| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Anion inhibition profiles of the complete domain of the η-carbonic anhydrase from Plasmodium falciparum
|
Del Prete, Sonia
|
|
2016
|
24 |
18 |
p. 4410-4414
5 p.
|
artikel
|
| 2 |
Antibacterial and anticancer activity of a series of novel peptides incorporating cyclic tetra-substituted Cα amino acids
|
Hicks, Rickey P.
|
|
2016
|
24 |
18 |
p. 4056-4065
10 p.
|
artikel
|
| 3 |
Anti-inflammatory properties of pterocarpanquinone LQB-118 in mice
|
Riça, Ingred G.
|
|
2016
|
24 |
18 |
p. 4415-4423
9 p.
|
artikel
|
| 4 |
Antileishmanial activity of new thiophene–indole hybrids: Design, synthesis, biological and cytotoxic evaluation, and chemometric studies
|
Félix, Mayara B.
|
|
2016
|
24 |
18 |
p. 3972-3977
6 p.
|
artikel
|
| 5 |
Antioxidant, anticancer activities and mechanistic studies of the flavone glycoside diosmin and its oxidovanadium(IV) complex. Interactions with bovine serum albumin
|
Naso, Luciana
|
|
2016
|
24 |
18 |
p. 4108-4119
12 p.
|
artikel
|
| 6 |
Arylazolyl(azinyl)thioacetanilides. Part 20: Discovery of novel purinylthioacetanilides derivatives as potent HIV-1 NNRTIs via a structure-based bioisosterism approach
|
Lu, Xueyi
|
|
2016
|
24 |
18 |
p. 4424-4433
10 p.
|
artikel
|
| 7 |
Bacterial versus human sphingosine-1-phosphate lyase (S1PL) in the design of potential S1PL inhibitors
|
Sanllehí, Pol
|
|
2016
|
24 |
18 |
p. 4381-4389
9 p.
|
artikel
|
| 8 |
Binding mode prediction of aplysiatoxin, a potent agonist of protein kinase C, through molecular simulation and structure–activity study on simplified analogs of the receptor-recognition domain
|
Ashida, Yoshiki
|
|
2016
|
24 |
18 |
p. 4218-4227
10 p.
|
artikel
|
| 9 |
Bortezomib inhibits bacterial and fungal β-carbonic anhydrases
|
Supuran, Claudiu T.
|
|
2016
|
24 |
18 |
p. 4406-4409
4 p.
|
artikel
|
| 10 |
Characterization of the action of tyrosinase on resorcinols
|
Garcia-Jimenez, Antonio
|
|
2016
|
24 |
18 |
p. 4434-4443
10 p.
|
artikel
|
| 11 |
Cholinesterase inhibitory activity of isoquinoline alkaloids from three Cryptocarya species (Lauraceae)
|
Wan Othman, Wan Nurul Nazneem
|
|
2016
|
24 |
18 |
p. 4464-4469
6 p.
|
artikel
|
| 12 |
Corrigendum to “Structural features underlying raloxifene’s biophysical interaction with bone matrix” [Bioorg. Med. Chem. 24 (2016) 759–767]
|
Bivi, Nicoletta
|
|
2016
|
24 |
18 |
p. 4516-
1 p.
|
artikel
|
| 13 |
Corrigendum to “Synthesis and evaluation of novel 1H-pyrrolo[2,3-b]pyridine-5-carboxamide derivatives as potent and orally efficacious immunomodulators targeting JAK3” [Bioorg. Med. Chem. 23 (2015) 4871–4883]
|
Nakajima, Yutaka
|
|
2016
|
24 |
18 |
p. 4517-
1 p.
|
artikel
|
| 14 |
Design and comparative anticonvulsant activity assessment of CNS-active alkyl-carbamoyl imidazole derivatives
|
Mawasi, Hafiz
|
|
2016
|
24 |
18 |
p. 4246-4253
8 p.
|
artikel
|
| 15 |
Design and development of new class of Mycobacterium tuberculosis l-alanine dehydrogenase inhibitors
|
Reshma, Rudraraju Srilakshmi
|
|
2016
|
24 |
18 |
p. 4499-4508
10 p.
