| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A series of nonsecosteroidal vitamin D receptor agonists for osteoporosis therapy
|
Kashiwagi, Hirotaka
|
|
2013
|
21 |
7 |
p. 1823-1833
11 p.
|
artikel
|
| 2 |
Bioorganic & Medicinal Chemistry Reviews and Perspectives
|
|
|
2013
|
21 |
7 |
p. I-III
nvt p.
|
artikel
|
| 3 |
Bromo-deaza-SAH: A potent and selective DOT1L inhibitor
|
Yu, Wenyu
|
|
2013
|
21 |
7 |
p. 1787-1794
8 p.
|
artikel
|
| 4 |
Corrigendum to “Identification and evaluation of antioxidant, analgesic/anti-inflammatory activity of the most active ninhydrin–phenol adducts synthesized” [Bioorg. Med. Chem. 14 (2006) 7113–7120]
|
Prabhakar, K.R.
|
|
2013
|
21 |
7 |
p. 2177-
1 p.
|
artikel
|
| 5 |
Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182
|
Mizuhara, Tsukasa
|
|
2013
|
21 |
7 |
p. 2079-2087
9 p.
|
artikel
|
| 6 |
Design and synthesis of 3,5-diaryl-4,5-dihydro-1H-pyrazoles as new tyrosinase inhibitors
|
Zhou, Zhixuan
|
|
2013
|
21 |
7 |
p. 2156-2162
7 p.
|
artikel
|
| 7 |
Design and synthesis of glycoprotein-based multivalent glyco-ligands for influenza hemagglutinin and human galectin-3
|
Wang, Helen
|
|
2013
|
21 |
7 |
p. 2037-2044
8 p.
|
artikel
|
| 8 |
Design, structure–activity relationship and in vivo efficacy of piperazine analogues of fenarimol as inhibitors of Trypanosoma cruzi
|
Keenan, Martine
|
|
2013
|
21 |
7 |
p. 1756-1763
8 p.
|
artikel
|
| 9 |
Design, synthesis, and binding mode prediction of 2-pyridone-based selective CB2 receptor agonists
|
Kusakabe, Ken-ichi
|
|
2013
|
21 |
7 |
p. 2045-2055
11 p.
|
artikel
|
| 10 |
Design, synthesis and pharmacological evaluation of omeprazole-like agents with anti-inflammatory activity
|
El-Nezhawy, Ahmed O.H.
|
|
2013
|
21 |
7 |
p. 1661-1670
10 p.
|
artikel
|
| 11 |
Development of silicon-containing bis-phenol derivatives as androgen receptor antagonists: Selectivity switching by C/Si exchange
|
Nakamura, Masaharu
|
|
2013
|
21 |
7 |
p. 1643-1651
9 p.
|
artikel
|
| 12 |
Discovery and structure–activity relationship of thienopyridine derivatives as bone anabolic agents
|
Saito, Keiji
|
|
2013
|
21 |
7 |
p. 1628-1642
15 p.
|
artikel
|
| 13 |
Discovery of dopamine D4 receptor antagonists with planar chirality
|
Sanna, Fabrizio
|
|
2013
|
21 |
7 |
p. 1680-1684
5 p.
|
artikel
|
| 14 |
Discovery of novel tricyclic indole derived inhibitors of HCV NS5B RNA dependent RNA polymerase
|
Venkatraman, Srikanth
|
|
2013
|
21 |
7 |
p. 2007-2017
11 p.
|
artikel
|
| 15 |
Discovery of potent dipeptidyl peptidase IV inhibitors through pharmacophore hybridization and hit-to-lead optimization
|
Zeng, Shaogao
|
|
2013
|
21 |
7 |
p. 1749-1755
7 p.
|
artikel
|
| 16 |
Editorial board
|
|
|
2013
|
21 |
7 |
p. IFC-
1 p.
|
artikel
|
| 17 |
Enantiomer and conformer recognition of (+) and (−)-disparlure and their analogs by the pheromone binding proteins of the gypsy moth, Lymantria dispar
|
Yu, Yang
|
|
2013
|
21 |
7 |
p. 1811-1822
12 p.
