| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A comparative study of ATP analogs for phosphorylation-dependent kinase–substrate crosslinking
|
Garre, Satish
|
|
2014
|
22 |
5 |
p. 1620-1625
6 p.
|
artikel
|
| 2 |
2-Acylamino-5-nitro-1,3-thiazoles: Preparation and in vitro bioevaluation against four neglected protozoan parasites
|
Nava-Zuazo, Carlos
|
|
2014
|
22 |
5 |
p. 1626-1633
8 p.
|
artikel
|
| 3 |
Anion inhibition study of the β-carbonic anhydrase (CahB1) from the cyanobacterium Coleofasciculus chthonoplastes (ex-Microcoleus chthonoplastes)
|
Vullo, Daniela
|
|
2014
|
22 |
5 |
p. 1667-1671
5 p.
|
artikel
|
| 4 |
Antiprotozoan lead discovery by aligning dry and wet screening: Prediction, synthesis, and biological assay of novel quinoxalinones
|
Martins Alho, Miriam A.
|
|
2014
|
22 |
5 |
p. 1568-1585
18 p.
|
artikel
|
| 5 |
Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, IX and XII with benzene sulfonamides incorporating 4- and 3-nitrophthalimide moieties
|
Sethi, Kalyan K.
|
|
2014
|
22 |
5 |
p. 1586-1595
10 p.
|
artikel
|
| 6 |
Chemical constituents of Plectranthus amboinicus and the synthetic analogs possessing anti-inflammatory activity
|
Chen, Yuan-Siao
|
|
2014
|
22 |
5 |
p. 1766-1772
7 p.
|
artikel
|
| 7 |
Design, synthesis and preliminary bioactivity studies of 1,2-dihydrobenzo[d]isothiazol-3-one-1,1-dioxide hydroxamic acid derivatives as novel histone deacetylase inhibitors
|
Han, Leiqiang
|
|
2014
|
22 |
5 |
p. 1529-1538
10 p.
|
artikel
|
| 8 |
Design, synthesis, radiolabeling and in vivo evaluation of potential positron emission tomography (PET) radioligands for brain imaging of the 5-HT7 receptor
|
Lacivita, Enza
|
|
2014
|
22 |
5 |
p. 1736-1750
15 p.
|
artikel
|
| 9 |
2,6-Diaminopurine nucleoside derivative of 9-ethyloxy-2-oxo-1,3-diazaphenoxazine (2-amino-Adap) for recognition of 8-oxo-dG in DNA
|
Taniguchi, Yosuke
|
|
2014
|
22 |
5 |
p. 1634-1641
8 p.
|
artikel
|
| 10 |
Discovery and optimization of a new class of pyruvate kinase inhibitors as potential therapeutics for the treatment of methicillin-resistant Staphylococcus aureus infections
|
Kumar, Nag S.
|
|
2014
|
22 |
5 |
p. 1708-1725
18 p.
|
artikel
|
| 11 |
Discovery and SAR study of hydroxyacetophenone derivatives as potent, non-steroidal farnesoid X receptor (FXR) antagonists
|
Liu, Peng
|
|
2014
|
22 |
5 |
p. 1596-1607
12 p.
|
artikel
|
| 12 |
Discovery of a novel series of indoline carbamate and indolinylpyrimidine derivatives as potent GPR119 agonists
|
Sato, Kenjiro
|
|
2014
|
22 |
5 |
p. 1649-1666
18 p.
|
artikel
|
| 13 |
Discovery of simplified N2-substituted pyrazolo[3,4-d]pyrimidine derivatives as novel adenosine receptor antagonists: Efficient synthetic approaches, biological evaluations and molecular docking studies
|
Venkatesan, Gopalakrishnan
|
|
2014
|
22 |
5 |
p. 1751-1765
15 p.
|
artikel
|
| 14 |
Editorial board
|
|
|
2014
|
22 |
5 |
p. IFC-
1 p.
|
artikel
|
| 15 |
Graphical contents list
|
|
|
2014
|
22 |
5 |
p. 1507-1514
8 p.
