| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Active immunisation of mice with GnRH lipopeptide vaccine candidates: Importance of T helper or multi-dimer GnRH epitope
|
Goodwin, Daryn
|
|
2014
|
22 |
17 |
p. 4848-4854
7 p.
|
artikel
|
| 2 |
Amine substitution of quinazolinones leads to selective nanomolar AChE inhibitors with ‘inverted’ binding mode
|
Darras, Fouad H.
|
|
2014
|
22 |
17 |
p. 4867-4881
15 p.
|
artikel
|
| 3 |
A new Rhodamine B-based ‘on–off’ chemical sensor with high selectivity and sensitivity toward Fe3+ and its imaging in living cells
|
Bao, Xiaofeng
|
|
2014
|
22 |
17 |
p. 4826-4835
10 p.
|
artikel
|
| 4 |
Antinociceptive and antidepressant-like action of endomorphin-2 analogs with proline surrogates in position 2
|
Perlikowska, Renata
|
|
2014
|
22 |
17 |
p. 4803-4809
7 p.
|
artikel
|
| 5 |
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents
|
Tonelli, Michele
|
|
2014
|
22 |
17 |
p. 4893-4909
17 p.
|
artikel
|
| 6 |
Apoptosis-inducing effect of a palladium(II) saccharinate complex of terpyridine on human breast cancer cells in vitro and in vivo
|
Ari, Ferda
|
|
2014
|
22 |
17 |
p. 4948-4954
7 p.
|
artikel
|
| 7 |
A semi-synthetic derivative of artemisinin, artesunate inhibits prostaglandin E2 production in LPS/IFNγ-activated BV2 microglia
|
Okorji, Uchechukwu P.
|
|
2014
|
22 |
17 |
p. 4726-4734
9 p.
|
artikel
|
| 8 |
‘Carba’-carfentanil (trans isomer): A μ opioid receptor (MOR) partial agonist with a distinct binding mode
|
Weltrowska, Grazyna
|
|
2014
|
22 |
17 |
p. 4581-4586
6 p.
|
artikel
|
| 9 |
Click approach to the discovery of 1,2,3-triazolylsalicylamides as potent Aurora kinase inhibitors
|
Song, Doohee
|
|
2014
|
22 |
17 |
p. 4855-4866
12 p.
|
artikel
|
| 10 |
Competitive antagonism of insect GABA receptors by 4-substituted 5-(4-piperidyl)-3-isothiazolols
|
Liu, Genyan
|
|
2014
|
22 |
17 |
p. 4637-4645
9 p.
|
artikel
|
| 11 |
Concise syntheses of 7-anilino-indoline-N-benzenesulfonamides as antimitotic and vascular disrupting agents
|
Mehndiratta, Samir
|
|
2014
|
22 |
17 |
p. 4917-4923
7 p.
|
artikel
|
| 12 |
Cyclic acyl guanidines bearing carbamate moieties allow potent and dirigible cholinesterase inhibition of either acetyl- or butyrylcholinesterase
|
Darras, Fouad H.
|
|
2014
|
22 |
17 |
p. 5020-5034
15 p.
|
artikel
|
| 13 |
Cytoprotective pyridinol antioxidants as potential therapeutic agents for neurodegenerative and mitochondrial diseases
|
Alam, Mohammad Parvez
|
|
2014
|
22 |
17 |
p. 4935-4947
13 p.
|
artikel
|
| 14 |
Cytotoxicity of synthesized 1,4-naphthoquinone analogues on selected human cancer cell lines
|
Kishore, Navneet
|
|
2014
|
22 |
17 |
p. 5013-5019
7 p.
|
artikel
|
| 15 |
Design of granulatimide and isogranulatimide analogues as potential Chk1 inhibitors: Study of amino-platforms for their synthesis
|
Lavrard, Hubert
|
|
2014
|
22 |
17 |
p. 4961-4967
7 p.
|
artikel
|
| 16 |
Design, stereoselective synthesis, configurational stability and biological activity of 7-chloro-9-(furan-3-yl)-2,3,3a,4-tetrahydro-1H-benzo[e]pyrrolo[2,1-c][1,2,4]thiadiazine 5,5-dioxide
|
Carrozzo, Marina Maria
|
|
2014
|
22 |
17 |
p. 4667-4676
10 p.
|
artikel
|
| 17 |
Design, synthesis, and biological evaluation of scaffold-based tripeptidomimetic antagonists for CXC chemokine receptor 4 (CXCR4)
|
Zachariassen, Zack G.
|
|
2014
|
22 |
17 |
p. 4759-4769
11 p.
|
artikel
|
| 18 |
Design, synthesis and biological evaluation of thienopyridinones as Chk1 inhibitors
|
Song, Pinrao
|
|
2014
|
22 |
17 |
p. 4882-4892
11 p.
