| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A fluorous and click approach for screening potential PET probes: Evaluation of potential hypoxia biomarkers
|
Bejot, Romain
|
|
2012
|
20 |
1 |
p. 324-329
6 p.
|
artikel
|
| 2 |
Amide-modified prenylcysteine based Icmt inhibitors: Structure–activity relationships, kinetic analysis and cellular characterization
|
Majmudar, Jaimeen D.
|
|
2012
|
20 |
1 |
p. 283-295
13 p.
|
artikel
|
| 3 |
Bisubstrate analogue inhibitors of 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase: New design with improved properties
|
Shi, Genbin
|
|
2012
|
20 |
1 |
p. 47-57
11 p.
|
artikel
|
| 4 |
Bivalent molecular probes for dopamine D 2-like receptors
|
Huber, Daniela
|
|
2012
|
20 |
1 |
p. 455-466
12 p.
|
artikel
|
| 5 |
Conjugation of a 3-(1H-phenanthro[9,10-d]imidazol-2-yl)-1H-indole intercalator to a triplex oligonucleotide and to a three-way junction
|
Fatthalla, Maha I.
|
|
2012
|
20 |
1 |
p. 207-214
8 p.
|
artikel
|
| 6 |
Corrigendum to “Chemistry of ecteinascidins. Part 3: Preparation of 2′-N-acyl derivatives of ecteinascidin 770 and evaluation of cytotoxicity” [Bioorg. Med. Chem. 19 (2011) 4421–4436]
|
Saktrakulkla, Panithi
|
|
2012
|
20 |
1 |
p. 531-
1 p.
|
artikel
|
| 7 |
Design and synthesis of novel β-diketo derivatives as HIV-1 integrase inhibitors
|
Hu, Liming
|
|
2012
|
20 |
1 |
p. 177-182
6 p.
|
artikel
|
| 8 |
Design and synthesis of 4,6-substituted-(diaphenylamino)quinazolines as potent EGFR inhibitors with antitumor activity
|
Li, Huan-Qiu
|
|
2012
|
20 |
1 |
p. 317-323
7 p.
|
artikel
|
| 9 |
Design, synthesis and biological activity of sphingosine kinase 2 selective inhibitors
|
Raje, Mithun R.
|
|
2012
|
20 |
1 |
p. 183-194
12 p.
|
artikel
|
| 10 |
Design, synthesis, and biological evaluation of novel (1-thioxo-1,2,3,4-tetrahydro-β-carbolin-9-yl)acetic acids as selective inhibitors for AKR1B1
|
Minehira, Daisuke
|
|
2012
|
20 |
1 |
p. 356-367
12 p.
|
artikel
|
| 11 |
Design, synthesis, and biological evaluation of 4-phenylpyrrole derivatives as novel androgen receptor antagonists
|
Yamamoto, Satoshi
|
|
2012
|
20 |
1 |
p. 422-434
13 p.
|
artikel
|
| 12 |
Design, synthesis, and evaluation of novel small molecule inhibitors of the influenza virus protein NS1
|
Jablonski, Joseph J.
|
|
2012
|
20 |
1 |
p. 487-497
11 p.
|
artikel
|
| 13 |
Design, synthesis and the effect of 1,2,3-triazole sialylmimetic neoglycoconjugates on Trypanosoma cruzi and its cell surface trans-sialidase
|
Campo, Vanessa L.
|
|
2012
|
20 |
1 |
p. 145-156
12 p.
|
artikel
|
| 14 |
Discovery of inhibitors and substrates of brassinin hydrolase: Probing selectivity with dithiocarbamate bioisosteres
|
Pedras, M. Soledade C.
|
|
2012
|
20 |
1 |
p. 225-233
9 p.
|
artikel
|
| 15 |
Discovery of pyrazolo[1,5-a]pyridines as p110α-selective PI3 kinase inhibitors
|
Kendall, Jackie D.
|
|
2012
|
20 |
1 |
p. 69-85
17 p.
|
artikel
|
| 16 |
Editorial board
|
|
|
2012
|
20 |
1 |
p. IFC-
1 p.
|
artikel
|
| 17 |
Efficient microwave-assisted synthesis, antibacterial activity and high fluorescence of 5 benzimidazolyl-2′-deoxyuridines
|
Krim, Jamal
|
|
2012
|
20 |
1 |
p. 480-486
7 p.
|
artikel
|
| 18 |
Elaborate ligand-based modeling and subsequent synthetic exploration unveil new nanomolar Ca2+/calmodulin-dependent protein kinase II inhibitory leads
|
Shahin, Rand
|
|
2012
|
20 |
1 |
p. 377-400
24 p.
|
artikel
|
| 19 |
Formation of ion-selective channel using cyclic tetrapeptides
|
Suga, Torao
|
|
2012
|
20 |
1 |
p. 42-46
5 p.
|
artikel
|
| 20 |
Graphical contents list
|
|
|
2012
|
20 |
1 |
p. 1-15
15 p.
