nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A new GLP-1 analogue with prolonged glucose-lowering activity in vivo via backbone-based modification at the N-terminus
|
Bai, Xiaohui |
|
2016 |
24 |
6 |
p. 1163-1170 8 p. |
artikel |
2 |
A photo-cleavable biotin affinity tag for the facile release of a photo-crosslinked carbohydrate-binding protein
|
Chang, Tsung-Che |
|
2016 |
24 |
6 |
p. 1216-1224 9 p. |
artikel |
3 |
A potent and selective inhibitor targeting human and murine 12/15-LOX
|
Armstrong, Michelle M. |
|
2016 |
24 |
6 |
p. 1183-1190 8 p. |
artikel |
4 |
Application of PEG-400 as a green biodegradable polymeric medium for the catalyst-free synthesis of spiro-dihydropyridines and their use as acetyl and butyrylcholinesterase inhibitors
|
Maryamabadi, Ammar |
|
2016 |
24 |
6 |
p. 1408-1417 10 p. |
artikel |
5 |
Candida albicans β-1,2 mannosyl transferase Bmt3: Preparation and evaluation of a β (1,2), α (1,2)-tetramannosyl fluorescent substrate
|
Cattiaux, Laurent |
|
2016 |
24 |
6 |
p. 1362-1368 7 p. |
artikel |
6 |
Design and synthesis of a series of serine derivatives as small molecule inhibitors of the SARS coronavirus 3CL protease
|
Konno, Hiroyuki |
|
2016 |
24 |
6 |
p. 1241-1254 14 p. |
artikel |
7 |
Design, RNA cleavage and antiviral activity of new artificial ribonucleases derived from mono-, di- and tripeptides connected by linkers of different hydrophobicity
|
Tamkovich, Nikolay |
|
2016 |
24 |
6 |
p. 1346-1355 10 p. |
artikel |
8 |
Design, synthesis and biological evaluation of dinucleotide mRNA cap analog containing propargyl moiety
|
Shanmugasundaram, Muthian |
|
2016 |
24 |
6 |
p. 1204-1208 5 p. |
artikel |
9 |
Design, synthesis and biological evaluation of imidazo[2,1-b]thiazole and benzo[d]imidazo[2,1-b]thiazole derivatives as Mycobacterium tuberculosis pantothenate synthetase inhibitors
|
Samala, Ganesh |
|
2016 |
24 |
6 |
p. 1298-1307 10 p. |
artikel |
10 |
Design, synthesis and biological evaluation of novel 4-phenoxy-6,7-disubstituted quinolines possessing (thio)semicarbazones as c-Met kinase inhibitors
|
Zhai, Xin |
|
2016 |
24 |
6 |
p. 1331-1345 15 p. |
artikel |
11 |
Development of 3-(4-aminosulphonyl)-phenyl-2-mercapto-3H-quinazolin-4-ones as inhibitors of carbonic anhydrase isoforms involved in tumorigenesis and glaucoma
|
Alafeefy, Ahmed M. |
|
2016 |
24 |
6 |
p. 1402-1407 6 p. |
artikel |
12 |
Discovery of human Golgi β-galactosidase with no identified glycosidase using a QMC substrate design platform for exo-glycosidase
|
Miura, Kazuki |
|
2016 |
24 |
6 |
p. 1369-1375 7 p. |
artikel |
13 |
Editorial board
|
|
|
2016 |
24 |
6 |
p. IFC- 1 p. |
artikel |
14 |
Flexible double-headed cytosine-linked 2′-deoxycytidine nucleotides. Synthesis, polymerase incorporation to DNA and interaction with DNA methyltransferases
|
Kielkowski, Pavel |
|
2016 |
24 |
6 |
p. 1268-1276 9 p. |
artikel |
15 |
From indole to pyrrole, furan, thiophene and pyridine: Search for novel small molecule inhibitors of bacterial transcription initiation complex formation
|
Thach, Oscar |
|
2016 |
24 |
6 |
p. 1171-1182 12 p. |
artikel |
16 |
Functionalized imidazolium and benzimidazolium salts as paraoxonase 1 inhibitors: Synthesis, characterization and molecular docking studies
|
Karataş, Mert Olgun |
|
2016 |
24 |
6 |
p. 1392-1401 10 p. |
artikel |
17 |
4H-Chromene-based anticancer agents towards multi-drug resistant HL60/MX2 human leukemia: SAR at the 4th and 6th positions
|
Puppala, Manohar |
|
2016 |
24 |
6 |
p. 1292-1297 6 p. |
artikel |
18 |
Identification of spirooxindole and dibenzoxazepine motifs as potent mineralocorticoid receptor antagonists
|
Lotesta, Stephen D. |
|
2016 |
24 |
6 |
p. 1384-1391 8 p. |
artikel |
19 |
99mTc-bioorthogonal click chemistry reagent for in vivo pretargeted imaging
|
García, María Fernanda |
|
2016 |
24 |
6 |
p. 1209-1215 7 p. |
artikel |
20 |
New derivative of 2-(2,4-dihydroxyphenyl)thieno-1,3-thiazin-4-one (BChTT) elicits antiproliferative effect via p38-mediated cell cycle arrest in cancer cells
|
Juszczak, Małgorzata |
|
2016 |
24 |
6 |
p. 1356-1361 6 p. |
artikel |
21 |
Recognition and detection of 8-oxo-rG in RNA using the DNA/OMeRNA chimera probes containing fluorescent adenosine-diazaphenoxazine analog
|
Koga, Yohei |
|
2016 |
24 |
6 |
p. 1308-1313 6 p. |
artikel |
22 |
Salicylanilide N-monosubstituted carbamates: Synthesis and in vitro antimicrobial activity
|
Krátký, Martin |
|
2016 |
24 |
6 |
p. 1322-1330 9 p. |
artikel |
23 |
2-Sulfonamidopyridine C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists
|
Ann, Jihyae |
|
2016 |
24 |
6 |
p. 1231-1240 10 p. |
artikel |
24 |
Synthesis and antibacterial evaluation of novel 4″-glycyl linked quinolyl-azithromycins with potent activity against macrolide-resistant pathogens
|
Pavlović, Dražen |
|
2016 |
24 |
6 |
p. 1255-1267 13 p. |
artikel |
25 |
Synthesis and biological evaluation of novel inhibitors against 1,3,8-trihydroxynaphthalene reductase from Magnaporthe grisea
|
Chen, Haifeng |
|
2016 |
24 |
6 |
p. 1225-1230 6 p. |
artikel |
26 |
Synthesis and evaluation of thiophene-based guanylhydrazones (iminoguanidines) efficient against panel of voriconazole-resistant fungal isolates
|
Ajdačić, Vladimir |
|
2016 |
24 |
6 |
p. 1277-1291 15 p. |
artikel |
27 |
Synthesis and pharmacological evaluation of nucleoside prodrugs designed to target siderophore biosynthesis in Mycobacterium tuberculosis
|
Dawadi, Surendra |
|
2016 |
24 |
6 |
p. 1314-1321 8 p. |
artikel |
28 |
Synthesis of fluorinated carbazoles via C–H arylation catalyzed by Pd/Cu bimetal system and their antibacterial activities
|
Kong, Xianqiang |
|
2016 |
24 |
6 |
p. 1376-1383 8 p. |
artikel |
29 |
The molecular structure of thio-ether fatty acids influences PPAR-dependent regulation of lipid metabolism
|
Lund, Jenny |
|
2016 |
24 |
6 |
p. 1191-1203 13 p. |
artikel |