| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Anion inhibitors of the β-carbonic anhydrase from the pathogenic bacterium responsible of tularemia, Francisella tularensis
|
Del Prete, Sonia
|
|
2017
|
25 |
17 |
p. 4800-4804
|
artikel
|
| 2 |
A novel antihypertension agent, sargachromenol D from marine brown algae, Sargassum siliquastrum, exerts dual action as an L-type Ca2+ channel blocker and endothelin A/B2 receptor antagonist
|
Park, Byong-Gon
|
|
2017
|
25 |
17 |
p. 4649-4655
|
artikel
|
| 3 |
Asymmetric synthesis and evaluation of epoxy-α-acyloxycarboxamides as selective inhibitors of cathepsin L
|
dos Santos, Deborah A.
|
|
2017
|
25 |
17 |
p. 4620-4627
|
artikel
|
| 4 |
Brassinolide-like activity of castasterone analogs with varied side chains against rice lamina inclination
|
Watanabe, Bunta
|
|
2017
|
25 |
17 |
p. 4566-4578
|
artikel
|
| 5 |
5-Bromoindirubin 3′-(O-oxiran-2-ylmethyl)oxime: A long-acting anticancer agent and a suicide inhibitor for epoxide hydrolase
|
Ichimaru, Yoshimi
|
|
2017
|
25 |
17 |
p. 4665-4676
|
artikel
|
| 6 |
Chiral-pool synthesis of 1,2,4-trisubstituted 1,4-diazepanes as novel σ1 receptor ligands
|
Fanter, Lena
|
|
2017
|
25 |
17 |
p. 4778-4799
|
artikel
|
| 7 |
Cycloalkane analogues of sinefungin as EHMT1/2 inhibitors
|
Liu, Qing
|
|
2017
|
25 |
17 |
p. 4579-4594
|
artikel
|
| 8 |
9,19-Cycloartenol glycoside G3 from Cimicifuga simplex regulates immune responses by modulating Th17/Treg ratio
|
Su, Yang
|
|
2017
|
25 |
17 |
p. 4917-4923
|
artikel
|
| 9 |
Design, synthesis and bioactivities of Celecoxib analogues or derivatives
|
Zhou, Shiyang
|
|
2017
|
25 |
17 |
p. 4887-4893
|
artikel
|
| 10 |
Design, synthesis, and pharmacological evaluation of a novel series of hormone sensitive lipase inhibitor
|
Ogiyama, Tomoko
|
|
2017
|
25 |
17 |
p. 4817-4828
|
artikel
|
| 11 |
Design, synthesis, molecular modeling and anti-hyperglycemic evaluation of quinazolin-4(3H)-one derivatives as potential PPARγ and SUR agonists
|
Ibrahim, Mohamed K.
|
|
2017
|
25 |
17 |
p. 4723-4744
|
artikel
|
| 12 |
Development of novel LP1-based analogues with enhanced delta opioid receptor profile
|
Pasquinucci, Lorella
|
|
2017
|
25 |
17 |
p. 4745-4752
|
artikel
|
| 13 |
Discovery of a low-systemic-exposure DGAT-1 inhibitor with a picolinoylpyrrolidine-2-carboxylic acid moiety
|
Yan, Jianwei
|
|
2017
|
25 |
17 |
p. 4701-4714
|
artikel
|
| 14 |
Discovery of a novel B-cell lymphoma 6 (BCL6)–corepressor interaction inhibitor by utilizing structure-based drug design
|
Yasui, Takeshi
|
|
2017
|
25 |
17 |
p. 4876-4886
|
artikel
|
| 15 |
Discovery of a tetrahydroisoquinoline-based HDAC inhibitor with improved plasma stability
|
Zhou, Nan
|
|
2017
|
25 |
17 |
p. 4614-4619
|
artikel
|
| 16 |
Discovery of new leads against Mycobacterium tuberculosis using scaffold hopping and shape based similarity
|
Wavhale, Ravindra D.