|
artikel
|
| 18 |
Five-membered iminocyclitol α-glucosidase inhibitors: Synthetic, biological screening and in silico studies
|
Guerreiro, Luis R.
|
|
2013
|
21 |
7 |
p. 1911-1917
7 p.
|
artikel
|
| 19 |
Fungal metabolites of xanthohumol with potent antiproliferative activity on human cancer cell lines in vitro
|
Tronina, Tomasz
|
|
2013
|
21 |
7 |
p. 2001-2006
6 p.
|
artikel
|
| 20 |
Graphical contents list
|
|
|
2013
|
21 |
7 |
p. 1583-1598
16 p.
|
artikel
|
| 21 |
Hit identification of novel heparanase inhibitors by structure- and ligand-based approaches
|
Gozalbes, Rafael
|
|
2013
|
21 |
7 |
p. 1944-1951
8 p.
|
artikel
|
| 22 |
Improvement of σ1 receptor affinity by late-stage C–H-bond arylation of spirocyclic lactones
|
Meyer, Christina
|
|
2013
|
21 |
7 |
p. 1844-1856
13 p.
|
artikel
|
| 23 |
Improving the inhibitory activity of arylidenaminoguanidine compounds at the N-methyl-d-aspartate receptor complex from a recursive computational-experimental structure–activity relationship study
|
Ring, Joshua R.
|
|
2013
|
21 |
7 |
p. 1764-1774
11 p.
|
artikel
|
| 24 |
Investigation of σ receptors agonist/antagonist activity through N-(6-methoxytetralin-1-yl)- and N-(6-methoxynaphthalen-1-yl)alkyl derivatives of polymethylpiperidines
|
Niso, Mauro
|
|
2013
|
21 |
7 |
p. 1865-1869
5 p.
|
artikel
|
| 25 |
Novel antiobesity agents: Synthesis and pharmacological evaluation of analogues of Rimonabant and of LH21
|
Alvarado, Mario
|
|
2013
|
21 |
7 |
p. 1708-1716
9 p.
|
artikel
|
| 26 |
Novel imidazophenoxazine-4-sulfonamides: Their synthesis and evaluation as potential inhibitors of PDE4
|
Reddy, Seelam Venkata
|
|
2013
|
21 |
7 |
p. 1952-1963
12 p.
|
artikel
|
| 27 |
Novel inhibitors of bacterial virulence: Development of 5,6-dihydrobenzo[h]quinazolin-4(3H)-ones for the inhibition of group A streptococcal streptokinase expression
|
Yestrepsky, Bryan D.
|
|
2013
|
21 |
7 |
p. 1880-1897
18 p.
|
artikel
|
| 28 |
Novel leucine ureido derivatives as inhibitors of aminopeptidase N (APN)
|
Ma, Chunhua
|
|
2013
|
21 |
7 |
p. 1621-1627
7 p.
|
artikel
|
| 29 |
Novel pseudopeptides incorporating a benzodiazepine-based turn mimetic—targeting Mycobacterium tuberculosis ribonucleotide reductase
|
Nurbo, Johanna
|
|
2013
|
21 |
7 |
p. 1992-2000
9 p.
|
artikel
|
| 30 |
Novel R-roscovitine NO-donor hybrid compounds as potential pro-resolution of inflammation agents
|
Montanaro, Gabriele
|
|
2013
|
21 |
7 |
p. 2107-2116
10 p.
|
artikel
|
| 31 |
Novel symmetrical ureas as modulators of protein arginine methyl transferases
|
Fontán, Noelia
|
|
2013
|
21 |
7 |
p. 2056-2067
12 p.
|
artikel
|
| 32 |
Olive secoiridoids and semisynthetic bioisostere analogues for the control of metastatic breast cancer
|
Busnena, Belnaser A.
|
|
2013
|
21 |
7 |
p. 2117-2127
11 p.
|
artikel
|
| 33 |
6-Oxo and 6-thio purine analogs as antimycobacterial agents
|
Pathak, Ashish K.
