| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A new class of aggregation inhibitor of amyloid-β peptide based on an O-acyl isopeptide
|
Kawashima, Hiroyuki
|
|
2013
|
21 |
21 |
p. 6323-6327
5 p.
|
artikel
|
| 2 |
A novel pH sensitive water soluble fluorescent nanomicellar sensor for potential biomedical applications
|
Georgiev, Nikolai I.
|
|
2013
|
21 |
21 |
p. 6292-6302
11 p.
|
artikel
|
| 3 |
Antimycobacterial and herbicidal activity of ring-substituted 1-hydroxynaphthalene-2-carboxanilides
|
Gonec, Tomas
|
|
2013
|
21 |
21 |
p. 6531-6541
11 p.
|
artikel
|
| 4 |
Arylamino methylene bisphosphonate derivatives as bone seeking matrix metalloproteinase inhibitors
|
Tauro, Marilena
|
|
2013
|
21 |
21 |
p. 6456-6465
10 p.
|
artikel
|
| 5 |
A synthetic compound, 4-acetyl-3-methyl-6-(3,4,5-trimethoxyphenyl)pyrano[3,4-c]pyran-1,8-dione, ameliorates ovalbumin-induced asthma
|
Chung, Hwan-Suck
|
|
2013
|
21 |
21 |
p. 6359-6365
7 p.
|
artikel
|
| 6 |
Bacterial neuraminidase inhibitory effects of prenylated isoflavones from roots of Flemingia philippinensis
|
Wang, Yan
|
|
2013
|
21 |
21 |
p. 6398-6404
7 p.
|
artikel
|
| 7 |
Binding mode characterization of 6α- and 6β-N-heterocyclic substituted naltrexamine derivatives via docking in opioid receptor crystal structures and site-directed mutagenesis studies: Application of the ‘message–address’ concept in development of mu opioid receptor selective antagonists
|
Zaidi, Saheem A.
|
|
2013
|
21 |
21 |
p. 6405-6413
9 p.
|
artikel
|
| 8 |
Biodistribution of vaccines comprised of hydrophobically-modified poly(γ-glutamic acid) nanoparticles and antigen proteins using fluorescence imaging
|
Toita, Riki
|
|
2013
|
21 |
21 |
p. 6608-6615
8 p.
|
artikel
|
| 9 |
‘Click’ synthesized sterol-based cationic lipids as gene carriers, and the effect of skeletons and headgroups on gene delivery
|
Sheng, Ruilong
|
|
2013
|
21 |
21 |
p. 6366-6377
12 p.
|
artikel
|
| 10 |
Colorimetric/fluorogenic detection of thiols by N-fused porphyrin in water
|
Ikawa, Yoshiya
|
|
2013
|
21 |
21 |
p. 6501-6505
5 p.
|
artikel
|
| 11 |
Conformational restriction approach to β-secretase (BACE1) inhibitors III: Effective investigation of the binding mode by combinational use of X-ray analysis, isothermal titration calorimetry and theoretical calculations
|
Yonezawa, Shuji
|
|
2013
|
21 |
21 |
p. 6506-6522
17 p.
|
artikel
|
| 12 |
Corrigendum to “Defining the key pharmacophore elements of PF-04620110: Discovery of a potent, orally-active, neutral DGAT-1 inhibitor” [Bioorg. Med. Chem. 21 (2013) 5081–5097]
|
Dow, Robert L.
|
|
2013
|
21 |
21 |
p. 6855-
1 p.
|
artikel
|
| 13 |
Corrigendum to “Synthesis and evaluation of coumarin derivatives as potential dual-action HIV-1 protease and reverse transcriptase inhibitors” [Bioorg. Med. Chem. 21 (2013) 1964–1971]
|
Olomola, Temitope O.
|
|
2013
|
21 |
21 |
p. 6856-
1 p.
|
artikel
|
| 14 |
Design and bio-evaluation of indole derivatives as potent Kv1.5 inhibitors
|
Guo, Xiaoke
|
|
2013
|
21 |
21 |
p. 6466-6476
11 p.
|
artikel
|
| 15 |
Design, synthesis and anticonvulsant properties of new N-Mannich bases derived from 3-phenylpyrrolidine-2,5-diones
|
Kamiński, Krzysztof
|
|
2013
|
21 |
21 |
p. 6821-6830
10 p.
|
artikel
|
| 16 |
Design, synthesis and biological evaluation of millepachine derivatives as a new class of tubulin polymerization inhibitors
|
Wang, Guangcheng
|
|
2013
|
21 |
21 |
p. 6844-6854
11 p.
