| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
An epigenetic modifier induces production of (10′S)-verruculide B, an inhibitor of protein tyrosine phosphatases by Phoma sp. nov. LG0217, a fungal endophyte of Parkinsonia microphylla
|
Gubiani, Juliana R.
|
|
2017
|
25 |
6 |
p. 1860-1866
7 p.
|
artikel
|
| 2 |
An in-tether sulfoxide chiral center influences the biophysical properties of the N-capped peptides
|
Li, Jingxu
|
|
2017
|
25 |
6 |
p. 1756-1761
6 p.
|
artikel
|
| 3 |
Antimicrobial activity of rhodanine-3-acetic acid derivatives
|
Krátký, Martin
|
|
2017
|
25 |
6 |
p. 1839-1845
7 p.
|
artikel
|
| 4 |
Benzimidazole inhibitors from the Niclosamide chemotype inhibit Wnt/β-catenin signaling with selectivity over effects on ATP homeostasis
|
Mook Jr., Robert A.
|
|
2017
|
25 |
6 |
p. 1804-1816
13 p.
|
artikel
|
| 5 |
Comparison of the anion inhibition profiles of the β- and γ-carbonic anhydrases from the pathogenic bacterium Burkholderia pseudomallei
|
Del Prete, Sonia
|
|
2017
|
25 |
6 |
p. 2010-2015
6 p.
|
artikel
|
| 6 |
Construction of a library of structurally diverse ribonucleopeptides with catalytic groups
|
Tamura, Tomoki
|
|
2017
|
25 |
6 |
p. 1881-1888
8 p.
|
artikel
|
| 7 |
Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A1 receptor antagonists and their biological evaluation
|
Koul, Summon
|
|
2017
|
25 |
6 |
p. 1963-1975
13 p.
|
artikel
|
| 8 |
Design, synthesis and biological evaluation of 2,4-disubstituted oxazole derivatives as potential PDE4 inhibitors
|
Li, Ya-Sheng
|
|
2017
|
25 |
6 |
p. 1852-1859
8 p.
|
artikel
|
| 9 |
Design, synthesis and preliminary biological evaluation of indole-3-carboxylic acid-based skeleton of Bcl-2/Mcl-1 dual inhibitors
|
Liu, Tingting
|
|
2017
|
25 |
6 |
p. 1939-1948
10 p.
|
artikel
|
| 10 |
Development of helix-stabilized cell-penetrating peptides containing cationic α,α-disubstituted amino acids as helical promoters
|
Yamashita, Hiroko
|
|
2017
|
25 |
6 |
p. 1846-1851
6 p.
|
artikel
|
| 11 |
Discovery and dimeric approach of novel Natriuretic Peptide Receptor A (NPR-A) agonists
|
Iwaki, Takehiko
|
|
2017
|
25 |
6 |
p. 1762-1769
8 p.
|
artikel
|
| 12 |
Discovery and optimization of benzimidazole derivatives as a novel chemotype of farnesoid X receptor (FXR) antagonists
|
Teno, Naoki
|
|
2017
|
25 |
6 |
p. 1787-1794
8 p.
|
artikel
|
| 13 |
Editorial board
|
|
|
2017
|
25 |
6 |
p. IFC-
1 p.
|
artikel
|
| 14 |
5-Ethynylarylnaphthalimides as antitumor agents: Synthesis and biological evaluation
|
Quintana-Espinoza, Patricia
|
|
2017
|
25 |
6 |
p. 1976-1983
8 p.
|
artikel
|
| 15 |
Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds
|
Krasavin, Mikhail
|
|
2017
|
25 |
6 |
p. 1914-1925
12 p.
|
artikel
|
| 16 |
Iminosugar-based ceramide mimicry for the design of new CERT START domain ligands
|
Santos, Cécile
|
|
2017
|
25 |
6 |
p. 1984-1989
6 p.
|
artikel
|
| 17 |
Incorporation of arginine mimetic residue into peptides for recognition of double stranded nucleic acid structure: Binding and aggregation studies
|
Li, Mao
|
|
2017
|
25 |
6 |
p. 1875-1880
6 p.
|
artikel
|
| 18 |
In vitro anticancer activity evaluation of new cationic platinum(II) complexes based on imidazole moiety
|
Rimoldi, Isabella
|
|
2017
|
25 |
6 |
p. 1907-1913
7 p.