|
|
2013
|
21 |
7 |
p. 1685-1695
11 p.
|
artikel
|
| 34 |
Peripherally acting novel lipo-endomorphin-1 peptides in neuropathic pain without producing constipation
|
Varamini, Pegah
|
|
2013
|
21 |
7 |
p. 1898-1904
7 p.
|
artikel
|
| 35 |
Preliminary biological evaluation and mechanism of action studies of selected 2-arylindoles against glioblastoma
|
Prabhu, Saurabh
|
|
2013
|
21 |
7 |
p. 1918-1924
7 p.
|
artikel
|
| 36 |
Probing functional diversity in pactamycin toward antibiotic, antitumor, and antiprotozoal activity
|
Hanessian, Stephen
|
|
2013
|
21 |
7 |
p. 1775-1786
12 p.
|
artikel
|
| 37 |
Quercetin–POC conjugates: Differential stability and bioactivity profiles between breast cancer (MCF-7) and colorectal carcinoma (HCT116) cell lines
|
Cho, Suh Young
|
|
2013
|
21 |
7 |
p. 1671-1679
9 p.
|
artikel
|
| 38 |
Selective aminopeptidase-N (CD13) inhibitors with relevance to cancer chemotherapy
|
Schmitt, Céline
|
|
2013
|
21 |
7 |
p. 2135-2144
10 p.
|
artikel
|
| 39 |
α-Selective glycosylation affords mucin-related GalNAc amino acids and diketopiperazines active on Trypanosoma cruzi
|
Martins-Teixeira, Maristela B.
|
|
2013
|
21 |
7 |
p. 1978-1987
10 p.
|
artikel
|
| 40 |
Semisynthetic studies identify mitochondria poisons from botanical dietary supplements—Geranyloxycoumarins from Aegle marmelos
|
Li, Jun
|
|
2013
|
21 |
7 |
p. 1795-1803
9 p.
|
artikel
|
| 41 |
Small-molecule inhibition of the uPAR·uPA interaction: Synthesis, biochemical, cellular, in vivo pharmacokinetics and efficacy studies in breast cancer metastasis
|
Mani, Timmy
|
|
2013
|
21 |
7 |
p. 2145-2155
11 p.
|
artikel
|
| 42 |
Small molecule inhibitors of PCNA/PIP-box interaction suppress translesion DNA synthesis
|
Actis, Marcelo
|
|
2013
|
21 |
7 |
p. 1972-1977
6 p.
|
artikel
|
| 43 |
Sponge-derived acetylenic alcohols, petrosiols, inhibit proliferation and migration of platelet-derived growth factor (PDGF)-induced vascular smooth muscle cells
|
Choi, Bong-Keun
|
|
2013
|
21 |
7 |
p. 1804-1810
7 p.
|
artikel
|
| 44 |
Stereoselective synthesis of a new class of potent and selective inhibitors of human Δ8,7-sterol isomerase
|
König, Mathias
|
|
2013
|
21 |
7 |
p. 1925-1943
19 p.
|
artikel
|
| 45 |
Substituted indolin-2-ones as p90 ribosomal S6 protein kinase 2 (RSK2) inhibitors: Molecular docking simulation and structure–activity relationship analysis
|
Zhong, Ye
|
|
2013
|
21 |
7 |
p. 1724-1734
11 p.
|
artikel
|
| 46 |
4-Substituted-2,3,5,6-tetrafluorobenzenesulfonamides as inhibitors of carbonic anhydrases I, II, VII, XII, and XIII
|
Dudutienė, Virginija
|
|
2013
|
21 |
7 |
p. 2093-2106
14 p.
|
artikel
|
| 47 |
Synthesis and biological activity of 5-chloro-N 4-substituted phenyl-9H-pyrimido[4,5-b]indole-2,4-diamines as vascular endothelial growth factor receptor-2 inhibitors and antiangiogenic agents
|
Gangjee, Aleem
|
|
2013
|
21 |
7 |
p. 1857-1864
8 p.
|
artikel
|
| 48 |
Synthesis and biological evaluation of helioxanthin analogues
|
Janmanchi, Damodar
|
|
2013
|
21 |
7 |
p. 2163-2176
14 p.
