| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Antiarrhythmic properties of phenylpiperazine derivatives of phenytoin with α1-adrenoceptor affinities
|
Handzlik, Jadwiga
|
|
2012
|
20 |
7 |
p. 2290-2303
14 p.
|
artikel
|
| 2 |
C–C bond formation at C-2 of a quinoline ring: Synthesis of 2-(1H-indol-3-yl)quinoline-3-carbonitrile derivatives as a new class of PDE4 inhibitors
|
Kumar, K. Shiva
|
|
2012
|
20 |
7 |
p. 2199-2207
9 p.
|
artikel
|
| 3 |
Corrigendum to “Generation of ‘Unnatural Natural Product’ library and identification of a small molecule inhibitor of XIAP” [Bioorg. Med. Chem. 19 (2011) 4377–4385]
|
Kawamura, Tatsuro
|
|
2012
|
20 |
7 |
p. 2479-
1 p.
|
artikel
|
| 4 |
Design and synthesis of thiourea compounds that inhibit transmembrane anchored carbonic anhydrases
|
Moeker, Janina
|
|
2012
|
20 |
7 |
p. 2392-2404
13 p.
|
artikel
|
| 5 |
Design, synthesis, and biological evaluation of 4-arylmethyl-1-phenylpyrazole and 4-aryloxy-1-phenylpyrazole derivatives as novel androgen receptor antagonists
|
Yamamoto, Satoshi
|
|
2012
|
20 |
7 |
p. 2338-2352
15 p.
|
artikel
|
| 6 |
Discovery of novel prostaglandin analogs as potent and selective EP2/EP4 dual agonists
|
Kambe, Tohru
|
|
2012
|
20 |
7 |
p. 2235-2251
17 p.
|
artikel
|
| 7 |
Editorial board
|
|
|
2012
|
20 |
7 |
p. IFC-
1 p.
|
artikel
|
| 8 |
Favourable involvement of α2A-adrenoreceptor antagonism in the I2-imidazoline binding sites-mediated morphine analgesia enhancement
|
Mammoli, Valerio
|
|
2012
|
20 |
7 |
p. 2259-2265
7 p.
|
artikel
|
| 9 |
Generation and exploration of new classes of antitubercular agents: The optimization of oxazolines, oxazoles, thiazolines, thiazoles to imidazo[1,2-a]pyridines and isomeric 5,6-fused scaffolds
|
Moraski, Garrett C.
|
|
2012
|
20 |
7 |
p. 2214-2220
7 p.
|
artikel
|
| 10 |
Graphical contents list
|
|
|
2012
|
20 |
7 |
p. 2191-2198
8 p.
|
artikel
|
| 11 |
Impact of stereochemistry on the biological activity of novel oleandomycin derivatives
|
Bauer, Jurica
|
|
2012
|
20 |
7 |
p. 2274-2281
8 p.
|
artikel
|
| 12 |
Indeno[1,2-b]indole derivatives as a novel class of potent human protein kinase CK2 inhibitors
|
Hundsdörfer, Claas
|
|
2012
|
20 |
7 |
p. 2282-2289
8 p.
|
artikel
|
| 13 |
In silico scaffold evaluation and solid phase approach to identify new gelatinase inhibitors
|
Topai, Alessandra
|
|
2012
|
20 |
7 |
p. 2323-2337
15 p.
|
artikel
|
| 14 |
Integrated structure-based activity prediction model of benzothiadiazines on various genotypes of HCV NS5b polymerase (1a, 1b and 4) and its application in the discovery of new derivatives
|
Ismail, Mohamed A.H.
|
|
2012
|
20 |
7 |
p. 2455-2478
24 p.
|
artikel
|
| 15 |
Intramolecular hydrogen bonding: A potential strategy for more bioavailable inhibitors of neuronal nitric oxide synthase
|
Labby, Kristin Jansen
|
|
2012
|
20 |
7 |
p. 2435-2443
9 p.
|
artikel
|
| 16 |
2-Morpholinoisoflav-3-enes as flexible intermediates in the synthesis of phenoxodiol, isophenoxodiol, equol and analogues: Vasorelaxant properties, estrogen receptor binding and Rho/RhoA kinase pathway inhibition
|
Tilley, Andrew J.