|
artikel
|
| 16 |
Lead modification: Amino acid appended indoles as highly effective 5-LOX inhibitors
|
Prasher, Parteek
|
|
2014
|
22 |
5 |
p. 1642-1648
7 p.
|
artikel
|
| 17 |
Reaction intermediate analogues as bisubstrate inhibitors of pantothenate synthetase
|
Xu, Zhixiang
|
|
2014
|
22 |
5 |
p. 1726-1735
10 p.
|
artikel
|
| 18 |
Structure activity relationship studies of 3-arylsulfonyl-pyrido[1,2-a]pyrimidin-4-imines as potent 5-HT6 antagonists
|
Hu, Shuanghua
|
|
2014
|
22 |
5 |
p. 1782-1790
9 p.
|
artikel
|
| 19 |
Structure-based optimization of cyclopropyl urea derivatives as potent soluble epoxide hydrolase inhibitors for potential decrease of renal injury without hypotensive action
|
Takai, Kentaro
|
|
2014
|
22 |
5 |
p. 1548-1557
10 p.
|
artikel
|
| 20 |
Synthesis and anticancer activity of focused compound libraries from the natural product lead, oroidin
|
Dyson, Lauren
|
|
2014
|
22 |
5 |
p. 1690-1699
10 p.
|
artikel
|
| 21 |
Synthesis and biological evaluation of 2,5-di(7-indolyl)-1,3,4-oxadiazoles, and 2- and 7-indolyl 2-(1,3,4-thiadiazolyl)ketones as antimicrobials
|
Kandemir, Hakan
|
|
2014
|
22 |
5 |
p. 1672-1679
8 p.
|
artikel
|
| 22 |
Synthesis, [18F] radiolabeling, and evaluation of poly (ADP-ribose) polymerase-1 (PARP-1) inhibitors for in vivo imaging of PARP-1 using positron emission tomography
|
Zhou, Dong
|
|
2014
|
22 |
5 |
p. 1700-1707
8 p.
|
artikel
|
| 23 |
Synthesis, nitric oxide release, and α-glucosidase inhibition of nitric oxide donating apigenin and chrysin derivatives
|
Wang, Qi-Qin
|
|
2014
|
22 |
5 |
p. 1515-1521
7 p.
|
artikel
|
| 24 |
Synthesis of a novel series of thiazole-based histone acetyltransferase inhibitors
|
Secci, Daniela
|
|
2014
|
22 |
5 |
p. 1680-1689
10 p.
|
artikel
|
| 25 |
Synthesis of 2,6-disubstituted benzylamine derivatives as reversible selective inhibitors of copper amine oxidases
|
Lucchesini, Francesco
|
|
2014
|
22 |
5 |
p. 1558-1567
10 p.
|
artikel
|
| 26 |
Synthesis of novel, peptidic kinase inhibitors with cytostatic/cytotoxic activity
|
Szymanski, Wiktor
|
|
2014
|
22 |
5 |
p. 1773-1781
9 p.
|
artikel
|
| 27 |
Synthesis of 6-tetrazolyl-substituted sulfocoumarins acting as highly potent and selective inhibitors of the tumor-associated carbonic anhydrase isoforms IX and XII
|
Grandane, Aiga
|
|
2014
|
22 |
5 |
p. 1522-1528
7 p.
|
artikel
|
| 28 |
Synthesis, selective cytotoxicities and probable mechanism of action of 7-methoxy-3-arylflavone-8-acetic acids
|
Zhou, Zhong-Zhen
|
|
2014
|
22 |
5 |
p. 1539-1547
9 p.
|
artikel
|
| 29 |
1,2,3-Triazole-, arylamino- and thio-substituted 1,4-naphthoquinones: Potent antitumor activity, electrochemical aspects, and bioisosteric replacement of C-ring-modified lapachones
|
da Cruz, Eduardo H.G.
|
|
2014
|
22 |
5 |
p. 1608-1619
12 p.
|
artikel
|
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