| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Acyclic phosph(on)ate inhibitors of Plasmodium falciparum hypoxanthine-guanine-xanthine phosphoribosyltransferase
|
Clinch, Keith
|
|
2013
|
21 |
17 |
p. 5629-5646
18 p.
|
artikel
|
| 2 |
A 2,6,9-hetero-trisubstituted purine inhibitor exhibits potent biological effects against multiple myeloma cells
|
Shahani, Vijay M.
|
|
2013
|
21 |
17 |
p. 5618-5628
11 p.
|
artikel
|
| 3 |
Analogs of iso-azepinomycin as potential transition-state analog inhibitors of guanase: Synthesis, biochemical screening, and structure–activity correlations of various selectively substituted imidazo[4,5-e][1,4]diazepines
|
Tantravedi, Saritha
|
|
2013
|
21 |
17 |
p. 4893-4903
11 p.
|
artikel
|
| 4 |
Anti-inflammatory and anti-apoptotic effects of (RS )-glucoraphanin bioactivated with myrosinase in murine sub-acute and acute MPTP-induced Parkinson’s disease
|
Galuppo, Maria
|
|
2013
|
21 |
17 |
p. 5532-5547
16 p.
|
artikel
|
| 5 |
Antiproliferative activity on human prostate carcinoma cell lines of new peptidomimetics containing the spiroazepinoindolinone scaffold
|
Pellegrino, Sara
|
|
2013
|
21 |
17 |
p. 5470-5479
10 p.
|
artikel
|
| 6 |
Antiprotozoal activity of bicyclic diamines with a N-methylpiperazinyl group at the bridgehead atom
|
Faist, Johanna
|
|
2013
|
21 |
17 |
p. 4988-4996
9 p.
|
artikel
|
| 7 |
Antitumor properties of substituted (αE)-α-(1H-indol-3-ylmethylene)benzeneacetic acids or amides
|
Forte, Giuseppe
|
|
2013
|
21 |
17 |
p. 5233-5245
13 p.
|
artikel
|
| 8 |
3-Aryl-4-acyloxyethoxyfuran-2(5H)-ones as inhibitors of tyrosyl-tRNA synthetase: Synthesis, molecular docking and antibacterial evaluation
|
Wang, Xu-Dong
|
|
2013
|
21 |
17 |
p. 4914-4922
9 p.
|
artikel
|
| 9 |
4β-[4′-(1-(Aryl)ureido)benzamide]podophyllotoxins as DNA topoisomerase I and IIα inhibitors and apoptosis inducing agents
|
Kamal, Ahmed
|
|
2013
|
21 |
17 |
p. 5198-5208
11 p.
|
artikel
|
| 10 |
A sphingosine 1-phosphate receptor 2 selective allosteric agonist
|
Satsu, Hideo
|
|
2013
|
21 |
17 |
p. 5373-5382
10 p.
|
artikel
|
| 11 |
Autotaxin inhibition: Development and application of computational tools to identify site-selective lead compounds
|
Norman, Derek D.
|
|
2013
|
21 |
17 |
p. 5548-5560
13 p.
|
artikel
|
| 12 |
Biodistribution of 125I-labeled polymeric vaccine carriers after subcutaneous injection
|
Toita, Riki
|
|
2013
|
21 |
17 |
p. 5310-5315
6 p.
|
artikel
|
| 13 |
Carbonic anhydrase inhibitors: Synthesis and inhibition of the cytosolic mammalian carbonic anhydrase isoforms I, II and VII with benzene sulfonamides incorporating 4,5,6,7-tetrachlorophthalimide moiety
|
Sethi, Kalyan K.
|
|
2013
|
21 |
17 |
p. 5168-5174
7 p.
|
artikel
|
| 14 |
3-Carboxamido-5-aryl-isoxazoles as new CB2 agonists for the treatment of colitis
|
Tourteau, Aurélien
|
|
2013
|
21 |
17 |
p. 5383-5394
12 p.
