nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A concise synthesis and evaluation of new malonamide derivatives as potential α-glucosidase inhibitors
|
Islam, Mohammad Shahidul |
|
2016 |
24 |
8 |
p. 1675-1682 8 p. |
artikel |
2 |
Antiretroviral (HIV-1) activity of azulene derivatives
|
Peet, Julia |
|
2016 |
24 |
8 |
p. 1653-1657 5 p. |
artikel |
3 |
C-3 benzoic acid derivatives of C-3 deoxybetulinic acid and deoxybetulin as HIV-1 maturation inhibitors
|
Liu, Zheng |
|
2016 |
24 |
8 |
p. 1757-1770 14 p. |
artikel |
4 |
Compound profiling and 3D-QSAR studies of hydrazone derivatives with activity against intracellular Trypanosoma cruzi
|
Costa, Lívia Bandeira |
|
2016 |
24 |
8 |
p. 1608-1618 11 p. |
artikel |
5 |
Design and evaluation of novel glutaminase inhibitors
|
McDermott, Lee A. |
|
2016 |
24 |
8 |
p. 1819-1839 21 p. |
artikel |
6 |
Design and synthesis of small molecule-sulfotyrosine mimetics that inhibit HIV-1 entry
|
Dogo-Isonagie, Cajetan |
|
2016 |
24 |
8 |
p. 1718-1728 11 p. |
artikel |
7 |
Design and synthesis of thiourea derivatives with sulfur-containing heterocyclic scaffolds as potential tyrosinase inhibitors
|
Liu, Pingping |
|
2016 |
24 |
8 |
p. 1866-1871 6 p. |
artikel |
8 |
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents
|
Waszkielewicz, A.M. |
|
2016 |
24 |
8 |
p. 1793-1810 18 p. |
artikel |
9 |
Design, synthesis and biological evaluation of N,N-3-phenyl-3-benzylaminopropanamide derivatives as novel cholesteryl ester transfer protein inhibitor
|
Zhao, Dongmei |
|
2016 |
24 |
8 |
p. 1589-1597 9 p. |
artikel |
10 |
Design, synthesis, and evaluation of 2-piperidone derivatives for the inhibition of β-amyloid aggregation and inflammation mediated neurotoxicity
|
Li, Lei |
|
2016 |
24 |
8 |
p. 1853-1865 13 p. |
artikel |
11 |
Design, synthesis of phenstatin/isocombretastatin-oxindole conjugates as antimitotic agents
|
Kumar, G. Bharath |
|
2016 |
24 |
8 |
p. 1729-1740 12 p. |
artikel |
12 |
Design, synthesis, topoisomerase I & II inhibitory activity, antiproliferative activity, and structure–activity relationship study of pyrazoline derivatives: An ATP-competitive human topoisomerase IIα catalytic inhibitor
|
Ahmad, Pervez |
|
2016 |
24 |
8 |
p. 1898-1908 11 p. |
artikel |
13 |
Development of a fluorescent cardiomyocyte specific binding probe
|
Pes, Lara |
|
2016 |
24 |
8 |
p. 1706-1717 12 p. |
artikel |
14 |
Development of a potent 2-oxoamide inhibitor of secreted phospholipase A2 guided by molecular docking calculations and molecular dynamics simulations
|
Vasilakaki, Sofia |
|
2016 |
24 |
8 |
p. 1683-1695 13 p. |
artikel |
15 |
Discovery of new low-molecular-weight p53–Mdmx disruptors and their anti-cancer activities
|
Uesato, Shinichi |
|
2016 |
24 |
8 |
p. 1919-1926 8 p. |
artikel |
16 |
Discovery of novel N,N-3-phenyl-3-benzylaminopropionanilides as potent inhibitors of cholesteryl ester transfer protein in vivo
|
Xie, Honglei |
|
2016 |
24 |
8 |
p. 1811-1818 8 p. |
artikel |
17 |
Donor substrate promiscuity of bacterial β1–3-N-acetylglucosaminyltransferases and acceptor substrate flexibility of β1–4-galactosyltransferases
|
Li, Yanhong |
|
2016 |
24 |
8 |
p. 1696-1705 10 p. |
