| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A CD4 mimic as an HIV entry inhibitor: Pharmacokinetics
|
Hashimoto, Chie
|
|
2013
|
21 |
24 |
p. 7884-7889
6 p.
|
artikel
|
| 2 |
A new peptidyl fluorescent chemosensors for the selective detection of mercury ions based on tetrapeptide
|
Thirupathi, Ponnaboina
|
|
2013
|
21 |
24 |
p. 7964-7970
7 p.
|
artikel
|
| 3 |
A novel nitro-substituted benzothiadiazole as fluorescent probe for tumor cells under hypoxic condition
|
Jiang, Qian
|
|
2013
|
21 |
24 |
p. 7735-7741
7 p.
|
artikel
|
| 4 |
Antioxidant action of propolis on mouse lungs exposed to short-term cigarette smoke
|
Lopes, Alan Aguiar
|
|
2013
|
21 |
24 |
p. 7570-7577
8 p.
|
artikel
|
| 5 |
Antioxidant activities of 5-hydroxyoxindole and its 3-hydroxy-3-phenacyl derivatives: The suppression of lipid peroxidation and intracellular oxidative stress
|
Yasuda, Daisuke
|
|
2013
|
21 |
24 |
p. 7709-7714
6 p.
|
artikel
|
| 6 |
Antiprion compounds that reduce PrPSc levels in dividing and stationary-phase cells
|
Silber, B. Michael
|
|
2013
|
21 |
24 |
p. 7999-8012
14 p.
|
artikel
|
| 7 |
Benzyloxybenzylammonium chlorides: Simple amine salts that display anticonvulsant activity
|
Lee, Hyosung
|
|
2013
|
21 |
24 |
p. 7655-7662
8 p.
|
artikel
|
| 8 |
Bioactive compounds from Stuhlmannia moavi from the Madagascar dry forest
|
Liu, Yixi
|
|
2013
|
21 |
24 |
p. 7591-7594
4 p.
|
artikel
|
| 9 |
Chromenylchalcones with inhibitory effects on monoamine oxidase B
|
Jo, Geunhyeong
|
|
2013
|
21 |
24 |
p. 7890-7897
8 p.
|
artikel
|
| 10 |
Design and synthesis of novel antimicrobials with activity against Gram-positive bacteria and mycobacterial species, including M. tuberculosis
|
Tiruveedhula, V.V.N. Phani Babu
|
|
2013
|
21 |
24 |
p. 7830-7840
11 p.
|
artikel
|
| 11 |
Design and synthesis of novel benzimidazole derivatives as phosphodiesterase 10A inhibitors with reduced CYP1A2 inhibition
|
Hamaguchi, Wataru
|
|
2013
|
21 |
24 |
p. 7612-7623
12 p.
|
artikel
|
| 12 |
Design, synthesis, and biological activities of novel hexahydropyrazino[1,2-a]indole derivatives as potent inhibitors of apoptosis (IAP) proteins antagonists with improved membrane permeability across MDR1 expressing cells
|
Shiokawa, Zenyu
|
|
2013
|
21 |
24 |
p. 7938-7954
17 p.
|
artikel
|
| 13 |
Design, synthesis and biological evaluation of novel 4-anilinoquinazolines with C-6 urea-linked side chains as inhibitors of the epidermal growth factor receptor
|
Zhang, Xu
|
|
2013
|
21 |
24 |
p. 7988-7998
11 p.
|
artikel
|
| 14 |
Design, synthesis, and biological evaluation of 1,2,4-triazole bearing 5-substituted biphenyl-2-sulfonamide derivatives as potential antihypertensive candidates
|
Liu, Jie
|
|
2013
|
21 |
24 |
p. 7742-7751
10 p.
|
artikel
|
| 15 |
Discovery and characterisation of hydrazines as inhibitors of the immune suppressive enzyme, indoleamine 2,3-dioxygenase 1 (IDO1)
|
Fung, Sai-Parng S.
|
|
2013
|
21 |
24 |
p. 7595-7603
9 p.
|
artikel
|
| 16 |
Discovery of a novel activator of 5-lipoxygenase from an anacardic acid derived compound collection
|
Wisastra, Rosalina
|
|
2013
|
21 |
24 |
p. 7763-7778
16 p.
|
artikel
|
| 17 |
Discovery of N-{5-[3-(3-hydroxypiperidin-1-yl)-1,2,4-oxadiazol-5-yl]-4-methyl-1,3-thiazol-2-yl}acetamide (TASP0415914) as an orally potent phosphoinositide 3-kinase γ inhibitor for the treatment of inflammatory diseases
|
Oka, Yusuke
|
|
2013
|
21 |
24 |
p. 7578-7583
6 p.
