| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A multi-endpoint matched molecular pair (MMP) analysis of 6-membered heterocycles
|
Chang, George
|
|
2017
|
25 |
1 |
p. 381-388
8 p.
|
artikel
|
| 2 |
An evaluation of central penetration from a peripherally administered oxytocin receptor selective antagonist in nonhuman primates
|
Smith, Aaron L.
|
|
2017
|
25 |
1 |
p. 305-315
11 p.
|
artikel
|
| 3 |
A new target for Parkinson’s disease: Small molecule SERCA activator CDN1163 ameliorates dyskinesia in 6-OHDA-lesioned rats
|
Dahl, Russell
|
|
2017
|
25 |
1 |
p. 53-57
5 p.
|
artikel
|
| 4 |
A novel adamantane thiadiazole derivative induces mitochondria-mediated apoptosis in lung carcinoma cell line
|
Ali, Ayat G.
|
|
2017
|
25 |
1 |
p. 241-253
13 p.
|
artikel
|
| 5 |
Antibacterial profiling of abietane-type diterpenoids
|
Helfenstein, Andreas
|
|
2017
|
25 |
1 |
p. 132-137
6 p.
|
artikel
|
| 6 |
A trans-platinum(II) complex induces apoptosis in cancer stem cells of breast cancer
|
Aztopal, Nazlihan
|
|
2017
|
25 |
1 |
p. 269-276
8 p.
|
artikel
|
| 7 |
Bioactivity of topologically confined gramicidin A dimers
|
Jadhav, Kirtikumar B.
|
|
2017
|
25 |
1 |
p. 261-268
8 p.
|
artikel
|
| 8 |
Bis(N-amidinohydrazones) and N-(amidino)-N′-aryl-bishydrazones: New classes of antibacterial/antifungal agents
|
Shrestha, Sanjib K.
|
|
2017
|
25 |
1 |
p. 58-66
9 p.
|
artikel
|
| 9 |
Design and synthesis of affinity chromatography ligands for the purification of 5-hydroxyeicosanoid dehydrogenase
|
Nagendra Reddy, Chintam
|
|
2017
|
25 |
1 |
p. 116-125
10 p.
|
artikel
|
| 10 |
Design and synthesis of novel N-sulfonyl-2-indoles that behave as 5-HT6 receptor ligands with significant selectivity for D3 over D2 receptors
|
Saavedra, Oscar M.
|
|
2017
|
25 |
1 |
p. 38-52
15 p.
|
artikel
|
| 11 |
Design, synthesis and biological evaluation of 4,5-dibromo-N-(thiazol-2-yl)-1H-pyrrole-2-carboxamide derivatives as novel DNA gyrase inhibitors
|
Tomašič, Tihomir
|
|
2017
|
25 |
1 |
p. 338-349
12 p.
|
artikel
|
| 12 |
Design, synthesis, biological evaluation, and molecular modeling studies of chalcone-rivastigmine hybrids as cholinesterase inhibitors
|
Wang, Ling
|
|
2017
|
25 |
1 |
p. 360-371
12 p.
|
artikel
|
| 13 |
Development of a novel series of non-natural triaryl agonists and antagonists of the Pseudomonas aeruginosa LasR quorum sensing receptor
|
Capilato, Joseph N.
|
|
2017
|
25 |
1 |
p. 153-165
13 p.
|
artikel
|
| 14 |
Discovery of novel curcumin derivatives targeting xanthine oxidase and urate transporter 1 as anti-hyperuricemic agents
|
Ao, Gui-Zhen
|
|
2017
|
25 |
1 |
p. 166-174
9 p.
|
artikel
|
| 15 |
Discovery of novel multi-target indole-based derivatives as potent and selective inhibitors of chikungunya virus replication
|
Scuotto, Maria
|
|
2017
|
25 |
1 |
p. 327-337
11 p.
