| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A fragment-based approach leading to the discovery of a novel binding site and the selective CK2 inhibitor CAM4066
|
De Fusco, Claudia
|
|
2017
|
25 |
13 |
p. 3471-3482
12 p.
|
artikel
|
| 2 |
Alkyne-linked reduction-activated protecting groups for diverse functionalization on the backbone of oligonucleotides
|
Saneyoshi, Hisao
|
|
2017
|
25 |
13 |
p. 3350-3356
7 p.
|
artikel
|
| 3 |
Antioxidant and anticholinesterase potential of diterpenoid alkaloids from Aconitum heterophyllum
|
Ahmad, Hanif
|
|
2017
|
25 |
13 |
p. 3368-3376
9 p.
|
artikel
|
| 4 |
C21-steroidal pregnane sapogenins and their derivatives as anti-inflammatory agents
|
Huang, Lie-Jun
|
|
2017
|
25 |
13 |
p. 3512-3524
13 p.
|
artikel
|
| 5 |
Design and optimization of purine derivatives as in vivo active PDE10A inhibitors
|
Chen, Liu
|
|
2017
|
25 |
13 |
p. 3315-3329
15 p.
|
artikel
|
| 6 |
Design and synthesis of novel photoinduced electron transfer-based hybridization probes
|
Yokoyama, Chika
|
|
2017
|
25 |
13 |
p. 3574-3582
9 p.
|
artikel
|
| 7 |
Design and synthesis of 1,2,3-triazolo linked benzo[d]imidazo[2,1-b]thiazole conjugates as tubulin polymerization inhibitors
|
Shaik, Siddiq Pasha
|
|
2017
|
25 |
13 |
p. 3285-3297
13 p.
|
artikel
|
| 8 |
Development of molecular tools based on the dopamine D3 receptor ligand FAUC 329 showing inhibiting effects on drug and food maintained behavior
|
Stößel, Anne
|
|
2017
|
25 |
13 |
p. 3491-3499
9 p.
|
artikel
|
| 9 |
Development of nonsteroidal glucocorticoid receptor modulators based on N-benzyl-N-(4-phenoxyphenyl)benzenesulfonamide scaffold
|
Yoshioka, Hiromasa
|
|
2017
|
25 |
13 |
p. 3461-3470
10 p.
|
artikel
|
| 10 |
Development of the optical sensor for discriminating isomers of fatty acids based on emissive network polymers composed of polyhedral oligomeric silsesquioxane
|
Narikiyo, Hayato
|
|
2017
|
25 |
13 |
p. 3431-3436
6 p.
|
artikel
|
| 11 |
Discovery and structure-guided fragment-linking of 4-(2,3-dichlorobenzoyl)-1-methyl-pyrrole-2-carboxamide as a pyruvate kinase M2 activator
|
Matsui, Yumi
|
|
2017
|
25 |
13 |
p. 3540-3546
7 p.
|
artikel
|
| 12 |
Discovery of indolin-2-one derivatives as potent PAK4 inhibitors: Structure-activity relationship analysis, biological evaluation and molecular docking study
|
Guo, Jing
|
|
2017
|
25 |
13 |
p. 3500-3511
12 p.
|
artikel
|
| 13 |
Dual functional small molecule fluorescent probes for image-guided estrogen receptor-specific targeting coupled potent antiproliferative potency for breast cancer therapy
|
Yang, Lu
|
|
2017
|
25 |
13 |
p. 3531-3539
9 p.
|
artikel
|
| 14 |
Editorial board
|
|
|
2017
|
25 |
13 |
p. IFC-
1 p.
|
artikel
|
| 15 |
Exploration of pyrrole derivatives to find an effective potassium-competitive acid blocker with moderately long-lasting suppression of gastric acid secretion
|
Nishida, Haruyuki
|
|
2017
|
25 |
13 |
p. 3447-3460
14 p.
|
artikel
|
| 16 |
Identification of a novel fluoropyrrole derivative as a potassium-competitive acid blocker with long duration of action
|
Nishida, Haruyuki
|
|
2017
|
25 |
13 |
p. 3298-3314
17 p.
|
artikel
|
| 17 |
Identification of novel 1,2,3,6-tetrahydropyridyl-substituted benzo[d]thiazoles: Lead generation and optimization toward potent and orally active EP1 receptor antagonists
|
Umei, Kentaro
|
|
2017
|
25 |
13 |
p. 3406-3430
25 p.
