| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Antileishmanial pharmacomodulation in 8-nitroquinolin-2(1H)-one series
|
Kieffer, Charline
|
|
2015
|
23 |
10 |
p. 2377-2386
10 p.
|
artikel
|
| 2 |
Anti-parallel triplexes: Synthesis of 8-aza-7-deazaadenine nucleosides with a 3-aminopropynyl side-chain and its corresponding LNA analog
|
Kosbar, Tamer R.
|
|
2015
|
23 |
10 |
p. 2458-2469
12 p.
|
artikel
|
| 3 |
Design, synthesis and biological evaluation of new hybrid anticonvulsants derived from N-benzyl-2-(2,5-dioxopyrrolidin-1-yl)propanamide and 2-(2,5-dioxopyrrolidin-1-yl)butanamide derivatives
|
Kamiński, Krzysztof
|
|
2015
|
23 |
10 |
p. 2548-2561
14 p.
|
artikel
|
| 4 |
Diarylsulfonamides and their bioisosteres as dual inhibitors of alkaline phosphatase and carbonic anhydrase: Structure activity relationship and molecular modelling studies
|
al-Rashida, Mariya
|
|
2015
|
23 |
10 |
p. 2435-2444
10 p.
|
artikel
|
| 5 |
Discovery of DS-5272 as a promising candidate: A potent and orally active p53–MDM2 interaction inhibitor
|
Miyazaki, Masaki
|
|
2015
|
23 |
10 |
p. 2360-2367
8 p.
|
artikel
|
| 6 |
Discovery of novel spiro 1,3,4-thiadiazolines as potent, orally bioavailable and brain penetrant KSP inhibitors
|
Mansoor, Umar Faruk
|
|
2015
|
23 |
10 |
p. 2424-2434
11 p.
|
artikel
|
| 7 |
Discovery of potent and selective urea-based ROCK inhibitors: Exploring the inhibitor’s potency and ROCK2/PKA selectivity by 3D-QSAR, molecular docking and molecular dynamics simulations
|
Mei, Ding
|
|
2015
|
23 |
10 |
p. 2505-2517
13 p.
|
artikel
|
| 8 |
Editorial board
|
|
|
2015
|
23 |
10 |
p. IFC-
1 p.
|
artikel
|
| 9 |
Exploration of benzamidochromenone derivatives with conformational restrictor as interleukin-5 inhibitors
|
Venkateswararao, Eeda
|
|
2015
|
23 |
10 |
p. 2498-2504
7 p.
|
artikel
|
| 10 |
Graphical contents list
|
|
|
2015
|
23 |
10 |
p. 2295-2302
8 p.
|
artikel
|
| 11 |
1-Heteroaryl-3-phenoxypropan-2-ones as inhibitors of cytosolic phospholipase A2α and fatty acid amide hydrolase: Effect of the replacement of the ether oxygen with sulfur and nitrogen moieties on enzyme inhibition and metabolic stability
|
Sundermann, Tom
|
|
2015
|
23 |
10 |
p. 2579-2592
14 p.
|
artikel
|
| 12 |
Identification of apoptosis signal-regulating kinase 1 (ASK1) inhibitors among the derivatives of benzothiazol-2-yl-3-hydroxy-5-phenyl-1,5-dihydro-pyrrol-2-one
|
Starosyla, Sergiy A.
|
|
2015
|
23 |
10 |
p. 2489-2497
9 p.
|
artikel
|
| 13 |
Identification of N-ethylmethylamine as a novel scaffold for inhibitors of soluble epoxide hydrolase by crystallographic fragment screening
|
Amano, Yasushi
|
|
2015
|
23 |
10 |
p. 2310-2317
8 p.
|
artikel
|
| 14 |
N-Acylsulfonamides strongly inhibit human carbonic anhydrase isoenzymes I and II
|
Yıldırım, Alper
|
|
2015
|
23 |
10 |
p. 2598-2605
8 p.
|
artikel
|
| 15 |
New indolizines with phenanthroline skeleton: Synthesis, structure, antimycobacterial and anticancer evaluation
|
Danac, Ramona
|
|
2015
|
23 |
10 |
p. 2318-2327
10 p.
