| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Antibacterial activities of Groebke–Blackburn–Bienaymé-derived imidazo[1,2-a]pyridin-3-amines
|
Shukla, Nikunj M.
|
|
2012
|
20 |
19 |
p. 5850-5863
14 p.
|
artikel
|
| 2 |
A sulfoximine-based inhibitor of human asparagine synthetase kills l-asparaginase-resistant leukemia cells
|
Ikeuchi, Hideyuki
|
|
2012
|
20 |
19 |
p. 5915-5927
13 p.
|
artikel
|
| 3 |
Bioorganic & Medicinal Chemistry Reviews and Perspectives
|
|
|
2012
|
20 |
19 |
p. I-III
nvt p.
|
artikel
|
| 4 |
Competitive antagonism of insect GABA receptors by iminopyridazine derivatives of GABA
|
Rahman, Mohammad Mostafizur
|
|
2012
|
20 |
19 |
p. 5957-5964
8 p.
|
artikel
|
| 5 |
Corrigendum to “Fluorescent ligands for the histamine H2 receptor: Synthesis and preliminary characterization” [Bioorg. Med. Chem. 12 (2004) 6495–6503
|
Malan, Sarel F.
|
|
2012
|
20 |
19 |
p. 6003-
1 p.
|
artikel
|
| 6 |
Design and synthesis of EGFR dimerization inhibitors and evaluation of their potential in the treatment of psoriasis
|
Petch, Donna
|
|
2012
|
20 |
19 |
p. 5901-5914
14 p.
|
artikel
|
| 7 |
Design, synthesis, and biological evaluation of the analogues of glaziovianin A, a potent antitumor isoflavone
|
Hayakawa, Ichiro
|
|
2012
|
20 |
19 |
p. 5745-5756
12 p.
|
artikel
|
| 8 |
Design, synthesis and evaluation of novel metalloproteinase inhibitors based on l-tyrosine scaffold
|
Cheng, Xian-Chao
|
|
2012
|
20 |
19 |
p. 5738-5744
7 p.
|
artikel
|
| 9 |
Development of a bifunctional chelating agent containing isothiocyanate residue for one step F-18 labeling of peptides and application for RGD labeling
|
Shetty, Dinesh
|
|
2012
|
20 |
19 |
p. 5941-5947
7 p.
|
artikel
|
| 10 |
Discovery and preclinical profile of teneligliptin (3-[(2S,4S)-4-[4-(3-methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]pyrrolidin-2-ylcarbonyl]thiazolidine): A highly potent, selective, long-lasting and orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes
|
Yoshida, Tomohiro
|
|
2012
|
20 |
19 |
p. 5705-5719
15 p.
|
artikel
|
| 11 |
Discovery of 3H-imidazo[4,5-c]quinolin-4(5H)-ones as potent and selective dipeptidyl peptidase IV (DPP-4) inhibitors
|
Ikuma, Yohei
|
|
2012
|
20 |
19 |
p. 5864-5883
20 p.
|
artikel
|
| 12 |
Discovery of 6-[4-(6-nitroxyhexanoyl)piperazin-1-yl)]-9H-purine, as pharmacological post-conditioning agent
|
Koufaki, Maria
|
|
2012
|
20 |
19 |
p. 5948-5956
9 p.
|
artikel
|
| 13 |
Editorial board
|
|
|
2012
|
20 |
19 |
p. OFC-
1 p.
|
artikel
|
| 14 |
Evaluation of dimerization–inhibitory activities of cyclic peptides containing a β-hairpin loop sequence of the EGF receptor
|
Mizuguchi, Takaaki
|
|
2012
|
20 |
19 |
p. 5730-5737
8 p.
|
artikel
|
| 15 |
[18F]FE@SNAP—A new PET tracer for the melanin concentrating hormone receptor 1 (MCHR1): Microfluidic and vessel-based approaches
|
Philippe, Cécile
|
|
2012
|
20 |
19 |
p. 5936-5940
5 p.
|
artikel
|
| 16 |
Graphical contents list
|
|
|
2012
|
20 |
19 |
p. 5669-5677
9 p.
|
artikel
|
| 17 |
Hybrid stereoisomers of a compact molecular probe based on a jasmonic acid glucoside: Syntheses and biological evaluations
|
Ueda, Minoru
|
|
2012
|
20 |
19 |
p. 5832-5843
12 p.
