| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Active site-directed plasmin inhibitors: Extension on the P2 residue
|
Hidaka, Koushi
|
|
2016
|
24 |
4 |
p. 545-553
9 p.
|
artikel
|
| 2 |
Allosteric inhibitors of Coxsackie virus A24 RNA polymerase
|
Schein, Catherine H.
|
|
2016
|
24 |
4 |
p. 570-577
8 p.
|
artikel
|
| 3 |
An appraisal on recent medicinal perspective of curcumin degradant: Dehydrozingerone (DZG)
|
Hampannavar, Girish A.
|
|
2016
|
24 |
4 |
p. 501-520
20 p.
|
artikel
|
| 4 |
A new chromanone derivative isolated from Hypericum lissophloeus (Hypericaceae) potentiates GABAA receptor currents in a subunit specific fashion
|
Crockett, Sara
|
|
2016
|
24 |
4 |
p. 681-685
5 p.
|
artikel
|
| 5 |
Cloning, characterization and anion inhibition studies of a γ-carbonic anhydrase from the Antarctic bacterium Colwellia psychrerythraea
|
De Luca, Viviana
|
|
2016
|
24 |
4 |
p. 835-840
6 p.
|
artikel
|
| 6 |
Cyclic RGD peptidomimetics containing 4- and 5-amino-cyclopropane pipecolic acid (CPA) templates as dual αVβ3 and α5β1 integrin ligands
|
Sernissi, Lorenzo
|
|
2016
|
24 |
4 |
p. 703-711
9 p.
|
artikel
|
| 7 |
Design and synthesis of an activity-based protein profiling probe derived from cinnamic hydroxamic acid
|
Ai, Teng
|
|
2016
|
24 |
4 |
p. 686-692
7 p.
|
artikel
|
| 8 |
Design and synthesis of calindol derivatives as potent and selective calcium sensing receptor agonists
|
Kiefer, Lionel
|
|
2016
|
24 |
4 |
p. 554-569
16 p.
|
artikel
|
| 9 |
Design and synthesis of novel androgen receptor antagonists via molecular modeling
|
Zhao, Chao
|
|
2016
|
24 |
4 |
p. 789-801
13 p.
|
artikel
|
| 10 |
Design, synthesis and biological evaluation of novel analgesic agents targeting both cyclooxygenase and TRPV1
|
Yan, Lin
|
|
2016
|
24 |
4 |
p. 849-857
9 p.
|
artikel
|
| 11 |
Design, synthesis, and docking studies of phenylpicolinamide derivatives bearing 1H-pyrrolo[2,3-b]pyridine moiety as c-Met inhibitors
|
Zhu, Wufu
|
|
2016
|
24 |
4 |
p. 812-819
8 p.
|
artikel
|
| 12 |
Design, synthesis and evaluation of novel 7-aminoalkyl-substituted flavonoid derivatives with improved cholinesterase inhibitory activities
|
Luo, Wen
|
|
2016
|
24 |
4 |
p. 672-680
9 p.
|
artikel
|
| 13 |
Development of acridine derivatives as selective Mycobacterium tuberculosis DNA gyrase inhibitors
|
Medapi, Brahmam
|
|
2016
|
24 |
4 |
p. 877-885
9 p.
|
artikel
|
| 14 |
2,3-Dihydrobenzofuran privileged structures as new bioinspired lead compounds for the design of mPGES-1 inhibitors
|
Di Micco, Simone
|
|
2016
|
24 |
4 |
p. 820-826
7 p.
|
artikel
|
| 15 |
Discovery of 2-(1H-indol-5-ylamino)-6-(2,4-difluorophenylsulfonyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one (7ao) as a potent selective inhibitor of Polo like kinase 2 (PLK2)
|
Reddy, M.V. Ramana
|
|
2016
|
24 |
4 |
p. 521-544
24 p.
|
artikel
|
| 16 |
DNA cleavage at the AP site via β-elimination mediated by the AP site-binding ligands
|
Abe, Yukiko S.
