| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
An altered zinc-binding site confers resistance to a covalent inactivator of New Delhi metallo-beta-lactamase-1 (NDM-1) discovered by high-throughput screening
|
Thomas, Pei W.
|
|
2013
|
21 |
11 |
p. 3138-3146
9 p.
|
artikel
|
| 2 |
Anti-inflammatory secondary metabolites from the leaves of Rosa laevigata
|
Yan, Min
|
|
2013
|
21 |
11 |
p. 3290-3297
8 p.
|
artikel
|
| 3 |
Antiproliferative homoscalarane sesterterpenes from two Madagascan sponges
|
Harinantenaina, Liva
|
|
2013
|
21 |
11 |
p. 2912-2917
6 p.
|
artikel
|
| 4 |
Benzimidazole-based antibacterial agents against Francisella tularensis
|
Kumar, Kunal
|
|
2013
|
21 |
11 |
p. 3318-3326
9 p.
|
artikel
|
| 5 |
Benzofuran-, benzothiophene-, indazole- and benzisoxazole-quinones: Excellent substrates for NAD(P)H:quinone oxidoreductase 1
|
Newsome, Jeffery J.
|
|
2013
|
21 |
11 |
p. 2999-3009
11 p.
|
artikel
|
| 6 |
Bioorganic & Medicinal Chemistry Reviews and Perspectives
|
|
|
2013
|
21 |
11 |
p. I-III
nvt p.
|
artikel
|
| 7 |
Design and syntheses of novel N′-((4-oxo-4H-chromen-3-yl)methylene)benzohydrazide as inhibitors of cyanobacterial fructose-1,6-/sedoheptulose-1,7-bisphosphatase
|
Tu, Qi-Dong
|
|
2013
|
21 |
11 |
p. 2826-2831
6 p.
|
artikel
|
| 8 |
Design and synthesis of 1-(benzothiazol-5-yl)-1H-1,2,4-triazol-5-ones as protoporphyrinogen oxidase inhibitors
|
Yang, Zuo
|
|
2013
|
21 |
11 |
p. 3245-3255
11 p.
|
artikel
|
| 9 |
Design and synthesis of l- and d-phenylalanine derived rhodanines with novel C5-arylidenes as inhibitors of HCV NS5B polymerase
|
Patel, Bhargav A.
|
|
2013
|
21 |
11 |
p. 3262-3271
10 p.
|
artikel
|
| 10 |
Design and synthesis of novel opioid ligands with an azabicyclo[2.2.2]octane skeleton having a 7-amide side chain and their pharmacologies
|
Watanabe, Yoshikazu
|
|
2013
|
21 |
11 |
p. 3032-3050
19 p.
|
artikel
|
| 11 |
Design, synthesis and antimicrobial activities evaluation of Schiff base derived from secnidazole derivatives as potential FabH inhibitors
|
Li, Yao
|
|
2013
|
21 |
11 |
p. 3120-3126
7 p.
|
artikel
|
| 12 |
Design, synthesis and biological evaluation of novel pyrimidine, 3-cyanopyridine and m-amino-N-phenylbenzamide based monocyclic EGFR tyrosine kinase inhibitors
|
Mao, Yongjun
|
|
2013
|
21 |
11 |
p. 3090-3104
15 p.
|
artikel
|
| 13 |
Design, synthesis and biological evaluation of novel 3,4,5-trisubstituted aminothiophenes as inhibitors of p53–MDM2 interaction. Part 2
|
Wang, Weisi
|
|
2013
|
21 |
11 |
p. 2886-2894
9 p.
|
artikel
|
| 14 |
Design, synthesis and biological evaluation of novel 3,4,5-trisubstituted aminothiophenes as inhibitors of p53–MDM2 interaction. Part 1
|
Wang, Weisi
|
|
2013
|
21 |
11 |
p. 2879-2885
7 p.
|
artikel
|
| 15 |
Design, synthesis and evaluation of 1,2-benzisothiazol-3-one derivatives as potent caspase-3 inhibitors
|
Liu, Dazhi
|
|
2013
|
21 |
11 |
p. 2960-2967
8 p.
