| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
α-Amino-β-fluorocyclopropanecarboxylic acids as a new tool for drug development: Synthesis of glutamic acid analogs and agonist activity towards metabotropic glutamate receptor 4
|
Lemonnier, Gérald
|
|
2012
|
20 |
15 |
p. 4716-4726
11 p.
|
artikel
|
| 2 |
C-6 aryl substituted 4-quinolone-3-carboxylic acids as inhibitors of hepatitis C virus
|
Chen, Yue-Lei
|
|
2012
|
20 |
15 |
p. 4790-4800
11 p.
|
artikel
|
| 3 |
Chemoenzymatic synthesis and biological evaluation of 2- and 3-hydroxypyridine derivatives against Leishmania mexicana
|
García Liñares, Guadalupe
|
|
2012
|
20 |
15 |
p. 4614-4624
11 p.
|
artikel
|
| 4 |
Corrigendum to “Cholinestrase inhibitory effects of geranylated flavonoids from Paulownia tomentosa fruits” [Bioorg. Med. Chem. 20 (2012) 2595–2602]
|
Cho, Jung Keun
|
|
2012
|
20 |
15 |
p. 4882-
1 p.
|
artikel
|
| 5 |
Corrigendum to “Novel diamino imidazole and pyrrole-containing polyamides: Synthesis and DNA binding studies of mono- and diamino-phenyl-ImPy*Im polyamides designed to target 5′-ACGCGT-3′” [Bioorg. Med. Chem. 20 (2012) 693–701]
|
Satam, Vijay
|
|
2012
|
20 |
15 |
p. 4881-
1 p.
|
artikel
|
| 6 |
Design and synthesis of novel DFG-out RAF/vascular endothelial growth factor receptor 2 (VEGFR2) inhibitors: 2. Synthesis and characterization of a novel imide-type prodrug for improving oral absorption
|
Okaniwa, Masanori
|
|
2012
|
20 |
15 |
p. 4680-4692
13 p.
|
artikel
|
| 7 |
Design, synthesis, and pharmacological evaluation of novel tetrahydroprotoberberine derivatives: Selective inhibitors of dopamine D1 receptor
|
Qian, Wangke
|
|
2012
|
20 |
15 |
p. 4862-4871
10 p.
|
artikel
|
| 8 |
Design, synthesis, biochemical studies, cellular characterization, and structure-based computational studies of small molecules targeting the urokinase receptor
|
Wang, Fang
|
|
2012
|
20 |
15 |
p. 4760-4773
14 p.
|
artikel
|
| 9 |
Development of novel antibacterial agents against methicillin-resistant Staphylococcus aureus
|
Chiu, Hao-Chieh
|
|
2012
|
20 |
15 |
p. 4653-4660
8 p.
|
artikel
|
| 10 |
Discovery and preliminary SAR of bisbenzylisoquinoline alkaloids as inducers of C/EBPα
|
Klausmeyer, Paul
|
|
2012
|
20 |
15 |
p. 4646-4652
7 p.
|
artikel
|
| 11 |
Discovery and SAR of orally efficacious tetrahydropyridopyridazinone PARP inhibitors for the treatment of cancer
|
Zhu, Gui-Dong
|
|
2012
|
20 |
15 |
p. 4635-4645
11 p.
|
artikel
|
| 12 |
DNA damage by C1027 involves hydrogen atom abstraction and addition to nucleobases
|
San Pedro, Joanna Maria N.
|
|
2012
|
20 |
15 |
p. 4744-4750
7 p.
|
artikel
|
| 13 |
Editorial board
|
|
|
2012
|
20 |
15 |
p. IFC-
1 p.
|
artikel
|
| 14 |
Experimental and ‘in silico’ analysis of the effect of pH on HIV-1 protease inhibitor affinity: Implications for the charge state of the protein ionogenic groups
|
Domínguez, José L.
|
|
2012
|
20 |
15 |
p. 4838-4847
10 p.
|
artikel
|
| 15 |
Exploration of the SAR of anti-invasive chalcones: Synthesis and biological evaluation of conformationally restricted analogues
|
Roman, Bart I.
|
|
2012
|
20 |
15 |
p. 4812-4819
8 p.
|
artikel
|
| 16 |
Graphical contents list
|
|
|
2012
|
20 |
15 |
p. 4599-4607
9 p.
|
artikel
|
| 17 |
Methylation of imidazoline related compounds leads to loss of α2-adrenoceptor affinity. Synthesis and biological evaluation of selective I1 imidazoline receptor ligands
|
Schann, Stephan
|
|
2012
|
20 |
15 |
p. 4710-4715
6 p.