|
artikel
|
| 16 |
Discovery of SMP-304, a novel benzylpiperidine derivative with serotonin transporter inhibitory activity and 5-HT1A weak partial agonistic activity showing the antidepressant-like effect
|
Yoshinaga, Hidefumi
|
|
2017
|
25 |
1 |
p. 293-304
12 p.
|
artikel
|
| 17 |
Editorial board
|
|
|
2017
|
25 |
1 |
p. IFC-
1 p.
|
artikel
|
| 18 |
Enhanced potency of bivalent small molecule gp41 inhibitors
|
Sofiyev, Vladimir
|
|
2017
|
25 |
1 |
p. 408-420
13 p.
|
artikel
|
| 19 |
Evaluation of known and novel inhibitors of Orai1-mediated store operated Ca2+ entry in MDA-MB-231 breast cancer cells using a Fluorescence Imaging Plate Reader assay
|
Azimi, Iman
|
|
2017
|
25 |
1 |
p. 440-449
10 p.
|
artikel
|
| 20 |
Folic acid conjugates with photosensitizers for cancer targeting in photodynamic therapy: Synthesis and photophysical properties
|
Stallivieri, Aurélie
|
|
2017
|
25 |
1 |
p. 1-10
10 p.
|
artikel
|
| 21 |
Gaining in pan-affinity towards sigma 1 and sigma 2 receptors. SAR studies on arylalkylamines
|
Rossi, Daniela
|
|
2017
|
25 |
1 |
p. 11-19
9 p.
|
artikel
|
| 22 |
Identification of 4-(2-furanyl)pyrimidin-2-amines as Janus kinase 2 inhibitors
|
Wang, Yazhou
|
|
2017
|
25 |
1 |
p. 75-83
9 p.
|
artikel
|
| 23 |
Improved binding affinities of pyrrolidine derivatives as Mcl-1 inhibitors by modifying amino acid side chains
|
Wan, Yichao
|
|
2017
|
25 |
1 |
p. 138-152
15 p.
|
artikel
|
| 24 |
Lipid-modified oligonucleotide conjugates: Insights into gene silencing, interaction with model membranes and cellular uptake mechanisms
|
Ugarte-Uribe, Begoña
|
|
2017
|
25 |
1 |
p. 175-186
12 p.
|
artikel
|
| 25 |
Modulating amyloid-β aggregation: The effects of peptoid side chain placement and chirality
|
Turner, J. Phillip
|
|
2017
|
25 |
1 |
p. 20-26
7 p.
|
artikel
|
| 26 |
Neo-tanshinlactone D-ring modified novel analogues induce apoptosis in human breast cancer cell via DNA damage
|
Banerji, Biswadip
|
|
2017
|
25 |
1 |
p. 202-212
11 p.
|
artikel
|
| 27 |
New glutathione peroxidase mimetics—Insights into antioxidant and cytotoxic activity
|
Pacuła, Agata J.
|
|
2017
|
25 |
1 |
p. 126-131
6 p.
|
artikel
|
| 28 |
Novel 5-nitropyrimidine derivatives bearing endo-azabicyclic alcohols/amines as potent GPR119 agonists
|
Fang, Yuanying
|
|
2017
|
25 |
1 |
p. 254-260
7 p.
|
artikel
|
| 29 |
NTS2-selective neurotensin mimetics with tetrahydrofuran amino acids
|
Simeth, Nadja A.
|
|
2017
|
25 |
1 |
p. 350-359
10 p.
|
artikel
|
| 30 |
Optimization and bioevaluation of Cdc37-derived peptides: An insight into Hsp90-Cdc37 protein-protein interaction modulators
|
Wang, Lei
|
|
2017
|
25 |
1 |
p. 233-240
8 p.
|
artikel
|
| 31 |
Polyfluorinated salicylic acid derivatives as analogs of known drugs: Synthesis, molecular docking and biological evaluation
|
Shchegol'kov, E.V.
|
|
2017
|
25 |
1 |
p. 91-99
9 p.
