| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Chemical synthesis and biological activity of novel brominated 7-deazaadenosine-3′,5′-cyclic monophosphate derivatives
|
Lelle, Marco
|
|
|
27 |
8 |
p. 1704-1713
|
artikel
|
| 2 |
Chemical synthesis and functional characterization of a new class of ceramide analogues as anti-cancer agents
|
Liu, Qianqian
|
|
|
27 |
8 |
p. 1489-1496
|
artikel
|
| 3 |
Designing of acyl sulphonamide based quinoxalinones as multifunctional aldose reductase inhibitors
|
Ji, Yunpeng
|
|
|
27 |
8 |
p. 1658-1669
|
artikel
|
| 4 |
Design, synthesis and activity evaluation of indole-based double – Branched HDAC1 inhibitors
|
Zhang, Qiuqiong
|
|
|
27 |
8 |
p. 1595-1604
|
artikel
|
| 5 |
Design, synthesis and biological evaluation of 2,5-dimethylfuran-3-carboxylic acid derivatives as potential IDO1 inhibitors
|
Yang, Xiaojun
|
|
|
27 |
8 |
p. 1605-1618
|
artikel
|
| 6 |
Discovery and development of novel rhodanine derivatives targeting enoyl-acyl carrier protein reductase
|
Xu, Jian-Fei
|
|
|
27 |
8 |
p. 1509-1516
|
artikel
|
| 7 |
Discovery of new ureido benzenesulfonamides incorporating 1,3,5-triazine moieties as carbonic anhydrase I, II, IX and XII inhibitors
|
Lolak, Nabih
|
|
|
27 |
8 |
p. 1588-1594
|
artikel
|
| 8 |
Discovery of novel selective Janus kinase 2 (JAK2) inhibitors bearing a 1H-pyrazolo[3,4-d]pyrimidin-4-amino scaffold
|
Yin, Yuan
|
|
|
27 |
8 |
p. 1562-1576
|
artikel
|
| 9 |
Editorial Board
|
|
|
|
27 |
8 |
p. ii
|
artikel
|
| 10 |
Effective syntheses of 2′,4′-BNANC monomers bearing adenine, guanine, thymine, and 5-methylcytosine, and the properties of oligonucleotides fully modified with 2′,4′-BNANC
|
Fujisaka, Aki
|
|
|
27 |
8 |
p. 1728-1741
|
artikel
|
| 11 |
Essential structure of orexin 1 receptor antagonist YNT-707, part III: Role of the 14-hydroxy and the 3-methoxy groups in antagonistic activity toward the orexin 1 receptor in YNT-707 derivatives lacking the 4,5-epoxy ring
|
Yamamoto, Naoshi
|
|
|
27 |
8 |
p. 1747-1758
|
artikel
|
| 12 |
Glucose-conjugated platinum(IV) complexes as tumor-targeting agents: design, synthesis and biological evaluation
|
Wang, Haifeng
|
|
|
27 |
8 |
p. 1639-1645
|
artikel
|
| 13 |
Graphical abstract TOC
|
|
|
|
27 |
8 |
p. OBC
|
artikel
|
| 14 |
Graphical abstract TOC
|
|
|
|
27 |
8 |
p. I-VII
|
artikel
|
| 15 |
Graphical abstract TOC
|
|
|
|
27 |
8 |
p. IBC
|
artikel
|
| 16 |
8-Hydroxy-2-(1H-1,2,3-triazol-1-yl)-1,4-naphtoquinone derivatives inhibited P2X7 Receptor-Induced dye uptake into murine Macrophages
|
Pacheco, P.A.F.
|
|
|
27 |
8 |
p. 1449-1455
|
artikel
|
| 17 |
Inhibition of the FAD containing ER oxidoreductin 1 (Ero1) protein by EN-460 as a strategy for treatment of multiple myeloma
|
Hayes, Karen E.