|
artikel
|
| 16 |
Novel pyrrole carboxamide inhibitors of JAK2 as potential treatment of myeloproliferative disorders
|
Brasca, Maria Gabriella
|
|
2015
|
23 |
10 |
p. 2387-2407
21 p.
|
artikel
|
| 17 |
Novel thiazolo[3,2-b]-1,2,4-triazoles derived from naproxen with analgesic/anti-inflammatory properties: Synthesis, biological evaluation and molecular modeling studies
|
Sarigol, Deniz
|
|
2015
|
23 |
10 |
p. 2518-2528
11 p.
|
artikel
|
| 18 |
Peptide based DNA nanocarriers incorporating a cell-penetrating peptide derived from neurturin protein and poly-l-lysine dendrons
|
Rosli, Nurlina
|
|
2015
|
23 |
10 |
p. 2470-2479
10 p.
|
artikel
|
| 19 |
Promising antiproliferative platinum(II) complexes based on imidazole moiety: synthesis, evaluation in HCT-116 cancer cell line and interaction with Ctr-1 Met-rich domain
|
Ferri, Nicola
|
|
2015
|
23 |
10 |
p. 2538-2547
10 p.
|
artikel
|
| 20 |
Structure activity relationship of selective GABA uptake inhibitors
|
Vogensen, Stine B.
|
|
2015
|
23 |
10 |
p. 2480-2488
9 p.
|
artikel
|
| 21 |
Structure–affinity relationship of the cocaine-binding aptamer with quinine derivatives
|
Slavkovic, Sladjana
|
|
2015
|
23 |
10 |
p. 2593-2597
5 p.
|
artikel
|
| 22 |
Structure-based discovery of small molecule hepsin and HGFA protease inhibitors: Evaluation of potency and selectivity derived from distinct binding pockets
|
Franco, Francisco M.
|
|
2015
|
23 |
10 |
p. 2328-2343
16 p.
|
artikel
|
| 23 |
Synthesis and biological evaluation of novel selective androgen receptor modulators (SARMs). Part I
|
Aikawa, Katsuji
|
|
2015
|
23 |
10 |
p. 2568-2578
11 p.
|
artikel
|
| 24 |
Synthesis and biological evaluation of open-chain analogs of cyclic peptides as inhibitors of cellular Shp2 activity
|
Zhen, Xiao-li
|
|
2015
|
23 |
10 |
p. 2562-2567
6 p.
|
artikel
|
| 25 |
Synthesis and evaluation of novel amide amino-β-lactam derivatives as cholesterol absorption inhibitors
|
Dražić, Tonko
|
|
2015
|
23 |
10 |
p. 2353-2359
7 p.
|
artikel
|
| 26 |
Synthesis, antinociceptive and anti-inflammatory effects of porphyrins
|
Alonso-Castro, Angel Josabad
|
|
2015
|
23 |
10 |
p. 2529-2537
9 p.
|
artikel
|
| 27 |
Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action
|
Bozdag, Murat
|
|
2015
|
23 |
10 |
p. 2368-2376
9 p.
|
artikel
|
| 28 |
Synthesis of new N-benzylpiperidine derivatives as cholinesterase inhibitors with β-amyloid anti-aggregation properties and beneficial effects on memory in vivo
|
Więckowska, Anna
|
|
2015
|
23 |
10 |
p. 2445-2457
13 p.
|
artikel
|
| 29 |
Systematic synthesis and anti-inflammatory activity of ω-carboxylated menaquinone derivatives—Investigations on identified and putative vitamin K2 metabolites
|
Fujii, Shinya
|
|
2015
|
23 |
10 |
p. 2344-2352
9 p.
|
artikel
|
| 30 |
The β-carbonic anhydrase from the malaria mosquito Anopheles gambiae is highly inhibited by sulfonamides
|
Syrjänen, Leo
|
|
2015
|
23 |
10 |
p. 2303-2309
7 p.
|
artikel
|
| 31 |
The design, synthesis and biological evaluation of conformationally restricted 4-substituted-2,6-dimethylfuro[2,3-d]pyrimidines as multi-targeted receptor tyrosine kinase and microtubule inhibitors as potential antitumor agents
|
Zhang, Xin
|
|
2015
|
23 |
10 |
p. 2408-2423
16 p.
|
artikel
|
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