nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A new potential approach to block HIV-1 replication via protein–protein interaction and strand-transfer inhibition
|
Ferro, Stefania |
|
2014 |
22 |
7 |
p. 2269-2279 11 p. |
artikel |
2 |
Antiproliferative activities of halogenated thieno[3,2-d]pyrimidines
|
Temburnikar, Kartik W. |
|
2014 |
22 |
7 |
p. 2113-2122 10 p. |
artikel |
3 |
Application of encoded library technology (ELT) to a protein–protein interaction target: Discovery of a potent class of integrin lymphocyte function-associated antigen 1 (LFA-1) antagonists
|
Kollmann, Christopher S. |
|
2014 |
22 |
7 |
p. 2353-2365 13 p. |
artikel |
4 |
Benzophenone C-glucosides and gallotannins from mango tree stem bark with broad-spectrum anti-viral activity
|
Abdel-Mageed, Wael M. |
|
2014 |
22 |
7 |
p. 2236-2243 8 p. |
artikel |
5 |
Binding free energies for nicotine analogs inhibiting cytochrome P450 2A6 by a combined use of molecular dynamics simulations and QM/MM-PBSA calculations
|
Lu, Haiting |
|
2014 |
22 |
7 |
p. 2149-2156 8 p. |
artikel |
6 |
Camphor-based symmetric diimines as inhibitors of influenza virus reproduction
|
Sokolova, Anastasiya S. |
|
2014 |
22 |
7 |
p. 2141-2148 8 p. |
artikel |
7 |
Characterization of the four isomers of 123I-CMICE-013: A potential SPECT myocardial perfusion imaging agent
|
Wei, Lihui |
|
2014 |
22 |
7 |
p. 2033-2044 12 p. |
artikel |
8 |
Chemically defined polyethylene glycol siRNA conjugates with enhanced gene silencing effect
|
Gaziova, Zuzana |
|
2014 |
22 |
7 |
p. 2320-2326 7 p. |
artikel |
9 |
Computer-aided identification of novel 3,5-substituted rhodanine derivatives with activity against Staphylococcus aureus DNA gyrase
|
Werner, Malela M. |
|
2014 |
22 |
7 |
p. 2176-2187 12 p. |
artikel |
10 |
Corrigendum to “Design, structure–activity relationship, and highly efficient asymmetric synthesis of 3-phenyl-4-benzylaminopiperidine derivatives as novel neurokinin-1 receptor antagonists” [Bioorg. Med. Chem. 19 (2011) 6430–6446]
|
Shirai, Junya |
|
2014 |
22 |
7 |
p. 2379- 1 p. |
artikel |
11 |
Decreasing acidity in a series of aldose reductase inhibitors: 2-Fluoro-4-(1H-pyrrol-1-yl)phenol as a scaffold for improved membrane permeation
|
Chatzopoulou, Maria |
|
2014 |
22 |
7 |
p. 2194-2207 14 p. |
artikel |
12 |
Design and synthesis of conformationally restricted inhibitors of active thrombin activatable fibrinolysis inhibitor (TAFIa)
|
Brink, Mikael |
|
2014 |
22 |
7 |
p. 2261-2268 8 p. |
artikel |
13 |
Design and synthesis of silicon-containing steroid sulfatase inhibitors possessing pro-estrogen antagonistic character
|
Kajita, Daisuke |
|
2014 |
22 |
7 |
p. 2244-2252 9 p. |
artikel |
14 |
Design, synthesis and biological evaluation of a series of pyrano chalcone derivatives containing indole moiety as novel anti-tubulin agents
|
Wang, Guangcheng |
|
2014 |
22 |
7 |
p. 2060-2079 20 p. |
artikel |
15 |
Design, synthesis and biological evaluation of new 5-nitro benzimidazole derivatives as AT1 antagonists with anti-hypertension activities
|
Zhu, Weibo |
|
2014 |
22 |
7 |
p. 2294-2302 9 p. |
artikel |
16 |
Design, synthesis and biological evaluation of novel 6-alkenylamides substituted of 4-anilinothieno[2,3-d]pyrimidines as irreversible epidermal growth factor receptor inhibitors
|
Ji, Xun |
|
2014 |
22 |
7 |
p. 2366-2378 13 p. |
artikel |
17 |
Discovery of 3-(4-methanesulfonylphenoxy)-N-[1-(2-methoxy-ethoxymethyl)-1H-pyrazol-3-yl]-5-(3-methylpyridin-2-yl)-benzamide as a novel glucokinase activator (GKA) for the treatment of type 2 diabetes mellitus
|
Park, Kaapjoo |
|
2014 |
22 |
7 |
p. 2280-2293 14 p. |
artikel |
18 |
[Dmt1]DALDA analogues with enhanced μ opioid agonist potency and with a mixed μ/κ opioid activity profile
|