|
artikel
|
| 49 |
Synthesis and biological evaluation of pyridazine derivatives as novel HIV-1 NNRTIs
|
Li, Dongyue
|
|
2013
|
21 |
7 |
p. 2128-2134
7 p.
|
artikel
|
| 50 |
Synthesis and biological evaluation of substituted imidazoquinoline derivatives as mPGES-1 inhibitors
|
Shiro, Tomoya
|
|
2013
|
21 |
7 |
p. 2068-2078
11 p.
|
artikel
|
| 51 |
Synthesis and discovery of novel piperidone-grafted mono- and bis-spirooxindole-hexahydropyrrolizines as potent cholinesterase inhibitors
|
Kia, Yalda
|
|
2013
|
21 |
7 |
p. 1696-1707
12 p.
|
artikel
|
| 52 |
Synthesis and evaluation of coumarin derivatives as potential dual-action HIV-1 protease and reverse transcriptase inhibitors
|
Olomola, Temitope O.
|
|
2013
|
21 |
7 |
p. 1964-1971
8 p.
|
artikel
|
| 53 |
Synthesis and in vitro evaluation of new derivatives of 2-substituted-6-fluorobenzo[d]thiazoles as cholinesterase inhibitors
|
Imramovský, Aleš
|
|
2013
|
21 |
7 |
p. 1735-1748
14 p.
|
artikel
|
| 54 |
Synthesis and properties of cationic oligopeptides with different side chain lengths that bind to RNA duplexes
|
Maeda, Yusuke
|
|
2013
|
21 |
7 |
p. 1717-1723
7 p.
|
artikel
|
| 55 |
Synthesis, characterization and Akt phosphorylation inhibitory activity of cyclopentanecarboxylate-substituted alkylphosphocholines
|
Alam, Md. Maqusood
|
|
2013
|
21 |
7 |
p. 2018-2024
7 p.
|
artikel
|
| 56 |
Synthesis of new fluorinated, 2-substituted 5-pyrrolidinylsulfonyl isatin derivatives as caspase-3 and caspase-7 inhibitors: Nonradioactive counterparts of putative PET-compatible apoptosis imaging agents
|
Limpachayaporn, Panupun
|
|
2013
|
21 |
7 |
p. 2025-2036
12 p.
|
artikel
|
| 57 |
Synthesis of novel azo compounds containing 5(4H)-oxazolone ring as potent tyrosinase inhibitors
|
Hamidian, Hooshang
|
|
2013
|
21 |
7 |
p. 2088-2092
5 p.
|
artikel
|
| 58 |
Synthesis of novel isoflavene–propranolol hybrids as anti-tumor agents
|
Yee, Eugene M.H.
|
|
2013
|
21 |
7 |
p. 1652-1660
9 p.
|
artikel
|
| 59 |
Thiazolidine-2,4-diones: Progress towards multifarious applications
|
Jain, Viral S.
|
|
2013
|
21 |
7 |
p. 1599-1620
22 p.
|
artikel
|
| 60 |
TOPS-MODE model of multiplexing neuroprotective effects of drugs and experimental-theoretic study of new 1,3-rasagiline derivatives potentially useful in neurodegenerative diseases
|
Luan, Feng
|
|
2013
|
21 |
7 |
p. 1870-1879
10 p.
|
artikel
|
| 61 |
Two-component covalent inhibitor
|
Cornett, Evan M.
|
|
2013
|
21 |
7 |
p. 1988-1991
4 p.
|
artikel
|
| 62 |
(+)-Usnic acid enamines with remarkable cicatrizing properties
|
Bruno, Michela
|
|
2013
|
21 |
7 |
p. 1834-1843
10 p.
|
artikel
|
| 63 |
Vavilosides A1/A2–B1/B2, new furostane glycosides from the bulbs of Allium vavilovii with cytotoxic activity
|
Zolfaghari, Behzad
|
|
2013
|
21 |
7 |
p. 1905-1910
6 p.
|
artikel
|
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