
| 16 |
Graphical abstract TOC
|
|
|
|
28 |
22 |
p.
|
artikel
|
| 17 |
Graphical abstract TOC
|
|
|
|
28 |
22 |
p.
|
artikel
|
| 18 |
Identification of diphenylalkylisoxazol-5-amine scaffold as novel activator of cardiac myosin
|
Boggu, Pulla Reddy
|
|
|
28 |
22 |
p.
|
artikel
|
| 19 |
Inhibition of Mycobacterium tuberculosis InhA: Design, synthesis and evaluation of new di-triclosan derivatives
|
Armstrong, Tom
|
|
|
28 |
22 |
p.
|
artikel
|
| 20 |
Lead optimization of 8-(methylamino)-2-oxo-1,2-dihydroquinolines as bacterial type II topoisomerase inhibitors
|
Ushiyama, Fumihito
|
|
|
28 |
22 |
p.
|
artikel
|
| 21 |
10-N-heterocylic aryl-isoxazole-amides (AIMs) have robust anti-tumor activity against breast and brain cancer cell lines and useful fluorescence properties
|
Weaver, Matthew J.
|
|
|
28 |
22 |
p.
|
artikel
|
| 22 |
Non-cytotoxic 1,2,3-triazole tethered fused heterocyclic ring derivatives display Tax protein inhibition and impair HTLV-1 infected cells
|
dos Santos, Daiane Fernanda
|
|
|
28 |
22 |
p.
|
artikel
|
| 23 |
N-phenyl ureidobenzenesulfonates, a novel class of promising human dihydroorotate dehydrogenase inhibitors
|
Bouzriba, Chahrazed
|
|
|
28 |
22 |
p.
|
artikel
|
| 24 |
Preparation and evaluation of soluble epoxide hydrolase inhibitors with improved physical properties and potencies for treating diabetic neuropathic pain
|
Lee, Kin Sing Stephen
|
|
|
28 |
22 |
p.
|
artikel
|
| 25 |
Protein synthesis with conformationally constrained cyclic dipeptides
|
Zhang, Chao
|
|
|
28 |
22 |
p.
|
artikel
|
| 26 |
Sequential dual site-selective protein labelling enabled by lysine modification
|
Matos, Maria J.
|
|
|
28 |
22 |
p.
|
artikel
|
| 27 |
Structure-based linker exploration: Discovery of 1-ethyl-1H-indole analogs as novel ATX inhibitors
|
Jia, Fang
|
|
|
28 |
22 |
p.
|
artikel
|
| 28 |
Synthesis and biological evaluation of novel flexible nucleoside analogues that inhibit flavivirus replication in vitro
|
Thames, Joy E.
|
|
|
28 |
22 |
p.
|
artikel
|
| 29 |
Synthesis and evaluation of etoposide and podophyllotoxin analogs against topoisomerase IIα and HCT-116 cells
|
Murphy, Matthew B.
|
|
|
28 |
22 |
p.
|
artikel
|
| 30 |
Synthesis and structure-activity relationships for tetrahydroisoquinoline-based inhibitors of Mycobacterium tuberculosis
|
Lu, Guo-Liang
|
|
|
28 |
22 |
p.
|
artikel
|
| 31 |
Tetrahydroquinolinyl phosphinamidates and phosphonamidates enhancing tolerance towards drought stress in crops via interaction with ABA receptor proteins
|
Frackenpohl, Jens
|
|
|
28 |
22 |
p.
|
artikel
|
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