| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Analysis of the aplyronine A-induced protein–protein interaction between actin and tubulin by surface plasmon resonance
|
Hirayama, Yuichiro
|
|
2016
|
24 |
12 |
p. 2809-2814
6 p.
|
artikel
|
| 2 |
Design and synthesis of peptide conjugates of phosphoramide mustard as prodrugs activated by prostate-specific antigen
|
Wu, Xinghua
|
|
2016
|
24 |
12 |
p. 2697-2706
10 p.
|
artikel
|
| 3 |
Design, synthesis, and biological evaluation of new arylamide derivatives possessing sulfonate or sulfamate moieties as steroid sulfatase enzyme inhibitors
|
El-Gamal, Mohammed I.
|
|
2016
|
24 |
12 |
p. 2762-2767
6 p.
|
artikel
|
| 4 |
Design, synthesis, and biological evaluation of substrate-competitive inhibitors of C-terminal Binding Protein (CtBP)
|
Korwar, Sudha
|
|
2016
|
24 |
12 |
p. 2707-2715
9 p.
|
artikel
|
| 5 |
Design, synthesis and preliminary biological evaluation of 4-aminopyrazole derivatives as novel and potent JAKs inhibitors
|
Liang, Xuewu
|
|
2016
|
24 |
12 |
p. 2660-2672
13 p.
|
artikel
|
| 6 |
Design, synthesis, structure–activity relationships, and docking studies of pyrazole-containing derivatives as a novel series of potent glucagon receptor antagonists
|
Shu, Shuangjie
|
|
2016
|
24 |
12 |
p. 2852-2863
12 p.
|
artikel
|
| 7 |
Development of cyanopyridine–triazine hybrids as lead multitarget anti-Alzheimer agents
|
Maqbool, Mudasir
|
|
2016
|
24 |
12 |
p. 2777-2788
12 p.
|
artikel
|
| 8 |
(7-Diethylaminocoumarin-4-yl)methyl ester of suberoylanilide hydroxamic acid as a caged inhibitor for photocontrol of histone deacetylase activity
|
Ieda, Naoya
|
|
2016
|
24 |
12 |
p. 2789-2793
5 p.
|
artikel
|
| 9 |
Discovery of 5-(methylthio)pyrimidine derivatives as L858R/T790M mutant selective epidermal growth factor receptor (EGFR) inhibitors
|
Xiao, Qiang
|
|
2016
|
24 |
12 |
p. 2673-2680
8 p.
|
artikel
|
| 10 |
Discovery of pyrazinone based compounds that potently inhibit the drug-resistant enzyme variant R155K of the hepatitis C virus NS3 protease
|
Belfrage, Anna Karin
|
|
2016
|
24 |
12 |
p. 2603-2620
18 p.
|
artikel
|
| 11 |
Discovery, synthesis, and structure–activity relationships of 20S-dammar-24-en-2α,3β,12β,20-tetrol (GP) derivatives as a new class of AMPKα2β1γ1 activators
|
Dong, Chenhuan
|
|
2016
|
24 |
12 |
p. 2688-2696
9 p.
|
artikel
|
| 12 |
Editorial board
|
|
|
2016
|
24 |
12 |
p. IFC-
1 p.
|
artikel
|
| 13 |
Evaluation of N-substituent structural variations in opioid receptor profile of LP1
|
Pasquinucci, Lorella
|
|
2016
|
24 |
12 |
p. 2832-2842
11 p.
|
artikel
|
| 14 |
Exploring new chemical functionalities to improve aromatase inhibition of steroids
|
Varela, Carla L.
|
|
2016
|
24 |
12 |
p. 2823-2831
9 p.
|
artikel
|
| 15 |
Exploring the 2- and 5-positions of the pyrazolo[4,3-d]pyrimidin-7-amino scaffold to target human A1 and A2A adenosine receptors
|
Squarcialupi, Lucia
|
|
2016
|
24 |
12 |
p. 2794-2808
15 p.