Bai, Longxiang |
|
2014 |
22 |
7 |
p. 2333-2338 6 p. |
artikel |
19 |
Editorial board
|
|
|
2014 |
22 |
7 |
p. IFC- 1 p. |
artikel |
20 |
Endomorphin analogues with mixed μ-opioid (MOP) receptor agonism/δ-opioid (DOP) receptor antagonism and lacking β-arrestin2 recruitment activity
|
Cai, Jun |
|
2014 |
22 |
7 |
p. 2208-2219 12 p. |
artikel |
21 |
Expanded potential of seleno-carbohydrates as a molecular tool for X-ray structural determination of a carbohydrate–protein complex with single/multi-wavelength anomalous dispersion phasing
|
Suzuki, Tatsuya |
|
2014 |
22 |
7 |
p. 2090-2101 12 p. |
artikel |
22 |
Facile synthesis, cytotoxicity and bioimaging of Fe3+ selective fluorescent chemosensor
|
Saleem, Muhammad |
|
2014 |
22 |
7 |
p. 2045-2051 7 p. |
artikel |
23 |
Fused heterocyclic compounds bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 1: Design, synthesis and biological evaluation of novel 5,7-disubstituted pyrazolo[1,5-a]pyrimidine derivatives
|
Tian, Ye |
|
2014 |
22 |
7 |
p. 2052-2059 8 p. |
artikel |
24 |
Graphical contents list
|
|
|
2014 |
22 |
7 |
p. 1973-1982 10 p. |
artikel |
25 |
N-Acyl-phosphoramidates as potential novel form of gemcitabine prodrugs
|
Baraniak, Janina |
|
2014 |
22 |
7 |
p. 2133-2140 8 p. |
artikel |
26 |
Novel nitroimidazole alkylsulfonamides as hypoxic cell radiosensitisers
|
Bonnet, Muriel |
|
2014 |
22 |
7 |
p. 2123-2132 10 p. |
artikel |
27 |
Pyrrolopyrimidine-inhibitors with hydantoin moiety as spacer can explore P4/S4 interaction on plasmin
|
Teno, Naoki |
|
2014 |
22 |
7 |
p. 2339-2352 14 p. |
artikel |
28 |
Recognition of RNA duplex by a neomycin–Hoechst 33258 conjugate
|
Willis, Bert |
|
2014 |
22 |
7 |
p. 2327-2332 6 p. |
artikel |
29 |
Some non-conventional biomolecular targets for diamidines. A short survey
|
Huang, Tien L. |
|
2014 |
22 |
7 |
p. 1983-1992 10 p. |
artikel |
30 |
Studies on the antiproliferative effects of tropolone derivatives in Jurkat T-lymphocyte cells
|
Ononye, Sophia N. |
|
2014 |
22 |
7 |
p. 2188-2193 6 p. |
artikel |
31 |
Synthesis and anticonvulsant activity of some new pyrazolo[3,4-b]pyrazines and related heterocycles
|
Farghaly, Abdel-Rahman |
|
2014 |
22 |
7 |
p. 2166-2175 10 p. |
artikel |
32 |
Synthesis and biological evaluation of new pyrazolone–pyridazine conjugates as anti-inflammatory and analgesic agents
|
Khalil, Nadia Abdalla |
|
2014 |
22 |
7 |
p. 2080-2089 10 p. |
artikel |
33 |
Synthesis and evaluation of effective photoaffinity probe molecule of furospinosulin-1, a hypoxia-selective growth inhibitor
|
Kotoku, Naoyuki |
|
2014 |
22 |
7 |
p. 2102-2112 11 p. |
artikel |
34 |
Synthesis and methemoglobinemia-inducing properties of benzocaine isosteres designed as humane rodenticides
|
Conole, Daniel |
|
2014 |
22 |
7 |
p. 2220-2235 16 p. |
artikel |
35 |
Synthesis, biological evaluation and 3D-QSAR studies of new chalcone derivatives as inhibitors of human P-glycoprotein
|
Parveen, Zahida |
|
2014 |
22 |
7 |
p. 2311-2319 9 p. |
artikel |
36 |
Synthetic approaches to the 2012 new drugs
|
Ding, Hong X. |
|
2014 |
22 |
7 |
p. 2005-2032 28 p. |
artikel |
37 |
The chemistry and biology of febrifugine and halofuginone
|
McLaughlin, Noel P. |
|
2014 |
22 |
7 |
p. 1993-2004 12 p. |
artikel |
38 |
The identification, analysis and structure-based development of novel inhibitors of 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase
|
Yun, Mi-Kyung |
|
2014 |
22 |
7 |
p. 2157-2165 9 p. |
artikel |
39 |
The identification of novel 5′-amino gemcitabine analogs as potent RRM1 inhibitors
|
Labroli, Marc A. |
|
2014 |
22 |
7 |
p. 2303-2310 8 p. |
artikel |
40 |
Using ‘biased-privileged’ scaffolds to identify lysine methyltransferase inhibitors
|
Kashyap, Sudhir |
|
2014 |
22 |
7 |
p. 2253-2260 8 p. |
artikel |