|
artikel
|
| 21 |
Heavy metal-free 19F NMR probes for quantitative measurements of glutathione reductase activity using silica nanoparticles as a signal quencher
|
Tanaka, Kazuo
|
|
2012
|
20 |
1 |
p. 96-100
5 p.
|
artikel
|
| 22 |
Investigation of chalcones and benzochalcones as inhibitors of breast cancer resistance protein
|
Juvale, Kapil
|
|
2012
|
20 |
1 |
p. 346-355
10 p.
|
artikel
|
| 23 |
Investigation of substituted 6-aminohexanoates as skin penetration enhancers
|
Brychtova, Katerina
|
|
2012
|
20 |
1 |
p. 86-95
10 p.
|
artikel
|
| 24 |
Layer-by-Layer coated tyrosinase: An efficient and selective synthesis of catechols
|
Guazzaroni, Melissa
|
|
2012
|
20 |
1 |
p. 157-166
10 p.
|
artikel
|
| 25 |
Marine sponge Hymeniacidon sp. amphilectane metabolites potently inhibit rat brain microglia thromboxane B2 generation
|
Mayer, Alejandro M.S.
|
|
2012
|
20 |
1 |
p. 279-282
4 p.
|
artikel
|
| 26 |
Mefloquine–oxazolidine derivatives, derived from mefloquine and arenecarbaldehydes: In vitro activity including against the multidrug-resistant tuberculosis strain T113
|
Gonçalves, Raoni S.B.
|
|
2012
|
20 |
1 |
p. 243-248
6 p.
|
artikel
|
| 27 |
Modification of HIV-1 reverse transcriptase and integrase activity by gold(III) complexes in direct biochemical assays
|
Mphahlele, Morore
|
|
2012
|
20 |
1 |
p. 401-407
7 p.
|
artikel
|
| 28 |
Molecular docking studies of a phlorotannin, dieckol isolated from Ecklonia cava with tyrosinase inhibitory activity
|
Kang, Sung-Myung
|
|
2012
|
20 |
1 |
p. 311-316
6 p.
|
artikel
|
| 29 |
NMR-based conformational analysis of sphingomyelin in bicelles
|
Yamaguchi, Toshiyuki
|
|
2012
|
20 |
1 |
p. 270-278
9 p.
|
artikel
|
| 30 |
Novel bioactive metabolites of dipyrone (metamizol)
|
Rogosch, Tobias
|
|
2012
|
20 |
1 |
p. 101-107
7 p.
|
artikel
|
| 31 |
Novel inhibitors of epidermal growth factor receptor: (4-(Arylamino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl)(1H-indol-2-yl)methanones and (1H-indol-2-yl)(4-(phenylamino)thieno[2,3-d]pyrimidin-6-yl)methanones
|
Beckers, Thomas
|
|
2012
|
20 |
1 |
p. 125-136
12 p.
|
artikel
|
| 32 |
Novel pyrazolo[1,5-a]pyridines as p110α-selective PI3 kinase inhibitors: Exploring the benzenesulfonohydrazide SAR
|
Kendall, Jackie D.
|
|
2012
|
20 |
1 |
p. 58-68
11 p.
|
artikel
|
| 33 |
N-4-t-Butylbenzyl 2-(4-methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure–activity relationships in the A-region
|
Kim, Yong Soo
|
|
2012
|
20 |
1 |
p. 215-224
10 p.
|
artikel
|
| 34 |
Nucleic acid probe containing fluorescent tricyclic base-linked acyclonucleoside for detection of single nucleotide polymorphisms
|
Furukawa, Kinji
|
|
2012
|
20 |
1 |
p. 16-24
9 p.
|
artikel
|
| 35 |
Optimizing thiadiazole analogues of resveratrol versus three chemopreventive targets
|
Mayhoub, Abdelrahman S.
|
|
2012
|
20 |
1 |
p. 510-520
11 p.
|
artikel
|
| 36 |
Persipeptides A and B, two cyclic peptides from Streptomyces sp. UTMC 1154
|
Mohammadipanah, Fatemeh
|
|
2012
|
20 |
1 |
p. 335-339
5 p.
|
artikel
|
| 37 |
Prediction of drug efficacy for cancer treatment based on comparative analysis of chemosensitivity and gene expression data
|
Wan, Peng
|
|
2012
|
20 |
1 |
p. 167-176
10 p.
|
artikel
|
| 38 |
Prediction of inhibitory activities of Hsp90 inhibitors
|
Swuec, Paolo
|
|
2012
|
20 |
1 |
p. 408-414
7 p.
|
artikel
|
| 39 |
Quantitative structure–activity relationships of 1,3,4-thiadiazol-2(3H)-ones and 1,3,4-oxadiazol-2(3H)-ones as human protoporphyrinogen oxidase inhibitors
|
Zuo, Yang
|
|
2012
|
20 |
1 |
p. 296-304
9 p.
|
artikel
|
| 40 |
Radiosynthesis of [13N]dantrolene, a positron emission tomography probe for breast cancer resistant protein, using no-carrier-added [13N]ammonia
|
Kumata, Katsushi
|
|
2012
|
20 |
1 |
p. 305-310
6 p.