|
|
2012
|
20 |
7 |
p. 2353-2361
9 p.
|
artikel
|
| 17 |
Mutation of active site residues Asn67 to Ile, Gln92 to Val and Leu204 to Ser in human carbonic anhydrase II: Influences on the catalytic activity and affinity for inhibitors
|
Turkoglu, Sumeyye
|
|
2012
|
20 |
7 |
p. 2208-2213
6 p.
|
artikel
|
| 18 |
N 4-(3-Bromophenyl)-7-(substituted benzyl) pyrrolo[2,3-d]pyrimidines as potent multiple receptor tyrosine kinase inhibitors: Design, synthesis, and in vivo evaluation
|
Gangjee, Aleem
|
|
2012
|
20 |
7 |
p. 2444-2454
11 p.
|
artikel
|
| 19 |
New retinoid derivatives as back-ups of Adarotene
|
Giannini, Giuseppe
|
|
2012
|
20 |
7 |
p. 2405-2415
11 p.
|
artikel
|
| 20 |
Novel coumarins and 2-thioxo-coumarins as inhibitors of the tumor-associated carbonic anhydrases IX and XII
|
Carta, Fabrizio
|
|
2012
|
20 |
7 |
p. 2266-2273
8 p.
|
artikel
|
| 21 |
Optimization of the aromatase inhibitory activities of pyridylthiazole analogues of resveratrol
|
Mayhoub, Abdelrahman S.
|
|
2012
|
20 |
7 |
p. 2427-2434
8 p.
|
artikel
|
| 22 |
Perturbing pro-survival proteins using quinoxaline derivatives: A structure–activity relationship study
|
Rajule, Rajkumar
|
|
2012
|
20 |
7 |
p. 2227-2234
8 p.
|
artikel
|
| 23 |
1,3-Phenylene bis(ketoacid) derivatives as inhibitors of Escherichia coli dihydrodipicolinate synthase
|
Boughton, Berin A.
|
|
2012
|
20 |
7 |
p. 2419-2426
8 p.
|
artikel
|
| 24 |
Proteasome inhibitors for cancer therapy
|
Iqbal, Mohamed
|
|
2012
|
20 |
7 |
p. 2362-2368
7 p.
|
artikel
|
| 25 |
Synthesis and evaluation of fluorobenzoylated di- and tripeptides as inhibitors of cyclooxygenase-2 (COX-2)
|
Sharma, Sai Kiran
|
|
2012
|
20 |
7 |
p. 2221-2226
6 p.
|
artikel
|
| 26 |
Synthesis and P2Y2 receptor agonist activities of uridine 5′-phosphonate analogues
|
Van Poecke, Sara
|
|
2012
|
20 |
7 |
p. 2304-2315
12 p.
|
artikel
|
| 27 |
Synthesis and structure–activity relationship of 4-amino-2-phenylpyrimidine derivatives as a series of novel GPR119 agonists
|
Negoro, Kenji
|
|
2012
|
20 |
7 |
p. 2369-2375
7 p.
|
artikel
|
| 28 |
Synthesis, antimicrobial and anticancer activities of a novel series of diphenyl 1-(pyridin-3-yl)ethylphosphonates
|
Abdel-Megeed, Mohamed F.
|
|
2012
|
20 |
7 |
p. 2252-2258
7 p.
|
artikel
|
| 29 |
Synthesis of macrocyclic bisbibenzyl derivatives and their anticancer effects as anti-tubulin agents
|
Jiang, Juan
|
|
2012
|
20 |
7 |
p. 2382-2391
10 p.
|
artikel
|
| 30 |
Tea catechins and flavonoids from the leaves of Camellia sinensis inhibit yeast alcohol dehydrogenase
|
Manir, Md. Maniruzzaman
|
|
2012
|
20 |
7 |
p. 2376-2381
6 p.
|
artikel
|
| 31 |
The synthesis of ethacrynic acid thiazole derivatives as glutathione S-transferase pi inhibitors
|
Li, Ting
|
|
2012
|
20 |
7 |
p. 2316-2322
7 p.
|
artikel
|
| 32 |
The synthesis of 2′-methylseleno adenosine and guanosine 5′-triphosphates
|
Santner, Tobias
|
|
2012
|
20 |
7 |
p. 2416-2418
3 p.
|
artikel
|
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