| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Activation of lysine-specific demethylase 1 inhibitor peptide by redox-controlled cleavage of a traceless linker
|
Amano, Yuichi
|
|
2017
|
25 |
3 |
p. 1227-1234
|
artikel
|
| 2 |
A one-pot laccase-catalysed synthesis of coumestan derivatives and their anticancer activity
|
Qwebani-Ogunleye, Tozama
|
|
2017
|
25 |
3 |
p. 1172-1182
|
artikel
|
| 3 |
Benzenesulfonamide bearing imidazothiadiazole and thiazolotriazole scaffolds as potent tumor associated human carbonic anhydrase IX and XII inhibitors
|
Kumar, Rajiv
|
|
2017
|
25 |
3 |
p. 1286-1293
|
artikel
|
| 4 |
Bifunctional conjugates with potent inhibitory activity towards cyclooxygenase and histone deacetylase
|
Raji, Idris
|
|
2017
|
25 |
3 |
p. 1202-1218
|
artikel
|
| 5 |
Construction of a 3D-shaped, natural product like fragment library by fragmentation and diversification of natural products
|
Prescher, Horst
|
|
2017
|
25 |
3 |
p. 921-925
|
artikel
|
| 6 |
Design and optimization of aspartate N-acetyltransferase inhibitors for the potential treatment of Canavan disease
|
Thangavelu, Bharani
|
|
2017
|
25 |
3 |
p. 870-885
|
artikel
|
| 7 |
Design and synthesis of new coumarin hybrids and insight into their mode of antiproliferative action
|
Elshemy, Heba A.H.
|
|
2017
|
25 |
3 |
p. 1066-1075
|
artikel
|
| 8 |
Design, synthesis and biological evaluation of 4′-aminochalcone-rivastigmine hybrids as multifunctional agents for the treatment of Alzheimer's disease
|
Xiao, Ganyuan
|
|
2017
|
25 |
3 |
p. 1030-1041
|
artikel
|
| 9 |
Design, synthesis and biological evaluation of 7-(aryl)-2,3-dihydro-[1,4]dioxino[2,3-g]quinoline derivatives as potential Hsp90 inhibitors and anticancer agents
|
Malayeri, Sina Omid
|
|
2017
|
25 |
3 |
p. 1294-1302
|
artikel
|
| 10 |
Design, synthesis and biological evaluation of (E)-3,4-dihydroxystyryl 4-acylaminophenethyl sulfone, sulfoxide derivatives as dual inhibitors of HIV-1 CCR5 and integrase
|
Sun, Yixing
|
|
2017
|
25 |
3 |
p. 1076-1084
|
artikel
|
| 11 |
Design, synthesis and biological evaluation of novel 4-(2-fluorophenoxy)quinoline derivatives as selective c-Met inhibitors
|
Wang, Xiaoqiang
|
|
2017
|
25 |
3 |
p. 886-896
|
artikel
|
| 12 |
Design, synthesis and in vitro biological evaluation of oligopeptides targeting E. coli type I signal peptidase (LepB)
|
De Rosa, Maria
|
|
2017
|
25 |
3 |
p. 897-911
|
artikel
|
| 13 |
Design, synthesis, in vitro characterization and preliminary imaging studies on fluorinated bile acid derivatives as PET tracers to study hepatic transporters
|
Testa, Andrea
|
|
2017
|
25 |
3 |
p. 963-976
|
artikel
|
| 14 |
Determination of binding modes and binding constants for the complexes of 6H-pyrido[4,3-b]carbazole derivatives with DNA
|
Shimazu, Akihito
|
|
2017
|
25 |
3 |
p. 1094-1112
|
artikel
|
| 15 |