|
artikel
|
| 18 |
Identification of novel α7 nicotinic receptor ligands by in silico screening against the crystal structure of a chimeric α7 receptor ligand binding domain
|
Akdemir, Atilla
|
|
2012
|
20 |
19 |
p. 5992-6002
11 p.
|
artikel
|
| 19 |
Novel interleukin-5 inhibitors based on hydroxyethylaminomethyl-4H-chromen-4-one scaffold
|
Joo, Cheonik
|
|
2012
|
20 |
19 |
p. 5757-5762
6 p.
|
artikel
|
| 20 |
O-Hydroxyl- or o-amino benzylamine-tacrine hybrids: Multifunctional biometals chelators, antioxidants, and inhibitors of cholinesterase activity and amyloid-β aggregation
|
Mao, Fei
|
|
2012
|
20 |
19 |
p. 5884-5892
9 p.
|
artikel
|
| 21 |
Phosphoramidate derivatives of acyclovir: Synthesis and antiviral activity in HIV-1 and HSV-1 models in vitro
|
Zakirova, Natalia F.
|
|
2012
|
20 |
19 |
p. 5802-5809
8 p.
|
artikel
|
| 22 |
Possible conformation of amphotericin B dimer in membrane-bound assembly as deduced from solid-state NMR
|
Umegawa, Yuichi
|
|
2012
|
20 |
19 |
p. 5699-5704
6 p.
|
artikel
|
| 23 |
Protective effects of caffeoylquinic acids on the aggregation and neurotoxicity of the 42-residue amyloid β-protein
|
Miyamae, Yusaku
|
|
2012
|
20 |
19 |
p. 5844-5849
6 p.
|
artikel
|
| 24 |
Studies on synthesis and activation mechanism of mitomycin dimers connected by 1,2-dithiolane and diol linkers
|
Kim, Hyoung Rae
|
|
2012
|
20 |
19 |
p. 5720-5729
10 p.
|
artikel
|
| 25 |
Synthesis and antiplasmodial activity of new heteroaryl derivatives of 7-chloro-4-aminoquinoline
|
Casagrande, Manolo
|
|
2012
|
20 |
19 |
p. 5965-5979
15 p.
|
artikel
|
| 26 |
Synthesis and biological evaluation of novel homochiral carbocyclic nucleosides from 1-amino-2-indanols
|
Ugliarolo, Esteban A.
|
|
2012
|
20 |
19 |
p. 5986-5991
6 p.
|
artikel
|
| 27 |
Synthesis and comparison of antiplasmodial activity of (+), (−) and racemic 7-chloro-4-(N-lupinyl)aminoquinoline
|
Rusconi, Chiara
|
|
2012
|
20 |
19 |
p. 5980-5985
6 p.
|
artikel
|
| 28 |
Synthesis and evaluation of novel heteroaromatic substrates of GABA aminotransferase
|
Hawker, Dustin D.
|
|
2012
|
20 |
19 |
p. 5763-5773
11 p.
|
artikel
|
| 29 |
Synthesis and evaluation of the anti-proliferative and NF-κB activities of a library of simplified tylophorine analogs
|
Niphakis, Micah J.
|
|
2012
|
20 |
19 |
p. 5893-5900
8 p.
|
artikel
|
| 30 |
Synthesis and structure–activity relationship of a novel class of 15-membered macrolide antibiotics known as ‘11a-azalides’
|
Sugimoto, Tomohiro
|
|
2012
|
20 |
19 |
p. 5787-5801
15 p.
|
artikel
|
| 31 |
Synthesis of novel ursolic acid heterocyclic derivatives with improved abilities of antiproliferation and induction of p53, p21waf1 and NOXA in pancreatic cancer cells
|
Leal, Ana S.
|
|
2012
|
20 |
19 |
p. 5774-5786
13 p.
|
artikel
|
| 32 |
Synthesis of quinolinomorphinan derivatives as highly selective δ opioid receptor ligands
|
Ida, Yoshihiro
|
|
2012
|
20 |
19 |
p. 5810-5831
22 p.
|
artikel
|
| 33 |
Tanshinones as selective and slow-binding inhibitors for SARS-CoV cysteine proteases
|
Park, Ji-Young
|
|
2012
|
20 |
19 |
p. 5928-5935
8 p.
|
artikel
|
| 34 |
The biology and chemistry of antifungal agents: A review
|
Kathiravan, Muthu K
|
|
2012
|
20 |
19 |
p. 5678-5698
21 p.
|
artikel
|
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