|
artikel
|
| 16 |
Design, synthesis and pharmacological characterization of analogs of 2-aminoethyl diphenylborinate (2-APB), a known store-operated calcium channel blocker, for inhibition of TRPV6-mediated calcium transport
|
Hofer, Alexandre
|
|
2013
|
21 |
11 |
p. 3202-3213
12 p.
|
artikel
|
| 17 |
Development of cell-active non-peptidyl inhibitors of cysteine cathepsins
|
Dana, Dibyendu
|
|
2013
|
21 |
11 |
p. 2975-2987
13 p.
|
artikel
|
| 18 |
Discovery and evaluation of piperid-4-one-containing mono-carbonyl analogs of curcumin as anti-inflammatory agents
|
Wu, Jianzhang
|
|
2013
|
21 |
11 |
p. 3058-3065
8 p.
|
artikel
|
| 19 |
Discovery of novel 4-(2-fluorophenoxy)quinoline derivatives bearing 4-oxo-1,4-dihydrocinnoline-3-carboxamide moiety as c-Met kinase inhibitors
|
Li, Sai
|
|
2013
|
21 |
11 |
p. 2843-2855
13 p.
|
artikel
|
| 20 |
Discovery of 3-phenyl-1H-5-pyrazolylamine derivatives containing a urea pharmacophore as potent and efficacious inhibitors of FMS-like tyrosine kinase-3 (FLT3)
|
Lin, Wen-Hsing
|
|
2013
|
21 |
11 |
p. 2856-2867
12 p.
|
artikel
|
| 21 |
Editorial board
|
|
|
2013
|
21 |
11 |
p. IFC-
1 p.
|
artikel
|
| 22 |
Enaminones 11. An examination of some ethyl ester enaminone derivatives as anticonvulsant agents
|
Alexander, Mariano S.
|
|
2013
|
21 |
11 |
p. 3272-3279
8 p.
|
artikel
|
| 23 |
Evaluation of N-phenyl homopiperazine analogs as potential dopamine D3 receptor selective ligands
|
Li, Aixiao
|
|
2013
|
21 |
11 |
p. 2988-2998
11 p.
|
artikel
|
| 24 |
Fluorescent properties of oligonucleotides doubly modified with an indole-fused cytosine analog and 2-aminopurine
|
Seio, Kohji
|
|
2013
|
21 |
11 |
p. 3197-3201
5 p.
|
artikel
|
| 25 |
Geranylated flavonoids displaying SARS-CoV papain-like protease inhibition from the fruits of Paulownia tomentosa
|
Cho, Jung Keun
|
|
2013
|
21 |
11 |
p. 3051-3057
7 p.
|
artikel
|
| 26 |
Graphical contents list
|
|
|
2013
|
21 |
11 |
p. 2779-2794
16 p.
|
artikel
|
| 27 |
4-(1H-Imidazo[4,5-f]-1,10-phenanthrolin-2-yl)phenol-based G-quadruplex DNA binding agents: Telomerase inhibition, cytotoxicity and DNA-binding studies
|
Wei, Chun-Ying
|
|
2013
|
21 |
11 |
p. 3379-3387
9 p.
|
artikel
|
| 28 |
Human acidic mammalian chitinase as a novel target for anti-asthma drug design using in silico screening
|
Wakasugi, Masaki
|
|
2013
|
21 |
11 |
p. 3214-3220
7 p.
|
artikel
|
| 29 |
Inhibition of VEGF expression in cancer cells and endothelial cell differentiation by synthetic stilbene derivatives
|
Martí-Centelles, Rosa
|
|
2013
|
21 |
11 |
p. 3010-3015
6 p.
|
artikel
|
| 30 |
Inhibitors for the hepatitis C virus RNA polymerase explored by SAR with advanced machine learning methods
|
Weidlich, Iwona E.
|
|
2013
|
21 |
11 |
p. 3127-3137
11 p.
|
artikel
|
| 31 |
Inulin-based glycopolymer: Its preparation, lectin-affinity and gellation property
|
Izawa, Kazumi
|
|
2013
|
21 |
11 |
p. 2895-2902
8 p.
