| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A bright approach to the immunoproteasome: Development of LMP2/β1i-specific imaging probes
|
Carmony, Kimberly Cornish
|
|
2012
|
20 |
2 |
p. 607-613
7 p.
|
artikel
|
| 2 |
A carbamate-based approach to primaquine prodrugs: Antimalarial activity, chemical stability and enzymatic activation
|
Mata, Graça
|
|
2012
|
20 |
2 |
p. 886-892
7 p.
|
artikel
|
| 3 |
Activity based subcellular resolution imaging of lipases
|
Viertler, Martin
|
|
2012
|
20 |
2 |
p. 628-632
5 p.
|
artikel
|
| 4 |
Alkyne derivatives of isocoumarins as clickable activity-based probes for serine proteases
|
Haedke, Ute
|
|
2012
|
20 |
2 |
p. 633-640
8 p.
|
artikel
|
| 5 |
4-Aminoethylpiperazinyl aryl ketones with 5-HT1A/5-HT7 selectivity
|
Kim, Mi Kyoung
|
|
2012
|
20 |
2 |
p. 1139-1148
10 p.
|
artikel
|
| 6 |
A new class of non-thiazolidinedione, non-carboxylic-acid-based highly selective peroxisome proliferator-activated receptor (PPAR) γ agonists: Design and synthesis of benzylpyrazole acylsulfonamides
|
Rikimaru, Kentaro
|
|
2012
|
20 |
2 |
p. 714-733
20 p.
|
artikel
|
| 7 |
An integrated computational workflow for efficient and quantitative modeling of renin inhibitors
|
Subramanian, Govindan
|
|
2012
|
20 |
2 |
p. 851-858
8 p.
|
artikel
|
| 8 |
Antidiabetogenic oligostilbenoids and 3-ethyl-4-phenyl-3,4-dihydroisocoumarins from the bark of Shorea roxburghii
|
Morikawa, Toshio
|
|
2012
|
20 |
2 |
p. 832-840
9 p.
|
artikel
|
| 9 |
Antioxidant properties of 4-quinolones and structurally related flavones
|
Greeff, Jane
|
|
2012
|
20 |
2 |
p. 809-818
10 p.
|
artikel
|
| 10 |
A para-nitrophenol phosphonate probe labels distinct serine hydrolases of Arabidopsis
|
Nickel, Sabrina
|
|
2012
|
20 |
2 |
p. 601-606
6 p.
|
artikel
|
| 11 |
Bacterial biofilm formation inhibitory activity revealed for plant derived natural compounds
|
Artini, M.
|
|
2012
|
20 |
2 |
p. 920-926
7 p.
|
artikel
|
| 12 |
Bioorthogonal proteomics of 15-hexadecynyloxyacetic acid chemical reporter reveals preferential targeting of fatty acid modified proteins and biosynthetic enzymes
|
Yount, Jacob S.
|
|
2012
|
20 |
2 |
p. 650-654
5 p.
|
artikel
|
| 13 |
Cell-based and in-silico studies on the high intrinsic activity of two boron-containing salbutamol derivatives at the human β2-adrenoceptor
|
Soriano-Ursúa, Marvin A.
|
|
2012
|
20 |
2 |
p. 933-941
9 p.
|
artikel
|
| 14 |
Chemical proteomics
|
Overkleeft, Herman
|
|
2012
|
20 |
2 |
p. 552-553
2 p.
|
artikel
|
| 15 |
Cleavable linkers in chemical biology
|
Leriche, Geoffray
|
|
2012
|
20 |
2 |
p. 571-582
12 p.
|
artikel
|
| 16 |
Cyclohexane 1,3-diones and their inhibition of mutant SOD1-dependent protein aggregation and toxicity in PC12 cells
|
Zhang, Wei
|
|
2012
|
20 |
2 |
p. 1029-1045
17 p.
|
artikel
|
| 17 |
Cyclolobatriene, a novel prenylated germacrene diterpene, from the soft coral Lobophytum pauciflorum
|
Govindam, Sudhakar V.S.
|
|
2012
|
20 |
2 |
p. 687-692
6 p.
|
artikel
|
| 18 |
Design and synthesis of benzo[c,d]indolone-pyrrolobenzodiazepine conjugates as potential anticancer agents
|
Kamal, Ahmed
|
|
2012
|
20 |
2 |
p. 789-800
12 p.