|
|
|
27 |
8 |
p. 1479-1488
|
artikel
|
| 18 |
Lead optimization of selective tubulin inhibitors as anti-trypanosomal agents
|
Zhao, Anran
|
|
|
27 |
8 |
p. 1517-1528
|
artikel
|
| 19 |
Model studies for isolation of G-quadruplex-forming DNA sequences through a pull-down strategy with macrocyclic polyoxazole
|
Iida, Keisuke
|
|
|
27 |
8 |
p. 1742-1746
|
artikel
|
| 20 |
Molecular recognition of a branched peptide with HIV-1 Rev Response Element (RRE) RNA
|
Dai, Yumin
|
|
|
27 |
8 |
p. 1759-1765
|
artikel
|
| 21 |
N-Acyl pyrazoles: Effective and tunable inhibitors of serine hydrolases
|
Otrubova, Katerina
|
|
|
27 |
8 |
p. 1693-1703
|
artikel
|
| 22 |
Novel nonapeptide GLP (28–36) amide derivatives with improved hypoglycemic and body weight lowering effects
|
Li, Leyao
|
|
|
27 |
8 |
p. 1670-1676
|
artikel
|
| 23 |
Raloxifene-encapsulated hyaluronic acid-decorated chitosan nanoparticles selectively induce apoptosis in lung cancer cells
|
Almutairi, Fahad M.
|
|
|
27 |
8 |
p. 1629-1638
|
artikel
|
| 24 |
Small structural alterations greatly influence the membrane affinity of lipophilic ligands: Membrane interactions of bafilomycin A1 and its desmethyl derivative bearing 19F-labeling
|
Hayashi, Tatsuru
|
|
|
27 |
8 |
p. 1677-1682
|
artikel
|
| 25 |
Structural requirement of tunicamycin V for MraY inhibition
|
Yamamoto, Kazuki
|
|
|
27 |
8 |
p. 1714-1719
|
artikel
|
| 26 |
Structure-based design and synthesis of pyrimidine-4,6-diamine derivatives as Janus kinase 3 inhibitors
|
Yu, Ru-Nan
|
|
|
27 |
8 |
p. 1646-1657
|
artikel
|
| 27 |
Synthesis and biological evaluation of novel cYY analogues targeting Mycobacterium tuberculosis CYP121A1
|
Kishk, Safaa M.
|
|
|
27 |
8 |
p. 1546-1561
|
artikel
|
| 28 |
Synthesis and biological evaluation of solubilized sulfonamide analogues of the phosphatidylinositol 3-kinase inhibitor ZSTK474
|
Giddens, Anna C.
|
|
|
27 |
8 |
p. 1529-1545
|
artikel
|
| 29 |
Synthesis and pharmacological evaluation of novel arylpiperazine oxicams derivatives as potent analgesics without ulcerogenicity
|
Szczęśniak-Sięga, Berenika M.
|
|
|
27 |
8 |
p. 1619-1628
|
artikel
|
| 30 |
Synthesis and radical-scavenging activity of C-methylated fisetin analogues
|
Imai, Kohei
|
|
|
27 |
8 |
p. 1720-1727
|
artikel
|
| 31 |
Synthesis and structure–activity relationships of pyrazine-2-carboxamide derivatives as novel echinoderm microtubule-associated protein-like 4 (EML4)–anaplastic lymphoma kinase (ALK) inhibitors
|
Iikubo, Kazuhiko
|
|
|
27 |
8 |
p. 1683-1692
|
artikel
|
| 32 |
The design of 1,4-naphthoquinone derivatives and mechanisms underlying apoptosis induction through ROS-dependent MAPK/Akt/STAT3 pathways in human lung cancer cells
|
Zhang, Yi
|
|
|
27 |
8 |
p. 1577-1587
|
artikel
|
| 33 |
The discovery of quinoline-3-carboxamides as hematopoietic prostaglandin D synthase (H-PGDS) inhibitors
|
Deaton, David N.
|
|
|
27 |
8 |
p. 1456-1478
|
artikel
|
| 34 |
The impact of binding site waters on the activity/selectivity trade-off of Janus kinase 2 (JAK2) inhibitors
|
Egyed, Attila
|
|
|
27 |
8 |
p. 1497-1508
|
artikel
|
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