|
artikel
|
| 41 |
Reactive metabolites of desipramine and clomipramine: The kinetics of formation and reactivity with DNA
|
Korobkova, Ekaterina A.
|
|
2012
|
20 |
1 |
p. 340-345
6 p.
|
artikel
|
| 42 |
Solid-phase synthesis of 2′-hydroxychalcones. Effects on cell growth inhibition, cell cycle and apoptosis of human tumor cell lines
|
Neves, Marta Perro
|
|
2012
|
20 |
1 |
p. 25-33
9 p.
|
artikel
|
| 43 |
Stereochemical diversity of AI-2 analogs modulates quorum sensing in Vibrio harveyi and Escherichia coli
|
Rui, Fabio
|
|
2012
|
20 |
1 |
p. 249-256
8 p.
|
artikel
|
| 44 |
Structure-based redesign of an edema toxin inhibitor
|
Chen, Deliang
|
|
2012
|
20 |
1 |
p. 368-376
9 p.
|
artikel
|
| 45 |
Studies of anti-fibrillogenic activity of phthalocyanines of zirconium containing out-of-plane ligands
|
Kovalska, Vladyslava
|
|
2012
|
20 |
1 |
p. 330-334
5 p.
|
artikel
|
| 46 |
Synthesis and biological activities of 2-[(heteroaryl)methyl]imidazolines
|
Saczewski, Jaroslaw
|
|
2012
|
20 |
1 |
p. 108-116
9 p.
|
artikel
|
| 47 |
Synthesis and biological evaluation of (4H-1,2,4-triazol-4-yl)isoquinoline derivatives as selective glycine transporter 1 inhibitors
|
Sugane, Takashi
|
|
2012
|
20 |
1 |
p. 34-41
8 p.
|
artikel
|
| 48 |
Synthesis and biological evaluation of sialic acid derivatives containing a long hydrophobic chain at the anomeric position and their C-5 linked polymers as potent influenza virus inhibitors
|
Suzuki, Kaori
|
|
2012
|
20 |
1 |
p. 446-454
9 p.
|
artikel
|
| 49 |
Synthesis and evaluation of novel 4-[(3H,3aH,6aH)-3-phenyl)-4,6-dioxo-2-phenyldihydro-2H-pyrrolo[3,4-d]isoxazol-5(3H,6H,6aH)-yl]benzoic acid derivatives as potent acetylcholinesterase inhibitors and anti-amnestic agents
|
Anand, Preet
|
|
2012
|
20 |
1 |
p. 521-530
10 p.
|
artikel
|
| 50 |
Synthesis, anti-inflammatory activity and ulcerogenic liability of novel nitric oxide donating/chalcone hybrids
|
Abuo-Rahma, Gamal El-Din A.A.
|
|
2012
|
20 |
1 |
p. 195-206
12 p.
|
artikel
|
| 51 |
Synthesis, antiproliferative activity and genotoxicity of novel anthracene-containing aminophosphonates and a new anthracene-derived Schiff base
|
Kraicheva, I.
|
|
2012
|
20 |
1 |
p. 117-124
8 p.
|
artikel
|
| 52 |
Synthesis, biological evaluation and molecular modeling of 1,2,3-triazole analogs of combretastatin A-1
|
Akselsen, Øyvind W.
|
|
2012
|
20 |
1 |
p. 234-242
9 p.
|
artikel
|
| 53 |
Synthesis of 5-aryl-1,4-benzodiazepine derivatives attached in resorcinaren-PAMAM dendrimers and their anti-cancer activity
|
Cortez-Maya, Sandra
|
|
2012
|
20 |
1 |
p. 415-421
7 p.
|
artikel
|
| 54 |
Synthesis of novel 3-cyclohexylpropanoic acid-derived nitrogen heterocyclic compounds and their evaluation for tuberculostatic activity
|
Gobis, Katarzyna
|
|
2012
|
20 |
1 |
p. 137-144
8 p.
|
artikel
|
| 55 |
Synthesis, radiofluorination and pharmacological evaluation of a fluoromethyl spirocyclic PET tracer for central σ1 receptors and comparison with fluoroalkyl homologs
|
Maisonial, Aurélie
|
|
2012
|
20 |
1 |
p. 257-269
13 p.
|
artikel
|
| 56 |
Synthetic studies of bi-fluorescence-labeled maltooligosaccharides as substrates for α-amylase on the basis of fluorescence resonance energy transfer (FRET)
|
Oka, Hiroyuki
|
|
2012
|
20 |
1 |
p. 435-445
11 p.
|
artikel
|
| 57 |
The design, synthesis and biological evaluations of C-6 or C-7 substituted 2-hydroxyisoquinoline-1,3-diones as inhibitors of hepatitis C virus
|
Chen, Yue-Lei
|
|
2012
|
20 |
1 |
p. 467-479
13 p.
|
artikel
|
| 58 |
The discovery of UK-369003, a novel PDE5 inhibitor with the potential for oral bioavailability and dose-proportional pharmacokinetics
|
Rawson, David J.
|
|
2012
|
20 |
1 |
p. 498-509
12 p.
|
artikel
|
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