|
artikel
|
| 19 |
Design, synthesis and evaluation of polar head group containing 2-keto-oxazole inhibitors of FAAH
|
Rusch, Marion
|
|
2012
|
20 |
2 |
p. 1100-1112
13 p.
|
artikel
|
| 20 |
Design, synthesis, biological evaluation and molecular modeling of 1,3,4-oxadiazoline analogs of combretastatin-A4 as novel antitubulin agents
|
Hu, Yang
|
|
2012
|
20 |
2 |
p. 903-909
7 p.
|
artikel
|
| 21 |
Development and characterization of improved β-lactone-based anti-virulence drugs targeting ClpP
|
Zeiler, Evelyn
|
|
2012
|
20 |
2 |
p. 583-591
9 p.
|
artikel
|
| 22 |
Diazirine based photoaffinity labeling
|
Dubinsky, Luba
|
|
2012
|
20 |
2 |
p. 554-570
17 p.
|
artikel
|
| 23 |
Editorial board
|
|
|
2012
|
20 |
2 |
p. IFC-
1 p.
|
artikel
|
| 24 |
Effective and reversible DNA condensation induced by bifunctional molecules containing macrocyclic polyamines and naphthyl moieties
|
Yan, Hao
|
|
2012
|
20 |
2 |
p. 801-808
8 p.
|
artikel
|
| 25 |
Enhancement of optical properties of dyes for bioprobes by freezing effect of molecular motion using POSS-core dendrimers
|
Tanaka, Kazuo
|
|
2012
|
20 |
2 |
p. 915-919
5 p.
|
artikel
|
| 26 |
Evaluation of sulfatase-directed quinone methide traps for proteomics
|
Lenger, Janina
|
|
2012
|
20 |
2 |
p. 622-627
6 p.
|
artikel
|
| 27 |
Facile synthesis and evaluation of C-functionalized benzyl-1-oxa-4,7,10-triazacyclododecane-N,N′,N″-triacetic acid as chelating agent for 111In-labeled polypeptides
|
Suzuki, Hiroyuki
|
|
2012
|
20 |
2 |
p. 978-984
7 p.
|
artikel
|
| 28 |
Febrifugine analogue compounds: Synthesis and antimalarial evaluation
|
Zhu, Shuren
|
|
2012
|
20 |
2 |
p. 927-932
6 p.
|
artikel
|
| 29 |
Graphical contents list
|
|
|
2012
|
20 |
2 |
p. 533-549
17 p.
|
artikel
|
| 30 |
Labeling and enrichment of Arabidopsis thaliana matrix metalloproteases using an active-site directed, marimastat-based photoreactive probe
|
Lenger, Janina
|
|
2012
|
20 |
2 |
p. 592-596
5 p.
|
artikel
|
| 31 |
N 4-Aryl-6-substitutedphenylmethyl-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamines as receptor tyrosine kinase inhibitors
|
Gangjee, Aleem
|
|
2012
|
20 |
2 |
p. 910-914
5 p.
|
artikel
|
| 32 |
Novel diamino imidazole and pyrrole-containing polyamides: Synthesis and DNA binding studies of mono- and diamino-phenyl-ImPy*Im polyamides designed to target 5′-ACGCGT-3′
|
Satam, Vijay
|
|
2012
|
20 |
2 |
p. 693-701
9 p.
|
artikel
|
| 33 |
Novel inhibitors of surface layer processing in Clostridium difficile
|
Tam Dang, T.H.
|
|
2012
|
20 |
2 |
p. 614-621
8 p.
|
artikel
|
| 34 |
Novel 3-phenylpiperidine-4-carboxamides as highly potent and orally long-acting neurokinin-1 receptor antagonists with reduced CYP3A induction
|
Shirai, Junya
|
|
2012
|
20 |
2 |
p. 962-977
16 p.
|
artikel
|
| 35 |
Novel (S)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids: Peroxisome proliferator-activated receptor γ selective agonists with protein-tyrosine phosphatase 1B inhibition
|
Otake, Kazuya
|
|
2012
|
20 |
2 |
p. 1060-1075
16 p.
