| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Active site mapping of trypsin, thrombin and matriptase-2 by sulfamoyl benzamidines
|
Dosa, Stefan
|
|
2012
|
20 |
21 |
p. 6489-6505
17 p.
|
artikel
|
| 2 |
Adamantyl carboxamides and acetamides as potent human 11β-hydroxysteroid dehydrogenase type 1 inhibitors
|
Su, Xiangdong
|
|
2012
|
20 |
21 |
p. 6394-6402
9 p.
|
artikel
|
| 3 |
A novel spirocyclic tropanyl-Δ2-isoxazoline derivative enhances citalopram and paroxetine binding to serotonin transporters as well as serotonin uptake
|
Dallanoce, Clelia
|
|
2012
|
20 |
21 |
p. 6344-6355
12 p.
|
artikel
|
| 4 |
1,3-Azoles from ortho-naphthoquinones: Synthesis of aryl substituted imidazoles and oxazoles and their potent activity against Mycobacterium tuberculosis
|
Moura, Kelly C.G.
|
|
2012
|
20 |
21 |
p. 6482-6488
7 p.
|
artikel
|
| 5 |
Bioorganic & Medicinal Chemistry Reviews and Perspectives
|
|
|
2012
|
20 |
21 |
p. I-III
nvt p.
|
artikel
|
| 6 |
Carbohydrate recognition by pentadecapeptide ligands for a series of sialylated oligosaccharides
|
Matsubara, Teruhiko
|
|
2012
|
20 |
21 |
p. 6452-6458
7 p.
|
artikel
|
| 7 |
Conformational analysis of two novel cytotoxic C2-substituted pyrrolo[2,3-f]quinolines in aqueous media, organic solvents, membrane bilayers and at the putative active site
|
Varvarigou, Nicole
|
|
2012
|
20 |
21 |
p. 6276-6284
9 p.
|
artikel
|
| 8 |
Design, synthesis and biological evaluation of heterocyclic azoles derivatives containing pyrazine moiety as potential telomerase inhibitors
|
Zhang, Yan-Bin
|
|
2012
|
20 |
21 |
p. 6356-6365
10 p.
|
artikel
|
| 9 |
Design, synthesis and in vitro evaluation of a series of α-substituted phenylpropanoic acid PPARγ agonists to further investigate the stereochemistry–activity relationship
|
Ohashi, Masao
|
|
2012
|
20 |
21 |
p. 6375-6383
9 p.
|
artikel
|
| 10 |
Development and characterization of endocannabinoid hydrolases FAAH and MAGL inhibitors bearing a benzotriazol-1-yl carboxamide scaffold
|
Morera, Ludovica
|
|
2012
|
20 |
21 |
p. 6260-6275
16 p.
|
artikel
|
| 11 |
Editorial board
|
|
|
2012
|
20 |
21 |
p. IFC-
1 p.
|
artikel
|
| 12 |
Graphical contents list
|
|
|
2012
|
20 |
21 |
p. 6199-6207
9 p.
|
artikel
|
| 13 |
Identification of a 2-phenyl-substituted octahydrobenzo[f]quinoline as a dopamine D3 receptor-selective full agonist ligand
|
Clark, Alia H.
|
|
2012
|
20 |
21 |
p. 6366-6374
9 p.
|
artikel
|
| 14 |
Improving the affinity of naphthalene diimide ligand to telomeric DNA by incorporating Zn2+ ions into its dipicolylamine groups
|
Czerwinska, Izabella
|
|
2012
|
20 |
21 |
p. 6416-6422
7 p.
|
artikel
|
| 15 |
Lead optimization studies towards the discovery of novel carbamates as potent AChE inhibitors for the potential treatment of Alzheimer’s disease
|
Roy, Kuldeep K.
|
|
2012
|
20 |
21 |
p. 6313-6320
8 p.
|
artikel
|
| 16 |
New prenylated isoflavonoids as protein tyrosine phosphatase 1B (PTP1B) inhibitors from Erythrina addisoniae
|
Nguyen, Phi Hung
|
|
2012
|
20 |
21 |
p. 6459-6464
6 p.
|
artikel
|
| 17 |
Novel multipotent phenylthiazole–tacrine hybrids for the inhibition of cholinesterase activity, β-amyloid aggregation and Ca2+ overload
|
Wang, Yue
|
|
2012
|
20 |
21 |
p. 6513-6522
10 p.