|
artikel
|
| 17 |
Design, synthesis and biological evaluation of novel anti-cytokine 1,2,4-triazine derivatives
|
Khoshneviszadeh, Mehdi
|
|
2013
|
21 |
21 |
p. 6708-6717
10 p.
|
artikel
|
| 18 |
Development of a novel fluorine-18 labeled deuterated fluororasagiline ([18F]fluororasagiline-D2) radioligand for PET studies of monoamino oxidase B (MAO-B)
|
Nag, S.
|
|
2013
|
21 |
21 |
p. 6634-6641
8 p.
|
artikel
|
| 19 |
Dimeric argininamide-type neuropeptide Y receptor antagonists: Chiral discrimination between Y1 and Y4 receptors
|
Keller, Max
|
|
2013
|
21 |
21 |
p. 6303-6322
20 p.
|
artikel
|
| 20 |
Discovery and characterization of NVP-QAV680, a potent and selective CRTh2 receptor antagonist suitable for clinical testing in allergic diseases
|
Sandham, David A.
|
|
2013
|
21 |
21 |
p. 6582-6591
10 p.
|
artikel
|
| 21 |
Discovery and characterization of synthetic 4′-hydroxyflavones—New CK2 inhibitors from flavone family
|
Golub, Andriy G.
|
|
2013
|
21 |
21 |
p. 6681-6689
9 p.
|
artikel
|
| 22 |
Divergent and convergent synthesis of polymannosylated dibranched antigenic peptide of the immunodominant epitope MBP(83–99)
|
Friligou, Irene
|
|
2013
|
21 |
21 |
p. 6718-6725
8 p.
|
artikel
|
| 23 |
Editorial board
|
|
|
2013
|
21 |
21 |
p. IFC-
1 p.
|
artikel
|
| 24 |
Evaluation of molecular model-based discovery of ecto-5′-nucleotidase inhibitors on the basis of X-ray structures
|
Furtmann, Norbert
|
|
2013
|
21 |
21 |
p. 6616-6622
7 p.
|
artikel
|
| 25 |
Further SAR studies on bicyclic basic merbarone analogues as potent antiproliferative agents
|
Spallarossa, Andrea
|
|
2013
|
21 |
21 |
p. 6328-6336
9 p.
|
artikel
|
| 26 |
α-Glucosidase-inhibitory iminosugars from the leaves of Suregada glomerulata
|
Yan, Ren-Yi
|
|
2013
|
21 |
21 |
p. 6796-6803
8 p.
|
artikel
|
| 27 |
Graphical contents list
|
|
|
2013
|
21 |
21 |
p. 6247-6263
17 p.
|
artikel
|
| 28 |
Hydroxyquinoline-derived compounds and analoguing of selective Mcl-1 inhibitors using a functional biomarker
|
Richard, David J.
|
|
2013
|
21 |
21 |
p. 6642-6649
8 p.
|
artikel
|
| 29 |
Identification, biological characterization and pharmacophoric analysis of a new potent and selective NK1 receptor antagonist clinical candidate
|
Di Fabio, Romano
|
|
2013
|
21 |
21 |
p. 6264-6273
10 p.
|
artikel
|
| 30 |
Identification of protein binding partners of ALK-5 kinase inhibitors
|
Ciayadi, Rudy
|
|
2013
|
21 |
21 |
p. 6496-6500
5 p.
|
artikel
|
| 31 |
Intermolecular interaction of voriconazole analogues with model membrane by DSC and NMR, and their antifungal activity using NMR based metabolic profiling
|
Kalamkar, Vaibhav
|
|
2013
|
21 |
21 |
p. 6753-6762
10 p.
|
artikel
|
| 32 |
99mTc-MORF oligomers specific for bacterial ribosomal RNA as potential specific infection imaging agents
|
Chen, Ling
|
|
2013
|
21 |
21 |
p. 6523-6530
8 p.
|
artikel
|
| 33 |
New derivatives of salicylamides: Preparation and antimicrobial activity against various bacterial species
|
Pauk, Karel
|
|
2013
|
21 |
21 |
p. 6574-6581
8 p.
|
artikel
|
| 34 |
New quaternary ammonium camphor derivatives and their antiviral activity, genotoxic effects and cytotoxicity
|
Sokolova, Anastasiya S.
|
|
2013
|
21 |
21 |
p. 6690-6698
9 p.
|
artikel
|
| 35 |
Novel BACE1 inhibitors with a non-acidic heterocycle at the P1′ position
|
Suzuki, Kenji
|
|
2013
|
21 |
21 |
p. 6665-6673
9 p.