|
|
2017
|
25 |
17 |
p. 4835-4844
|
artikel
|
| 17 |
Discovery of spiro[indole-3,2′-pyrrolidin]-2(1H)-one based inhibitors targeting Brr2, a core component of the U5 snRNP
|
Ito, Masahiro
|
|
2017
|
25 |
17 |
p. 4753-4767
|
artikel
|
| 18 |
Editorial board
|
|
|
2017
|
25 |
17 |
p. IFC
|
artikel
|
| 19 |
Fluoro and pentafluorothio analogs of the antitumoral curcuminoid EF24 with superior antiangiogenic and vascular-disruptive effects
|
Schmitt, Florian
|
|
2017
|
25 |
17 |
p. 4894-4903
|
artikel
|
| 20 |
Isolation and lipolytic activity of eurycomanone and its epoxy derivative from Eurycoma longifolia
|
Lahrita, Lucy
|
|
2017
|
25 |
17 |
p. 4829-4834
|
artikel
|
| 21 |
KBE009: An antimalarial bestatin-like inhibitor of the Plasmodium falciparum M1 aminopeptidase discovered in an Ugi multicomponent reaction-derived peptidomimetic library
|
González-Bacerio, Jorge
|
|
2017
|
25 |
17 |
p. 4628-4636
|
artikel
|
| 22 |
New prodrugs of two pyrimidine acyclic nucleoside phosphonates: Synthesis and antiviral activity
|
Krečmerová, Marcela
|
|
2017
|
25 |
17 |
p. 4637-4648
|
artikel
|
| 23 |
5- or/and 20-O-alkyl-2,3-dehydrosilybins: Synthesis and biological profiles on prostate cancer cell models
|
Vue, Bao
|
|
2017
|
25 |
17 |
p. 4845-4854
|
artikel
|
| 24 |
3-O-Substituted-3′,4′,5′-trimethoxyflavonols: Synthesis and cell-based evaluation as anti-prostate cancer agents
|
Li, Xiang
|
|
2017
|
25 |
17 |
p. 4768-4777
|
artikel
|
| 25 |
1,3-Oxazole-based selective picomolar inhibitors of cytosolic human carbonic anhydrase II alleviate ocular hypertension in rabbits: Potency is supported by X-ray crystallography of two leads
|
Ferraroni, Marta
|
|
2017
|
25 |
17 |
p. 4560-4565
|
artikel
|
| 26 |
pH responsive biodegradable nanogels for sustained release of bleomycin
|
Sahu, Prashant
|
|
2017
|
25 |
17 |
p. 4595-4613
|
artikel
|
| 27 |
Platinum(IV) complexes conjugated with phenstatin analogue as inhibitors of microtubule polymerization and reverser of multidrug resistance
|
Huang, Xiaochao
|
|
2017
|
25 |
17 |
p. 4686-4700
|
artikel
|
| 28 |
Recent synthetic and medicinal perspectives of tryptanthrin
|
Kaur, Ramandeep
|
|
2017
|
25 |
17 |
p. 4533-4552
|
artikel
|
| 29 |
Structure based drug design of Pim-1 kinase followed by pharmacophore guided synthesis of quinolone-based inhibitors
|
Swellmeen, Lubna
|
|
2017
|
25 |
17 |
p. 4855-4875
|
artikel
|
| 30 |
Synthesis and biological evaluation in vitro and in mammalian cells of new heteroaryl carboxyamides as HIV-protease inhibitors
|
Funicello, M.
|
|
2017
|
25 |
17 |
p. 4715-4722
|
artikel
|
| 31 |
Synthesis and biological evaluation of fluoro-substituted 3,4-dihydroquinazoline derivatives for cytotoxic and analgesic effects
|
Kim, Jin Han
|
|
2017
|
25 |
17 |
p. 4656-4664
|
artikel
|
| 32 |
Synthesis and biological investigation of tetrahydropyridopyrimidinone derivatives as potential multireceptor atypical antipsychotics
|
Xiamuxi, Hainimu
|
|
2017
|
25 |
17 |
p. 4904-4916
|
artikel
|
| 33 |
Synthesis and diabetic neuropathic pain-alleviating effects of 2N-(pyrazol-3-yl)methylbenzo[d]isothiazole-1,1-dioxide derivatives
|
Hong, Jin Ri
|
|
2017
|
25 |
17 |
p. 4677-4685
|
artikel
|
| 34 |
Synthesis and evaluation of osimertinib derivatives as potent EGFR inhibitors
|
Gao, Hongying
|
|
2017
|
25 |
17 |
p. 4553-4559
|
artikel
|
| 35 |
Synthesis of different heterocycles-linked chalcone conjugates as cytotoxic agents and tubulin polymerization inhibitors
|
Shankaraiah, Nagula
|
|
2017
|
25 |
17 |
p. 4805-4816
|
artikel
|
Tijdschrift beschrijving