|
artikel
|
| 18 |
Optimization of anti-Trypanosoma cruzi oxadiazoles leads to identification of compounds with efficacy in infected mice
|
dos Santos Filho, José Maurício
|
|
2012
|
20 |
21 |
p. 6423-6433
11 p.
|
artikel
|
| 19 |
Potent small molecule Hedgehog agonists induce VEGF expression in vitro
|
Seifert, Katrin
|
|
2012
|
20 |
21 |
p. 6465-6481
17 p.
|
artikel
|
| 20 |
Pyrido[1,2-a]pyrimidin-4-ones as antiplasmodial falcipain-2 inhibitors
|
Mane, U.R.
|
|
2012
|
20 |
21 |
p. 6296-6304
9 p.
|
artikel
|
| 21 |
Role of the side chain stereochemistry in the α-glucosidase inhibitory activity of kotalanol, a potent natural α-glucosidase inhibitor. Part 2
|
Tanabe, Genzoh
|
|
2012
|
20 |
21 |
p. 6321-6334
14 p.
|
artikel
|
| 22 |
Search for anticonvulsant and analgesic active derivatives of dihydrofuran-2(3H)-one
|
Więckowski, Krzysztof
|
|
2012
|
20 |
21 |
p. 6533-6544
12 p.
|
artikel
|
| 23 |
Small-molecular inhibitors of Ca2+-induced mitochondrial permeability transition (MPT) derived from muscle relaxant dantrolene
|
Murasawa, Shinpei
|
|
2012
|
20 |
21 |
p. 6384-6393
10 p.
|
artikel
|
| 24 |
Structure–activity relationship study of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives for potent anti-HIV agents
|
Mizuhara, Tsukasa
|
|
2012
|
20 |
21 |
p. 6434-6441
8 p.
|
artikel
|
| 25 |
Synthesis and antifungal activity of diverse C-2 pyridinyl and pyridinylvinyl substituted quinolines
|
Kouznetsov, Vladimir V.
|
|
2012
|
20 |
21 |
p. 6506-6512
7 p.
|
artikel
|
| 26 |
Synthesis and biological evaluation of a series of podophyllotoxins derivatives as a class of potent antitubulin agents
|
Liu, Yingqian
|
|
2012
|
20 |
21 |
p. 6285-6295
11 p.
|
artikel
|
| 27 |
Synthesis and structure–activity relationship of fused-pyrimidine derivatives as a series of novel GPR119 agonists
|
Negoro, Kenji
|
|
2012
|
20 |
21 |
p. 6442-6451
10 p.
|
artikel
|
| 28 |
Synthesis, biological activity and structure–activity relationship of endomorphin-1/substance P derivatives
|
Varamini, Pegah
|
|
2012
|
20 |
21 |
p. 6335-6343
9 p.
|
artikel
|
| 29 |
Synthesis of a potent photoreactive acidic γ-secretase modulator for target identification in cells
|
Rennhack, Andreas
|
|
2012
|
20 |
21 |
p. 6523-6532
10 p.
|
artikel
|
| 30 |
Synthesis of 1,5-diarylhaloimidazole analogs and their inhibitory activities against PGE2 production from LPS-treated RAW 264.7 cells
|
Yang, Zunhua
|
|
2012
|
20 |
21 |
p. 6256-6259
4 p.
|
artikel
|
| 31 |
Synthesis of imidacloprid derivatives with a chiral alkylated imidazolidine ring and evaluation of their insecticidal activity and affinity to the nicotinic acetylcholine receptor
|
Nishiwaki, Hisashi
|
|
2012
|
20 |
21 |
p. 6305-6312
8 p.
|
artikel
|
| 32 |
Synthesis of Staphylococcus aureus type 5 capsular polysaccharide repeating unit using novel l-FucNAc and d-FucNAc synthons and immunochemical evaluation
|
Danieli, Elisa
|
|
2012
|
20 |
21 |
p. 6403-6415
13 p.
|
artikel
|
| 33 |
Tandem photoaffinity labeling–bioorthogonal conjugation in medicinal chemistry
|
Lapinsky, David J.
|
|
2012
|
20 |
21 |
p. 6237-6247
11 p.
|
artikel
|
| 34 |
The antitumor agent doxorubicin binds to Fanconi anemia group F protein
|
Kusayanagi, Tomoe
|
|
2012
|
20 |
21 |
p. 6248-6255
8 p.
|
artikel
|
| 35 |
The therapeutic journey of benzimidazoles: A review
|
Bansal, Yogita
|
|
2012
|
20 |
21 |
p. 6208-6236
29 p.
|
artikel
|
Tijdschrift beschrijving