|
|
2016
|
24 |
4 |
p. 910-914
5 p.
|
artikel
|
| 17 |
Editorial board
|
|
|
2016
|
24 |
4 |
p. IFC-
1 p.
|
artikel
|
| 18 |
Expanding the structural diversity of diarylureas as multi-target tyrosine kinase inhibitors
|
Shan, Yuanyuan
|
|
2016
|
24 |
4 |
p. 750-758
9 p.
|
artikel
|
| 19 |
Ferulic acid–carbazole hybrid compounds: Combination of cholinesterase inhibition, antioxidant and neuroprotection as multifunctional anti-Alzheimer agents
|
Fang, Lei
|
|
2016
|
24 |
4 |
p. 886-893
8 p.
|
artikel
|
| 20 |
Fluorinated matrix metalloproteinases inhibitors—Phosphonate based potential probes for positron emission tomography
|
Beutel, Bernd
|
|
2016
|
24 |
4 |
p. 902-909
8 p.
|
artikel
|
| 21 |
Hydroxylated chalcones with dual properties: Xanthine oxidase inhibitors and radical scavengers
|
Hofmann, Emily
|
|
2016
|
24 |
4 |
p. 578-587
10 p.
|
artikel
|
| 22 |
Identification of B. anthracis N5-carboxyaminoimidazole ribonucleotide mutase (PurE) active site binding compounds via fragment library screening
|
Lei, Hao
|
|
2016
|
24 |
4 |
p. 596-605
10 p.
|
artikel
|
| 23 |
Illuminating the binding interactions of galactonoamidines during the inhibition of β-galactosidase (E. coli)
|
Fan, Qiu-Hua
|
|
2016
|
24 |
4 |
p. 661-671
11 p.
|
artikel
|
| 24 |
Investigating molecular dynamics-guided lead optimization of EGFR inhibitors
|
Lavecchia, Martin J.
|
|
2016
|
24 |
4 |
p. 768-778
11 p.
|
artikel
|
| 25 |
N-(3,4-Dimethylisoxazol-5-yl)piperazine-4-[4-(2-fluoro-4-[11C]methylphenyl)thiazol-2-yl]-1-carboxamide: A promising positron emission tomography ligand for fatty acid amide hydrolase
|
Shimoda, Yoko
|
|
2016
|
24 |
4 |
p. 627-634
8 p.
|
artikel
|
| 26 |
New hybrid molecules with anticonvulsant and antinociceptive activity derived from 3-methyl- or 3,3-dimethyl-1-[1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl]pyrrolidine-2,5-diones
|
Kamiński, Krzysztof
|
|
2016
|
24 |
4 |
p. 606-618
13 p.
|
artikel
|
| 27 |
New MKLP-2 inhibitors in the paprotrain series: Design, synthesis and biological evaluations
|
Labrière, Christophe
|
|
2016
|
24 |
4 |
p. 721-734
14 p.
|
artikel
|
| 28 |
Novel triazolothiadiazines act as potent anticancer agents in liver cancer cells through Akt and ASK-1 proteins
|
Aytaç, Peri S.
|
|
2016
|
24 |
4 |
p. 858-872
15 p.
|
artikel
|
| 29 |
Phytochemical meanings of tetrahydro-β-carboline moiety in strictosidine derivatives
|
Sudžuković, Nicole
|
|
2016
|
24 |
4 |
p. 588-595
8 p.
|
artikel
|
| 30 |
Semisynthetic routes to PF1022H—A precursor for new derivatives of the anthelmintic cyclooctadepsipeptide PF1022A
|
Sivanathan, Sivatharushan
|
|
2016
|
24 |
4 |
p. 873-876
4 p.
|
artikel
|
| 31 |
Structural features underlying raloxifene’s biophysical interaction with bone matrix
|
Bivi, Nicoletta
|
|
2016
|
24 |
4 |
p. 759-767
9 p.
