| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Benzene-1,3-dicarboxylic acid 2,5-dimethylpyrrole derivatives as multiple inhibitors of bacterial Mur ligases (MurC–MurF)
|
Perdih, Andrej
|
|
2014
|
22 |
15 |
p. 4124-4134
11 p.
|
artikel
|
| 2 |
Benzoquinones as inhibitors of botulinum neurotoxin serotype A
|
Bremer, Paul T.
|
|
2014
|
22 |
15 |
p. 3971-3981
11 p.
|
artikel
|
| 3 |
Bicyclic tetrapeptides as potent HDAC inhibitors: Effect of aliphatic loop position and hydrophobicity on inhibitory activity
|
Islam, Md. Nurul
|
|
2014
|
22 |
15 |
p. 3862-3870
9 p.
|
artikel
|
| 4 |
Bradykinin antagonists and thiazolidinone derivatives as new potential anti-cancer compounds
|
Avdieiev, Stanislav
|
|
2014
|
22 |
15 |
p. 3815-3823
9 p.
|
artikel
|
| 5 |
Corrigendum to “4-Quinolone-3-carboxylic acids as cell-permeable inhibitors of protein tyrosine phosphatase 1B” [Bioorg. Med. Chem. 22 (2014) 3670–3683]
|
Zhi, Ying
|
|
2014
|
22 |
15 |
p. 4347-
1 p.
|
artikel
|
| 6 |
Coumarin hybrids as novel therapeutic agents
|
Sandhu, Sonali
|
|
2014
|
22 |
15 |
p. 3806-3814
9 p.
|
artikel
|
| 7 |
Design and synthesis of 5-[(2-chloro-6-fluorophenyl)acetylamino]-3-(4-fluorophenyl)-4-(4-pyrimidinyl)isoxazole (AKP-001), a novel inhibitor of p38 MAP kinase with reduced side effects based on the antedrug concept
|
Hasumi, Koichi
|
|
2014
|
22 |
15 |
p. 4162-4176
15 p.
|
artikel
|
| 8 |
Design and synthesis of 8-hydroxyquinoline-based radioprotective agents
|
Ariyasu, Shinya
|
|
2014
|
22 |
15 |
p. 3891-3905
15 p.
|
artikel
|
| 9 |
Design, synthesis and biological evaluation of (E)-3-(3,4-dihydroxyphenyl)acrylylpiperazine derivatives as a new class of tubulin polymerization inhibitors
|
Yin, Yong
|
|
2014
|
22 |
15 |
p. 4285-4292
8 p.
|
artikel
|
| 10 |
Development of potent antagonists for formyl peptide receptor 1 based on Boc-Phe-d-Leu-Phe-d-Leu-Phe-OH
|
Hayashi, Ryo
|
|
2014
|
22 |
15 |
p. 3824-3828
5 p.
|
artikel
|
| 11 |
Development of radamide analogs as Grp94 inhibitors
|
Muth, Aaron
|
|
2014
|
22 |
15 |
p. 4083-4098
16 p.
|
artikel
|
| 12 |
2,2′-Dihydroxybenzophenones and their carbonyl N-analogues as inhibitor scaffolds for MDR-involved human glutathione transferase isoenzyme A1-1
|
Perperopoulou, Fereniki D.
|
|
2014
|
22 |
15 |
p. 3957-3970
14 p.
|
artikel
|
| 13 |
Discovery of novel inhibitors of vascular endothelial growth factor-A–Neuropilin-1 interaction by structure-based virtual screening
|
Starzec, Anna
|
|
2014
|
22 |
15 |
p. 4042-4048
7 p.
|
artikel
|
| 14 |
Discovery of potent and selective spiroindolinone MDM2 inhibitor, RO8994, for cancer therapy
|
Zhang, Zhuming
|
|
2014
|
22 |
15 |
p. 4001-4009
9 p.
