| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
3-Amino-thieno[2,3-b]pyridines as microtubule-destabilising agents: Molecular modelling and biological evaluation in the sea urchin embryo and human cancer cells
|
Eurtivong, Chatchakorn
|
|
2017
|
25 |
2 |
p. 658-664
7 p.
|
artikel
|
| 2 |
Anion inhibition profiles of the γ-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei responsible of melioidosis and highly drug resistant to common antibiotics
|
Del Prete, Sonia
|
|
2017
|
25 |
2 |
p. 575-580
6 p.
|
artikel
|
| 3 |
A novel curcumin derivative which inhibits P-glycoprotein, arrests cell cycle and induces apoptosis in multidrug resistance cells
|
Lopes-Rodrigues, Vanessa
|
|
2017
|
25 |
2 |
p. 581-596
16 p.
|
artikel
|
| 4 |
Anti-inflammatory tetraquinane diterpenoids from a Crinipellis species
|
Rohr, Markus
|
|
2017
|
25 |
2 |
p. 514-522
9 p.
|
artikel
|
| 5 |
Biotransformation of rutabaga phytoalexins by the fungus Alternaria brassicicola: Unveiling the first hybrid metabolite derived from a phytoalexin and a fungal polyketide
|
Pedras, M. Soledade C.
|
|
2017
|
25 |
2 |
p. 557-567
11 p.
|
artikel
|
| 6 |
Cellular uptake of glucoheptoamidated poly(amidoamine) PAMAM G3 dendrimer with amide-conjugated biotin, a potential carrier of anticancer drugs
|
Uram, Łukasz
|
|
2017
|
25 |
2 |
p. 706-713
8 p.
|
artikel
|
| 7 |
Coating lanthanide nanoparticles with carbohydrate ligands elicits affinity for HeLa and RAW264.7 cells, enhancing their photodamaging effect
|
Kanamori, Takashi
|
|
2017
|
25 |
2 |
p. 743-749
7 p.
|
artikel
|
| 8 |
Computer design, synthesis, and bioactivity analyses of drugs like fingolimod used in the treatment of multiple sclerosis
|
Turgut, Gurbet Çelik
|
|
2017
|
25 |
2 |
p. 483-495
13 p.
|
artikel
|
| 9 |
Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity
|
Bozdag, Murat
|
|
2017
|
25 |
2 |
p. 677-683
7 p.
|
artikel
|
| 10 |
Cyclic citrullinated MBP87–99 peptide stimulates T cell responses: Implications in triggering disease
|
Apostolopoulos, Vasso
|
|
2017
|
25 |
2 |
p. 528-538
11 p.
|
artikel
|
| 11 |
Design and synthesis of phosphoryl-substituted diphenylpyrimidines (Pho-DPPYs) as potent Bruton’s tyrosine kinase (BTK) inhibitors: Targeted treatment of B lymphoblastic leukemia cell lines
|
Ge, Yang
|
|
2017
|
25 |
2 |
p. 765-772
8 p.
|
artikel
|
| 12 |
Design, synthesis and analgesic/anti-inflammatory evaluation of novel diarylthiazole and diarylimidazole derivatives towards selective COX-1 inhibitors with better gastric profile
|
Abdelazeem, Ahmed H.
|
|
2017
|
25 |
2 |
p. 665-676
12 p.
|
artikel
|
| 13 |
Design, synthesis and antithrombotic evaluation of novel non-peptide thrombin inhibitors
|
Chen, Dongxing
|
|
2017
|
25 |
2 |
p. 458-470
13 p.
|
artikel
|
| 14 |
Design, synthesis and biological evaluation of alkylamino biphenylamides as Hsp90 C-terminal inhibitors
|
Garg, Gaurav
|
|
2017
|
25 |
2 |
p. 451-457
7 p.
|
artikel
|
| 15 |
Design, synthesis and pharmacological evaluation of 4-hydroxyphenylglycine and 4-hydroxyphenylglycinol derivatives as GPR88 agonists
|
Jin, Chunyang
|
|
2017
|
25 |
2 |
p. 805-812
8 p.
|
artikel
|
| 16 |
Discovery and preclinical evaluation of 7-benzyl-N-(substituted)-pyrrolo[3,2-d]pyrimidin-4-amines as single agents with microtubule targeting effects along with triple-acting angiokinase inhibition as antitumor agents
|
Pavana, Roheeth Kumar
|
|
2017
|
25 |
2 |
p. 545-556
12 p.
|
artikel
|
| 17 |
Discovery of biphenyl imidazole derivatives as potent antifungal agents: Design, synthesis, and structure-activity relationship studies
|
Zhao, Dongmei
|
|
2017
|
25 |
2 |
p. 750-758
9 p.
|
artikel
|
| 18 |
Discovery of 4-sulfamoyl-phenyl-β-lactams as a new class of potent carbonic anhydrase isoforms I, II, IV and VII inhibitors: The first example of subnanomolar CA IV inhibitors
|
Angapelly, Srinivas
|
|
2017
|
25 |
2 |
p. 539-544
6 p.
|
artikel
|
| 19 |
Editorial board
|
|
|
2017
|
25 |
2 |
p. IFC-
1 p.