|
artikel
|
| 15 |
Catalytic asymmetric total synthesis of (S)-(−)-zearalenone, a novel lipoxygenase inhibitor
|
Baggelaar, Marc P.
|
|
2013
|
21 |
17 |
p. 5271-5274
4 p.
|
artikel
|
| 16 |
Cembrane diterpenoids from the soft coral Sarcophyton trocheliophorum Marenzeller as a new class of PTP1B inhibitors
|
Liang, Lin-Fu
|
|
2013
|
21 |
17 |
p. 5076-5080
5 p.
|
artikel
|
| 17 |
C-Glucosides with heteroaryl thiophene as novel sodium-dependent glucose cotransporter 2 inhibitors
|
Koga, Yuichi
|
|
2013
|
21 |
17 |
p. 5561-5572
12 p.
|
artikel
|
| 18 |
Corrigendum to “Integrated structure-based activity prediction model of benzothiadiazines on various genotypes of HCV NS5b polymerase (1a, 1b and 4) and its application in the discovery of new derivatives” [Bioorg. Med. Chem. 20(7) (2012) 2455–2478]
|
Ismail, Mohamed A.H.
|
|
2013
|
21 |
17 |
p. 5647-
1 p.
|
artikel
|
| 19 |
Corrigendum to “Nucleic acid changes during photodynamic inactivation of bacteria by cationic porphyrins” [Bioorg. Med. Chem. 21 (2013) 4311–4318]
|
Alves, Eliana
|
|
2013
|
21 |
17 |
p. 5648-
1 p.
|
artikel
|
| 20 |
Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: Identification of an efficient lead for potent inhibitors of GABA transports
|
Nakada, Kazuaki
|
|
2013
|
21 |
17 |
p. 4938-4950
13 p.
|
artikel
|
| 21 |
Defining the key pharmacophore elements of PF-04620110: Discovery of a potent, orally-active, neutral DGAT-1 inhibitor
|
Dow, Robert L.
|
|
2013
|
21 |
17 |
p. 5081-5097
17 p.
|
artikel
|
| 22 |
Design and synthesis of 6,7-methylenedioxy-4-substituted phenylquinolin-2(1H)-one derivatives as novel anticancer agents that induce apoptosis with cell cycle arrest at G2/M phase
|
Chen, Yi-Fong
|
|
2013
|
21 |
17 |
p. 5064-5075
12 p.
|
artikel
|
| 23 |
Design and synthesis of novel 1,25-dihydroxyvitamin D3 analogues having a spiro-oxetane fused at the C2 position in the A-ring
|
Fujishima, Toshie
|
|
2013
|
21 |
17 |
p. 5209-5217
9 p.
|
artikel
|
| 24 |
Design and synthesis of novel series of 5-HT6 receptor ligands having indole, a central aromatic core and 1-amino-4 methyl piperazine as a positive ionizable group
|
Hayat, Faisal
|
|
2013
|
21 |
17 |
p. 5573-5582
10 p.
|
artikel
|
| 25 |
Design, synthesis and in vitro evaluation against human cancer cells of 5-methyl-5-styryl-2,5-dihydrofuran-2-ones, a new series of goniothalamin analogues
|
Bruder, Marjorie
|
|
2013
|
21 |
17 |
p. 5107-5117
11 p.
|
artikel
|
| 26 |
Design, synthesis and pharmacological evaluation of (E)-3,4-dihydroxy styryl sulfonamides derivatives as multifunctional neuroprotective agents against oxidative and inflammatory injury
|
Ning, Xianling
|
|
2013
|
21 |
17 |
p. 5589-5597
9 p.
|
artikel
|
| 27 |
Design, synthesis and structure–activity relationships of some novel, highly potent anti-invasive (E)- and (Z)-stilbenes
|
Roman, Bart I.
|
|
2013
|
21 |
17 |
p. 5054-5063
10 p.
|
artikel
|
| 28 |
Discovery and optimization of novel 4-phenoxy-6,7-disubstituted quinolines possessing semicarbazones as c-Met kinase inhibitors
|
Qi, Baohui
|
|
2013
|
21 |
17 |
p. 5246-5260
15 p.