|
artikel
|
| 16 |
Hydraphiles enhance antimicrobial potency against Escherichia coli, Pseudomonas aeruginosa, and Bacillus subtilis
|
Patel, Mohit B.
|
|
2016
|
24 |
12 |
p. 2864-2870
7 p.
|
artikel
|
| 17 |
Identification of 1,2,3-triazole derivatives that protect pancreatic β cells against endoplasmic reticulum stress-mediated dysfunction and death through the inhibition of C/EBP-homologous protein expression
|
Duan, Hongliang
|
|
2016
|
24 |
12 |
p. 2621-2630
10 p.
|
artikel
|
| 18 |
Molecular design, synthesis and anticoagulant activity evaluation of fluorinated dabigatran analogues
|
Wang, Fei
|
|
2016
|
24 |
12 |
p. 2739-2753
15 p.
|
artikel
|
| 19 |
Plasmid DNA delivery by arginine-rich cell-penetrating peptides containing unnatural amino acids
|
Kato, Takuma
|
|
2016
|
24 |
12 |
p. 2681-2687
7 p.
|
artikel
|
| 20 |
Selectivity of 3-bromo-isoxazoline inhibitors between human and Plasmodium falciparum glyceraldehyde-3-phosphate dehydrogenases
|
Bruno, Stefano
|
|
2016
|
24 |
12 |
p. 2654-2659
6 p.
|
artikel
|
| 21 |
Structure-guided development of dual β2 adrenergic/dopamine D2 receptor agonists
|
Weichert, Dietmar
|
|
2016
|
24 |
12 |
p. 2641-2653
13 p.
|
artikel
|
| 22 |
Sulfone-stabilized carbanions for the reversible covalent capture of a posttranslationally-generated cysteine oxoform found in protein tyrosine phosphatase 1B (PTP1B)
|
Parsons, Zachary D.
|
|
2016
|
24 |
12 |
p. 2631-2640
10 p.
|
artikel
|
| 23 |
Synthesis and bioevaluation of substituted chalcones, coumaranones and other flavonoids as anti-HIV agents
|
Cole, Amy L.
|
|
2016
|
24 |
12 |
p. 2768-2776
9 p.
|
artikel
|
| 24 |
Synthesis and biological evaluation of 1,2-dithiol-3-thiones and pyrrolo[1,2-a]pyrazines as novel hypoxia inducible factor-1 (HIF-1) inhibitor
|
Lee, Young Hun
|
|
2016
|
24 |
12 |
p. 2843-2851
9 p.
|
artikel
|
| 25 |
Synthesis and characterization of a fluorescent probe for α-tocopherol suitable for fluorescence microscopy
|
Ghelfi, Mikel
|
|
2016
|
24 |
12 |
p. 2754-2761
8 p.
|
artikel
|
| 26 |
Synthesis and inhibitory evaluation of 3-linked imipramines for the exploration of the S2 site of the human serotonin transporter
|
Brinkø, Anne
|
|
2016
|
24 |
12 |
p. 2725-2738
14 p.
|
artikel
|
| 27 |
Synthesis and in vitro growth inhibitory activity of novel silyl- and trityl-modified nucleosides
|
Panayides, Jenny-Lee
|
|
2016
|
24 |
12 |
p. 2716-2724
9 p.
|
artikel
|
| 28 |
Synthesis, anticancer activity, and SAR analyses of compounds containing the 5:7-fused 4,6,8-triaminoimidazo[4,5-e][1,3]diazepine ring system
|
Xie, Min
|
|
2016
|
24 |
12 |
p. 2595-2602
8 p.
|
artikel
|
| 29 |
The 5-aromatic hydantoin-3-acetate derivatives as inhibitors of the tumour multidrug resistance efflux pump P-glycoprotein (ABCB1): Synthesis, crystallographic and biological studies
|
Żesławska, Ewa
|
|
2016
|
24 |
12 |
p. 2815-2822
8 p.
|
artikel
|
Tijdschrift beschrijving