|
artikel
|
| 16 |
Design of cyclic RGD-conjugated Aib-containing amphipathic helical peptides for targeted delivery of small interfering RNA
|
Wada, Shun-ichi
|
|
2016
|
24 |
18 |
p. 4478-4485
8 p.
|
artikel
|
| 17 |
Design, synthesis and anti-P. falciparum activity of pyrazolopyridine–sulfonamide derivatives
|
Silva, Thais B.
|
|
2016
|
24 |
18 |
p. 4492-4498
7 p.
|
artikel
|
| 18 |
Design, synthesis, and evaluation of Trolox-conjugated amyloid-β C-terminal peptides for therapeutic intervention in an in vitro model of Alzheimer’s disease
|
Arai, Takuya
|
|
2016
|
24 |
18 |
p. 4138-4143
6 p.
|
artikel
|
| 19 |
Design, synthesis, and mode of action studies of a mitomycin tetramer inducing double activations with a single probe
|
Kim, Hyoung Rae
|
|
2016
|
24 |
18 |
p. 4023-4031
9 p.
|
artikel
|
| 20 |
Design, synthesis, molecular docking and biological evaluation of thiophen-2-iminothiazolidine derivatives for use against Trypanosoma cruzi
|
Silva-Júnior, E.F.
|
|
2016
|
24 |
18 |
p. 4228-4240
13 p.
|
artikel
|
| 21 |
Detection of l-alanylaminopeptidase activity in microorganisms using fluorogenic self-immolative enzyme substrates
|
Cellier, Marie
|
|
2016
|
24 |
18 |
p. 4066-4074
9 p.
|
artikel
|
| 22 |
Development of ethynyl-2′-deoxyuridine chemical probes for cell proliferation
|
Lovitt, Carrie J.
|
|
2016
|
24 |
18 |
p. 4272-4280
9 p.
|
artikel
|
| 23 |
Dideoxy nucleoside triphosphate (ddNTP) analogues: Synthesis and polymerase substrate activities of pyrrolidinyl nucleoside triphosphates (prNTPs)
|
Gade, Chandrasekhar Reddy
|
|
2016
|
24 |
18 |
p. 4016-4022
7 p.
|
artikel
|
| 24 |
Discovery and optimization of a series of imidazo[4,5-b]pyrazine derivatives as highly potent and exquisitely selective inhibitors of the mesenchymal–epithelial transition factor (c-Met) protein kinase
|
Zhao, Fei
|
|
2016
|
24 |
18 |
p. 4281-4290
10 p.
|
artikel
|
| 25 |
Discovery of a new type of scaffold for the creation of novel tyrosinase inhibitors
|
Oyama, Takahiro
|
|
2016
|
24 |
18 |
p. 4509-4515
7 p.
|
artikel
|
| 26 |
Discovery of a potent and highly selective transforming growth factor β receptor-associated kinase 1 (TAK1) inhibitor by structure based drug design (SBDD)
|
Muraoka, Terushige
|
|
2016
|
24 |
18 |
p. 4206-4217
12 p.
|
artikel
|
| 27 |
Dual and antagonic therapeutic effects of sulfated glycans
|
Pomin, Vitor H.
|
|
2016
|
24 |
18 |
p. 3965-3971
7 p.
|
artikel
|
| 28 |
Editorial board
|
|
|
2016
|
24 |
18 |
p. IFC-
1 p.
|
artikel
|
| 29 |
Effects of stereochemistry, saturation, and hydrocarbon chain length on the ability of synthetic constrained azacyclic sphingolipids to trigger nutrient transporter down-regulation, vacuolation, and cell death
|
Perryman, Michael S.
|
|
2016
|
24 |
18 |
p. 4390-4397
8 p.
|
artikel
|
| 30 |
Exploring new scaffolds for angiotensin II receptor antagonism
|
Kritsi, Eftichia
|
|
2016
|
24 |
18 |
p. 4444-4451
8 p.
|
artikel
|
| 31 |
Functional foldamers that target bacterial membranes: The effect of charge, amphiphilicity and conformation
|
Patil-Sen, Yogita
|
|
2016
|
24 |
18 |
p. 4241-4245
5 p.
|
artikel
|
| 32 |
Identification of the first small-molecule inhibitor of the REV7 DNA repair protein interaction
|
Actis, Marcelo L.
|
|
2016
|
24 |
18 |
p. 4339-4346
8 p.
