no |
title |
author |
magazine |
year |
volume |
issue |
page(s) |
type |
1 |
Activation studies with amines and amino acids of the α-carbonic anhydrase from the pathogenic protozoan Trypanosoma cruzi
|
Angeli, Andrea |
|
|
26 |
14 |
p. 4187-4190 |
article |
2 |
Activity of steroid 4 and derivatives 4a–4f as inhibitors of the enzyme 5α-reductase 1
|
Arellano, Yazmín |
|
|
26 |
14 |
p. 4058-4064 |
article |
3 |
Anti-acute myeloid leukemia activity of 2-chloro-3-alkyl-1,4-naphthoquinone derivatives through inducing mtDNA damage and GSH depletion
|
Li, Kun |
|
|
26 |
14 |
p. 4191-4200 |
article |
4 |
A short synthesis of Dronedarone
|
Piotrkowska, Barbara |
|
|
26 |
14 |
p. 4330-4335 |
article |
5 |
Corrigendum to “Exploration of multi-target potential of chromen-4-one based compounds in Alzheimer’s disease: Design, synthesis and biological evaluations” [Bioorg. Med. Chem. 25 (2017) 6273–6285]
|
Singh, Manjinder |
|
|
26 |
14 |
p. 4360-4361 |
article |
6 |
Curcumin derivatives and Aβ-fibrillar aggregates: An interactions’ study for diagnostic/therapeutic purposes in neurodegenerative diseases
|
Orteca, Giulia |
|
|
26 |
14 |
p. 4288-4300 |
article |
7 |
Design and biological evaluation of novel hybrids of 1, 5-diarylpyrazole and Chrysin for selective COX-2 inhibition
|
Ren, Shen-Zhen |
|
|
26 |
14 |
p. 4264-4275 |
article |
8 |
Design and synthesis of alkyl substituted pyridino[2,3-D]pyrimidine compounds as PI3Kα/mTOR dual inhibitors with improved pharmacokinetic properties and potent in vivo antitumor activity
|
Liu, Yinyin |
|
|
26 |
14 |
p. 3992-4000 |
article |
9 |
Design and synthesis of novel pyrimido[5,4-d]pyrimidine derivatives as GPR119 agonist for treatment of type 2 diabetes
|
Fang, Yuanying |
|
|
26 |
14 |
p. 4080-4087 |
article |
10 |
Design, synthesis and anticancer evaluation of acridine hydroxamic acid derivatives as dual Topo and HDAC inhibitors
|
Chen, Jiwei |
|
|
26 |
14 |
p. 3958-3966 |
article |
11 |
Design, synthesis and biological evaluation of nitric oxide releasing derivatives of dapagliflozin as potential anti-diabetic and anti-thrombotic agents
|
Li, Zheng |
|
|
26 |
14 |
p. 3947-3952 |
article |
12 |
Design, synthesis, and biological evaluation of novel oxadiazole- and thiazole-based histamine H3R ligands
|
Khanfar, Mohammad A. |
|
|
26 |
14 |
p. 4034-4046 |
article |
13 |
Design, synthesis and biological evaluation of novel series of 2H-benzo[b][1,4]oxazin-3(4H)-one and 2H-benzo[b][1,4]oxazine scaffold derivatives as PI3Kα inhibitors
|
Dong, Fu-Dan |
|
|
26 |
14 |
p. 3982-3991 |
article |
14 |
Design, synthesis and biological evaluation of novel spiro-pentacylamides as acetyl-CoA carboxylase inhibitors
|
Wei, Qiangqiang |
|
|
26 |
14 |
p. 3866-3874 |
article |
15 |
Design, synthesis and biological evaluation of piperazino-enaminones as novel suppressants of pro-Inflammatory cytokines
|
Ghoneim, Ola M. |
|
|
26 |
14 |
p. 3890-3898 |
article |
16 |
Design, synthesis and docking study of 4-arylpiperazine carboxamides as monoamine neurotransmitters reuptake inhibitors
|
Paudel, Suresh |
|
|
26 |
14 |
p. 4127-4135 |
article |
17 |
Design, synthesis, and evaluation of novel l-phenylglycine derivatives as potential PPARγ lead compounds
|
Liu, Jinyu |
