| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Application of in-vitro screening methods on hypoxia inducible factor prolyl hydroxylase inhibitors
|
Wu, Yue
|
|
2017
|
25 |
15 |
p. 3891-3899
|
artikel
|
| 2 |
BACE1 inhibitory activity and molecular docking analysis of meroterpenoids from Sargassum serratifolium
|
Seong, Su Hui
|
|
2017
|
25 |
15 |
p. 3964-3970
|
artikel
|
| 3 |
Cyclic MOG35 – 55 ameliorates clinical and neuropathological features of experimental autoimmune encephalomyelitis
|
Lourbopoulos, Athanasios
|
|
2017
|
25 |
15 |
p. 4163-4174
|
artikel
|
| 4 |
Design, synthesis and biological evaluation of renin inhibitors guided by simulated annealing of chemical potential simulations
|
Cloudsdale, Ian S.
|
|
2017
|
25 |
15 |
p. 3947-3963
|
artikel
|
| 5 |
Design, synthesis and biological evaluation of sulfonamide-substituted diphenylpyrimidine derivatives (Sul-DPPYs) as potent focal adhesion kinase (FAK) inhibitors with antitumor activity
|
Qu, Menghua
|
|
2017
|
25 |
15 |
p. 3989-3996
|
artikel
|
| 6 |
Design, synthesis, and evaluation of DNA topoisomerase II-targeted nucleosides
|
Matsumoto, Hironobu
|
|
2017
|
25 |
15 |
p. 4133-4144
|
artikel
|
| 7 |
Design, synthesis and tumor cell growth inhibitory activity of 3-nitro-2H-cheromene derivatives as histone deacetylaes inhibitors
|
Tan, Shuai
|
|
2017
|
25 |
15 |
p. 4123-4132
|
artikel
|
| 8 |
Discovery of novel 5-oxa-2,6-diazaspiro[3.4]oct-6-ene derivatives as potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonists for treatment of type 2 diabetes mellitus
|
Hirose, Hideki
|
|
2017
|
25 |
15 |
p. 4175-4193
|
artikel
|
| 9 |
Discovery of novel quinazoline-2,4(1H,3H)-dione derivatives as potent PARP-2 selective inhibitors
|
Zhao, Hailong
|
|
2017
|
25 |
15 |
p. 4045-4054
|
artikel
|
| 10 |
Discovery of novel somatostatin receptor subtype 5 (SSTR5) antagonists: Pharmacological studies and design to improve pharmacokinetic profiles and human Ether-a-go-go-related gene (hERG) inhibition
|
Yamasaki, Takeshi
|
|
2017
|
25 |
15 |
p. 4153-4162
|
artikel
|
| 11 |
Discovery of simplified leucyladenylate sulfamates as novel leucyl-tRNA synthetase (LRS)-targeted mammalian target of rapamycin complex 1 (mTORC1) inhibitors
|
Yoon, Suyoung
|
|
2017
|
25 |
15 |
p. 4145-4152
|
artikel
|
| 12 |
Editorial board
|
|
|
2017
|
25 |
15 |
p. IFC
|
artikel
|
| 13 |
Isolation, structure elucidation, and synthesis of antiplasmodial quinolones from Crinum firmifolium
|
Presley, Christopher C.