|
artikel
|
| 15 |
Dual-stage triterpenoids from an African medicinal plant targeting the malaria parasite
|
Ramalhete, Cátia
|
|
2014
|
22 |
15 |
p. 3887-3890
4 p.
|
artikel
|
| 16 |
Editorial board
|
|
|
2014
|
22 |
15 |
p. IFC-
1 p.
|
artikel
|
| 17 |
Effect of p-aminophenols on tyrosinase activity
|
Komori, Yu
|
|
2014
|
22 |
15 |
p. 3994-4000
7 p.
|
artikel
|
| 18 |
Facile synthesis, optical and conformational characteristics, and efficient intracellular delivery of a peptide–DNA conjugate
|
Lee, Mun-kyung
|
|
2014
|
22 |
15 |
p. 4204-4209
6 p.
|
artikel
|
| 19 |
Fragment-based hit discovery and structure-based optimization of aminotriazoloquinazolines as novel Hsp90 inhibitors
|
Casale, Elena
|
|
2014
|
22 |
15 |
p. 4135-4150
16 p.
|
artikel
|
| 20 |
Furazan and furoxan sulfonamides are strong α-carbonic anhydrase inhibitors and potential antiglaucoma agents
|
Chegaev, Konstantin
|
|
2014
|
22 |
15 |
p. 3913-3921
9 p.
|
artikel
|
| 21 |
Glucopyranosylidene-spiro-iminothiazolidinone, a new bicyclic ring system: Synthesis, derivatization, and evaluation for inhibition of glycogen phosphorylase by enzyme kinetic and crystallographic methods
|
Czifrák, Katalin
|
|
2014
|
22 |
15 |
p. 4028-4041
14 p.
|
artikel
|
| 22 |
Graphical contents list
|
|
|
2014
|
22 |
15 |
p. 3791-3805
15 p.
|
artikel
|
| 23 |
Identification and development of 2-methylimidazo[1,2-a]pyridine-3-carboxamides as Mycobacterium tuberculosis pantothenate synthetase inhibitors
|
Samala, Ganesh
|
|
2014
|
22 |
15 |
p. 4223-4232
10 p.
|
artikel
|
| 24 |
Inhibitory and mechanistic investigations of oxo-lipids with human lipoxygenase isozymes
|
Armstrong, Michelle M.
|
|
2014
|
22 |
15 |
p. 4293-4297
5 p.
|
artikel
|
| 25 |
Lead identification of benzimidazolone and azabenzimidazolone arylsulfonamides as CC-chemokine receptor 4 (CCR4) antagonists
|
Miah, Afjal H.
|
|
2014
|
22 |
15 |
p. 4298-4311
14 p.
|
artikel
|
| 26 |
Melleolides induce rapid cell death in human primary monocytes and cancer cells
|
Bohnert, Markus
|
|
2014
|
22 |
15 |
p. 3856-3861
6 p.
|
artikel
|
| 27 |
Molecular mechanism of Symplectoteuthis bioluminescence—Part 4: Chromophore exchange and oxidation of the cysteine residue
|
Chou, Chun-Ming
|
|
2014
|
22 |
15 |
p. 4177-4188
12 p.
|
artikel
|
| 28 |
Novel pyrazoline derivatives as bi-inhibitor of COX-2 and B-Raf in treating cervical carcinoma
|
Yu, Minmin
|
|
2014
|
22 |
15 |
p. 4109-4118
10 p.
|
artikel
|
| 29 |
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines
|
Bukhari, Syed Nasir Abbas
|
|
2014
|
22 |
15 |
p. 4151-4161
11 p.
|
artikel
|
| 30 |
Position-specific modification with imidazolyl group on10–23 DNAzyme realized catalytic activity enhancement
|
Li, Zhiwen
|
|
2014
|
22 |
15 |
p. 4010-4017
8 p.
|
artikel
|
| 31 |
Potential C-terminal-domain inhibitors of heat shock protein 90 derived from a C-terminal peptide helix
|
Gavenonis, Jason
|
|
2014
|
22 |
15 |
p. 3989-3993
5 p.