|
|
26 |
14 |
p. 4153-4167 |
article |
18 |
Design, synthesis and evaluation of novel sophoridinic imine derivatives containing conjugated planar structure as potent anticancer agents
|
Xu, Yiming |
|
|
26 |
14 |
p. 4136-4144 |
article |
19 |
Design, synthesis and pharmacology of aortic-selective acyl-CoA: Cholesterol O-acyltransferase (ACAT/SOAT) inhibitors
|
Shibuya, Kimiyuki |
|
|
26 |
14 |
p. 4001-4013 |
article |
20 |
Design, synthesis, in vitro and in vivo evaluation, and structure-activity relationship (SAR) discussion of novel dipeptidyl boronic acid proteasome inhibitors as orally available anti-cancer agents for the treatment of multiple myeloma and mechanism studies
|
Lei, Meng |
|
|
26 |
14 |
p. 3975-3981 |
article |
21 |
Development of efficient one-pot three-component assembly of trityl olmesartan medoxomil
|
Toplak Časar, Renata |
|
|
26 |
14 |
p. 4348-4359 |
article |
22 |
Discovery of novel leucyladenylate sulfamate surrogates as leucyl-tRNA synthetase (LRS)-targeted mammalian target of rapamycin complex 1 (mTORC1) inhibitors
|
Yoon, Suyoung |
|
|
26 |
14 |
p. 4073-4079 |
article |
23 |
Editorial Board
|
|
|
|
26 |
14 |
p. ii |
article |
24 |
Facile construction of fused benzimidazole-isoquinolinones that induce cell-cycle arrest and apoptosis in colorectal cancer cells
|
He, Liu-Jun |
|
|
26 |
14 |
p. 3899-3908 |
article |
25 |
Forewords BMC
|
Gallou, Fabrice |
|
|
26 |
14 |
p. 4329 |
article |
26 |
Graphical abstract TOC
|
|
|
|
26 |
14 |
p. IBC |
article |
27 |
Graphical abstract TOC
|
|
|
|
26 |
14 |
p. I-XII |
article |
28 |
Graphical abstract TOC
|
|
|
|
26 |
14 |
p. OBC |
article |
29 |
Identification by Inverse Virtual Screening of magnolol-based scaffold as new tankyrase-2 inhibitors
|
Di Micco, Simone |
|
|
26 |
14 |
p. 3953-3957 |
article |
30 |
Identification of natural product compounds as quorum sensing inhibitors in Pseudomonas fluorescens P07 through virtual screening
|
Ding, Ting |
|
|
26 |
14 |
p. 4088-4099 |
article |
31 |
Identification of PKMYT1 inhibitors by screening the GSK published protein kinase inhibitor set I and II
|
Platzer, Charlott |
|
|
26 |
14 |
p. 4014-4024 |
article |
32 |
Indenone derivatives as inhibitor of human DNA dealkylation repair enzyme AlkBH3
|
Nigam, Richa |
|
|
26 |
14 |
p. 4100-4112 |
article |
33 |
Mechanism underlying inhibitory effect of six dicaffeoylquinic acid isomers on melanogenesis and the computational molecular modeling studies
|
Ha, Ji Hoon |
|
|
26 |
14 |
p. 4201-4208 |
article |
34 |
7β-Methyl substituent is a structural locus associated with activity cliff for nepenthone analogues
|
Sun, Hui-jiao |
|
|
26 |
14 |
p. 4254-4263 |
article |
35 |
Novel amino acid-substituted diphenylpyrimidine derivatives as potent BTK inhibitors against B cell lymphoma cell lines
|
Wang, Changyuan |
|
|
26 |
14 |
p. 4179-4186 |
article |
36 |
Optimization and in vivo evaluation of pyrazolopyridines as a potent and selective PI3Kδ inhibitor
|
Hamajima, Toshihiro |
|
|
26 |
14 |
p. 3917-3924 |
article |
37 |
Quinoxaline derivatives as potential antitrypanosomal and antileishmanial agents
|
Cogo, Juliana |
|
|
26 |
14 |
p. 4065-4072 |
article |
38 |
Rational design of novel irreversible inhibitors for human arginase
