| no |
title |
author |
magazine |
year |
volume |
issue |
page(s) |
type |
| 1 |
Advances in the structural studies of antibiotic potentiators against Escherichia coli
|
Blankson, Gifty A.
|
|
2019
|
27 |
15 |
p. 3254-3278
|
article
|
| 2 |
Anti-atherosclerosis effect of H2S donors based on nicotinic acid and chlorfibrate structures
|
Bai, Zhongjie
|
|
2019
|
27 |
15 |
p. 3307-3318
|
article
|
| 3 |
Bypassing lantibiotic resistance by an effective nisin derivative
|
Zaschke-Kriesche, Julia
|
|
2019
|
27 |
15 |
p. 3454-3462
|
article
|
| 4 |
Chemical modification-mediated optimisation of bronchodilatory activity of mepenzolate, a muscarinic receptor antagonist with anti-inflammatory activity
|
Yamashita, Yasunobu
|
|
2019
|
27 |
15 |
p. 3339-3346
|
article
|
| 5 |
Designed P-glycoprotein inhibitors with triazol-tetrahydroisoquinoline-core increase doxorubicin-induced mortality in multidrug resistant K562/A02 cells
|
Kairuki, Mutta
|
|
2019
|
27 |
15 |
p. 3347-3357
|
article
|
| 6 |
Design, synthesis and biological evaluation of novel 2,3-indolinedione derivatives against mantle cell lymphoma
|
Yu, Shengping
|
|
2019
|
27 |
15 |
p. 3319-3327
|
article
|
| 7 |
Design, synthesis and fungicidal activity evaluation of novel pyrimidinamine derivatives containing phenyl-thiazole/oxazole moiety
|
Yan, Zhongzhong
|
|
2019
|
27 |
15 |
p. 3218-3228
|
article
|
| 8 |
Design, synthesis and molecular modelling of new bulky Fananserin derivatives with altered pharmacological profile as potential antidepressants
|
Zaręba, Przemysław
|
|
2019
|
27 |
15 |
p. 3396-3407
|
article
|
| 9 |
Discovery and Biological evaluation of pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-dione derivatives as potent Bruton’s tyrosine kinase inhibitors
|
Diao, Yanyan
|
|
2019
|
27 |
15 |
p. 3390-3395
|
article
|
| 10 |
Discovery and development of DNA polymerase IIIC inhibitors to treat Gram-positive infections
|
Xu, Wei-Chu
|
|
2019
|
27 |
15 |
p. 3209-3217
|
article
|
| 11 |
Discovery of a pyrazolo[1,5-a]pyrimidine derivative (MT-3014) as a highly selective PDE10A inhibitor via core structure transformation from the stilbene moiety
|
Koizumi, Yuuki
|
|
2019
|
27 |
15 |
p. 3440-3450
|
article
|
| 12 |
Discovery of DC_H31 as potential mutant IDH1 inhibitor through NADPH-based high throughput screening
|
Duan, Zhe
|
|
2019
|
27 |
15 |
p. 3229-3236
|
article
|
| 13 |
Editorial Board
|
|
|
2019
|
27 |
15 |
p. ii
|
article
|
| 14 |
Expanding chemogenomic space using chemoproteomics
|
Jones, Lyn H.
|
|
2019
|
27 |
15 |
p. 3451-3453
|
article
|
| 15 |
Graphical abstract TOC
|
|
|
2019
|
27 |
15 |
p. I-VII
|
article
|
| 16 |
Graphical abstract TOC
|
|
|
2019
|
27 |
15 |
p. IBC
|
article
|
| 17 |
Graphical abstract TOC
|
|
|
2019
|
27 |
15 |
p. OBC
|
article
|
| 18 |
Highly diverse cembranoids from the South China Sea soft coral Sinularia scabra as a new class of potential immunosuppressive agents
|
Yang, Min
|
|
2019
|
27 |
15 |
p. 3469-3476
|
article
|
| 19 |
Identification of topoisomerases as molecular targets of cytosporolide C and its analog
|
Otake, Keisuke
|
|
2019
|
27 |
15 |
p. 3334-3338
|
article
|
| 20 |
Inhibition of polypeptide N-acetyl-α-galactosaminyltransferases is an underlying mechanism of dietary polyphenols preventing colorectal tumorigenesis
|
Liu, Feng
|
|
2019
|
27 |
15 |
p. 3372-3382
|
article
|
| 21 |
Multicomponent synthesis of α-acylamino and α-acyloxy amide derivatives of desmycosin and their activity against gram-negative bacteria
|
Budragchaa, Tuvshinjargal
|
|
2019
|
27 |
15 |
p. 3237-3247
|
article
|
| 22 |
New sensible method to quantize the intestinal absorption of receptor ligands
|
Buccioni, Michela
|
|
2019
|
27 |
15 |
p. 3328-3333
|
article
|
| 23 |
Novel meriolin derivatives as rapid apoptosis inducers
|
Drießen, Daniel
|
|
2019
|
27 |
15 |
p. 3463-3468
|
article
|
| 24 |
Opportunities and challenges for the development of covalent chemical immunomodulators
|
Backus, Keriann M.
|
|
2019
|
27 |
15 |
p. 3421-3439
|
article
|
| 25 |
Polybenzyls from Gastrodia elata, their agonistic effects on melatonin receptors and structure-activity relationships
|
Chen, Si-Yue
|
|
2019
|
27 |
15 |
p. 3299-3306
|
article
|
| 26 |
Structure-activity relationship study of thiazolyl-hydroxamate derivatives as selective histone deacetylase 6 inhibitors
|
Nam, Gibeom
|
|
2019
|
27 |
15 |
p. 3408-3420
|
article
|
| 27 |
Synthesis and bioactivity of 1,3-thiazolidine-2-thione derivatives against type III secretion system of Xanthomonas oryzae
|
Tao, Hui
|
|
2019
|
27 |
15 |
p. 3364-3371
|
article
|
| 28 |
Synthesis and biological evaluation of glucose conjugated phthalocyanine as a second-generation photosensitizer
|
Uruma, Yoshiyuki
|
|
2019
|
27 |
15 |
p. 3279-3284
|
article
|
| 29 |
Synthesis and in vitro cytotoxicity evaluation of β-carboline-combretastatin carboxamides as apoptosis inducing agents: DNA intercalation and topoisomerase-II inhibition
|
Jadala, Chetna
|
|
2019
|
27 |
15 |
p. 3285-3298
|
article
|
| 30 |
Synthesis and molecular modeling of novel non-sulfonylureas as hypoglycemic agents and selective ALR2 inhibitors
|
Salem, Manar G.
|
|
2019
|
27 |
15 |
p. 3383-3389
|
article
|
| 31 |
Synthesis and preliminary in vitro evaluation of DOTA-Tenatumomab conjugates for theranostic applications in tenascin expressing tumors
|
Giannini, Giuseppe
|
|
2019
|
27 |
15 |
p. 3248-3253
|
article
|
| 32 |
Synthesis of oxytocin derivatives lipidated via a carbonate or carbamate linkage as a long-acting therapeutic agent for social impairment-like behaviors
|
Cherepanov, Stanislav M.
|
|
2019
|
27 |
15 |
p. 3358-3363
|
article
|
Journal description