|
artikel
|
| 33 |
Identification of the minimum pharmacophore of lipid–phosphatidylserine (PS) binding peptide–peptoid hybrid PPS1D1
|
Singh, Jaspal
|
|
2016
|
24 |
18 |
p. 4470-4477
8 p.
|
artikel
|
| 34 |
Inhibitors for the bacterial ectonucleotidase Lp1NTPDase from Legionella pneumophila
|
Fiene, Amelie
|
|
2016
|
24 |
18 |
p. 4363-4371
9 p.
|
artikel
|
| 35 |
Introduction of perfluoroalkyl chain into the esterifying moiety of bacteriochlorophyll c in the green sulfur photosynthetic bacterium Chlorobaculum tepidum by pigment biosynthesis
|
Saga, Yoshitaka
|
|
2016
|
24 |
18 |
p. 4165-4170
6 p.
|
artikel
|
| 36 |
Kinetic and structural insights into the binding of histone deacetylase 1 and 2 (HDAC1, 2) inhibitors
|
Wagner, Florence F.
|
|
2016
|
24 |
18 |
p. 4008-4015
8 p.
|
artikel
|
| 37 |
Multiantigenic peptide–polymer conjugates as therapeutic vaccines against cervical cancer
|
Hussein, Waleed M.
|
|
2016
|
24 |
18 |
p. 4372-4380
9 p.
|
artikel
|
| 38 |
Novel FXR (farnesoid X receptor) modulators: Potential therapies for cholesterol gallstone disease
|
Yu, Donna D.
|
|
2016
|
24 |
18 |
p. 3986-3993
8 p.
|
artikel
|
| 39 |
Oxa-Pictet–Spengler reaction as key step in the synthesis of novel σ receptor ligands with 2-benzopyran structure
|
Knappmann, Inga
|
|
2016
|
24 |
18 |
p. 4045-4055
11 p.
|
artikel
|
| 40 |
Robust design of some selective matrix metalloproteinase-2 inhibitors over matrix metalloproteinase-9 through in silico/fragment-based lead identification and de novo lead modification: Syntheses and biological assays
|
Adhikari, Nilanjan
|
|
2016
|
24 |
18 |
p. 4291-4309
19 p.
|
artikel
|
| 41 |
Similarities and differences in affinity and binding modes of tricyclic pyrimido- and pyrazinoxanthines at human and rat adenosine receptors
|
Szymańska, Ewa
|
|
2016
|
24 |
18 |
p. 4347-4362
16 p.
|
artikel
|
| 42 |
Simple and accurate single base resolution analysis of 5-hydroxymethylcytosine by catalytic oxidative bisulfite sequencing using micelle incarcerated oxidants
|
Fukuzawa, Seketsu
|
|
2016
|
24 |
18 |
p. 4254-4262
9 p.
|
artikel
|
| 43 |
Small molecule non-peptide inhibitors of botulinum neurotoxin serotype E: Structure–activity relationship and a pharmacophore model
|
Kumar, Gyanendra
|
|
2016
|
24 |
18 |
p. 3978-3985
8 p.
|
artikel
|
| 44 |
Solution-phase microwave assisted parallel synthesis, biological evaluation and in silico docking studies of N,N′-disubstituted thioureas derived from 3-chlorobenzoic acid
|
Rauf, Muhammad Khawar
|
|
2016
|
24 |
18 |
p. 4452-4463
12 p.
|
artikel
|
| 45 |
Steric structure–activity relationship of cyproheptadine derivatives as inhibitors of histone methyltransferase Set7/9
|
Fujiwara, Takashi
|
|
2016
|
24 |
18 |
p. 4318-4323
6 p.
|
artikel
|
| 46 |
Strand-invading linear probe combined with unmodified PNA
|
Asanuma, Hiroyuki
|
|
2016
|
24 |
18 |
p. 4129-4137
9 p.
|
artikel
|
| 47 |
Structure elucidation of anti-methicillin resistant Staphylococcus aureus (MRSA) flavonoids from balsam poplar buds
|
Simard, François
|
|
2016
|
24 |
18 |
p. 4188-4198
11 p.