|
Guo, Xuefeng |
|
|
26 |
14 |
p. 3939-3946 |
article |
39 |
Regio- and stereospecific synthesis of rac-carbasugar-based cyclohexane pentols; Investigations of their α- and β-glucosidase inhibitions
|
Karakılıç, Emel |
|
|
26 |
14 |
p. 4276-4287 |
article |
40 |
Route design, the foundation of successful chemical development
|
Cornwall, Philip |
|
|
26 |
14 |
p. 4336-4347 |
article |
41 |
Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs
|
Tber, Zahira |
|
|
26 |
14 |
p. 4310-4319 |
article |
42 |
Senolytic activity of piperlongumine analogues: Synthesis and biological evaluation
|
Liu, Xingui |
|
|
26 |
14 |
p. 3925-3938 |
article |
43 |
SIRT4 is the last puzzle of mitochondrial sirtuins
|
Li, Yan |
|
|
26 |
14 |
p. 3861-3865 |
article |
44 |
Small molecule scaffolds that disrupt the Rev1-CT/RIR protein-protein interaction
|
Ozen, Zuleyha |
|
|
26 |
14 |
p. 4301-4309 |
article |
45 |
Stereospecific reduction of the butenolide in strigolactones in plants
|
Yamauchi, Misa |
|
|
26 |
14 |
p. 4225-4233 |
article |
46 |
Structural optimization and in vitro profiling of N-phenylbenzamide-based farnesoid X receptor antagonists
|
Schmidt, Jurema |
|
|
26 |
14 |
p. 4240-4253 |
article |
47 |
Synthesis and anticancer activity of novel bisindolylhydroxymaleimide derivatives with potent GSK-3 kinase inhibition
|
Winfield, Hannah J. |
|
|
26 |
14 |
p. 4209-4224 |
article |
48 |
Synthesis and antitumor activity of bis(hydroxymethyl)propionate analogs of pterostilbene in cisplatin-resistant human oral cancer cells
|
Hsieh, Min-Tsang |
|
|
26 |
14 |
p. 3909-3916 |
article |
49 |
Synthesis and biological properties of aryl methyl sulfones
|
Navarro, Lorena |
|
|
26 |
14 |
p. 4113-4126 |
article |
50 |
Synthesis and characterization of some atypical sphingoid bases
|
Saied, Essa M. |
|
|
26 |
14 |
p. 4047-4057 |
article |
51 |
Synthesis and hybridizing properties of isoDNAs including 3′-O,4′-C-ethyleneoxy-bridged 5-methyluridine derivatives
|
Osawa, Takashi |
|
|
26 |
14 |
p. 3875-3881 |
article |
52 |
Synthesis and pharmacological evaluation of pyrazolo[4,3-c]quinolinones as high affinity GABAA-R ligands and potential anxiolytics
|
López Rivilli, Marisa J. |
|
|
26 |
14 |
p. 3967-3974 |
article |
53 |
Synthesis, antitumor activity evaluation and mechanistic study of novel hederacolchiside A1 derivatives bearing an aryl triazole moiety
|
Li, Hui-ning |
|
|
26 |
14 |
p. 4025-4033 |
article |
54 |
Synthetic molecules for disruption of the MYC protein-protein interface
|
Jacob, Nicholas T. |
|
|
26 |
14 |
p. 4234-4239 |
article |
55 |
Terpenoids with vasorelaxant effects from the Chinese liverwort Scapania carinthiaca
|
Qiao, Yanan |
|
|
26 |
14 |
p. 4320-4328 |
article |
56 |
The genome-wide sequence specificity of DNA cleavage by bleomycin analogues in human cells
|
Murray, Vincent |
|
|
26 |
14 |
p. 4168-4178 |
article |
57 |
The synthesis and evaluation of phenoxyacylhydroxamic acids as potential agents for Helicobacter pylori infections
|
Ni, Wei-Wei |
|
|
26 |
14 |
p. 4145-4152 |
article |
58 |
The tyrosinase inhibitory effects of isoxazolone derivatives with a (Z)-β-phenyl-α, β-unsaturated carbonyl scaffold
|
Kim, Su Jeong |
|
|
26 |
14 |
p. 3882-3889 |
article |