|
artikel
|
| 32 |
Sulfamide derivatives with selective carbonic anhydrase VII inhibitory action
|
Villalba, Maria Luisa
|
|
2016
|
24 |
4 |
p. 894-901
8 p.
|
artikel
|
| 33 |
Sulfonamides incorporating heteropolycyclic scaffolds show potent inhibitory action against carbonic anhydrase isoforms I, II, IX and XII
|
Barresi, Elisabetta
|
|
2016
|
24 |
4 |
p. 921-927
7 p.
|
artikel
|
| 34 |
Synthesis and anti-tuberculosis activity of glycitylamines
|
Corkran, Hilary M.
|
|
2016
|
24 |
4 |
p. 693-702
10 p.
|
artikel
|
| 35 |
Synthesis and biological activity of ferrocenyl indeno[1,2-c]isoquinolines as topoisomerase II inhibitors
|
Wambang, Nathalie
|
|
2016
|
24 |
4 |
p. 651-660
10 p.
|
artikel
|
| 36 |
Synthesis and biological evaluation of disubstituted amidoxanthones as potential telomeric G-quadruplex DNA-binding and apoptosis-inducing agents
|
Shen, Rui
|
|
2016
|
24 |
4 |
p. 619-626
8 p.
|
artikel
|
| 37 |
Synthesis and biological evaluation of novel 5-hydroxylaminoisoxazole derivatives as lipoxygenase inhibitors and metabolism enhancing agents
|
Averina, Elena B.
|
|
2016
|
24 |
4 |
p. 712-720
9 p.
|
artikel
|
| 38 |
Synthesis and biological evaluation of 3-tetrazolo steroidal analogs: Novel class of 5α-reductase inhibitors
|
Aggarwal, Saurabh
|
|
2016
|
24 |
4 |
p. 779-788
10 p.
|
artikel
|
| 39 |
Synthesis and evaluation of styrylpyran fluorophores for noninvasive detection of cerebral β-amyloid deposits
|
Zhu, Bi-yue
|
|
2016
|
24 |
4 |
p. 827-834
8 p.
|
artikel
|
| 40 |
Synthesis and immunological evaluation of N-acyl modified Tn analogues as anticancer vaccine candidates
|
Song, Chengcheng
|
|
2016
|
24 |
4 |
p. 915-920
6 p.
|
artikel
|
| 41 |
Synthesis, antimicrobial evaluation and molecular modeling of 5-hydroxyisoquinolinium salt series; the effect of the hydroxyl moiety
|
Soukup, Ondrej
|
|
2016
|
24 |
4 |
p. 841-848
8 p.
|
artikel
|
| 42 |
Synthesis, characterization and antimicrobial activities of novel silver(I) complexes with coumarin substituted N-heterocyclic carbene ligands
|
Karataş, Mert Olgun
|
|
2016
|
24 |
4 |
p. 643-650
8 p.
|
artikel
|
| 43 |
Synthesis, isomerization and biological activity of novel 2-selenohydantoin derivatives
|
Ivanenkov, Yan A.
|
|
2016
|
24 |
4 |
p. 802-811
10 p.
|
artikel
|
| 44 |
Synthesis of novel polybrominated benzimidazole derivatives—potential CK2 inhibitors with anticancer and proapoptotic activity
|
Łukowska-Chojnacka, Edyta
|
|
2016
|
24 |
4 |
p. 735-741
7 p.
|
artikel
|
| 45 |
Synthesis, structure, and evaluation of a β-cyclodextrin-artificial carbohydrate conjugate for use as a doxorubicin-carrying molecule
|
Yamanoi, Takashi
|
|
2016
|
24 |
4 |
p. 635-642
8 p.
|
artikel
|
| 46 |
Three new double-headed nucleotides with additional nucleobases connected to C-5 of pyrimidines; synthesis, duplex and triplex studies
|
Kumar, Pawan
|
|
2016
|
24 |
4 |
p. 742-749
8 p.
|
artikel
|
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