|
artikel
|
| 20 |
Effects of new fluorinated analogues of GABA, pregabalin bioisosters, on the ambient level and exocytotic release of [3H]GABA from rat brain nerve terminals
|
Borisova, T.
|
|
2017
|
25 |
2 |
p. 759-764
6 p.
|
artikel
|
| 21 |
Influence of chain length on the activity of tripeptidomimetic antagonists for CXC chemokine receptor 4 (CXCR4)
|
Baumann, Markus
|
|
2017
|
25 |
2 |
p. 646-657
12 p.
|
artikel
|
| 22 |
Multitarget drug design strategy against Alzheimer’s disease: Homoisoflavonoid Mannich base derivatives serve as acetylcholinesterase and monoamine oxidase B dual inhibitors with multifunctional properties
|
Li, Yan
|
|
2017
|
25 |
2 |
p. 714-726
13 p.
|
artikel
|
| 23 |
N-Propargylpiperidines with naphthalene-2-carboxamide or naphthalene-2-sulfonamide moieties: Potential multifunctional anti-Alzheimer’s agents
|
Košak, Urban
|
|
2017
|
25 |
2 |
p. 633-645
13 p.
|
artikel
|
| 24 |
α-Pyrone derivatives, tetra/hexahydroxanthones, and cyclodepsipeptides from two freshwater fungi
|
El-Elimat, Tamam
|
|
2017
|
25 |
2 |
p. 795-804
10 p.
|
artikel
|
| 25 |
SRC2-3 binds to vitamin D receptor with high sensitivity and strong affinity
|
Egawa, Daichi
|
|
2017
|
25 |
2 |
p. 568-574
7 p.
|
artikel
|
| 26 |
Structure-activity relationship of the inhibitory effects of flavonoids on nitric oxide production in RAW264.7 cells
|
Jiang, Wen-Jun
|
|
2017
|
25 |
2 |
p. 779-788
10 p.
|
artikel
|
| 27 |
Structure-activity relationship study of a small cyclic peptide H-c[Lys-Pro-Glu]-Arg-OH: a potent inhibitor of Vascular Endothelial Growth Factor interaction with Neuropilin-1
|
Grabowska, Karolina
|
|
2017
|
25 |
2 |
p. 597-602
6 p.
|
artikel
|
| 28 |
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH3 or 2-CH3
|
Gunia-Krzyżak, Agnieszka
|
|
2017
|
25 |
2 |
p. 471-482
12 p.
|
artikel
|
| 29 |
Synthesis and binding monitoring of a new nanomolar PAMAM-based matrix metalloproteinases inhibitor (MMPIs)
|
Cerofolini, Linda
|
|
2017
|
25 |
2 |
p. 523-527
5 p.
|
artikel
|
| 30 |
Synthesis and biological evaluation of phosphate isosters of fosmidomycin and analogs as inhibitors of Escherichia coli and Mycobacterium smegmatis 1-deoxyxylulose 5-phosphate reductoisomerases
|
Munier, Mathilde
|
|
2017
|
25 |
2 |
p. 684-689
6 p.
|
artikel
|
| 31 |
Synthesis and characterization of novel, conjugated, fluorescent DNJ derivatives for α-glucosidase recognition
|
Hatano, Akihiko
|
|
2017
|
25 |
2 |
p. 773-778
6 p.
|
artikel
|
| 32 |
Synthesis and evaluation of a 68Ga-labeled bradykinin B1 receptor agonist for imaging with positron emission tomography
|
Amouroux, Guillaume
|
|
2017
|
25 |
2 |
p. 690-696
7 p.
|
artikel
|
| 33 |
Synthesis and immunological evaluation of a low molecular weight saccharide with TLR-4 agonist activity
|
Basava, Vikram
|
|
2017
|
25 |
2 |
p. 697-705
9 p.
|
artikel
|
| 34 |
Synthesis and optimization of novel α-phenylglycinamides as selective TRPM8 antagonists
|
Kobayashi, Jun-ichi
|
|
2017
|
25 |
2 |
p. 727-742
16 p.
|
artikel
|
| 35 |
Synthesis, antioxidant and antichagasic properties of a selected series of hydroxy-3-arylcoumarins
|
Robledo-O’Ryan, Natalia
|
|
2017
|
25 |
2 |
p. 621-632
12 p.
|
artikel
|
| 36 |
Synthesis, evaluation and molecular modelling studies of 2-(carbazol-3-yl)-2-oxoacetamide analogues as a new class of potential pancreatic lipase inhibitors
|
Sridhar, S.N.C.
|
|
2017
|
25 |
2 |
p. 609-620
12 p.
|
artikel
|
| 37 |
Synthesis of a biological active β-hairpin peptide by addition of two structural motifs
|
Fischer, Sabrina
|
|
2017
|
25 |
2 |
p. 603-608
6 p.
|
artikel
|
| 38 |
Synthesis of novel C4-benzazole naphthalimide derivatives with potent anti-tumor properties against murine melanoma
|
Lu, Yen-Ta
|
|
2017
|
25 |
2 |
p. 789-794
6 p.
|
artikel
|
| 39 |
Triazolopyridine ethers as potent, orally active mGlu2 positive allosteric modulators for treating schizophrenia
|
Higgins, Mendi A.
|
|
2017
|
25 |
2 |
p. 496-513
18 p.
|
artikel
|
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