|
|
2017
|
25 |
15 |
p. 4203-4211
|
artikel
|
| 14 |
Novel pyridyl nitrofuranyl isoxazolines show antibacterial activity against multiple drug resistant Staphylococcus species
|
Picconi, Pietro
|
|
2017
|
25 |
15 |
p. 3971-3979
|
artikel
|
| 15 |
Olaparib hydroxamic acid derivatives as dual PARP and HDAC inhibitors for cancer therapy
|
Yuan, Zigao
|
|
2017
|
25 |
15 |
p. 4100-4109
|
artikel
|
| 16 |
Synthesis and biological activity of peptide proline-boronic acids as proteasome inhibitors
|
Han, Liqiang
|
|
2017
|
25 |
15 |
p. 4031-4044
|
artikel
|
| 17 |
Synthesis and biological evaluation of JL-A7 derivatives as potent ABCB1 inhibitors
|
Pan, Miaobo
|
|
2017
|
25 |
15 |
p. 4194-4202
|
artikel
|
| 18 |
Synthesis and evaluation of symmetric acyclic nucleoside bisphosphonates as inhibitors of the Plasmodium falciparum, Plasmodium vivax and human 6-oxopurine phosphoribosyltransferases and the antimalarial activity of their prodrugs
|
Špaček, Petr
|
|
2017
|
25 |
15 |
p. 4008-4030
|
artikel
|
| 19 |
Synthesis and pharmacological evaluation of glycine amide derivatives as novel vascular adhesion protein-1 inhibitors without CYP3A4 and CYP2C19 inhibition
|
Yamaki, Susumu
|
|
2017
|
25 |
15 |
p. 4110-4122
|
artikel
|
| 20 |
Synthesis, antiviral evaluation and molecular docking studies of N 4-aryl substituted/unsubstituted thiosemicarbazones derived from 1-indanones as potent anti-bovine viral diarrhea virus agents
|
Soraires Santacruz, María C.
|
|
2017
|
25 |
15 |
p. 4055-4063
|
artikel
|
| 21 |
Synthesis, biological evaluation and molecular modeling of imidazo[1,2-a]pyridine derivatives as potent antitubulin agents
|
Liu, Jin
|
|
2017
|
25 |
15 |
p. 4088-4099
|
artikel
|
| 22 |
Synthesis, docking study and neuroprotective effects of some novel pyrano[3,2-c]chromene derivatives bearing morpholine/phenylpiperazine moiety
|
Sameem, Bilqees
|
|
2017
|
25 |
15 |
p. 3980-3988
|
artikel
|
| 23 |
Synthesis, molecular docking, and biological activity of polyfluoroalkyl dihydroazolo[5,1-c][1,2,4]triazines as selective carboxylesterase inhibitors
|
Shchegol'kov, Evgeny V.
|
|
2017
|
25 |
15 |
p. 3997-4007
|
artikel
|
| 24 |
Synthesis, molecular modelling and CYP24A1 inhibitory activity of novel of (E)-N-(2-(1H-imidazol-1-yl)-2-(phenylethyl)-3/4-styrylbenzamides
|
Taban, Ismail M.
|
|
2017
|
25 |
15 |
p. 4076-4087
|
artikel
|
| 25 |
The selective cytotoxicity of new triazene compounds to human melanoma cells
|
Sousa, Ana
|
|
2017
|
25 |
15 |
p. 3900-3910
|
artikel
|
| 26 |
The synthesis and evaluation of triazolopyrimidines as anti-tubercular agents
|
Zuniga, Edison S.
|
|
2017
|
25 |
15 |
p. 3922-3946
|
artikel
|
| 27 |
The tobacco cembranoid (1S,2E,4S,7E,11E)-2,7,11-cembratriene-4,6-diol as a novel angiogenesis inhibitory lead for the control of breast malignancies
|
Hailat, Mohammad M.
|
|
2017
|
25 |
15 |
p. 3911-3921
|
artikel
|
| 28 |
1,2,4-Triazole and 1,3,4-oxadiazole analogues: Synthesis, MO studies, in silico molecular docking studies, antimalarial as DHFR inhibitor and antimicrobial activities
|
Thakkar, Sampark S.
|
|
2017
|
25 |
15 |
p. 4064-4075
|
artikel
|
| 29 |
Ultrasound-dependent cytoplasmic internalization of a peptide-sonosensitizer conjugate
|
Inaba, Yuki
|
|
2017
|
25 |
15 |
p. 4212-4217
|
artikel
|
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