| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Bivalent O-glycoside mimetics with S/disulfide/Se substitutions and aromatic core: Synthesis, molecular modeling and inhibitory activity on biomedically relevant lectins in assays of increasing physiological relevance
|
Kaltner, Herbert
|
|
2017
|
25 |
12 |
p. 3158-3170
|
artikel
|
| 2 |
Catabolism of antibody drug conjugates and characterization methods
|
Shadid, Mohammad
|
|
2017
|
25 |
12 |
p. 2933-2945
|
artikel
|
| 3 |
Covalent inhibitors of LgtC: A blueprint for the discovery of non-substrate-like inhibitors for bacterial glycosyltransferases
|
Xu, Yong
|
|
2017
|
25 |
12 |
p. 3182-3194
|
artikel
|
| 4 |
Derivatives of caffeic acid, a natural antioxidant, as the basis for the discovery of novel nonpeptidic neurotrophic agents
|
Moosavi, Fatemeh
|
|
2017
|
25 |
12 |
p. 3235-3246
|
artikel
|
| 5 |
Design and synthesis of pyrazolo[3,4-d]pyrimidines: Nitric oxide releasing compounds targeting hepatocellular carcinoma
|
Elshaier, Yaseen A.M.M.
|
|
2017
|
25 |
12 |
p. 2956-2970
|
artikel
|
| 6 |
Design, synthesis and anti-tumor activity study of novel histone deacetylase inhibitors containing isatin-based caps and o-phenylenediamine-based zinc binding groups
|
Gao, Shuai
|
|
2017
|
25 |
12 |
p. 2981-2994
|
artikel
|
| 7 |
Design, synthesis and biological evaluation of 3,4-dihydro-2(1H)-quinoline-O-alkylamine derivatives as new multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer’s disease
|
Sang, Zhipei
|
|
2017
|
25 |
12 |
p. 3006-3017
|
artikel
|
| 8 |
Design, synthesis, and docking studies of quinazoline analogues bearing aryl semicarbazone scaffolds as potent EGFR inhibitors
|
Tu, Yuanbiao
|
|
2017
|
25 |
12 |
p. 3148-3157
|
artikel
|
| 9 |
Design, synthesis, and evaluation of multitarget-directed ligands against Alzheimer’s disease based on the fusion of donepezil and curcumin
|
Yan, Jun
|
|
2017
|
25 |
12 |
p. 2946-2955
|
artikel
|
| 10 |
Design, synthesis, and pharmacological evaluation of 4-azolyl-benzamide derivatives as novel GPR52 agonists
|
Tokumaru, Kazuyuki
|
|
2017
|
25 |
12 |
p. 3098-3115
|
artikel
|
| 11 |
Dimeric isoxazolyl-1,4-dihydropyridines have enhanced binding at the multi-drug resistance transporter
|
Steiger, Scott A.
|
|
2017
|
25 |
12 |
p. 3223-3234
|
artikel
|
| 12 |
Dual 7-ethyl-10-hydroxycamptothecin conjugated phospholipid prodrug assembled liposomes with in vitro anticancer effects
|
Du, Yawei
|
|
2017
|
25 |
12 |
p. 3247-3258
|
artikel
|
| 13 |
Editorial board
|
|
|
2017
|
25 |
12 |
p. IFC
|
artikel
|
| 14 |
Effect of natural and semi-synthetic cadinanes from Heterotheca inuloides on NF-κB, Nrf2 and STAT3 signaling pathways and evaluation of their in vitro cytotoxicity in human cancer cell lines
|
Egas, Verónica
|
|
2017
|
25 |
12 |
p. 3135-3147
|
artikel
|
| 15 |
Effect of 1,2,3-triazole salts, non-classical bioisosteres of miltefosine, on Leishmania amazonensis
|
Stroppa, Pedro H.F.