|
artikel
|
| 19 |
In vivo instability of platensimycin and platencin: Synthesis and biological evaluation of urea- and carbamate-platensimycin
|
Dong, Liao-Bin
|
|
2017
|
25 |
6 |
p. 1990-1996
7 p.
|
artikel
|
| 20 |
Mechanisms of action and structure-activity relationships of cytotoxic flavokawain derivatives
|
Thieury, Charlotte
|
|
2017
|
25 |
6 |
p. 1817-1829
13 p.
|
artikel
|
| 21 |
Multifunctional thioxanthone derivatives with acetylcholinesterase, monoamine oxidases and β-amyloid aggregation inhibitory activities as potential agents against Alzheimer’s disease
|
Luo, Li
|
|
2017
|
25 |
6 |
p. 1997-2009
13 p.
|
artikel
|
| 22 |
Mycobacterium tuberculosis chorismate mutase: A potential target for TB
|
Khanapur, Manjulatha
|
|
2017
|
25 |
6 |
p. 1725-1736
12 p.
|
artikel
|
| 23 |
New nitrofurans amenable by isocyanide multicomponent chemistry are active against multidrug-resistant and poly-resistant Mycobacterium tuberculosis
|
Krasavin, Mikhail
|
|
2017
|
25 |
6 |
p. 1867-1874
8 p.
|
artikel
|
| 24 |
Novel 6-methoxycarbonyl indolinones bearing a pyrrole Mannich base moiety as angiokinase inhibitors
|
Qin, Mingze
|
|
2017
|
25 |
6 |
p. 1778-1786
9 p.
|
artikel
|
| 25 |
Piperazines as nootropic agents: New derivatives of the potent cognition-enhancer DM235 carrying hydrophilic substituents
|
Martino, Maria Vittoria
|
|
2017
|
25 |
6 |
p. 1795-1803
9 p.
|
artikel
|
| 26 |
Syntheses and mucosal adjuvant activity of simplified oleanolic acid saponins possessing cinnamoyl ester
|
Shirahata, Tatsuya
|
|
2017
|
25 |
6 |
p. 1747-1755
9 p.
|
artikel
|
| 27 |
Synthesis and biological evaluation of novel N3-substituted dihydropyrimidine derivatives as T-type calcium channel blockers and their efficacy as analgesics in mouse models of inflammatory pain
|
Teleb, Mohamed
|
|
2017
|
25 |
6 |
p. 1926-1938
13 p.
|
artikel
|
| 28 |
Synthesis and biological evaluation of potential inhibitors of the cysteine proteases cruzain and rhodesain designed by molecular simplification
|
Braga, Saulo Fehelberg Pinto
|
|
2017
|
25 |
6 |
p. 1889-1900
12 p.
|
artikel
|
| 29 |
Synthesis and evaluation of N-(benzofuran-5-yl)aromaticsulfonamide derivatives as novel HIF-1 inhibitors that possess anti-angiogenic potential
|
Wei, Jinlian
|
|
2017
|
25 |
6 |
p. 1737-1746
10 p.
|
artikel
|
| 30 |
Synthesis and pharmacological evaluation of pyrazolo[1,5-a]pyrimidin-7(4H)-one derivatives as potential GABAA-R ligands
|
Guerrini, Gabriella
|
|
2017
|
25 |
6 |
p. 1901-1906
6 p.
|
artikel
|
| 31 |
Synthesis of 1,3,5-trisubstituted pyrazolines as potential antimalarial and antimicrobial agents
|
Mishra, Vikash K.
|
|
2017
|
25 |
6 |
p. 1949-1962
14 p.
|
artikel
|
| 32 |
Synthetic analogs of rhamnolipids modulate structured biofilms formed by rhamnolipid-nonproducing mutant of Pseudomonas aeruginosa
|
Zheng, Hewen
|
|
2017
|
25 |
6 |
p. 1830-1838
9 p.
|
artikel
|
| 33 |
The role of cell cycle progression for the apoptosis of cancer cells induced by palladium(II)-saccharinate complexes of terpyridine
|
Kacar, Omer
|
|
2017
|
25 |
6 |
p. 1770-1777
8 p.
|
artikel
|
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