| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
(+)-Altholactone exhibits broad spectrum immune modulating activity by inhibiting the activation of pro-inflammatory cytokines in RAW 264.7 cell lines
|
Johnson, Tyler A.
|
|
2013
|
21 |
14 |
p. 4358-4364
7 p.
|
artikel
|
| 2 |
Antagonism of L-type Ca2+ channels CaV1.3 and CaV1.2 by 1,4-dihydropyrimidines and 4H-pyrans as dihydropyridine mimics
|
Kang, Soosung
|
|
2013
|
21 |
14 |
p. 4365-4373
9 p.
|
artikel
|
| 3 |
Anti-leishmanial evaluation of C2-aryl quinolines: Mechanistic insight on bioenergetics and sterol biosynthetic pathway of Leishmania braziliensis
|
Bompart, Daznia
|
|
2013
|
21 |
14 |
p. 4426-4431
6 p.
|
artikel
|
| 4 |
Australian marine sponge alkaloids as a new class of glycine-gated chloride channel receptor modulator
|
Balansa, Walter
|
|
2013
|
21 |
14 |
p. 4420-4425
6 p.
|
artikel
|
| 5 |
Benzimidazole-2-one: A novel anchoring principle for antagonizing p53-Mdm2
|
Wang, Wei
|
|
2013
|
21 |
14 |
p. 3982-3995
14 p.
|
artikel
|
| 6 |
Bioorganic & Medicinal Chemistry Reviews and Perspectives
|
|
|
2013
|
21 |
14 |
p. I-III
nvt p.
|
artikel
|
| 7 |
Brassinolide-2,3-acetonide: A brassinolide-induced rice lamina joint inclination antagonist
|
Muto, Takuya
|
|
2013
|
21 |
14 |
p. 4413-4419
7 p.
|
artikel
|
| 8 |
C3′-endo-puckered pyrrolidine containing PNA has favorable geometry for RNA binding: Novel ethano locked PNA (ethano-PNA)
|
Banerjee, Anjan
|
|
2013
|
21 |
14 |
p. 4092-4101
10 p.
|
artikel
|
| 9 |
Chromenylchalcones showing cytotoxicity on human colon cancer cell lines and in silico docking with aurora kinases
|
Shin, Soon Young
|
|
2013
|
21 |
14 |
p. 4250-4258
9 p.
|
artikel
|
| 10 |
Design, synthesis and biological activity evaluation of desloratadine analogues as H1 receptor antagonists
|
Lin, Yan
|
|
2013
|
21 |
14 |
p. 4178-4185
8 p.
|
artikel
|
| 11 |
Design, synthesis and biological evaluation of enzymatically cleavable NSAIDs prodrugs derived from self-immolative dendritic scaffolds for the treatment of inflammatory diseases
|
Wei, Jinbao
|
|
2013
|
21 |
14 |
p. 4192-4200
9 p.
|
artikel
|
| 12 |
Design, synthesis and evaluation of retinoids with novel bulky hydrophobic partial structures
|
Amano, Yohei
|
|
2013
|
21 |
14 |
p. 4342-4350
9 p.
|
artikel
|
| 13 |
Development and characterization of a promising fluorine-18 labelled radiopharmaceutical for in vivo imaging of fatty acid amide hydrolase
|
Sadovski, Oleg
|
|
2013
|
21 |
14 |
p. 4351-4357
7 p.
|
artikel
|
| 14 |
Development of time resolved fluorescence resonance energy transfer-based assay for FXR antagonist discovery
|
Yu, Donna D.
|
|
2013
|
21 |
14 |
p. 4266-4278
13 p.
|
artikel
|
| 15 |
1,4-Diaryl-substituted triazoles as cyclooxygenase-2 inhibitors: Synthesis, biological evaluation and molecular modeling studies
|
Kaur, Jatinder
|
|
2013
|
21 |
14 |
p. 4288-4295
8 p.
|
artikel
|
| 16 |
Direct targeting of β-catenin: Inhibition of protein–protein interactions for the inactivation of Wnt signaling
|
Hahne, Gernot
|
|
2013
|
21 |
14 |
p. 4020-4026
7 p.
|
artikel
|
| 17 |
Discovery of novel series of 6-benzyl substituted 4-aminocarbonyl-1,4-diazepane-2,5-diones as human chymase inhibitors using structure-based drug design
|
Tanaka, Taisaku
|
|
2013
|
21 |
14 |
p. 4233-4249
17 p.
|
artikel
|
| 18 |
Editorial board
|
|
|
2013
|
21 |
14 |
p. IFC-
1 p.