|
artikel
|
| 32 |
Preliminary SAR and biological evaluation of antitubercular triazolothiadiazine derivatives against drug-susceptible and drug-resistant Mtb strains
|
Li, Ziqiang
|
|
2017
|
25 |
1 |
p. 213-220
8 p.
|
artikel
|
| 33 |
Rational design, synthesis, and structure–activity relationships of 5-amino-1H-pyrazole-4-carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors
|
Basu, Sujay
|
|
2017
|
25 |
1 |
p. 67-74
8 p.
|
artikel
|
| 34 |
Strategy for designing selective α-l-rhamnosidase inhibitors: Synthesis and biological evaluation of l-DMDP cyclic isothioureas
|
Miyawaki, Shota
|
|
2017
|
25 |
1 |
p. 107-115
9 p.
|
artikel
|
| 35 |
Structure-activity relationship-based screening of antibiotics against Gram-negative Acinetobacter baumannii
|
Lee, Jee-Young
|
|
2017
|
25 |
1 |
p. 372-380
9 p.
|
artikel
|
| 36 |
Structure-activity relationship study towards non-peptidic positron emission tomography (PET) radiotracer for gastrin releasing peptide receptors: Development of [18F] (S)-3-(1H-indol-3-yl)-N-[1-[5-(2-fluoroethoxy)pyridin-2-yl]cyclohexylmethyl]-2-methyl-2-[3-(4-nitrophenyl)ureido]propionamide
|
Lacivita, Enza
|
|
2017
|
25 |
1 |
p. 277-292
16 p.
|
artikel
|
| 37 |
Synthesis and biological evaluation of hesperetin derivatives as agents inducing apoptosis
|
Jung, Kang-Yeoun
|
|
2017
|
25 |
1 |
p. 397-407
11 p.
|
artikel
|
| 38 |
Synthesis and evaluation of naphthyl bearing 1,2,3-triazole analogs as antiplasmodial agents, cytotoxicity and docking studies
|
Balabadra, Saikrishna
|
|
2017
|
25 |
1 |
p. 221-232
12 p.
|
artikel
|
| 39 |
Synthesis and investigation of novel 6-(1,2,3-triazol-4-yl)-4-aminoquinazolin derivatives possessing hydroxamic acid moiety for cancer therapy
|
Ding, Chao
|
|
2017
|
25 |
1 |
p. 27-37
11 p.
|
artikel
|
| 40 |
Synthesis and in vitro antikinetoplastid activity of polyamine–hydroxybenzotriazole conjugates
|
Jagu, Elodie
|
|
2017
|
25 |
1 |
p. 84-90
7 p.
|
artikel
|
| 41 |
Synthesis and structure activity relationships of glycine amide derivatives as novel Vascular Adhesion Protein-1 inhibitors
|
Yamaki, Susumu
|
|
2017
|
25 |
1 |
p. 187-201
15 p.
|
artikel
|
| 42 |
Synthesis, anticancer, and docking studies of salicyl-hydrazone analogues: A novel series of small potent tropomyosin receptor kinase A inhibitors
|
Alam, Mohammad Sayed
|
|
2017
|
25 |
1 |
p. 389-396
8 p.
|
artikel
|
| 43 |
Synthesis, anti-proliferative activity, SAR study, and preliminary in vivo toxicity study of substituted N,N′-bis(arylmethyl)benzimidazolium salts against a panel of non-small cell lung cancer cell lines
|
Shelton, Kerri L.
|
|
2017
|
25 |
1 |
p. 421-439
19 p.
|
artikel
|
| 44 |
Synthesis, COX-1/2 inhibition activities and molecular docking study of isothiazolopyridine derivatives
|
Świątek, Piotr
|
|
2017
|
25 |
1 |
p. 316-326
11 p.
|
artikel
|
| 45 |
Synthesis, structure–activity relationship and molecular docking of 3-oxoaurones and 3-thioaurones as acetylcholinesterase and butyrylcholinesterase inhibitors
|
Mughal, Ehsan Ullah
|
|
2017
|
25 |
1 |
p. 100-106
7 p.
|
artikel
|
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