artikel |
18 |
Editorial board
|
|
|
2016 |
24 |
8 |
p. IFC- 1 p. |
artikel |
19 |
Evaluation of the anti-inflammatory action of curcumin analog (DM1): Effect on iNOS and COX-2 gene expression and autophagy pathways
|
Paulino, Niraldo |
|
2016 |
24 |
8 |
p. 1927-1935 9 p. |
artikel |
20 |
Exploration of 2-benzylbenzimidazole scaffold as novel inhibitor of NF-κB
|
Boggu, PullaReddy |
|
2016 |
24 |
8 |
p. 1872-1878 7 p. |
artikel |
21 |
Investigation of 4-amino-5-alkynylpyrimidine-2(1H)-ones as anti-mycobacterial agents
|
Garg, Gaurav |
|
2016 |
24 |
8 |
p. 1771-1777 7 p. |
artikel |
22 |
In vivo phase II-enzymes inducers, as potential chemopreventive agents, based on the chalcone and furoxan skeletons
|
Cabrera, Mauricio |
|
2016 |
24 |
8 |
p. 1665-1674 10 p. |
artikel |
23 |
Isatin analogs as novel inhibitors of Candida spp. β-carbonic anhydrase enzymes
|
Akdemir, Atilla |
|
2016 |
24 |
8 |
p. 1648-1652 5 p. |
artikel |
24 |
Molecular simulation of cyclohexanyl nucleic acid (CNA) duplexes with CNA, DNA and RNA and CNA triloop and tetraloop hairpin structures
|
Froeyen, Matheus |
|
2016 |
24 |
8 |
p. 1778-1785 8 p. |
artikel |
25 |
Novel indole-based melatonin analogues: Evaluation of antioxidant activity and protective effect against amyloid β-induced damage
|
Gurer-Orhan, Hande |
|
2016 |
24 |
8 |
p. 1658-1664 7 p. |
artikel |
26 |
Novel nicotine analogues with potential anti-mycobacterial activity
|
Gandhi, Paresh T. |
|
2016 |
24 |
8 |
p. 1637-1647 11 p. |
artikel |
27 |
Novel squaramides with in vitro liver stage antiplasmodial activity
|
Ribeiro, Carlos J.A. |
|
2016 |
24 |
8 |
p. 1786-1792 7 p. |
artikel |
28 |
Novel tricyclic pyrazolo[1,5-d][1,4]benzoxazepin-5(6H)-one: Design, synthesis, model and use as hMAO-B inhibitors
|
Chen, Rui |
|
2016 |
24 |
8 |
p. 1741-1748 8 p. |
artikel |
29 |
Quinoxalinone (Part II). Discovery of (Z)-3-(2-(pyridin-4-yl)vinyl)quinoxalinone derivates as potent VEGFR-2 kinase inhibitors
|
Shi, Leilei |
|
2016 |
24 |
8 |
p. 1840-1852 13 p. |
artikel |
30 |
Rational design, synthesis and biological evaluation of 1,3,4-oxadiazole pyrimidine derivatives as novel pyruvate dehydrogenase complex E1 inhibitors
|
He, Haifeng |
|
2016 |
24 |
8 |
p. 1879-1888 10 p. |
artikel |
31 |
Synthesis, and anticonvulsant activity of new amides derived from 3-methyl- or 3-ethyl-3-methyl-2,5-dioxo-pyrrolidin-1-yl-acetic acids
|
Obniska, Jolanta |
|
2016 |
24 |
8 |
p. 1598-1607 10 p. |
artikel |
32 |
Synthesis and biological evaluation of quinoline derivatives as potential anti-prostate cancer agents and Pim-1 kinase inhibitors
|
Li, Kun |
|
2016 |
24 |
8 |
p. 1889-1897 9 p. |
artikel |
33 |
Synthesis, and docking studies of phenylpyrimidine-carboxamide derivatives bearing 1H-pyrrolo[2,3-b]pyridine moiety as c-Met inhibitors
|
Zhu, Wufu |
|
2016 |
24 |
8 |
p. 1749-1756 8 p. |
artikel |
34 |
Thiadiazole derivatives as New Class of β-glucuronidase inhibitors
|
Salar, Uzma |
|
2016 |
24 |
8 |
p. 1909-1918 10 p. |
artikel |
35 |
1,2,4-Triazolyl octahydropyrrolo[2,3-b]pyrroles: A new series of potent and selective dopamine D3 receptor antagonists
|
Micheli, Fabrizio |
|
2016 |
24 |
8 |
p. 1619-1636 18 p. |
artikel |