|
artikel
|
| 29 |
Discovery of 2-methyl-1-{1-[(5-methyl-1H-indol-2-yl)carbonyl]piperidin-4-yl}propan-2-ol: A novel, potent and selective type 5 17β-hydroxysteroid dehydrogenase inhibitor
|
Watanabe, Kazushi
|
|
2013
|
21 |
17 |
p. 5261-5270
10 p.
|
artikel
|
| 30 |
Discovery of two new inhibitors of Botrytis cinerea chitin synthase by a chemical library screening
|
Magellan, Hervé
|
|
2013
|
21 |
17 |
p. 4997-5003
7 p.
|
artikel
|
| 31 |
Editorial board
|
|
|
2013
|
21 |
17 |
p. IFC-
1 p.
|
artikel
|
| 32 |
Effect of ring-constrained phenylpropyloxyethylamines on sigma receptors
|
Stavitskaya, Lidiya
|
|
2013
|
21 |
17 |
p. 4923-4927
5 p.
|
artikel
|
| 33 |
Effect of single pyrrole replacement with β-alanine on DNA binding affinity and sequence specificity of hairpin pyrrole/imidazole polyamides targeting 5′-GCGC-3′
|
Han, Yong-Woon
|
|
2013
|
21 |
17 |
p. 5436-5441
6 p.
|
artikel
|
| 34 |
Evaluation of novel aryloxyalkyl derivatives of imidazole and 1,2,4-triazole as heme oxygenase-1 (HO-1) inhibitors and their antitumor properties
|
Salerno, Loredana
|
|
2013
|
21 |
17 |
p. 5145-5153
9 p.
|
artikel
|
| 35 |
Exploring pyrimidine-substituted curcumin analogues: Design, synthesis and effects on EGFR signaling
|
Qiu, Peiju
|
|
2013
|
21 |
17 |
p. 5012-5020
9 p.
|
artikel
|
| 36 |
Fluorescent probes for investigation of isoprenoid configuration and size discrimination by bactoprenol-utilizing enzymes
|
Mostafavi, Anahita Z.
|
|
2013
|
21 |
17 |
p. 5428-5435
8 p.
|
artikel
|
| 37 |
Fluorescent rhodanine-3-acetic acids visualize neurofibrillary tangles in Alzheimer’s disease brains
|
Anumala, Upendra Rao
|
|
2013
|
21 |
17 |
p. 5139-5144
6 p.
|
artikel
|
| 38 |
Functionalized hydroxyethylamine based peptide nanostructures as potential inhibitors of falcipain-3, an essential proteases of Plasmodium falciparum
|
Rathi, Brijesh
|
|
2013
|
21 |
17 |
p. 5503-5509
7 p.
|
artikel
|
| 39 |
Gene suppression via U1 small nuclear RNA interference (U1i) machinery using oligonucleotides containing 2′-modified-4′-thionucleosides
|
Kikuchi, Yusaku
|
|
2013
|
21 |
17 |
p. 5292-5296
5 p.
|
artikel
|
| 40 |
Graphical contents list
|
|
|
2013
|
21 |
17 |
p. 4853-4873
21 p.
|
artikel
|
| 41 |
1-Hydroxypyrazole as a bioisostere of the acetic acid moiety in a series of aldose reductase inhibitors
|
Papastavrou, Nikolaos
|
|
2013
|
21 |
17 |
p. 4951-4957
7 p.
|
artikel
|
| 42 |
Improved synthesis of 17β-hydroxy-16α-iodo-wortmannin, 17β-hydroxy-16α-iodoPX866, and the [131I] analogue as useful PET tracers for PI3-kinase
|
Sun, Duoli
|
|
2013
|
21 |
17 |
p. 5182-5187
6 p.
|
artikel
|
| 43 |
Inhibition of Mycobacterium tuberculosis strains H37Rv and MDR MS-115 by a new set of C5 modified pyrimidine nucleosides
|
Shmalenyuk, Eduard R.