|
artikel
|
| 48 |
Synthesis and anticancer potential of novel xanthone derivatives with 3,6-substituted chains
|
Liu, Chaomei
|
|
2016
|
24 |
18 |
p. 4263-4271
9 p.
|
artikel
|
| 49 |
Synthesis and biological evaluation of analogues of the potent ADAM8 inhibitor cyclo(RLsKDK) for the treatment of inflammatory diseases and cancer metastasis
|
Yim, Victor
|
|
2016
|
24 |
18 |
p. 4032-4037
6 p.
|
artikel
|
| 50 |
Synthesis and biological evaluation of Oblongifolin C derivatives as c-Met inhibitors
|
Wang, Liping
|
|
2016
|
24 |
18 |
p. 4120-4128
9 p.
|
artikel
|
| 51 |
Synthesis and biological evaluation of 3-substituted 5-benzylidene-1-methyl-2-thiohydantoins as potent NADPH oxidase (NOX) inhibitors
|
Bae, Yun Soo
|
|
2016
|
24 |
18 |
p. 4144-4151
8 p.
|
artikel
|
| 52 |
Synthesis and biological investigation of new equatorial (β) stereoisomers of 3-aminotropane arylamides with atypical antipsychotic profile
|
Stefanowicz, Jacek
|
|
2016
|
24 |
18 |
p. 3994-4007
14 p.
|
artikel
|
| 53 |
Synthesis and evaluation of multi-target-directed ligands for the treatment of Alzheimer’s disease based on the fusion of donepezil and melatonin
|
Wang, Jin
|
|
2016
|
24 |
18 |
p. 4324-4338
15 p.
|
artikel
|
| 54 |
Synthesis and in vitro reactivation study of isonicotinamide derivatives of 2-(hydroxyimino)-N-(pyridin-3-yl)acetamide as reactivators of Sarin and VX inhibited human acetylcholinesterase (hAChE)
|
Karade, Hitendra N.
|
|
2016
|
24 |
18 |
p. 4171-4176
6 p.
|
artikel
|
| 55 |
Synthesis and potent antiprotozoal activity of mono/di amidino 2-anilinobenzimidazoles versus Plasmodium falciparum and Trypanosoma brucei rhodesiense
|
Karaaslan, Cigdem
|
|
2016
|
24 |
18 |
p. 4038-4044
7 p.
|
artikel
|
| 56 |
Synthesis and properties of peptide nucleic acid labeled at the N-terminus with HiLyte Fluor 488 fluorescent dye
|
Hnedzko, Dziyana
|
|
2016
|
24 |
18 |
p. 4199-4205
7 p.
|
artikel
|
| 57 |
Synthesis, antiproliferative and pro-apoptotic activity of 2-phenylindoles
|
Kelly, Patrick M.
|
|
2016
|
24 |
18 |
p. 4075-4099
25 p.
|
artikel
|
| 58 |
Synthesis 4-[2-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-ethyl]-benzenesulfonamides with subnanomolar carbonic anhydrase II and XII inhibitory properties
|
Bozdag, Murat
|
|
2016
|
24 |
18 |
p. 4100-4107
8 p.
|
artikel
|
| 59 |
Synthesis of alanyl nucleobase amino acids and their incorporation into proteins
|
Talukder, Poulami
|
|
2016
|
24 |
18 |
p. 4177-4187
11 p.
|
artikel
|
| 60 |
Synthesis of asymmetric zinc(II) phthalocyanines with two different functional groups & spectroscopic properties and photodynamic activity for photodynamic therapy
|
Göksel, Meltem
|
|
2016
|
24 |
18 |
p. 4152-4164
13 p.
|
artikel
|
| 61 |
The development of peptide ligands that target helix 69 rRNA of bacterial ribosomes
|
Dremann, Danielle N.
|
|
2016
|
24 |
18 |
p. 4486-4491
6 p.
|
artikel
|
| 62 |
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation
|
Zhou, Yang
|
|
2016
|
24 |
18 |
p. 4310-4317
8 p.
|
artikel
|
| 63 |
Zinc-mediated binding of a low-molecular-weight stabilizer of the host anti-viral factor apolipoprotein B mRNA-editing enzyme, catalytic polypeptide-like 3G
|
Radwan, Mohamed O.
|
|
2016
|
24 |
18 |
p. 4398-4405
8 p.
|
artikel
|
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