|
artikel
|
| 36 |
Oxidative folding of lysozyme with aromatic dithiols, and aliphatic and aromatic monothiols
|
Patel, Amar S.
|
|
2012
|
20 |
2 |
p. 1020-1028
9 p.
|
artikel
|
| 37 |
Prediction of sites of metabolism in a substrate molecule, instanced by carbamazepine oxidation by CYP3A4
|
Yuki, Hitomi
|
|
2012
|
20 |
2 |
p. 775-783
9 p.
|
artikel
|
| 38 |
Protein enrichment by capture–release based on strain-promoted cycloaddition of azide with bicyclononyne (BCN)
|
Temming, Rinske P.
|
|
2012
|
20 |
2 |
p. 655-661
7 p.
|
artikel
|
| 39 |
Publisher’s Note
|
|
|
2012
|
20 |
2 |
p. 550-551
2 p.
|
artikel
|
| 40 |
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase
|
Manfroni, Giuseppe
|
|
2012
|
20 |
2 |
p. 866-876
11 p.
|
artikel
|
| 41 |
Pyrrolo- and pyrazolo-[3,4-e][1,2,4]triazolo[1,5-c]pyrimidines as adenosine receptor antagonists
|
Baraldi, Pier Giovanni
|
|
2012
|
20 |
2 |
p. 1046-1059
14 p.
|
artikel
|
| 42 |
Pyrrolo[1,2-b]pyridazines, pyrrolo[2,1-f]triazin-4(3H)-ones, and related compounds as novel corticotropin-releasing factor 1 (CRF1) receptor antagonists
|
Saito, Tetsuji
|
|
2012
|
20 |
2 |
p. 1122-1138
17 p.
|
artikel
|
| 43 |
Resin-based investigation of acyl carrier protein interaction networks in Escherichia coli
|
Rothmann, Michael
|
|
2012
|
20 |
2 |
p. 667-671
5 p.
|
artikel
|
| 44 |
Resveratrol as a k cat type inhibitor for tyrosinase: Potentiated melanogenesis inhibitor
|
Satooka, Hiroki
|
|
2012
|
20 |
2 |
p. 1090-1099
10 p.
|
artikel
|
| 45 |
Selective inhibition of plant serine hydrolases by agrochemicals revealed by competitive ABPP
|
Kaschani, Farnusch
|
|
2012
|
20 |
2 |
p. 597-600
4 p.
|
artikel
|
| 46 |
Semisynthetic neoboutomellerone derivatives as ubiquitin-proteasome pathway inhibitors
|
Beck, Joséphine
|
|
2012
|
20 |
2 |
p. 819-831
13 p.
|
artikel
|
| 47 |
STAT6 phosphorylation inhibitors block eotaxin-3 secretion in bronchial epithelial cells
|
Zhou, Li
|
|
2012
|
20 |
2 |
p. 750-758
9 p.
|
artikel
|
| 48 |
Structure–activity relationship of α hormones, the mating factors of phytopathogen Phytophthora
|
Molli, Shylaja D.
|
|
2012
|
20 |
2 |
p. 681-686
6 p.
|
artikel
|
| 49 |
Structure–activity relationships for naturally occurring coumarins as β-secretase inhibitor
|
Marumoto, Shinsuke
|
|
2012
|
20 |
2 |
p. 784-788
5 p.
|
artikel
|
| 50 |
Structure–activity relationships of 2-amino-3-aroyl-4-[(4-arylpiperazin-1-yl)methyl]thiophenes. Part 2: Probing the influence of diverse substituents at the phenyl of the arylpiperazine moiety on allosteric enhancer activity at the A1 adenosine receptor
|
Romagnoli, Romeo
|
|
2012
|
20 |
2 |
p. 996-1007
12 p.
|
artikel
|
| 51 |
Studies on the biosynthesis of the lipodepsipeptide antibiotic Ramoplanin A2
|
Hoertz, Amanda J.
|
|
2012
|
20 |
2 |
p. 859-865
7 p.
|
artikel
|
| 52 |
Switchable MRI contrast agents based on morphological changes of pH-responsive polymers
|
Okada, Satoshi
|
|
2012
|
20 |
2 |
p. 769-774
6 p.