|
|
2013
|
21 |
17 |
p. 4874-4884
11 p.
|
artikel
|
| 44 |
Inhibition of tumor-associated human carbonic anhydrase isozymes IX and XII by a new class of substituted-phenylacetamido aromatic sulfonamides
|
Akdemir, Atilla
|
|
2013
|
21 |
17 |
p. 5228-5232
5 p.
|
artikel
|
| 45 |
In search of potent and selective inhibitors of neuronal nitric oxide synthase with more simple structures
|
Jing, Qing
|
|
2013
|
21 |
17 |
p. 5323-5331
9 p.
|
artikel
|
| 46 |
Investigations on synthesis and structure elucidation of novel [1,2,4]triazolo[1,2-a]pyridazine-1-thiones and their inhibitory activity against inducible nitric oxide synthase
|
Schulz, Ulrike
|
|
2013
|
21 |
17 |
p. 5518-5531
14 p.
|
artikel
|
| 47 |
Isoswinholide B and swinholide K, potently cytotoxic dimeric macrolides from Theonella swinhoei
|
Sinisi, Annamaria
|
|
2013
|
21 |
17 |
p. 5332-5338
7 p.
|
artikel
|
| 48 |
Lipophilic derivatives of natural chlorins: Synthesis, mixed micelles with phospholipids, and uptake by cultured cells
|
Ponomarev, Gelii V.
|
|
2013
|
21 |
17 |
p. 5420-5427
8 p.
|
artikel
|
| 49 |
Liver-targeting of primaquine-(poly-γ-glutamic acid) and its degradation in rat hepatocytes
|
Tomiya, Noboru
|
|
2013
|
21 |
17 |
p. 5275-5281
7 p.
|
artikel
|
| 50 |
Macamides and their synthetic analogs: Evaluation of in vitro FAAH inhibition
|
Wu, Hui
|
|
2013
|
21 |
17 |
p. 5188-5197
10 p.
|
artikel
|
| 51 |
Modular construction of quaternary hemiaminal-based inhibitor candidates and their in cellulo assessment with HIV-1 protease
|
Gros, Guillaume
|
|
2013
|
21 |
17 |
p. 5407-5413
7 p.
|
artikel
|
| 52 |
5-Nitro-2-furfuriliden derivatives as potential anti-Trypanosoma cruzi agents: Design, synthesis, bioactivity evaluation, cytotoxicity and exploratory data analysis
|
Palace-Berl, Fanny
|
|
2013
|
21 |
17 |
p. 5395-5406
12 p.
|
artikel
|
| 53 |
Novel N-hydroxyfurylacrylamide-based histone deacetylase (HDAC) inhibitors with branched CAP group (Part 2)
|
Feng, Taotao
|
|
2013
|
21 |
17 |
p. 5339-5354
16 p.
|
artikel
|
| 54 |
One-pot tandem Hurtley–retro-Claisen–cyclisation reactions in the synthesis of 3-substituted analogues of 5-aminoisoquinolin-1-one (5-AIQ), a water-soluble inhibitor of PARPs
|
Woon, Esther C.Y.
|
|
2013
|
21 |
17 |
p. 5218-5227
10 p.
|
artikel
|
| 55 |
Oxazolopyridines and thiazolopyridines as monoamine oxidase B inhibitors for the treatment of Parkinson’s disease
|
Park, Hye Ri
|
|
2013
|
21 |
17 |
p. 5480-5487
8 p.
|
artikel
|
| 56 |
Quantification of free ligand conformational preferences by NMR and their relationship to the bioactive conformation
|
Blundell, Charles D.
|
|
2013
|
21 |
17 |
p. 4976-4987
12 p.
|
artikel
|
| 57 |
Rapid modifications of N-substitution in iminosugars: Development of new β-glucocerebrosidase inhibitors and pharmacological chaperones for Gaucher disease
|
Cheng, Wei-Chieh
|
|
2013
|
21 |
17 |
p. 5021-5028
8 p.