|
artikel
|
| 19 |
Effects on polo-like kinase 1 polo-box domain binding affinities of peptides incurred by structural variation at the phosphoamino acid position
|
Qian, Wenjian
|
|
2013
|
21 |
14 |
p. 3996-4003
8 p.
|
artikel
|
| 20 |
Exploring DOXP-reductoisomerase binding limits using phosphonated N-aryl and N-heteroarylcarboxamides as DXR inhibitors
|
Bodill, Taryn
|
|
2013
|
21 |
14 |
p. 4332-4341
10 p.
|
artikel
|
| 21 |
Functional consequences of retro-inverso isomerization of a miniature protein inhibitor of the p53–MDM2 interaction
|
Li, Chong
|
|
2013
|
21 |
14 |
p. 4045-4050
6 p.
|
artikel
|
| 22 |
Graphical contents list
|
|
|
2013
|
21 |
14 |
p. 3967-3980
14 p.
|
artikel
|
| 23 |
Identification of 1,6-dihydropyrazolo[4,3-c]carbazoles and 3,6-dihydropyrazolo[3,4-c]carbazoles as new Pim kinase inhibitors
|
Suchaud, Virginie
|
|
2013
|
21 |
14 |
p. 4102-4111
10 p.
|
artikel
|
| 24 |
Inhibition and stabilization of protein–protein interactions
|
Ottmann, Christian
|
|
2013
|
21 |
14 |
p. 3981-
1 p.
|
artikel
|
| 25 |
Inhibition of HIV-1 integrase dimerization and activity with crosslinked interfacial peptides
|
Zhao, Lei
|
|
2013
|
21 |
14 |
p. 4041-4044
4 p.
|
artikel
|
| 26 |
Large conductance Ca2+-activated K+ channel (BKCa) activating properties of a series of novel N-arylbenzamides: Channel subunit dependent effects
|
Kirby, R.W.
|
|
2013
|
21 |
14 |
p. 4186-4191
6 p.
|
artikel
|
| 27 |
Long-chain triazolyl acids as inhibitors of osteoclastogenesis
|
Marshall, Andrew J.
|
|
2013
|
21 |
14 |
p. 4112-4119
8 p.
|
artikel
|
| 28 |
6′-Methyl-5′-homoaristeromycin: A structural variation of the anti-orthopox virus candidate 5′-homoaristeromycin
|
Yang, Minmin
|
|
2013
|
21 |
14 |
p. 4374-4377
4 p.
|
artikel
|
| 29 |
Microwave assisted solid phase synthesis of highly functionalized N-alkylated oligobenzamide α-helix mimetics
|
Long, Kérya
|
|
2013
|
21 |
14 |
p. 4034-4040
7 p.
|
artikel
|
| 30 |
Novel artemisinin derivatives with potential usefulness against liver/colon cancer and viral hepatitis
|
Blazquez, Alba G.
|
|
2013
|
21 |
14 |
p. 4432-4441
10 p.
|
artikel
|
| 31 |
Novel inhibitors of a Grb2 SH3C domain interaction identified by a virtual screen
|
Simister, Philip C.
|
|
2013
|
21 |
14 |
p. 4027-4033
7 p.
|
artikel
|
| 32 |
Novel synthetic acridine derivatives as potent DNA-binding and apoptosis-inducing antitumor agents
|
Lang, Xuliang
|
|
2013
|
21 |
14 |
p. 4170-4177
8 p.
|
artikel
|
| 33 |
Nucleic acid changes during photodynamic inactivation of bacteria by cationic porphyrins
|
Alves, Eliana
|
|
2013
|
21 |
14 |
p. 4311-4318
8 p.
|
artikel
|
| 34 |
Peptidomimetic modification improves cell permeation of bivalent farnesyltransferase inhibitors
|
Machida, Shinnosuke
|
|
2013
|
21 |
14 |
p. 4004-4010
7 p.
|
artikel
|
| 35 |
Plucking the high hanging fruit: A systematic approach for targeting protein–protein interactions
|
Raj, Monika
|
|
2013
|
21 |
14 |
p. 4051-4057
7 p.
|
artikel
|
| 36 |
Potent suppression of c-di-GMP synthesis via I-site allosteric inhibition of diguanylate cyclases with 2′-F-c-di-GMP
|
Zhou, Jie
|
|
2013
|
21 |
14 |
p. 4396-4404
9 p.
|
artikel
|
| 37 |
Pt(II) complexes with (N,N′) or (C,N,E)− (E=N,S) ligands: Cytotoxic studies, effect on DNA tertiary structure and structure–activity relationships
|
Albert, Joan
|
|
2013
|
21 |
14 |
p. 4210-4217
8 p.
|
artikel
|
| 38 |
Recent syntheses of PI3K/Akt/mTOR signaling pathway inhibitors
|
Welker, Mark E.