Development of new inhibitors for N-acylethanolamine-hydrolyzing acid amidase as promising tool against bladder cancer
|
Vago, Riccardo
|
|
2017
|
25 |
3 |
p. 1242-1249
|
artikel
|
| 16 |
Development of new PTK7-targeting aptamer-fluorescent and -radiolabelled probes for evaluation as molecular imaging agents: Lymphoma and melanoma in vivo proof of concept
|
Calzada, Victoria
|
|
2017
|
25 |
3 |
p. 1163-1171
|
artikel
|
| 17 |
Development of radioiodinated acridine derivatives for in vivo imaging of prion deposits in the brain
|
Kawasaki, Masao
|
|
2017
|
25 |
3 |
p. 1085-1093
|
artikel
|
| 18 |
Discovery of hepatitis B virus capsid assembly inhibitors leading to a heteroaryldihydropyrimidine based clinical candidate (GLS4)
|
Ren, Qingyun
|
|
2017
|
25 |
3 |
p. 1042-1056
|
artikel
|
| 19 |
Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa
|
Vullo, Daniela
|
|
2017
|
25 |
3 |
p. 1260-1265
|
artikel
|
| 20 |
Editorial board
|
|
|
2017
|
25 |
3 |
p. IFC
|
artikel
|
| 21 |
1-Heteroarylpropan-2-ones as inhibitors of fatty acid amide hydrolase: Studies on structure-activity relationships and metabolic stability
|
Zahov, Stefan
|
|
2017
|
25 |
3 |
p. 825-837
|
artikel
|
| 22 |
Hetero-Diels-Alder approach to Bis(indolyl)methanes
|
Grosso, Carla
|
|
2017
|
25 |
3 |
p. 1122-1131
|
artikel
|
| 23 |
Highly predictive and interpretable models for PAMPA permeability
|
Sun, Hongmao
|
|
2017
|
25 |
3 |
p. 1266-1276
|
artikel
|
| 24 |
Identification of a melampomagnolide B analog as a potential lead molecule for treatment of acute myelogenous leukemia
|
Albayati, Zaineb A.F.
|
|
2017
|
25 |
3 |
p. 1235-1241
|
artikel
|
| 25 |
Lycopene pretreatment improves hepatotoxicity induced by acetaminophen in C57BL/6 mice
|
Bandeira, Ana Carla Balthar
|
|
2017
|
25 |
3 |
p. 1057-1065
|
artikel
|
| 26 |
Macrocyclic MEK1/2 inhibitor with efficacy in a mouse model of cardiomyopathy caused by lamin A/C gene mutation
|
Wu, Wei
|
|
2017
|
25 |
3 |
p. 1004-1013
|
artikel
|
| 27 |
Neuritogenic activity of bi-functional bis-tryptoline triazole
|
Jiaranaikulwanitch, Jutamas
|
|
2017
|
25 |
3 |
p. 1195-1201
|
artikel
|
| 28 |
New derivatives of 7-chloroquinolin-4-amine with antiprotozoal activity
|
Faist, Johanna
|
|
2017
|
25 |
3 |
p. 941-948
|
artikel
|
| 29 |
New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies
|
Intagliata, Sebastiano
|
|
2017
|
25 |
3 |
p. 1250-1259
|
artikel
|
| 30 |
Novel thrombopoietin mimetic peptides bind c-Mpl receptor: Synthesis, biological evaluation and molecular modeling
|
Liu, Yaquan
|
|
2017
|
25 |
3 |
p. 1113-1121
|
artikel
|
| 31 |
2-Oxoamides based on dipeptides as selective calcium-independent phospholipase A2 inhibitors
|
Smyrniotou, Anneta
|
|
2017
|
25 |
3 |
p. 926-940
|
artikel
|
| 32 |
Practical synthesis of capromorelin, a growth hormone secretagogue, via a crystallization-induced dynamic resolution
|
Rose, Colin R.