|
artikel
|
| 18 |
Inhibition of amyloid β aggregation and protective effect on SH-SY5Y cells by triterpenoid saponins from the cactus Polaskia chichipe
|
Fujihara, Koji
|
|
2017
|
25 |
13 |
p. 3377-3383
7 p.
|
artikel
|
| 19 |
Kinetic properties and affinities for sulfonamide inhibitors of an α-carbonic anhydrase (CruCA4) involved in coral biomineralization in the Mediterranean red coral Corallium rubrum
|
Del Prete, Sonia
|
|
2017
|
25 |
13 |
p. 3525-3530
6 p.
|
artikel
|
| 20 |
Lathyrol and epoxylathyrol derivatives: Modulation of Cdr1p and Mdr1p drug-efflux transporters of Candida albicans in Saccharomyces cerevisiae model
|
Mónico, Andreia
|
|
2017
|
25 |
13 |
p. 3278-3284
7 p.
|
artikel
|
| 21 |
Lipase-catalyzed kinetic resolution as key step in the synthesis of enantiomerically pure σ ligands with 2-benzopyran structure
|
Knappmann, Inga
|
|
2017
|
25 |
13 |
p. 3384-3395
12 p.
|
artikel
|
| 22 |
Medicinal chemistry of antischistosomal drugs: Praziquantel and oxamniquine
|
da Silva, Vinícius Barros Ribeiro
|
|
2017
|
25 |
13 |
p. 3259-3277
19 p.
|
artikel
|
| 23 |
N-Substituted and ring opened saccharin derivatives selectively inhibit transmembrane, tumor-associated carbonic anhydrases IX and XII
|
Ivanova, Jekaterīna
|
|
2017
|
25 |
13 |
p. 3583-3589
7 p.
|
artikel
|
| 24 |
Potential anti-gout constituents as xanthine oxidase inhibitor from the fruits of Stauntonia brachyanthera
|
Liu, Dan
|
|
2017
|
25 |
13 |
p. 3562-3566
5 p.
|
artikel
|
| 25 |
Potential inhibitors of human carbonic anhydrase isozymes I and II: Design, synthesis and docking studies of new 1,3,4-thiadiazole derivatives
|
Altıntop, Mehlika Dilek
|
|
2017
|
25 |
13 |
p. 3547-3554
8 p.
|
artikel
|
| 26 |
Sulfonamide inhibition profiles of the β-carbonic anhydrase from the pathogenic bacterium Francisella tularensis responsible of the febrile illness tularemia
|
Del Prete, Sonia
|
|
2017
|
25 |
13 |
p. 3555-3561
7 p.
|
artikel
|
| 27 |
Synthesis and biological activity of new phthalimides as potential anti-inflammatory agents
|
Bach, Duc-Hiep
|
|
2017
|
25 |
13 |
p. 3396-3405
10 p.
|
artikel
|
| 28 |
Synthesis and biological evaluation of novel selective androgen receptor modulators (SARMs) Part III: Discovery of 4-(5-oxopyrrolidine-1-yl)benzonitrile derivative 2f as a clinical candidate
|
Aikawa, Katsuji
|
|
2017
|
25 |
13 |
p. 3330-3349
20 p.
|
artikel
|
| 29 |
Synthesis and biological research of novel azaacridine derivatives as potent DNA-binding ligands and topoisomerase II inhibitors
|
Li, Dan
|
|
2017
|
25 |
13 |
p. 3437-3446
10 p.
|
artikel
|
| 30 |
Synthesis and cytotoxic activity of new artemisinin hybrid molecules against human leukemia cells
|
Letis, Antonios S.
|
|
2017
|
25 |
13 |
p. 3357-3367
11 p.
|
artikel
|
| 31 |
Synthesis of novel acyl selenoureido benzensulfonamides as carbonic anhydrase I, II, VII and IX inhibitors
|
Angeli, Andrea
|
|
2017
|
25 |
13 |
p. 3567-3573
7 p.
|
artikel
|
| 32 |
Zinc complex of tryptophan appended 1,4,7,10-tetraazacyclododecane as potential anticancer agent: Synthesis and evaluation
|
Adhikari, Anupriya
|
|
2017
|
25 |
13 |
p. 3483-3490
8 p.
|
artikel
|
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