|
artikel
|
| 18 |
ortho-Carbaborane derivatives of indomethacin as cyclooxygenase (COX)-2 selective inhibitors
|
Scholz, Matthias
|
|
2012
|
20 |
15 |
p. 4830-4837
8 p.
|
artikel
|
| 19 |
PEGylation of Neuromedin U yields a promising candidate for the treatment of obesity and diabetes
|
Ingallinella, Paolo
|
|
2012
|
20 |
15 |
p. 4751-4759
9 p.
|
artikel
|
| 20 |
Rational drug design for anti-cancer chemotherapy: Multi-target QSAR models for the in silico discovery of anti-colorectal cancer agents
|
Speck-Planche, Alejandro
|
|
2012
|
20 |
15 |
p. 4848-4855
8 p.
|
artikel
|
| 21 |
Reduced glutathione-resisting 19F NMR sensors for detecting HNO
|
Kitamura, Narufumi
|
|
2012
|
20 |
15 |
p. 4668-4674
7 p.
|
artikel
|
| 22 |
Short synthesis and antimalarial activity of fagaronine
|
Rivaud, M.
|
|
2012
|
20 |
15 |
p. 4856-4861
6 p.
|
artikel
|
| 23 |
Synthesis and anticonvulsant activity of new N-Mannich bases derived from 3-(2-fluorophenyl)- and 3-(2-bromophenyl)-pyrrolidine-2,5-diones. Part II
|
Obniska, Jolanta
|
|
2012
|
20 |
15 |
p. 4872-4880
9 p.
|
artikel
|
| 24 |
Synthesis and antiviral properties of novel 7-heterocyclic substituted 7-deaza-adenine nucleoside inhibitors of Hepatitis C NS5B polymerase
|
Di Francesco, M. Emilia
|
|
2012
|
20 |
15 |
p. 4801-4811
11 p.
|
artikel
|
| 25 |
Synthesis and biological evaluation of 4′-[(benzimidazole-1-yl)methyl]biphenyl-2-sulfonamide derivatives as dual angiotensin II/endothelin A receptor antagonists
|
Bai, Renren
|
|
2012
|
20 |
15 |
p. 4661-4667
7 p.
|
artikel
|
| 26 |
Synthesis and biological evaluation of new N-acyl-homoserine-lactone analogues, based on triazole and tetrazole scaffolds, acting as LuxR-dependent quorum sensing modulators
|
Sabbah, Mohamad
|
|
2012
|
20 |
15 |
p. 4727-4736
10 p.
|
artikel
|
| 27 |
Synthesis and evaluation of the quorum sensing inhibitory effect of substituted triazolyldihydrofuranones
|
Brackman, Gilles
|
|
2012
|
20 |
15 |
p. 4737-4743
7 p.
|
artikel
|
| 28 |
Synthesis and in vitro antiproliferative activity of new 11-aminoalkylamino-substituted 5H- and 6H-indolo[2,3-b]quinolines; structure–activity relationships of neocryptolepines and 6-methyl congeners
|
Wang, Li
|
|
2012
|
20 |
15 |
p. 4820-4829
10 p.
|
artikel
|
| 29 |
Synthesis and in vitro evaluation of α-synuclein ligands
|
Yu, Lihai
|
|
2012
|
20 |
15 |
p. 4625-4634
10 p.
|
artikel
|
| 30 |
Synthesis, antimalarial activity and cytotoxicity of 10-aminoethylether derivatives of artemisinin
|
Cloete, Theunis T.
|
|
2012
|
20 |
15 |
p. 4701-4709
9 p.
|
artikel
|
| 31 |
Synthesis, cytotoxic activities and cell cycle arrest profiles of half-sandwich N-sulfonamide based dithio-o-carborane metal complexes
|
Dou, Huan
|
|
2012
|
20 |
15 |
p. 4693-4700
8 p.
|
artikel
|
| 32 |
Synthesis of N2 -modified 7-methylguanosine 5′-monophosphates as nematode translation inhibitors
|
Piecyk, Karolina
|
|
2012
|
20 |
15 |
p. 4781-4789
9 p.
|
artikel
|
| 33 |
The cell adhesion and proliferation activities of a peptide derived from human tenascin-C are dependent on two Ile residues
|
Hayashi, Ryo
|
|
2012
|
20 |
15 |
p. 4608-4613
6 p.
|
artikel
|
| 34 |
Total synthesis of grassystatin A, a probe for cathepsin E function
|
Yang, Siming
|
|
2012
|
20 |
15 |
p. 4774-4780
7 p.
|
artikel
|
| 35 |
Tumor cell-specific prodrugs using arsonic acid-presenting iron oxide nanoparticles with high sensitivity
|
Minehara, Hiroki
|
|
2012
|
20 |
15 |
p. 4675-4679
5 p.
|
artikel
|
Tijdschrift beschrijving