|
artikel
|
| 53 |
Synthesis and biochemical analysis of 2,2,3,3,4,4,5,5,6,6,7,7-dodecafluoro-N-hydroxy-octanediamides as inhibitors of human histone deacetylases
|
Henkes, Leonhard M.
|
|
2012
|
20 |
2 |
p. 985-995
11 p.
|
artikel
|
| 54 |
Synthesis and biological evaluation of 4-[3-chloro-4-(3-fluorobenzyloxy)anilino]-6-(3-substituted-phenoxy)pyrimidines as dual EGFR/ErbB-2 kinase inhibitors
|
Li, Siyuan
|
|
2012
|
20 |
2 |
p. 877-885
9 p.
|
artikel
|
| 55 |
Synthesis and evaluation of novel modified γ-lactam prostanoids as EP4 subtype-selective agonists
|
Kambe, Tohru
|
|
2012
|
20 |
2 |
p. 702-713
12 p.
|
artikel
|
| 56 |
Synthesis, biological evaluation and mechanistic studies of totarol amino alcohol derivatives as potential antimalarial agents
|
Tacon, Claire
|
|
2012
|
20 |
2 |
p. 893-902
10 p.
|
artikel
|
| 57 |
Synthesis, biological evaluation and molecular docking studies of resveratrol derivatives possessing curcumin moiety as potent antitubulin agents
|
Ruan, Ban-Feng
|
|
2012
|
20 |
2 |
p. 1113-1121
9 p.
|
artikel
|
| 58 |
Synthesis of benzopolycyclic cage amines: NMDA receptor antagonist, trypanocidal and antiviral activities
|
Torres, Eva
|
|
2012
|
20 |
2 |
p. 942-948
7 p.
|
artikel
|
| 59 |
Synthesis of deguelin–biotin conjugates and investigation into deguelin’s interactions
|
Garcia, José
|
|
2012
|
20 |
2 |
p. 672-680
9 p.
|
artikel
|
| 60 |
Synthesis of 9-phosphonoalkyl and 9-phosphonoalkoxyalkyl purines: Evaluation of their ability to act as inhibitors of Plasmodium falciparum, Plasmodium vivax and human hypoxanthine–guanine–(xanthine) phosphoribosyltransferases
|
Česnek, Michal
|
|
2012
|
20 |
2 |
p. 1076-1089
14 p.
|
artikel
|
| 61 |
Synthesis of quinolinomorphinan-4-ol derivatives as δ opioid receptor agonists
|
Ida, Yoshihiro
|
|
2012
|
20 |
2 |
p. 949-961
13 p.
|
artikel
|
| 62 |
Synthesis physicochemical profile and PAMPA study of new NO-donor edaravone co-drugs
|
Rolando, Barbara
|
|
2012
|
20 |
2 |
p. 841-850
10 p.
|
artikel
|
| 63 |
Synthesis, SAR, and preliminary mechanistic evaluation of novel antiproliferative N 6,5′-bis-ureido- and 5′-carbamoyl-N 6-ureidoadenosine derivatives
|
Shelton, Jadd R.
|
|
2012
|
20 |
2 |
p. 1008-1019
12 p.
|
artikel
|
| 64 |
Towards a stable noeuromycin analog with a d-manno configuration: Synthesis and glycosidase inhibition of d-manno-like tri- and tetrahydroxylated azepanes
|
Deschamp, Julia
|
|
2012
|
20 |
2 |
p. 641-649
9 p.
|
artikel
|
| 65 |
Two-step bioorthogonal activity-based proteasome profiling using copper-free click reagents: A comparative study
|
van der Linden, Wouter A.
|
|
2012
|
20 |
2 |
p. 662-666
5 p.
|
artikel
|
| 66 |
Ultrasound mediated catalyst free synthesis of 6H-1-benzopyrano[4,3-b]quinolin-6-ones leading to novel quinoline derivatives: Their evaluation as potential anti-cancer agents
|
Mulakayala, Naveen
|
|
2012
|
20 |
2 |
p. 759-768
10 p.
|
artikel
|
| 67 |
Weight loss effects of quaternary salts of 5-amino-1-(chloromethyl)-1,2-dihydro-3H-benz[e]indoles; structure–activity relationships
|
Tercel, Moana
|
|
2012
|
20 |
2 |
p. 734-749
16 p.
|
artikel
|
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