| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
6-Aryl-4-amino-pyrimido[4,5-b]indole 2′-deoxyribonucleoside triphosphates (benzo-fused 7-deaza-dATP analogues): Synthesis, fluorescent properties, enzymatic incorporation into DNA and DNA-protein binding study
|
Bosáková, Andrea
|
|
2016
|
24 |
19 |
p. 4528-4535
8 p.
|
artikel
|
| 2 |
3-Arylpropionylhydroxamic acid derivatives as Helicobacter pylori urease inhibitors: Synthesis, molecular docking and biological evaluation
|
Shi, Wei-Kang
|
|
2016
|
24 |
19 |
p. 4519-4527
9 p.
|
artikel
|
| 3 |
Ca-asp bound X-ray structure and inhibition of Bacillus anthracis dihydroorotase (DHOase)
|
Rice, Amy J.
|
|
2016
|
24 |
19 |
p. 4536-4543
8 p.
|
artikel
|
| 4 |
Coumarin derivatives as potential inhibitors of acetylcholinesterase: Synthesis, molecular docking and biological studies
|
Singla, Shaffali
|
|
2016
|
24 |
19 |
p. 4587-4599
13 p.
|
artikel
|
| 5 |
CpG methylation increases the DNA binding of 9-aminoacridine carboxamide Pt analogues
|
Kava, Hieronimus W.
|
|
2016
|
24 |
19 |
p. 4701-4710
10 p.
|
artikel
|
| 6 |
Design, synthesis, and biological evaluation of 1,9-diheteroarylnona-1,3,6,8-tetraen-5-ones as a new class of anti-prostate cancer agents
|
Zhang, Xiaojie
|
|
2016
|
24 |
19 |
p. 4692-4700
9 p.
|
artikel
|
| 7 |
Design, synthesis and biological evaluation of novel hamamelitannin analogues as potentiators for vancomycin in the treatment of biofilm related Staphylococcus aureus infections
|
Vermote, Arno
|
|
2016
|
24 |
19 |
p. 4563-4575
13 p.
|
artikel
|
| 8 |
Design, synthesis, and evaluation of 4,6-diaminonicotinamide derivatives as novel and potent immunomodulators targeting JAK3
|
Nakajima, Yutaka
|
|
2016
|
24 |
19 |
p. 4711-4722
12 p.
|
artikel
|
| 9 |
Discovery and antiparasitic activity of AZ960 as a Trypanosoma brucei ERK8 inhibitor
|
Valenciano, Ana L.
|
|
2016
|
24 |
19 |
p. 4647-4651
5 p.
|
artikel
|
| 10 |
Discovery and synthetic optimization of a novel scaffold for hydrophobic tunnel-targeted autotaxin inhibition
|
Ragle, Lauren E.
|
|
2016
|
24 |
19 |
p. 4660-4674
15 p.
|
artikel
|
| 11 |
Discovery of a 7-arylaminobenzimidazole series as novel CRF1 receptor antagonists
|
Mochizuki, Michiyo
|
|
2016
|
24 |
19 |
p. 4675-4691
17 p.
|
artikel
|
| 12 |
Discovery of N-(benzyloxy)-1,3-diphenyl-1H-pyrazole-4-carboxamide derivatives as potential antiproliferative agents by inhibiting MEK
|
Lv, Xian-Hai
|
|
2016
|
24 |
19 |
p. 4652-4659
8 p.
|
artikel
|
| 13 |
Editorial board
|
|
|
2016
|
24 |
19 |
p. IFC-
1 p.
|
artikel
|
| 14 |
2-(4-Fluorophenyl)-quinazolin-4(3H)-one as a novel tyrosinase inhibitor: Synthesis, inhibitory activity, and mechanism
|
Wang, Rui
|
|
2016
|
24 |
19 |
p. 4620-4625
6 p.
|
artikel
|
| 15 |
In vitro cytotoxicity of novel 2,5,7-tricarbo-substituted indoles derived from 2-amino-5-bromo-3-iodoacetophenone
|
Mphahlele, Malose J.
|
|
2016
|
24 |
19 |
p. 4576-4586
11 p.
|
artikel
|
| 16 |
New antiproliferative 7-(4-(N-substituted carbamoylmethyl)piperazin-1-yl) derivatives of ciprofloxacin induce cell cycle arrest at G2/M phase
|
Mohammed, Hamada H.H.
|
|
2016
|
24 |
19 |
p. 4636-4646
11 p.
|
artikel
|
| 17 |
Novel small molecule binders of human N-glycanase 1, a key player in the endoplasmic reticulum associated degradation pathway
|
Srinivasan, Bharath
|
|
2016
|
24 |
19 |
p. 4750-4758
9 p.
|
artikel
|
| 18 |
Novel tricyclic poly (ADP-ribose) polymerase-1/2 inhibitors with potent anticancer chemopotentiating activity: Design, synthesis and biological evaluation
|
Li, Hui
|
|
2016
|
24 |
19 |
p. 4731-4740
10 p.
|
artikel
|
| 19 |
Oleanolic acid-NO donor-platinum(II) trihybrid molecules: Targeting cytotoxicity on hepatoma cells with combined action mode and good safety
|
Fang, Lei
|
|
2016
|
24 |
19 |
p. 4611-4619
9 p.
|
artikel
|
| 20 |
2-Oxoamide inhibitors of cytosolic group IVA phospholipase A2 with reduced lipophilicity
|
Antonopoulou, Georgia
|
|
2016
|
24 |
19 |
p. 4544-4554
11 p.
|
artikel
|
| 21 |
Structure–activity relationship of Garcinia xanthones analogues: Potent Hsp90 inhibitors with cytotoxicity and antiangiogenesis activity
|
Xu, Xiaoli
|
|
2016
|
24 |
19 |
p. 4626-4635
10 p.
|
artikel
|
| 22 |
Synthesis and aromatase inhibitory evaluation of 4-N-nitrophenyl substituted amino-4H-1,2,4-triazole derivatives
|
Song, Zhidan
|
|
2016
|
24 |
19 |
p. 4723-4730
8 p.
|
artikel
|
| 23 |
Synthesis and evaluation of 8-hydroxyquinolin derivatives substituted with (benzo[d][1,2]selenazol-3(2H)-one) as effective inhibitor of metal-induced Aβ aggregation and antioxidant
|
Wang, Bo
|
|
2016
|
24 |
19 |
p. 4741-4749
9 p.
|
artikel
|
| 24 |
The human tyrosine kinase Kit and its gatekeeper mutant T670I, show different kinetic properties: Implications for drug design
|
Kissova, Miroslava
|
|
2016
|
24 |
19 |
p. 4555-4562
8 p.
|
artikel
|
| 25 |
Toward chelerythrine optimization: Analogues designed by molecular simplification exhibit selective growth inhibition in non-small-cell lung cancer cells
|
Yang, Rosania
|
|
2016
|
24 |
19 |
p. 4600-4610
11 p.
|
artikel
|
| 26 |
Towards the PET radiotracer for p75 neurotrophin receptor: [11C]LM11A-24 shows biological activity in vitro, but unfavorable ex vivo and in vivo profile
|
Gibon, Julien
|
|
2016
|
24 |
19 |
p. 4759-4765
7 p.
|
artikel
|
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