|
|
2013
|
21 |
14 |
p. 4063-4091
29 p.
|
artikel
|
| 39 |
Small-molecule modulators of 14-3-3 protein–protein interactions
|
Ottmann, Christian
|
|
2013
|
21 |
14 |
p. 4058-4062
5 p.
|
artikel
|
| 40 |
Small molecules inhibit the interaction of Nrf2 and the Keap1 Kelch domain through a non-covalent mechanism
|
Marcotte, Douglas
|
|
2013
|
21 |
14 |
p. 4011-4019
9 p.
|
artikel
|
| 41 |
20(S)-Protopanaxadiol (PPD) analogues chemosensitize multidrug-resistant cancer cells to clinical anticancer drugs
|
Liu, Junhua
|
|
2013
|
21 |
14 |
p. 4279-4287
9 p.
|
artikel
|
| 42 |
1-substituted apomorphines as potent dopamine agonists
|
Reinart-Okugbeni, Reet
|
|
2013
|
21 |
14 |
p. 4143-4150
8 p.
|
artikel
|
| 43 |
Synthesis and antibacterial activity of novel phosphonium salts on the basis of pyridoxine
|
Pugachev, Mikhail V.
|
|
2013
|
21 |
14 |
p. 4388-4395
8 p.
|
artikel
|
| 44 |
Synthesis and anti-HCMV activity of 1-[ω-(phenoxy)alkyl]uracil derivatives and analogues thereof
|
Novikov, Mikhail S.
|
|
2013
|
21 |
14 |
p. 4151-4157
7 p.
|
artikel
|
| 45 |
Synthesis and bioactive evaluation of novel hybrids of metronidazole and berberine as new type of antimicrobial agents and their transportation behavior by human serum albumin
|
Zhang, Ling
|
|
2013
|
21 |
14 |
p. 4158-4169
12 p.
|
artikel
|
| 46 |
Synthesis and biological evaluation of a targeted DNA-binding transcriptional activator with HDAC8 inhibitory activity
|
Saha, Abhijit
|
|
2013
|
21 |
14 |
p. 4201-4209
9 p.
|
artikel
|
| 47 |
Synthesis and biological evaluation of 4,5-dihydro-1H-pyrazole derivatives as potential nNOS/iNOS selective inhibitors. Part 2: Influence of diverse substituents in both the phenyl moiety and the acyl group
|
Carrión, M. Dora
|
|
2013
|
21 |
14 |
p. 4132-4142
11 p.
|
artikel
|
| 48 |
Synthesis and biological evaluation of novel tamoxifen analogues
|
Christodoulou, Michael S.
|
|
2013
|
21 |
14 |
p. 4120-4131
12 p.
|
artikel
|
| 49 |
Synthesis and evaluation of novel orally active p53–MDM2 interaction inhibitors
|
Miyazaki, Masaki
|
|
2013
|
21 |
14 |
p. 4319-4331
13 p.
|
artikel
|
| 50 |
Synthesis and functional analysis of deferriferrichrysin derivatives: Application to colorimetric pH indicators
|
Kobayashi, Yuka
|
|
2013
|
21 |
14 |
p. 4296-4300
5 p.
|
artikel
|
| 51 |
Synthesis and in vitro evaluation of glycosyl derivatives of luteinizing hormone-releasing hormone (LHRH)
|
Moradi, Shayli Varasteh
|
|
2013
|
21 |
14 |
p. 4259-4265
7 p.
|
artikel
|
| 52 |
Synthesis and preliminary biological evaluation of a compound library of triazolylcyclitols
|
Carrau, Gonzalo
|
|
2013
|
21 |
14 |
p. 4225-4232
8 p.
|
artikel
|
| 53 |
Synthesis and properties of thymidines with six-membered amide bridge
|
Hari, Yoshiyuki
|
|
2013
|
21 |
14 |
p. 4405-4412
8 p.
|
artikel
|
| 54 |
Synthesis, biological evaluation and molecular modeling of substituted 2-aminobenzimidazoles as novel inhibitors of acetylcholinesterase and butyrylcholinesterase
|
Zhu, Jinmei
|
|
2013
|
21 |
14 |
p. 4218-4224
7 p.
|
artikel
|
| 55 |
Synthesis of organic nitrates of luteolin as a novel class of potent aldose reductase inhibitors
|
Wang, Qi-Qin
|
|
2013
|
21 |
14 |
p. 4301-4310
10 p.
|
artikel
|
| 56 |
The synthesis of neurotensin antagonist SR 48692 for prostate cancer research
|
Baxendale, I.R.
|
|
2013
|
21 |
14 |
p. 4378-4387
10 p.
|
artikel
|
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