| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
An aza-nucleoside, fragment-like inhibitor of the DNA repair enzyme alkyladenine glycosylase (AAG)
|
Mas Claret, Eduard
|
|
|
28 |
11 |
p.
|
artikel
|
| 2 |
A novel Golgi mannosidase inhibitor: Molecular design, synthesis, enzyme inhibition, and inhibition of spheroid formation
|
Koyama, Ryosuke
|
|
|
28 |
11 |
p.
|
artikel
|
| 3 |
Benzoxepinones: A new isoform-selective class of tumor associated carbonic anhydrase inhibitors
|
Grandane, Aiga
|
|
|
28 |
11 |
p.
|
artikel
|
| 4 |
Cytotoxicity of 4-substituted quinoline derivatives: Anticancer and antileishmanial potential
|
Costa, Claudia A.
|
|
|
28 |
11 |
p.
|
artikel
|
| 5 |
Design and synthesis of 1,3-benzothiazinone derivatives as potential anti-inflammatory agents
|
Li, Junfang
|
|
|
28 |
11 |
p.
|
artikel
|
| 6 |
Design and synthesis of novel pyrrolo[2,3-b]pyridine derivatives targeting V600EBRAF
|
Abdel-Maksoud, Mohammed S.
|
|
|
28 |
11 |
p.
|
artikel
|
| 7 |
Design, synthesis and acaricidal activities of Cyflumetofen analogues based on carbon-silicon isosteric replacement
|
Zhou, Cong
|
|
|
28 |
11 |
p.
|
artikel
|
| 8 |
Deuteration of the farnesyl terminal methyl groups of δ-tocotrienol and its effects on the metabolic stability and ability of inducing G-CSF production
|
Liu, Xingui
|
|
|
28 |
11 |
p.
|
artikel
|
| 9 |
Discovery of a new potent inhibitor of mushroom tyrosinase (Agaricus bisporus) containing 4-(4-hydroxyphenyl)piperazin-1-yl moiety
|
De Luca, Laura
|
|
|
28 |
11 |
p.
|
artikel
|
| 10 |
Discovery of novel, potent, and orally bioavailable pyrido[2,3-d][1]benzazepin-6-one antagonists for parathyroid hormone receptor 1
|
Arai, Yoshikazu
|
|
|
28 |
11 |
p.
|
artikel
|
| 11 |
Editorial Board
|
|
|
|
28 |
11 |
p.
|
artikel
|
| 12 |
Enzymatic synthesis of biphenyl-DNA oligonucleotides
|
Röthlisberger, Pascal
|
|
|
28 |
11 |
p.
|
artikel
|
| 13 |
Exploratory studies on CA-15L, an anti-HIV active HIV-1 capsid fragment
|
Tsuji, Kohei
|
|
|
28 |
11 |
p.
|
artikel
|
| 14 |
Graphical Abstract Contents Continued
|
|
|
|
28 |
11 |
p.
|
artikel
|
| 15 |
Graphical abstract TOC
|
|
|
|
28 |
11 |
p.
|
artikel
|
| 16 |
Graphical abstract TOC
|
|
|
|
28 |
11 |
p.
|
artikel
|
| 17 |
Induction of enantio-selective apoptosis in human leukemia HL-60 cells by (S)-erypoegin K, an isoflavone isolated from Erythrina poeppigiana
|
Hikita, Kiyomi
|
|
|
28 |
11 |
p.
|
artikel
|
| 18 |
Inhibition of bacterial growth and galactosyltransferase activity of WbwC by α, ω-bis(3-alkyl-1H-imidazolium)alkane salts: Effect of varying carbon content
|
Kocev, Alexander
|
|
|
28 |
11 |
p.
|
artikel
|
| 19 |
Microbial transformation of glycyrrhetinic acid derivatives by Bacillus subtilis ATCC 6633 and Bacillus megaterium CGMCC 1.1741
|
Shen, Pingping
|
|
|
28 |
11 |
p.
|
artikel
|
| 20 |
Optimization and biological evaluation of imidazopyridine derivatives as a novel scaffold for γ-secretase modulators with oral efficacy against cognitive deficits in Alzheimer’s disease model mice
|
Sekioka, Ryuichi
|
|
|
28 |
11 |
p.
|
artikel
|
| 21 |
Progress towards drug discovery for Friedreich’s Ataxia: Identifying synthetic oligonucleotides that more potently activate expression of human frataxin protein
|
Shen, Xiulong
|
|
|
28 |
11 |
p.
|
artikel
|
| 22 |
Secondary metabolites from Isodon ternifolius (D. Don) Kudo and their anticancer activity as DNA topoisomerase IB and Tyrosyl-DNA phosphodiesterase 1 inhibitors
|
Zhang, Hong-Li
|
|
|
28 |
11 |
p.
|
artikel
|
| 23 |
Structural modifications of indolinones bearing a pyrrole moiety and discovery of a multi-kinase inhibitor with potent antitumor activity
|
Qin, Mingze
|
|
|
28 |
11 |
p.
|
artikel
|
| 24 |
Structure-activity relationship studies on the inhibition of the bacterial translation of novel Odilorhabdins analogues
|
Loza, Einars
|
|
|
28 |
11 |
p.
|
artikel
|
| 25 |
Syntheses and pharmacokinetic evaluations of four metabolites of 2-(4-(2-((1H-benzo[d]imidazol-2-yl)thio)ethyl)piperazin-1-yl)-N-(6-methyl-2,4-bis-(methylthio)pyridin-3-yl)acetamide hydrochloride [K-604], an acyl-CoA:cholesterol O-acyltransferase-1 inhibitor
|
Shibuya, Kimiyuki
|
|
|
28 |
11 |
p.
|
artikel
|
| 26 |
Syntheses, in vitro α-amylase and α-glucosidase dual inhibitory activities of 4-amino-1,2,4-triazole derivatives their molecular docking and kinetic studies
|
Yeye, Emmanuel Oloruntoba
|
|
|
28 |
11 |
p.
|
artikel
|
| 27 |
Synthesis and cytotoxic effects of 2-thio-3,4-dihydroquinazoline derivatives as novel T-type calcium channel blockers
|
Nam, Yunchan
|
|
|
28 |
11 |
p.
|
artikel
|
| 28 |
Synthesis and evaluation of 7-azaindole derivatives bearing benzocycloalkanone motifs as protein kinase inhibitors
|
Qhobosheane, Malikotsi A.
|
|
|
28 |
11 |
p.
|
artikel
|
| 29 |
Synthesis and structure-activity relationships of thieno[2,3-d]pyrimidines as atypical protein kinase C inhibitors to control retinal vascular permeability and cytokine-induced edema
|
Liu, Xuwen
|
|
|
28 |
11 |
p.
|
artikel
|
| 30 |
Synthesis, state-of-the-art NMR-binding and molecular modeling study of new benzimidazole core derivatives as Pin1 inhibitors: Targeting breast cancer
|
Nashaat, Samira
|
|
|
28 |
11 |
p.
|
artikel
|
| 31 |
Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activity
|
Brizzi, Antonella
|
|
|
28 |
11 |
p.
|
artikel
|
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