|
artikel
|
| 58 |
Solid phase synthesis of Smac/DIABLO-derived peptides using a ‘Safety-Catch’ resin: Identification of potent XIAP BIR3 antagonists
|
Elsawy, Mohamed A.
|
|
2013
|
21 |
17 |
p. 5004-5011
8 p.
|
artikel
|
| 59 |
Solid-phase synthesis of 5′-triphosphate 2′-5′-oligoadenylates analogs with 3′-O-biolabile groups and their evaluation as RNase L activators and antiviral drugs
|
Thillier, Yann
|
|
2013
|
21 |
17 |
p. 5461-5469
9 p.
|
artikel
|
| 60 |
Structure–activity relationships for ketamine esters as short-acting anaesthetics
|
Jose, Jiney
|
|
2013
|
21 |
17 |
p. 5098-5106
9 p.
|
artikel
|
| 61 |
Structure–activity relationship studies of Niemann-Pick type C1-like 1 (NPC1L1) ligands identified by screening assay monitoring pharmacological chaperone effect
|
Karaki, Fumika
|
|
2013
|
21 |
17 |
p. 5297-5309
13 p.
|
artikel
|
| 62 |
2-Substituted 4-hydroxybutanamides as potential inhibitors of γ-aminobutyric acid transporters mGAT1–mGAT4: Synthesis and biological evaluation
|
Kowalczyk, Paula
|
|
2013
|
21 |
17 |
p. 5154-5167
14 p.
|
artikel
|
| 63 |
5-Substituted-(1,2,3-triazol-4-yl)thiophene-2-sulfonamides strongly inhibit human carbonic anhydrases I, II, IX and XII: Solution and X-ray crystallographic studies
|
Leitans, Janis
|
|
2013
|
21 |
17 |
p. 5130-5138
9 p.
|
artikel
|
| 64 |
Synthesis and bioevaluation of some new isoniazid derivatives
|
Matei, Lilia
|
|
2013
|
21 |
17 |
p. 5355-5361
7 p.
|
artikel
|
| 65 |
Synthesis and biological activity of benzo-fused 7-deazaadenosine analogues. 5- and 6-substituted 4-amino- or 4-alkylpyrimido[4,5-b]indole ribonucleosides
|
Tichý, Michal
|
|
2013
|
21 |
17 |
p. 5362-5372
11 p.
|
artikel
|
| 66 |
Synthesis and biological evaluation of novobiocin analogues as potential heat shock protein 90 inhibitors
|
Gunaherath, G.M. Kamal B.
|
|
2013
|
21 |
17 |
p. 5118-5129
12 p.
|
artikel
|
| 67 |
Synthesis and biological evaluation of potential threonine synthase inhibitors: Rhizocticin A and Plumbemycin A
|
Gahungu, Mathias
|
|
2013
|
21 |
17 |
p. 4958-4967
10 p.
|
artikel
|
| 68 |
Synthesis and Characterization of Time-resolved Fluorescence Probes for Evaluation of Competitive Binding to Melanocortin Receptors
|
Alleti, Ramesh
|
|
2013
|
21 |
17 |
p. 5029-5038
10 p.
|
artikel
|
| 69 |
Synthesis and evaluation of 1-[2-(4-[11C]methoxyphenyl)phenyl]piperazine for imaging of the serotonin 5-HT7 receptor in the rat brain
|
Shimoda, Yoko
|
|
2013
|
21 |
17 |
p. 5316-5322
7 p.
|
artikel
|
| 70 |
Synthesis and α-glucosidase inhibitory activity evaluation of N-substituted aminomethyl-β-d-glucopyranosides
|
Bian, Xiaoli
|
|
2013
|
21 |
17 |
p. 5442-5450
9 p.
|
artikel
|
| 71 |
Synthesis and initial in vitro biological evaluation of two new zinc-chelating compounds: Comparison with TPEN and PAC-1
|
Åstrand, O. Alexander H.