|
artikel
|
| 18 |
Discovery of XEN445: A potent and selective endothelial lipase inhibitor raises plasma HDL-cholesterol concentration in mice
|
Sun, Shaoyi
|
|
2013
|
21 |
24 |
p. 7724-7734
11 p.
|
artikel
|
| 19 |
Editorial board
|
|
|
2013
|
21 |
24 |
p. IFC-
1 p.
|
artikel
|
| 20 |
Effect of Ala replacement with Aib in amphipathic cell-penetrating peptide on oligonucleotide delivery into cells
|
Wada, Shun-ichi
|
|
2013
|
21 |
24 |
p. 7669-7673
5 p.
|
artikel
|
| 21 |
Further discovery of caffeic acid derivatives as novel influenza neuraminidase inhibitors
|
Xie, Yuanchao
|
|
2013
|
21 |
24 |
p. 7715-7723
9 p.
|
artikel
|
| 22 |
Graphical contents list
|
|
|
2013
|
21 |
24 |
p. 7549-7561
13 p.
|
artikel
|
| 23 |
Heptaoxygenated xanthones as anti-austerity agents from Securidaca longepedunculata
|
Dibwe, Dya Fita
|
|
2013
|
21 |
24 |
p. 7663-7668
6 p.
|
artikel
|
| 24 |
Inhibitors of tissue-nonspecific alkaline phosphatase: Design, synthesis, kinetics, biomineralization and cellular tests
|
Debray, Julien
|
|
2013
|
21 |
24 |
p. 7981-7987
7 p.
|
artikel
|
| 25 |
Investigation of quinazolines as inhibitors of breast cancer resistance protein (ABCG2)
|
Juvale, Kapil
|
|
2013
|
21 |
24 |
p. 7858-7873
16 p.
|
artikel
|
| 26 |
Isoquinoline derivatives as potent CRTH2 antagonists: Design, synthesis and SAR
|
Nishikawa-Shimono, Rie
|
|
2013
|
21 |
24 |
p. 7674-7685
12 p.
|
artikel
|
| 27 |
Novel method of the synthesis and hybridization properties of an oligonucleotide containing non-ionic diisopropylsilyl internucleotide linkage
|
Moriguchi, Tomohisa
|
|
2013
|
21 |
24 |
p. 8013-8018
6 p.
|
artikel
|
| 28 |
Pivaloylcodeine, a new codeine derivative, for the inhibition of morphine glucuronidation. An in vitro study in the rat
|
Antonilli, Letizia
|
|
2013
|
21 |
24 |
p. 7955-7963
9 p.
|
artikel
|
| 29 |
Potent and broad-spectrum antibacterial activity of indole-based bisamidine antibiotics: Synthesis and SAR of novel analogs of MBX 1066 and MBX 1090
|
Williams, John D.
|
|
2013
|
21 |
24 |
p. 7790-7806
17 p.
|
artikel
|
| 30 |
Structure-based design, synthesis, and evaluation of imidazo[1,2-b]pyridazine and imidazo[1,2-a]pyridine derivatives as novel dual c-Met and VEGFR2 kinase inhibitors
|
Matsumoto, Shigemitsu
|
|
2013
|
21 |
24 |
p. 7686-7698
13 p.
|
artikel
|
| 31 |
Sulphonamide 1,4-dithia-7-azaspiro[4,4]nonane derivatives as gelatinase A inhibitors
|
Shi, Leilei
|
|
2013
|
21 |
24 |
p. 7752-7762
11 p.
|
artikel
|
| 32 |
Synthesis and biological evaluation of 3-hydroxymethyl-5-(1H-1,2,3-triazol) isoxazolidines
|
Romeo, Roberto
|
|
2013
|
21 |
24 |
p. 7929-7937
9 p.
|
artikel
|
| 33 |
Synthesis and biological evaluation of substituted 1,2,3-benzotriazines and pyrido[3,2-d]-1,2,3-triazines as inhibitors of vascular endothelial growth factor receptor-2
|
Zhao, Xing-Wang
|
|
2013
|
21 |
24 |
p. 7807-7815
9 p.
|
artikel
|
| 34 |
Synthesis and cytotoxicity of pyranonaphthoquinone natural product analogues under bioreductive conditions
|
Heapy, Amanda M.