|
artikel
|
| 32 |
Lead optimization of 5-amino-6-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)-4-hydroxyhexanamides to reduce a cardiac safety issue: Discovery of DS-8108b, an orally active renin inhibitor
|
Nakamura, Yuji
|
|
2013
|
21 |
11 |
p. 3175-3196
22 p.
|
artikel
|
| 33 |
2-(2-Methylfuran-3-carboxamido)-3-phenylpropanoic acid, a potential CYP26A1 inhibitor to enhance all-trans retinoic acid-induced leukemia cell differentiation based on virtual screening and biological evaluation
|
Li, Fengrong
|
|
2013
|
21 |
11 |
p. 3256-3261
6 p.
|
artikel
|
| 34 |
Microwave assisted synthesis, cholinesterase enzymes inhibitory activities and molecular docking studies of new pyridopyrimidine derivatives
|
Basiri, Alireza
|
|
2013
|
21 |
11 |
p. 3022-3031
10 p.
|
artikel
|
| 35 |
Modification of agonist binding moiety in hybrid derivative 5/7-{[2-(4-aryl-piperazin-1-yl)-ethyl]-propyl-amino}-5,6,7,8-tetrahydro-naphthalen-1-ol/-2-amino versions: Impact on functional activity and selectivity for dopamine D2/D3 receptors
|
Gopishetty, Bhaskar
|
|
2013
|
21 |
11 |
p. 3164-3174
11 p.
|
artikel
|
| 36 |
Modulation of acridine mutagen ICR191 intercalation to DNA by methylxanthines—Analysis with mathematical models
|
Gołuński, Grzegorz
|
|
2013
|
21 |
11 |
p. 3280-3289
10 p.
|
artikel
|
| 37 |
Multidimensional optimization of promising antitumor xanthone derivatives
|
Azevedo, Carlos M.G.
|
|
2013
|
21 |
11 |
p. 2941-2959
19 p.
|
artikel
|
| 38 |
Novel imidazole-functionalized cyclen cationic lipids: Synthesis and application as non-viral gene vectors
|
Liu, Qiang
|
|
2013
|
21 |
11 |
p. 3105-3113
9 p.
|
artikel
|
| 39 |
Novel isoquinoline derivatives as antimicrobial agents
|
Galán, Abraham
|
|
2013
|
21 |
11 |
p. 3221-3230
10 p.
|
artikel
|
| 40 |
Palladium(II) saccharinate complexes with bis(2-pyridylmethyl)amine induce cell death by apoptosis in human breast cancer cells in vitro
|
Ari, Ferda
|
|
2013
|
21 |
11 |
p. 3016-3021
6 p.
|
artikel
|
| 41 |
7-Phenyl-imidazoquinolin-4(5H)-one derivatives as selective and orally available mPGES-1 inhibitors
|
Shiro, Tomoya
|
|
2013
|
21 |
11 |
p. 2868-2878
11 p.
|
artikel
|
| 42 |
Probes for narcotic receptor mediated phenomena. 47.1 Novel C4a- and N-substituted-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ols
|
Iyer, Malliga R.
|
|
2013
|
21 |
11 |
p. 3298-3309
12 p.
|
artikel
|
| 43 |
RCAI-61 and related 6′-modified analogs of KRN7000: Their synthesis and bioactivity for mouse lymphocytes to produce interferon-γ in vivo
|
Tashiro, Takuya
|
|
2013
|
21 |
11 |
p. 3066-3079
14 p.
|
artikel
|
| 44 |
Selective CB2 agonists with anti-pruritic activity: Discovery of potent and orally available bicyclic 2-pyridones
|
Kusakabe, Ken-ichi
|
|
2013
|
21 |
11 |
p. 3154-3163
10 p.
|
artikel
|
| 45 |
Structure–activity relationships for 4-anilinoquinoline derivatives as inhibitors of the DNA methyltransferase enzyme DNMT1
|
Gamage, Swarna A.
|
|
2013
|
21 |
11 |
p. 3147-3153
7 p.
|
artikel
|
| 46 |
Sugar-attached upconversion lanthanide nanoparticles: A novel tool for high-throughput lectin assay
|
Liu, Yu
|
|
2013
|
21 |
11 |
p. 2832-2842
11 p.