|
artikel
|
| 36 |
Novel complex crystal structure of prolyl hydroxylase domain-containing protein 2 (PHD2): 2,8-Diazaspiro[4.5]decan-1-ones as potent, orally bioavailable PHD2 inhibitors
|
Deng, Guanghui
|
|
2013
|
21 |
21 |
p. 6349-6358
10 p.
|
artikel
|
| 37 |
Novel 3-nitro-1H-1,2,4-triazole-based piperazines and 2-amino-1,3-benzothiazoles as antichagasic agents
|
Papadopoulou, Maria V.
|
|
2013
|
21 |
21 |
p. 6600-6607
8 p.
|
artikel
|
| 38 |
Phenyl substituted 3-hydroxypyridin-2(1H)-ones: Inhibitors of influenza A endonuclease
|
Parhi, Ajit K.
|
|
2013
|
21 |
21 |
p. 6435-6446
12 p.
|
artikel
|
| 39 |
Quinazolino linked 4β-amidopodophyllotoxin conjugates regulate angiogenic pathway and control breast cancer cell proliferation
|
Kamal, Ahmed
|
|
2013
|
21 |
21 |
p. 6414-6426
13 p.
|
artikel
|
| 40 |
Radiochemical and radiobiological assessment of a pyridyl-S-cysteine functionalized bombesin derivative labeled with the 99mTc ( CO ) 3 + core
|
Bouziotis, Penelope
|
|
2013
|
21 |
21 |
p. 6699-6707
9 p.
|
artikel
|
| 41 |
Rv1268c protein peptide inhibiting Mycobacterium tuberculosis H37Rv entry to target cells
|
Ocampo, Marisol
|
|
2013
|
21 |
21 |
p. 6650-6656
7 p.
|
artikel
|
| 42 |
Selective inhibition of heme oxygenase-2 activity by analogs of 1-(4-chlorobenzyl)-2-(pyrrolidin-1-ylmethyl)-1H-benzimidazole (clemizole): Exploration of the effects of substituents at the N-1 position
|
Vlahakis, Jason Z.
|
|
2013
|
21 |
21 |
p. 6788-6795
8 p.
|
artikel
|
| 43 |
Structural study of the location of the phenyl tail of benzene sulfonamides and the effect on human carbonic anhydrase inhibition
|
Güzel-Akdemir, Özlen
|
|
2013
|
21 |
21 |
p. 6674-6680
7 p.
|
artikel
|
| 44 |
Structure–activity relationships of 2-aminothiazoles effective against Mycobacterium tuberculosis
|
Meissner, Anja
|
|
2013
|
21 |
21 |
p. 6385-6397
13 p.
|
artikel
|
| 45 |
Subcellular localization of proflavine derivative and induction of oxidative stress—In vitro studies
|
Ipóthová, Z.
|
|
2013
|
21 |
21 |
p. 6726-6731
6 p.
|
artikel
|
| 46 |
Synthesis and antioxidant activity of novel Mannich base of 1,3,4-oxadiazole derivatives possessing 1,4-benzodioxan
|
Ma, Liang
|
|
2013
|
21 |
21 |
p. 6763-6770
8 p.
|
artikel
|
| 47 |
Synthesis and antiprotozoal activity of dicationic 2,6-diphenylpyrazines and aza-analogues
|
Hu, Laixing
|
|
2013
|
21 |
21 |
p. 6732-6741
10 p.
|
artikel
|
| 48 |
Synthesis and anti-Trypanosoma cruzi activity of naphthoquinone-containing triazoles: Electrochemical studies on the effects of the quinoidal moiety
|
Diogo, Emilay B.T.
|
|
2013
|
21 |
21 |
p. 6337-6348
12 p.
|
artikel
|
| 49 |
Synthesis and anti-tumor activity of carbohydrate analogues of the tetrahydrofuran containing acetogenins
|
Bachan, Stewart
|
|
2013
|
21 |
21 |
p. 6554-6564
11 p.
|
artikel
|
| 50 |
Synthesis and biological evaluation of 2-amino-5-aryl-3-benzylthiopyridine scaffold based potent c-Met inhibitors
|
Zhang, Dengyou
|
|
2013
|
21 |
21 |
p. 6804-6820
17 p.
|
artikel
|
| 51 |
Synthesis and biological evaluation of indole-based, anti-cancer agents inspired by the vascular disrupting agent 2-(3′-hydroxy-4′-methoxyphenyl)-3-(3″,4″,5″-trimethoxybenzoyl)-6-methoxyindole (OXi8006)
|
MacDonough, Matthew T.