|
artikel
|
| 32 |
Pyridine analogues of spirocyclic σ1 receptor ligands
|
Miyata, Kengo
|
|
2014
|
22 |
15 |
p. 4277-4284
8 p.
|
artikel
|
| 33 |
Pyrrolo- and pyridomorphinans: Non-selective opioid antagonists and delta opioid agonists/mu opioid partial agonists
|
Kumar, V.
|
|
2014
|
22 |
15 |
p. 4067-4072
6 p.
|
artikel
|
| 34 |
Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery
|
Tykvart, Jan
|
|
2014
|
22 |
15 |
p. 4099-4108
10 p.
|
artikel
|
| 35 |
RETRACTED: Design and synthesis of CHAP31, trapoxin B and HC-toxin based bicyclic tetrapeptides disulfide as potent histone deacetylase inhibitors
|
Hoque, Md. Ashraful
|
|
2014
|
22 |
15 |
p. 3850-3855
6 p.
|
artikel
|
| 36 |
SAR studies of differently functionalized chalcones based hydrazones and their cyclized derivatives as inhibitors of mammalian cathepsin B and cathepsin H
|
Raghav, Neera
|
|
2014
|
22 |
15 |
p. 4233-4245
13 p.
|
artikel
|
| 37 |
Selective inhibition of human carbonic anhydrases by novel amide derivatives of probenecid: Synthesis, biological evaluation and molecular modelling studies
|
D’Ascenzio, Melissa
|
|
2014
|
22 |
15 |
p. 3982-3988
7 p.
|
artikel
|
| 38 |
Spectroscopic investigations of the binding mechanisms between antimicrobial peptides and membrane models of Pseudomonas aeruginosa and Klebsiella pneumoniae
|
Chai, Hanbo
|
|
2014
|
22 |
15 |
p. 4210-4222
13 p.
|
artikel
|
| 39 |
Straightforward entry to pyrido[2,3-d]pyrimidine-2,4(1H,3H)-diones and their ADME properties
|
Jatczak, Martyna
|
|
2014
|
22 |
15 |
p. 3947-3956
10 p.
|
artikel
|
| 40 |
Structure-based optimization and biological evaluation of trisubstituted pyrazole as a core structure of potent ROS1 kinase inhibitors
|
Park, Byung Sun
|
|
2014
|
22 |
15 |
p. 3871-3878
8 p.
|
artikel
|
| 41 |
Synthesis and antibacterial activity of catecholate–ciprofloxacin conjugates
|
Fardeau, Sylvain
|
|
2014
|
22 |
15 |
p. 4049-4060
12 p.
|
artikel
|
| 42 |
Synthesis and biological activity of new salicylanilide N,N-disubstituted carbamates and thiocarbamates
|
Krátký, Martin
|
|
2014
|
22 |
15 |
p. 4073-4082
10 p.
|
artikel
|
| 43 |
Synthesis and biological evaluation of 2-anilino-4-substituted-7H-pyrrolopyrimidines as PDK1 inhibitors
|
O’Brien, Nathan J.
|
|
2014
|
22 |
15 |
p. 3879-3886
8 p.
|
artikel
|
| 44 |
Synthesis and biological evaluation of bivalent cannabinoid receptor ligands based on hCB2R selective benzimidazoles reveal unexpected intrinsic properties
|
Nimczick, Martin
|
|
2014
|
22 |
15 |
p. 3938-3946
9 p.
|
artikel
|
| 45 |
Synthesis and biological evaluation of novel radioiodinated imidazopyridine derivatives for amyloid-β imaging in Alzheimer’s disease
|
Chen, Chun-Jen
|
|
2014
|
22 |
15 |
p. 4189-4197
9 p.
|
artikel
|
| 46 |
Synthesis and cholinesterase inhibition of cativic acid derivatives
|
Alza, Natalia P.