|
artikel
|
| 47 |
Synthesis and biological evaluation against Leishmania amazonensis of a series of alkyl-substituted benzophenones
|
Maciel-Rezende, Claudia Mara
|
|
2013
|
21 |
11 |
p. 3114-3119
6 p.
|
artikel
|
| 48 |
Synthesis and biological evaluation of Esaprazole analogues showing σ1 binding and neuroprotective properties in vitro
|
Kelly, Nicholas M.
|
|
2013
|
21 |
11 |
p. 3334-3347
14 p.
|
artikel
|
| 49 |
Synthesis and biological evaluation of fluoro analogues of antimitotic phenstatin
|
Ghinet, Alina
|
|
2013
|
21 |
11 |
p. 2932-2940
9 p.
|
artikel
|
| 50 |
Synthesis and biological evaluation of novel styryl benzimidazole derivatives as probes for imaging of neurofibrillary tangles in Alzheimer’s disease
|
Matsumura, Kenji
|
|
2013
|
21 |
11 |
p. 3356-3362
7 p.
|
artikel
|
| 51 |
Synthesis and biology of oligoethylene glycol linked naphthoxylosides
|
Holmqvist, Karin
|
|
2013
|
21 |
11 |
p. 3310-3317
8 p.
|
artikel
|
| 52 |
Synthesis and carbonic anhydrase inhibitory properties of sulfamides structurally related to dopamine
|
Aksu, Kadir
|
|
2013
|
21 |
11 |
p. 2925-2931
7 p.
|
artikel
|
| 53 |
Synthesis and characterization of 123I-CMICE-013: A potential SPECT myocardial perfusion imaging agent
|
Wei, Lihui
|
|
2013
|
21 |
11 |
p. 2903-2911
9 p.
|
artikel
|
| 54 |
Synthesis and cytotoxicity of oligomycin A derivatives modified in the side chain
|
Lysenkova, Lyudmila N.
|
|
2013
|
21 |
11 |
p. 2918-2924
7 p.
|
artikel
|
| 55 |
Synthesis and evaluation of 7-chloro-4-(piperazin-1-yl)quinoline-sulfonamide as hybrid antiprotozoal agents
|
Salahuddin, Attar
|
|
2013
|
21 |
11 |
p. 3080-3089
10 p.
|
artikel
|
| 56 |
Synthesis and evaluation of N-substituted nipecotic acid derivatives with an unsymmetrical bis-aromatic residue attached to a vinyl ether spacer as potential GABA uptake inhibitors
|
Quandt, Gabriele
|
|
2013
|
21 |
11 |
p. 3363-3378
16 p.
|
artikel
|
| 57 |
Synthesis of the (1→6)-linked thiodisaccharide of galactofuranose: Inhibitory activity against a β-galactofuranosidase
|
Repetto, Evangelina
|
|
2013
|
21 |
11 |
p. 3327-3333
7 p.
|
artikel
|
| 58 |
Synthetic approaches to the 2011 new drugs
|
Ding, Hong X.
|
|
2013
|
21 |
11 |
p. 2795-2825
31 p.
|
artikel
|
| 59 |
The discovery of colchicine-SAHA hybrids as a new class of antitumor agents
|
Zhang, Xuan
|
|
2013
|
21 |
11 |
p. 3240-3244
5 p.
|
artikel
|
| 60 |
The effects and mechanism of flavonoid–rePON1 interactions. Structure–activity relationship study
|
Atrahimovich, Dana
|
|
2013
|
21 |
11 |
p. 3348-3355
8 p.
|
artikel
|
| 61 |
The kinetic deuterium isotope effect as applied to metabolic deactivation of imatinib to the des-methyl metabolite, CGP74588
|
Manley, Paul W.
|
|
2013
|
21 |
11 |
p. 3231-3239
9 p.
|
artikel
|
| 62 |
The systematic structure–activity relationship to predict how flavones bind to human androgen receptor for their antagonistic activity
|
Tamura, Hiroto
|
|
2013
|
21 |
11 |
p. 2968-2974
7 p.
|
artikel
|
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