|
artikel
|
| 19 |
Design, synthesis and evaluation of rivastigmine and curcumin hybrids as site-activated multitarget-directed ligands for Alzheimer’s disease therapy
|
Li, Yujie
|
|
2014
|
22 |
17 |
p. 4717-4725
9 p.
|
artikel
|
| 20 |
Design, synthesis, and in vitro evaluation of an activity-based protein profiling (ABPP) probe targeting agmatine deiminases
|
Thomson, Andrew
|
|
2014
|
22 |
17 |
p. 4602-4608
7 p.
|
artikel
|
| 21 |
Design, synthesis, biological evaluation of substituted benzofurans as DNA gyraseB inhibitors of Mycobacterium tuberculosis
|
Renuka, Janupally
|
|
2014
|
22 |
17 |
p. 4924-4934
11 p.
|
artikel
|
| 22 |
Development of novel membrane active lipidated peptidomimetics active against drug resistant clinical isolates
|
Lohan, Sandeep
|
|
2014
|
22 |
17 |
p. 4544-4552
9 p.
|
artikel
|
| 23 |
Discovery of inhibitors of the mitotic kinase TTK based on N-(3-(3-sulfamoylphenyl)-1H-indazol-5-yl)-acetamides and carboxamides
|
Laufer, Radoslaw
|
|
2014
|
22 |
17 |
p. 4968-4997
30 p.
|
artikel
|
| 24 |
Discovery of quinazolin-4-amines bearing benzimidazole fragments as dual inhibitors of c-Met and VEGFR-2
|
Shi, Lei
|
|
2014
|
22 |
17 |
p. 4735-4744
10 p.
|
artikel
|
| 25 |
Discovery, structure–activity relationship studies, and anti-nociceptive effects of 1-phenyl-3,6,6-trimethyl-1,5,6,7-tetrahydro-4H-indazol-4-one as novel opioid receptor agonists
|
Cheng, Ming-Fu
|
|
2014
|
22 |
17 |
p. 4694-4703
10 p.
|
artikel
|
| 26 |
Editorial board
|
|
|
2014
|
22 |
17 |
p. IFC-
1 p.
|
artikel
|
| 27 |
Endoperoxide polyketides from a Chinese Plakortis simplex: Further evidence of the impact of stereochemistry on antimalarial activity of simple 1,2-dioxanes
|
Chianese, Giuseppina
|
|
2014
|
22 |
17 |
p. 4572-4580
9 p.
|
artikel
|
| 28 |
Ethyl 2-(benzylidene)-7-methyl-3-oxo-2,3-dihydro-5H-thiazolo[3,2-a]pyrimidine-6-carboxylate analogues as a new scaffold for protein kinase casein kinase 2 inhibitor
|
Jin, Cheng-Hao
|
|
2014
|
22 |
17 |
p. 4553-4565
13 p.
|
artikel
|
| 29 |
Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands
|
Sancineto, Luca
|
|
2014
|
22 |
17 |
p. 4658-4666
9 p.
|
artikel
|
| 30 |
Formation of the carboxamidine precursor of cyanuric acid from guanine oxidative lesion dehydro-guanidinohydantoin
|
Irvoas, Joris
|
|
2014
|
22 |
17 |
p. 4711-4716
6 p.
|
artikel
|
| 31 |
Graphical contents list
|
|
|
2014
|
22 |
17 |
p. 4523-4536
14 p.
|
artikel
|
| 32 |
Identification of novel inhibitors of phospho-MurNAc-pentapeptide translocase MraY from library screening: Isoquinoline alkaloid michellamine B and xanthene dye phloxine B
|
Mihalyi, Agnes
|
|
2014
|
22 |
17 |
p. 4566-4571
6 p.
|
artikel
|
| 33 |
Inhibitory effects of p-alkylaminophenol on melanogenesis
|
Takahashi, Noriko
|
|
2014
|
22 |
17 |
p. 4677-4683
7 p.
|
artikel
|
| 34 |
Mono- and di-halogenated histamine, histidine and carnosine derivatives are potent carbonic anhydrase I, II, VII, XII and XIV activators
|
Saada, Mohamed-Chiheb
|
|
2014
|
22 |
17 |
p. 4752-4758
7 p.
|
artikel
|
| 35 |
Novel 3,6-bis(imidazolidine)acridines as effective photosensitizers for photodynamic therapy
|
Čižeková, L.
|
|
2014
|
22 |
17 |
p. 4684-4693
10 p.
|
artikel
|
| 36 |
Novel N-biphenyl-2-ylmethyl 2-methoxyphenylpiperazinylalkanamides as 5-HT7R antagonists for the treatment of depression
|
Kim, Youngjae
|
|
2014
|
22 |
17 |
p. 4587-4596
10 p.