|
|
2014
|
22 |
15 |
p. 3838-3849
12 p.
|
artikel
|
| 47 |
Synthesis and evaluation of N 6-substituted apioadenosines as potential adenosine A3 receptor modulators
|
Toti, Kiran S.
|
|
2014
|
22 |
15 |
p. 4257-4268
12 p.
|
artikel
|
| 48 |
Synthesis and evaluation of the novel 2-[18F]fluoro-3-propoxy-triazole-pyridine-substituted losartan for imaging AT1 receptors
|
Arksey, Natasha
|
|
2014
|
22 |
15 |
p. 3931-3937
7 p.
|
artikel
|
| 49 |
Synthesis and fungicidal activity of quinolin-6-yloxyacetamides, a novel class of tubulin polymerization inhibitors
|
Lamberth, Clemens
|
|
2014
|
22 |
15 |
p. 3922-3930
9 p.
|
artikel
|
| 50 |
Synthesis and SAR studies of benzyl ether derivatives as potent orally active S1P1 agonists
|
Tsuji, Takashi
|
|
2014
|
22 |
15 |
p. 4246-4256
11 p.
|
artikel
|
| 51 |
Synthesis and structure–activity relationship of thiobarbituric acid derivatives as potent inhibitors of urease
|
Khan, Khalid Mohammed
|
|
2014
|
22 |
15 |
p. 4119-4123
5 p.
|
artikel
|
| 52 |
Synthesis and structure–activity relationships of new carbonyl guanidine derivatives as novel dual 5-HT2B and 5-HT7 receptor antagonists. Part 2
|
Moritomo, Ayako
|
|
2014
|
22 |
15 |
p. 4323-4337
15 p.
|
artikel
|
| 53 |
Synthesis, antioxidant and cytoprotective evaluation of potential antiatherogenic phenolic hydrazones. A structure–activity relationship insight
|
Vanucci-Bacqué, Corinne
|
|
2014
|
22 |
15 |
p. 4269-4276
8 p.
|
artikel
|
| 54 |
Synthesis, biological evaluation and molecular modeling of 1,3,4-thiadiazol-2-amide derivatives as novel antitubulin agents
|
Li, Yu-Jing
|
|
2014
|
22 |
15 |
p. 4312-4322
11 p.
|
artikel
|
| 55 |
Synthesis of new compounds with promising antiviral properties against group A and B Human Rhinoviruses
|
Bernard, Angela M.
|
|
2014
|
22 |
15 |
p. 4061-4066
6 p.
|
artikel
|
| 56 |
Synthesis, reactivity and biological activity of N(4)-boronated derivatives of 2′-deoxycytidine
|
Nizioł, Joanna
|
|
2014
|
22 |
15 |
p. 3906-3912
7 p.
|
artikel
|
| 57 |
Target evaluation of deoxyhypusine synthase from Theileria parva the neglected animal parasite and its relationship to Plasmodium
|
Njuguna, James T.
|
|
2014
|
22 |
15 |
p. 4338-4346
9 p.
|
artikel
|
| 58 |
The development of new molecular tools containing a chemically synthesized carbohydrate ligand for the elucidation of carbohydrate roles via photoaffinity labeling: Carbohydrate–protein interactions are affected by the structures of the glycosidic bonds and the reducing-end sugar
|
Ohtsuka, Isao
|
|
2014
|
22 |
15 |
p. 3829-3837
9 p.
|
artikel
|
| 59 |
Topoisomerase II inhibitors from the roots of Stellera chamaejasme L.
|
Liu, Li-Ping
|
|
2014
|
22 |
15 |
p. 4198-4203
6 p.
|
artikel
|
| 60 |
Triazolopyridyl ketones as a novel class of antileishmanial agents. DNA binding and BSA interaction
|
Adam, Rosa
|
|
2014
|
22 |
15 |
p. 4018-4027
10 p.
|
artikel
|
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