|
|
2017
|
25 |
12 |
p. 3034-3045
|
artikel
|
| 16 |
Exploring the influence of indololactone structure on selectivity for binding to the C1 domains of PKCα, PKCε, and RasGRP
|
Elhalem, Eleonora
|
|
2017
|
25 |
12 |
p. 2971-2980
|
artikel
|
| 17 |
Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure–activity relationship study of 4-epi-jaspine B
|
Ohno, Hiroaki
|
|
2017
|
25 |
12 |
p. 3046-3052
|
artikel
|
| 18 |
N-(Aroyl)-N-(arylmethyloxy)-α-alanines: Selective inhibitors of aldose reductase
|
Nencetti, Susanna
|
|
2017
|
25 |
12 |
p. 3068-3076
|
artikel
|
| 19 |
Ortho group activation of a bromopyrrole ester in Suzuki-Miyaura cross-coupling reactions: Application to the synthesis of new microtubule depolymerizing agents with potent cytotoxic activities
|
Gupton, John T.
|
|
2017
|
25 |
12 |
p. 3206-3214
|
artikel
|
| 20 |
Small molecules inhibit STAT3 activation, autophagy, and cancer cell anchorage-independent growth
|
Zhou, Donghui
|
|
2017
|
25 |
12 |
p. 2995-3005
|
artikel
|
| 21 |
Stereospecific cholinesterase inhibition by O,S-diethylphenylphosphonothioate
|
Mohammed, Ahmed
|
|
2017
|
25 |
12 |
p. 3053-3058
|
artikel
|
| 22 |
Structure of a Myeloid cell leukemia-1 (Mcl-1) inhibitor bound to drug site 3 of Human Serum Albumin
|
Zhao, Bin
|
|
2017
|
25 |
12 |
p. 3087-3092
|
artikel
|
| 23 |
Studies of CDK 8/19 inhibitors: Discovery of novel and selective CDK8/19 dual inhibitors and elimination of their CYP3A4 time-dependent inhibition potential
|
Fujimoto, Jun
|
|
2017
|
25 |
12 |
p. 3018-3033
|
artikel
|
| 24 |
Synthesis and biological evaluation of largazole zinc-binding group analogs
|
Kim, Bumki
|
|
2017
|
25 |
12 |
p. 3077-3086
|
artikel
|
| 25 |
Synthesis and biological evaluation of N-(carbobenzyloxy)-l-phenylalanine and N-(carbobenzyloxy)-l-aspartic acid-β-benzyl ester derivatives as potent topoisomerase IIα inhibitors
|
Han, Xiaoyan
|
|
2017
|
25 |
12 |
p. 3116-3126
|
artikel
|
| 26 |
Synthesis and biological evaluation of novel aromatic and heterocyclic bis-sulfonamide Schiff bases as carbonic anhydrase I, II, VII and IX inhibitors
|
Akocak, Suleyman
|
|
2017
|
25 |
12 |
p. 3093-3097
|
artikel
|
| 27 |
Synthesis and biological evaluation of selective tubulin inhibitors as anti-trypanosomal agents
|
Bobba, Viharika
|
|
2017
|
25 |
12 |
p. 3215-3222
|
artikel
|
| 28 |
Synthesis and evaluation of a series of pyridine and pyrimidine derivatives as type II c-Met inhibitors
|
Zhao, Yanmei
|
|
2017
|
25 |
12 |
p. 3195-3205
|
artikel
|
| 29 |
Synthesis, biochemical evaluation, and molecular modeling studies of aryl and arylalkyl di-n-butyl phosphates, effective butyrylcholinesterase inhibitors
|
Nakayama, Kensaku
|
|
2017
|
25 |
12 |
p. 3171-3181
|
artikel
|
| 30 |
Synthesis of benzoxazole derivatives as interleukin-6 antagonists
|
Kim, Darong
|
|
2017
|
25 |
12 |
p. 3127-3134
|
artikel
|
| 31 |
The synthesis and evaluation of new butadiene derivatives as tubulin polymerization inhibitors
|
Pang, Yanqing
|
|
2017
|
25 |
12 |
p. 3059-3067
|
artikel
|
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