|
|
2013
|
21 |
21 |
p. 6831-6843
13 p.
|
artikel
|
| 52 |
Synthesis and biological evaluation of N-(2-fluorophenyl)-2β-deoxyfuconojirimycin acetamide as a potent inhibitor for α-l-fucosidases
|
Kato, Atsushi
|
|
2013
|
21 |
21 |
p. 6565-6573
9 p.
|
artikel
|
| 53 |
Synthesis and biological evaluation of novel acylhydrazone derivatives as potential antitumor agents
|
Congiu, Cenzo
|
|
2013
|
21 |
21 |
p. 6592-6599
8 p.
|
artikel
|
| 54 |
Synthesis and biological evaluation of novel C-aryl d-glucofuranosides as sodium-dependent glucose co-transporter 2 inhibitors
|
Lin, Tzung-Sheng
|
|
2013
|
21 |
21 |
p. 6282-6291
10 p.
|
artikel
|
| 55 |
Synthesis and enzymatic evaluation of phosphoramidon and its β anomer: Anomerization of α-l-rhamnose triacetate upon phosphitylation
|
Sun, Qi
|
|
2013
|
21 |
21 |
p. 6778-6787
10 p.
|
artikel
|
| 56 |
Synthesis and evaluation of novel azetidine analogs as potent inhibitors of vesicular [3H]dopamine uptake
|
Ding, Derong
|
|
2013
|
21 |
21 |
p. 6771-6777
7 p.
|
artikel
|
| 57 |
Synthesis and pharmacological evaluation of novel N-aryl-3,4-dihydro-1′H-spiro[chromene-2,4′-piperidine]-1′-carboxamides as TRPM8 antagonists
|
Chaudhari, Sachin S.
|
|
2013
|
21 |
21 |
p. 6542-6553
12 p.
|
artikel
|
| 58 |
Synthesis and structure–activity relationship of 2-phenyliminochromene derivatives as inhibitors for aldo–keto reductase (AKR) 1B10
|
Endo, Satoshi
|
|
2013
|
21 |
21 |
p. 6378-6384
7 p.
|
artikel
|
| 59 |
Synthesis and study of antiproliferative, antitopoisomerase II, DNA-intercalating and DNA-damaging activities of arylnaphthalimides
|
Quintana-Espinoza, Patricia
|
|
2013
|
21 |
21 |
p. 6484-6495
12 p.
|
artikel
|
| 60 |
Synthesis, DNA/protein binding and in vitro cytotoxic studies of new palladium metallothiosemicarbazones
|
Prabhakaran, R.
|
|
2013
|
21 |
21 |
p. 6742-6752
11 p.
|
artikel
|
| 61 |
Synthesis of amino-hydroxy-benzocycloheptenones as potent, selective, non-peptidic dinuclear zinc metalloaminopeptidase inhibitors
|
Al-Lakkis-Wehbe, Mira
|
|
2013
|
21 |
21 |
p. 6447-6455
9 p.
|
artikel
|
| 62 |
Synthesis of sterically encumbered 11β-aminoprogesterone derivatives and evaluation as 11β-hydroxysteroid dehydrogenase inhibitors and mineralocorticoid receptor antagonists
|
Pandya, Keyur
|
|
2013
|
21 |
21 |
p. 6274-6281
8 p.
|
artikel
|
| 63 |
Synthesis, structural characterization and cell death-inducing effect of novel palladium(II) and platinum(II) saccharinate complexes with 2-(hydroxymethyl)pyridine and 2-(2-hydroxyethyl)pyridine on cancer cells in vitro
|
Ari, Ferda
|
|
2013
|
21 |
21 |
p. 6427-6434
8 p.
|
artikel
|
| 64 |
The synthesis and anticancer activity of analogs of the indole phytoalexins brassinin, 1-methoxyspirobrassinol methyl ether and cyclobrassinin
|
Budovská, Mariana
|
|
2013
|
21 |
21 |
p. 6623-6633
11 p.
|
artikel
|
| 65 |
Towards new C6-rigid S-DABO HIV-1 reverse transcriptase inhibitors: Synthesis, biological investigation and molecular modeling studies
|
Wu, Hai-Qiu
|
|
2013
|
21 |
21 |
p. 6477-6483
7 p.
|
artikel
|
| 66 |
TRPV1 antagonist with high analgesic efficacy: 2-Thio pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides
|
Ha, Tae-Hwan
|
|
2013
|
21 |
21 |
p. 6657-6664
8 p.
|
artikel
|
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