|
artikel
|
| 37 |
2-Phenylaminonaphthoquinones and related compounds: Synthesis, trypanocidal and cytotoxic activities
|
Sieveking, Ivan
|
|
2014
|
22 |
17 |
p. 4609-4620
12 p.
|
artikel
|
| 38 |
Pyrrole-3-carboxamides as potent and selective JAK2 inhibitors
|
Brasca, Maria Gabriella
|
|
2014
|
22 |
17 |
p. 4998-5012
15 p.
|
artikel
|
| 39 |
Ricinine: A pyridone alkaloid from Ricinus communis that activates the Wnt signaling pathway through casein kinase 1α
|
Ohishi, Kensuke
|
|
2014
|
22 |
17 |
p. 4597-4601
5 p.
|
artikel
|
| 40 |
Sequence-specific DNA alkylation and transcriptional inhibition by long-chain hairpin pyrrole–imidazole polyamide–chlorambucil conjugates targeting CAG/CTG trinucleotide repeats
|
Asamitsu, Sefan
|
|
2014
|
22 |
17 |
p. 4646-4657
12 p.
|
artikel
|
| 41 |
Stereoselective synthesis of lanthionine derivatives in aqueous solution and their incorporation into the peptidoglycan of Escherichia coli
|
Denoël, Thibaut
|
|
2014
|
22 |
17 |
p. 4621-4628
8 p.
|
artikel
|
| 42 |
Structural optimization of a retrograde trafficking inhibitor that protects cells from infections by human polyoma- and papillomaviruses
|
Carney, Daniel W.
|
|
2014
|
22 |
17 |
p. 4836-4847
12 p.
|
artikel
|
| 43 |
Structure–affinity relationships and pharmacological characterization of new alkyl-resorcinol cannabinoid receptor ligands: Identification of a dual cannabinoid receptor/TRPA1 channel agonist
|
Brizzi, Antonella
|
|
2014
|
22 |
17 |
p. 4770-4783
14 p.
|
artikel
|
| 44 |
Structure based inhibitor design targeting glycogen phosphorylase b. Virtual screening, synthesis, biochemical and biological assessment of novel N-acyl-β-d-glucopyranosylamines
|
Parmenopoulou, Vanessa
|
|
2014
|
22 |
17 |
p. 4810-4825
16 p.
|
artikel
|
| 45 |
Sulfonamide inhibition study of the carbonic anhydrases from the bacterial pathogen Porphyromonas gingivalis: The β-class (PgiCAb) versus the γ-class (PgiCA) enzymes
|
Prete, Sonia Del
|
|
2014
|
22 |
17 |
p. 4537-4543
7 p.
|
artikel
|
| 46 |
Syntheses of coumarin–tacrine hybrids as dual-site acetylcholinesterase inhibitors and their activity against butylcholinesterase, Aβ aggregation, and β-secretase
|
Sun, Qi
|
|
2014
|
22 |
17 |
p. 4784-4791
8 p.
|
artikel
|
| 47 |
Synthesis and antifungal activity of substituted salicylaldehyde hydrazones, hydrazides and sulfohydrazides
|
Backes, Gregory L.
|
|
2014
|
22 |
17 |
p. 4629-4636
8 p.
|
artikel
|
| 48 |
Synthesis and biological evaluation of new simple indolic non peptidic HIV Protease inhibitors: The effect of different substitution patterns
|
Bonini, C.
|
|
2014
|
22 |
17 |
p. 4792-4802
11 p.
|
artikel
|
| 49 |
Synthesis and biological evaluation of pyrido[2,3-d]pyrimidine-2,4-dione derivatives as eEF-2K inhibitors
|
Edupuganti, Ramakrishna
|
|
2014
|
22 |
17 |
p. 4910-4916
7 p.
|
artikel
|
| 50 |
Synthesis of fluorinated agonist of sphingosine-1-phosphate receptor 1
|
Aliouane, Lucie
|
|
2014
|
22 |
17 |
p. 4955-4960
6 p.
|
artikel
|
| 51 |
Synthesis of protoporphyrin–lipids and biological evaluation of micelles and liposomes
|
Tachikawa, Shoji
|
|
2014
|
22 |
17 |
p. 4745-4751
7 p.
|
artikel
|
| 52 |
Synthesis of pyrazolo[4,3-a]phenanthridines, a new scaffold for Pim kinase inhibition
|
Suchaud, Virginie
|
|
2014
|
22 |
17 |
p. 4704-4710
7 p.
|
artikel
|
| 53 |
The Nagoya Medal of Organic Chemistry 2014
|
|
|
2014
|
22 |
17 |
p. I-
1 p.
|
artikel
|
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