|
|
2017
|
25 |
3 |
p. 1000-1003
|
artikel
|
| 33 |
Quercetin-glutamic acid conjugate with a non-hydrolysable linker; a novel scaffold for multidrug resistance reversal agents through inhibition of P-glycoprotein
|
Kim, Mi Kyoung
|
|
2017
|
25 |
3 |
p. 1219-1226
|
artikel
|
| 34 |
Quinolines: Microwave-assisted synthesis and their antifungal, anticancer and radical scavenger properties
|
Liberto, Natália Aparecida
|
|
2017
|
25 |
3 |
p. 1153-1162
|
artikel
|
| 35 |
Rickettsia prowazekii methionine aminopeptidase as a promising target for the development of antibacterial agents
|
Helgren, Travis R.
|
|
2017
|
25 |
3 |
p. 813-824
|
artikel
|
| 36 |
Small molecule mimics of DFTamP1, a database designed anti-Staphylococcal peptide
|
Dong, Yuxiang
|
|
2017
|
25 |
3 |
p. 864-869
|
artikel
|
| 37 |
Structure-guided development of covalent TAK1 inhibitors
|
Tan, Li
|
|
2017
|
25 |
3 |
p. 838-846
|
artikel
|
| 38 |
5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with effective carbonic anhydrase inhibitory activity: Solution and crystallographic investigations
|
Ivanova, Jekaterīna
|
|
2017
|
25 |
3 |
p. 857-863
|
artikel
|
| 39 |
Synthesis and biological evaluation of cis-restricted triazole/tetrazole mimics of combretastatin-benzothiazole hybrids as tubulin polymerization inhibitors and apoptosis inducers
|
Subba Rao, A.V.
|
|
2017
|
25 |
3 |
p. 977-999
|
artikel
|
| 40 |
Synthesis and evaluation of 1-(cyclopropylmethyl)-4-(4-[11C]methoxyphenyl)-piperidin-1-yl-2-oxo-1,2-dihydropyridine-3-carbonitrile ([11C]CMDC) for PET imaging of metabotropic glutamate receptor 2 in the rat brain
|
Ma, Yufei
|
|
2017
|
25 |
3 |
p. 1014-1021
|
artikel
|
| 41 |
Synthesis and evaluation of frentizole-based indolyl thiourea analogues as MAO/ABAD inhibitors for Alzheimer’s disease treatment
|
Hroch, Lukas
|
|
2017
|
25 |
3 |
p. 1143-1152
|
artikel
|
| 42 |
Synthesis, docking, cytotoxicity, and LTA4H inhibitory activity of new gingerol derivatives as potential colorectal cancer therapy
|
El-Naggar, Mai H.
|
|
2017
|
25 |
3 |
p. 1277-1285
|
artikel
|
| 43 |
Synthesis, functionalization and biological activity of arylated derivatives of (+)-estrone
|
Ivanov, Anton
|
|
2017
|
25 |
3 |
p. 949-962
|
artikel
|
| 44 |
Synthesis of antimicrobial glucosamides as bacterial quorum sensing mechanism inhibitors
|
Biswas, Nripendra N.
|
|
2017
|
25 |
3 |
p. 1183-1194
|
artikel
|
| 45 |
Synthesis of seleno-fucose compounds and their application to the X-ray structural determination of carbohydrate-lectin complexes using single/multi-wavelength anomalous dispersion phasing
|
Shimabukuro, Junpei
|
|
2017
|
25 |
3 |
p. 1132-1142
|
artikel
|
| 46 |
Synthesis, physicochemical and biological studies of technetium-99m labeled tacrine derivative as a diagnostic tool for evaluation of cholinesterase level
|
Gniazdowska, Ewa
|
|
2017
|
25 |
3 |
p. 912-920
|
artikel
|
| 47 |
Synthesis, X-ray molecular structure, biological evaluation and molecular docking studies of some N4-benzyl substituted 5-nitroisatin-3-thiosemicarbazones
|
Pervez, Humayun
|
|
2017
|
25 |
3 |
p. 1022-1029
|
artikel
|
| 48 |
Towards the development of activity-based probes for detection of lysine-specific demethylase-1 activity
|
Ourailidou, Maria E.
|
|
2017
|
25 |
3 |
p. 847-856
|
artikel
|
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