|
|
2013
|
21 |
24 |
p. 7971-7980
10 p.
|
artikel
|
| 35 |
Synthesis and evaluation of stability of m3G-CAP analogues in serum-supplemented medium and cytosolic extract
|
Honcharenko, Malgorzata
|
|
2013
|
21 |
24 |
p. 7921-7928
8 p.
|
artikel
|
| 36 |
Synthesis and pharmacological characterization of benzenesulfonamides as dual species inhibitors of human and murine mPGES-1
|
Hanke, Thomas
|
|
2013
|
21 |
24 |
p. 7874-7883
10 p.
|
artikel
|
| 37 |
Synthesis and pharmacological evaluation of novel bisindolylalkanes analogues
|
Song, Ya-Li
|
|
2013
|
21 |
24 |
p. 7624-7627
4 p.
|
artikel
|
| 38 |
Synthesis and structure–activity relationships of new carbonyl guanidine derivatives as novel dual 5-HT2B and 5-HT7 receptor antagonists
|
Moritomo, Ayako
|
|
2013
|
21 |
24 |
p. 7841-7852
12 p.
|
artikel
|
| 39 |
Synthesis, cytotoxic evaluation and molecular docking study of 2-alkylthio-4-(2,3,4-trimethoxyphenyl)-5-aryl-thiazoles as tubulin polymerization inhibitors
|
Salehi, Marjan
|
|
2013
|
21 |
24 |
p. 7648-7654
7 p.
|
artikel
|
| 40 |
Synthesis, docking and pharmacological evaluation of novel homo- and hetero-bis 3-piperazinylpropylindole derivatives at SERT and 5-HT1A receptor
|
Pessoa-Mahana, Hernán
|
|
2013
|
21 |
24 |
p. 7604-7611
8 p.
|
artikel
|
| 41 |
Synthesis of structurally diverse benzosuberene analogues and their biological evaluation as anti-cancer agents
|
Tanpure, Rajendra P.
|
|
2013
|
21 |
24 |
p. 8019-8032
14 p.
|
artikel
|
| 42 |
Synthesis of vitamin D3 analogues with A-ring modifications to directly measure vitamin D levels in biological samples
|
Hernández-Martín, Alba
|
|
2013
|
21 |
24 |
p. 7779-7789
11 p.
|
artikel
|
| 43 |
Synthesis, radiosynthesis and first in vitro evaluation of novel PET-tracers for the dopamine transporter: [11C]IPCIT and [18F]FE@IPCIT
|
Rami-Mark, Christina
|
|
2013
|
21 |
24 |
p. 7562-7569
8 p.
|
artikel
|
| 44 |
Tackling the conformational sampling of larger flexible compounds and macrocycles in pharmacology and drug discovery
|
Chen, I-Jen
|
|
2013
|
21 |
24 |
p. 7898-7920
23 p.
|
artikel
|
| 45 |
The most effective influence of 17-(3-ethoxypropyl) substituent on the binding affinity and the agonistic activity in KNT-127 derivatives, δ opioid receptor agonists
|
Nemoto, Toru
|
|
2013
|
21 |
24 |
p. 7628-7647
20 p.
|
artikel
|
| 46 |
The synthesis and biodistribution of [11C]metformin as a PET probe to study hepatobiliary transport mediated by the multi-drug and toxin extrusion transporter 1 (MATE1) in vivo
|
Hume, W. Ewan
|
|
2013
|
21 |
24 |
p. 7584-7590
7 p.
|
artikel
|
| 47 |
Towards tropomyosin-related kinase B (TrkB) receptor ligands for brain imaging with PET: Radiosynthesis and evaluation of 2-(4-[18F]fluorophenyl)-7,8-dihydroxy-4H-chromen-4-one and 2-(4-([N-methyl-11C]-dimethylamino)phenyl)-7,8-dihydroxy-4H-chromen-4-one
|
Bernard-Gauthier, Vadim
|
|
2013
|
21 |
24 |
p. 7816-7829
14 p.
|
artikel
|
| 48 |
Transnitrosation of alicyclic N-nitrosamines containing a sulfur atom
|
Inami, Keiko
|
|
2013
|
21 |
24 |
p. 7853-7857
5 p.
|
artikel
|
| 49 |
Tyrosinase and Layer-by-Layer supported tyrosinases in the synthesis of lipophilic catechols with antiinfluenza activity
|
Bozzini, Tiziana
|
|
2013
|
21 |
24 |
p. 7699-7708
10 p.
|
artikel
|
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