|
|
2013
|
21 |
17 |
p. 5175-5181
7 p.
|
artikel
|
| 72 |
Synthesis and insecticidal activities of 2,3-dihydroquinazolin-4(1H)-one derivatives targeting calcium channel
|
Zhou, Yunyun
|
|
2013
|
21 |
17 |
p. 4968-4975
8 p.
|
artikel
|
| 73 |
Synthesis and in vitro cytostatic activity of 1,2- and 1,3-diacylglycerophosphates of clofarabine
|
Tsybulskaya, Ilona
|
|
2013
|
21 |
17 |
p. 5414-5419
6 p.
|
artikel
|
| 74 |
Synthesis and in vivo evaluation of [18F]2-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)-4-methyl-1,2,4-triazine-3,5(2H,4H)-dione ([18F]FECUMI-101) as an imaging probe for 5-HT1A receptor agonist in nonhuman primates
|
Majo, Vattoly J.
|
|
2013
|
21 |
17 |
p. 5598-5604
7 p.
|
artikel
|
| 75 |
Synthesis and tubulin-binding properties of non-symmetrical click C5-curcuminoids
|
Caldarelli, Antonio
|
|
2013
|
21 |
17 |
p. 5510-5517
8 p.
|
artikel
|
| 76 |
Synthesis, biological activity and molecular modeling studies on 1H-benzimidazole derivatives as acetylcholinesterase inhibitors
|
Alpan, Ayşe Selcen
|
|
2013
|
21 |
17 |
p. 4928-4937
10 p.
|
artikel
|
| 77 |
Synthesis, evaluation and molecular dynamics study of some new 4-aminopyridine semicarbazones as an antiamnesic and cognition enhancing agents
|
Sinha, Saurabh K.
|
|
2013
|
21 |
17 |
p. 5451-5460
10 p.
|
artikel
|
| 78 |
Synthesis of novel isothiazolopyridines and their in vitro evaluation against Mycobacterium and Propionibacterium acnes
|
Malinka, Wiesław
|
|
2013
|
21 |
17 |
p. 5282-5291
10 p.
|
artikel
|
| 79 |
Synthesis of novel psoralen analogues and their in vitro antitumor activity
|
Francisco, Carla S.
|
|
2013
|
21 |
17 |
p. 5047-5053
7 p.
|
artikel
|
| 80 |
Synthesis of polysubstituted benzofuran derivatives as novel inhibitors of parasitic growth
|
Thévenin, Marion
|
|
2013
|
21 |
17 |
p. 4885-4892
8 p.
|
artikel
|
| 81 |
Synthesis, pH-dependent, and plasma stability of meropenem prodrugs for potential use against drug-resistant tuberculosis
|
Teitelbaum, Aaron M.
|
|
2013
|
21 |
17 |
p. 5605-5617
13 p.
|
artikel
|
| 82 |
Synthetic studies of centromere-associated protein-E (CENP-E) inhibitors: 1.Exploration of fused bicyclic core scaffolds using electrostatic potential map
|
Hirayama, Takaharu
|
|
2013
|
21 |
17 |
p. 5488-5502
15 p.
|
artikel
|
| 83 |
Tetrazole-based deoxyamodiaquines: Synthesis, ADME/PK profiling and pharmacological evaluation as potential antimalarial agents
|
Tukulula, Matshawandile
|
|
2013
|
21 |
17 |
p. 4904-4913
10 p.
|
artikel
|
| 84 |
Tocopheramines and tocotrienamines as antioxidants: ESR spectroscopy, rapid kinetics and DFT calculations
|
Bamonti, Luca
|
|
2013
|
21 |
17 |
p. 5039-5046
8 p.
|
artikel
|
| 85 |
Triplex-forming ability of oligonucleotides containing 1-aryl-1,2,3-triazole nucleobases linked via a two atom-length spacer
|
Hari, Yoshiyuki
|
|
2013
|
21 |
17 |
p. 5583-5588
6 p.
|
artikel
|
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