nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A structure–activity relationship of non-peptide macrocyclic histone deacetylase inhibitors and their anti-proliferative and anti-inflammatory activities
|
Tapadar, Subhasish |
|
2015 |
23 |
24 |
p. 7543-7564 22 p. |
artikel |
2 |
Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity
|
Bozdag, Murat |
|
2015 |
23 |
24 |
p. 7751-7764 14 p. |
artikel |
3 |
Corrigendum to “2-Arylquinazolin-4(3H)-ones: A new class of α-glucosidase inhibitors” [Bioorg. Med. Chem. 23 (2015) 7417–7421]
|
Javaid, Kulsoom |
|
2015 |
23 |
24 |
p. 7786- 1 p. |
artikel |
4 |
Corrigendum to “Inhibition of human topoisomerase I and II and anti-proliferative effects on MCF-7 cells by new titanocene complexes” [Bioorg. Med. Chem. 23 (2015) 7302–7312]
|
Chimento, Adele |
|
2015 |
23 |
24 |
p. 7785- 1 p. |
artikel |
5 |
Design, synthesis and evaluation of antiestrogen and histone deacetylase inhibitor molecular hybrids
|
Mendoza-Sanchez, Rodrigo |
|
2015 |
23 |
24 |
p. 7597-7606 10 p. |
artikel |
6 |
Design, synthesis and preliminary biological studies of pyrrolidine derivatives as Mcl-1 inhibitors
|
Wan, Yichao |
|
2015 |
23 |
24 |
p. 7685-7693 9 p. |
artikel |
7 |
Development of 68Ga-labeled multivalent nitroimidazole derivatives for hypoxia imaging
|
Seelam, Sudhakara Reddy |
|
2015 |
23 |
24 |
p. 7743-7750 8 p. |
artikel |
8 |
Discovery of 2-aryloxy-4-amino-quinazoline derivatives as novel protease-activated receptor 2 (PAR2) antagonists
|
Cho, Nam-Chul |
|
2015 |
23 |
24 |
p. 7717-7727 11 p. |
artikel |
9 |
Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure–activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-d-ribose 2′-oxidase
|
Landge, Sudhir |
|
2015 |
23 |
24 |
p. 7694-7710 17 p. |
artikel |
10 |
Discovery of novel quinoline-based mTOR inhibitors via introducing intra-molecular hydrogen bonding scaffold (iMHBS): The design, synthesis and biological evaluation
|
Ma, Xiaodong |
|
2015 |
23 |
24 |
p. 7585-7596 12 p. |
artikel |
11 |
(E)-2-Cyano-3-(substituted phenyl)acrylamide analogs as potent inhibitors of tyrosinase: A linear β-phenyl-α,β-unsaturated carbonyl scaffold
|
Son, Sujin |
|
2015 |
23 |
24 |
p. 7728-7734 7 p. |
artikel |
12 |
Editorial board
|
|
|
2015 |
23 |
24 |
p. IFC- 1 p. |
artikel |
13 |
Graphical contents list
|
|
|
2015 |
23 |
24 |
p. 7489-7496 8 p. |
artikel |
14 |
Identification of dual PPARα/γ agonists and their effects on lipid metabolism
|
Gao, Quanqing |
|
2015 |
23 |
24 |
p. 7676-7684 9 p. |
artikel |
15 |
Localization-dependent cell-killing effects of protoporphyrin (PPIX)-lipid micelles and liposomes in photodynamic therapy
|
Tachikawa, Shoji |
|
2015 |
23 |
24 |
p. 7578-7584 7 p. |
artikel |
16 |
Modification of a dihydropyrrolopyrimidine phosphoinositide 3-kinase (PI3K) inhibitor to improve oral bioavailability
|
Kawada, Hatsuo |
|
2015 |
23 |
24 |
p. 7650-7660 11 p. |
artikel |
17 |
Phenolic group on A-ring is key for dracoflavan B as a selective noncompetitive inhibitor of α-amylase
|
Toh, Zhi Siang |
|
2015 |
23 |
24 |
p. 7641-7649 9 p. |
artikel |
18 |
Pyrazole clubbed triazolo[1,5-a]pyrimidine hybrids as an anti-tubercular agents: Synthesis, in vitro screening and molecular docking study
|
Bhatt, Jaimin D. |
|
2015 |
23 |
24 |
p. 7711-7716 6 p. |
artikel |
19 |
Searching for novel applications of the benzohomoadamantane scaffold in medicinal chemistry: Synthesis of novel 11β-HSD1 inhibitors
|
Valverde, Elena |
|
2015 |
23 |
24 |
p. 7607-7617 11 p. |
artikel |
20 |
Singlet oxygen oxidation products of biliverdin IXα dimethyl ester
|
Dorazio, Sarina J. |
|
2015 |
23 |
24 |
p. 7671-7675 5 p. |
artikel |
21 |
Small molecules enhance functional O-mannosylation of Alpha-dystroglycan
|
Lv, Fengping |
|
2015 |
23 |
24 |
p. 7661-7670 10 p. |
artikel |
22 |
Structural interrogation of benzosuberene-based inhibitors of tubulin polymerization
|
Herdman, Christine A. |
|
2015 |
23 |
24 |
p. 7497-7520 24 p. |
artikel |
23 |
Synthesis and activity of novel 16-dehydropregnenolone acetate derivatives as inhibitors of type 1 5α-reductase and on cancer cell line SK-LU-1
|
Silva-Ortiz, Aylin Viviana |
|
2015 |
23 |
24 |
p. 7535-7542 8 p. |
artikel |
24 |
Synthesis and antitumor activity evaluation of PI3K inhibitors containing 3-substituted quinazolin-4(3H)-one moiety
|
Zhang, Hao |
|
2015 |
23 |
24 |
p. 7765-7776 12 p. |
artikel |
25 |
Synthesis and bio-evaluation of novel quinolino-stilbene derivatives as potential anticancer agents
|
Srivastava, Vandana |
|
2015 |
23 |
24 |
p. 7629-7640 12 p. |
artikel |
26 |
Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin
|
Martin, Benjamin P. |
|
2015 |
23 |
24 |
p. 7529-7534 6 p. |
artikel |
27 |
Synthesis and evaluation of 3-hydroxy-3-phenylpropanoate ester–AZT conjugates as potential dual-action HIV-1 Integrase and Reverse Transcriptase inhibitors
|
Manyeruke, Meloddy H. |
|
2015 |
23 |
24 |
p. 7521-7528 8 p. |
artikel |
28 |
Synthesis, antiviral activity and resistance of a novel small molecule HIV-1 entry inhibitor
|
Curreli, Francesca |
|
2015 |
23 |
24 |
p. 7618-7628 11 p. |
artikel |
29 |
Synthesis, structure–activity relationship and biological evaluation of novel arylpiperzines as α1A/1D-AR subselective antagonists for BPH
|
Xu, Fang |
|
2015 |
23 |
24 |
p. 7735-7742 8 p. |
artikel |
30 |
Targeting quorum sensing by designing azoline derivatives to inhibit the N-hexanoyl homoserine lactone-receptor CviR: Synthesis as well as biological and theoretical evaluations
|
Bucio-Cano, Alejandro |
|
2015 |
23 |
24 |
p. 7565-7577 13 p. |
artikel |
31 |
1,2,3-Triazolyl-4-oxoquinolines: A feasible beginning for promising chemical structures to inhibit oseltamivir-resistant influenza A and B viruses
|
Boechat, Fernanda da C.S. |
|
2015 |
23 |
24 |
p. 7777-7784 8 p. |
artikel |