| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Anti-proliferative activity and structure-activity relationship of honokiol derivatives
|
Lin, Ding
|
|
2019
|
27 |
16 |
p. 3729-3734
|
artikel
|
| 2 |
2-Aryladenine derivatives as a potent scaffold for A1, A3 and dual A1/A3 adenosine receptor antagonists: Synthesis and structure-activity relationships
|
Areias, Filipe
|
|
2019
|
27 |
16 |
p. 3551-3558
|
artikel
|
| 3 |
Biological evaluation of molecules of the azaBINOL class as antiviral agents: Inhibition of HIV-1 RNase H activity by 7-isopropoxy-8-(naphth-1-yl)quinoline
|
Overacker, Ross D.
|
|
2019
|
27 |
16 |
p. 3595-3604
|
artikel
|
| 4 |
2-(Bipiperidin-1-yl)-5-(nitroaryl)-1,3,4-thiadiazoles: Synthesis, evaluation of in vitro leishmanicidal activity, and mechanism of action
|
Mojallal-Tabatabaei, Zahra
|
|
2019
|
27 |
16 |
p. 3682-3691
|
artikel
|
| 5 |
Design, synthesis, and evaluation of novel N-(4-phenoxybenzyl)aniline derivatives targeting acetylcholinesterase, β-amyloid aggregation and oxidative stress to treat Alzheimer’s disease
|
Srivastava, Pavan
|
|
2019
|
27 |
16 |
p. 3650-3662
|
artikel
|
| 6 |
Design, synthesis, and in vitro bioactivity evaluation of fluorine-containing analogues for sphingosine-1-phosphate 2 receptor
|
Luo, Zonghua
|
|
2019
|
27 |
16 |
p. 3619-3631
|
artikel
|
| 7 |
Development of novel lithocholic acid derivatives as vitamin D receptor agonists
|
Masuno, Hiroyuki
|
|
2019
|
27 |
16 |
p. 3674-3681
|
artikel
|
| 8 |
Editorial Board
|
|
|
2019
|
27 |
16 |
p. ii
|
artikel
|
| 9 |
18F-labeled benzimidazopyridine derivatives for PET imaging of tau pathology in Alzheimer’s disease
|
Kaide, Sho
|
|
2019
|
27 |
16 |
p. 3587-3594
|
artikel
|
| 10 |
Functionalized 6-(piperidin-1-yl)-8,9-diphenyl purines as inverse agonists of the CB1 receptor – SAR efforts towards selectivity and peripheralization
|
Amato, George
|
|
2019
|
27 |
16 |
p. 3632-3649
|
artikel
|
| 11 |
Graphical abstract TOC
|
|
|
2019
|
27 |
16 |
p. IBC
|
artikel
|
| 12 |
Graphical abstract TOC
|
|
|
2019
|
27 |
16 |
p. I-V
|
artikel
|
| 13 |
Graphical abstract TOC
|
|
|
2019
|
27 |
16 |
p. OBC
|
artikel
|
| 14 |
Green synthesis, biological evaluation, molecular docking studies and 3D-QSAR analysis of novel phenylalanine linked quinazoline-4(3H)-one-sulphonamide hybrid entities distorting the malarial reductase activity in folate pathway
|
Patel, Tarosh S.
|
|
2019
|
27 |
16 |
p. 3574-3586
|
artikel
|
| 15 |
Introducing a new category of activity cliffs with chemical modifications at multiple sites and rationalizing contributions of individual substitutions
|
Stumpfe, Dagmar
|
|
2019
|
27 |
16 |
p. 3605-3612
|
artikel
|
| 16 |
Melanogenic inhibitory effects of Triangularin in B16F0 melanoma cells, in vitro and molecular docking studies
|
Santi, María D.
|
|
2019
|
27 |
16 |
p. 3722-3728
|
artikel
|
| 17 |
Modification of the 4-phenylbutyl side chain of potent 3-benzazepine-based GluN2B receptor antagonists
|
Wagner, Marina
|
|
2019
|
27 |
16 |
p. 3559-3567
|
artikel
|
| 18 |
New insights into the binding mode of pyridine-3-carboxamide inhibitors of E. coli DNA gyrase
|
Narramore, Sarah
|
|
2019
|
27 |
16 |
p. 3546-3550
|
artikel
|
| 19 |
Radiosynthesis and evaluation of a novel monoacylglycerol lipase radiotracer: 1,1,1,3,3,3-hexafluoropropan-2-yl-3-(1-benzyl-1H-pyrazol-3-yl)azetidine-1-[11C]carboxylate
|
Mori, Wakana
|
|
2019
|
27 |
16 |
p. 3568-3573
|
artikel
|
| 20 |
Rational approaches, design strategies, structure activity relationship and mechanistic insights for therapeutic coumarin hybrids
|
Singh, Harbinder
|
|
2019
|
27 |
16 |
p. 3477-3510
|
artikel
|
| 21 |
Small molecule inhibition of microRNA-21 expression reduces cell viability and microtumor formation
|
Ankenbruck, Nicholas
|
|
2019
|
27 |
16 |
p. 3735-3743
|
artikel
|
| 22 |
Synthesis and biological evaluation of 1-alkylaminomethyl-1,1-bisphosphonic acids against Trypanosoma cruzi and Toxoplasma gondii
|
Galaka, Tamila
|
|
2019
|
27 |
16 |
p. 3663-3673
|
artikel
|
| 23 |
Synthesis of an amphiphilic tetrazine derivative and its application as a liposomal component to accelerate release of encapsulated drugs
|
Kannaka, Kento
|
|
2019
|
27 |
16 |
p. 3613-3618
|
artikel
|
| 24 |
Synthesis, pharmacological evaluation, and mechanistic study of adefovir mixed phosphonate derivatives bearing cholic acid and l-amino acid moieties for the treatment of HBV
|
Li, Tao
|
|
2019
|
27 |
16 |
p. 3707-3721
|
artikel
|
| 25 |
Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors
|
Chino, Ayaka
|
|
2019
|
27 |
16 |
p. 3692-3706
|
artikel
|
| 26 |
The synthesis and evaluation of quinolinequinones as anti-mycobacterial agents
|
Santoso, Kristiana T.
|
|
2019
|
27 |
16 |
p. 3532-3545
|
artikel
|
| 27 |
1,2,3-Triazole-containing hybrids as leads in medicinal chemistry: A recent overview
|
Bozorov, Khurshed
|
|
2019
|
27 |
16 |
p. 3511-3531
|
artikel
|
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