| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
2-Aminomethylphenylamine as a novel scaffold for factor Xa inhibitor
|
Mochizuki, Akiyoshi
|
|
2011
|
19 |
5 |
p. 1623-1642
20 p.
|
artikel
|
| 2 |
An automated, polymer-assisted strategy for the preparation of urea and thiourea derivatives of 15-membered azalides as potential antimalarial chemotherapeutics
|
Hutinec, Antun
|
|
2011
|
19 |
5 |
p. 1692-1701
10 p.
|
artikel
|
| 3 |
Antitumor agents 283. Further elaboration of Desmosdumotin C analogs as potent antitumor agents: Activation of spindle assembly checkpoint as possible mode of action
|
Nakagawa-Goto, Kyoko
|
|
2011
|
19 |
5 |
p. 1816-1822
7 p.
|
artikel
|
| 4 |
Biological activity and ligand binding mode to the progesterone receptor of A-homo analogues of progesterone
|
Alvarez, Lautaro D.
|
|
2011
|
19 |
5 |
p. 1683-1691
9 p.
|
artikel
|
| 5 |
‘Click peptide’ using production of monomer Aβ from the O-acyl isopeptide: Application to assay system of aggregation inhibitors and cellular cytotoxicity
|
Sohma, Youhei
|
|
2011
|
19 |
5 |
p. 1729-1733
5 p.
|
artikel
|
| 6 |
Cofactor-type inhibitors of inosine monophosphate dehydrogenase via modular approach: Targeting the pyrophosphate binding sub-domain
|
Felczak, Krzysztof
|
|
2011
|
19 |
5 |
p. 1594-1605
12 p.
|
artikel
|
| 7 |
Cytotoxic 3,6-bis((imidazolidinone)imino)acridines: Synthesis, DNA binding and molecular modeling
|
Janovec, Ladislav
|
|
2011
|
19 |
5 |
p. 1790-1801
12 p.
|
artikel
|
| 8 |
Design, synthesis, and in vitro characterization of novel hybrid peptidomimetic inhibitors of STAT3 protein
|
Shahani, Vijay M.
|
|
2011
|
19 |
5 |
p. 1823-1838
16 p.
|
artikel
|
| 9 |
Discovery of novel (4-piperidinyl)-piperazines as potent and orally active acetyl-CoA carboxylase 1/2 non-selective inhibitors: F-Boc and triF-Boc groups are acid-stable bioisosteres for the Boc group
|
Chonan, Tomomichi
|
|
2011
|
19 |
5 |
p. 1580-1593
14 p.
|
artikel
|
| 10 |
Editorial board
|
|
|
2011
|
19 |
5 |
p. IFC-
1 p.
|
artikel
|
| 11 |
Enhanced reactivity of Lys182 explains the limited efficacy of biogenic amines in preventing the inactivation of glucose-6-phosphate dehydrogenase by methylglyoxal
|
Flores-Morales, Patricio
|
|
2011
|
19 |
5 |
p. 1613-1622
10 p.
|
artikel
|
| 12 |
Graphical contents list
|
|
|
2011
|
19 |
5 |
p. 1563-1570
8 p.
|
artikel
|
| 13 |
Huprines as a new family of dual acting trypanocidal–antiplasmodial agents
|
Defaux, Julien
|
|
2011
|
19 |
5 |
p. 1702-1707
6 p.
|
artikel
|
| 14 |
Identification of new GATA4-small molecule inhibitors by structure-based virtual screening
|
El-Hachem, Nehmé
|
|
2011
|
19 |
5 |
p. 1734-1742
9 p.
|
artikel
|
| 15 |
17,20-Lyase inhibitors. Part 4: Design, synthesis and structure–activity relationships of naphthylmethylimidazole derivatives as novel 17,20-lyase inhibitors
|
Kaku, Tomohiro
|
|
2011
|
19 |
5 |
p. 1751-1770
20 p.
|
artikel
|
| 16 |
Radiosynthesis and in vivo evaluation of [11C]MP-10 as a PET probe for imaging PDE10A in rodent and non-human primate brain
|
Tu, Zhude
|
|
2011
|
19 |
5 |
p. 1666-1673
8 p.
|
artikel
|
| 17 |
Radiosynthesis, biodistribution and micro-SPECT imaging study of dendrimer–avidin conjugate
|
Xu, Xiaoping
|
|
2011
|
19 |
5 |
p. 1643-1648
6 p.
|
artikel
|
| 18 |
Structure–activity relationships in glycosylated 2-phenyl-indoles, 2-phenyl-benzo[b]thiophenes and 2-phenyl-benzo[b]furans as DNA binding and potential antitumor agents
|
Shi, Wei
|
|
2011
|
19 |
5 |
p. 1779-1789
11 p.
|
artikel
|
| 19 |
Structure based design of heat shock protein 90 inhibitors acting as anticancer agents
|
Doddareddy, Munikumar Reddy
|
|
2011
|
19 |
5 |
p. 1714-1720
7 p.
|
artikel
|
| 20 |
Synthesis and biological activity of amino acid conjugates of abscisic acid
|
Todoroki, Yasushi
|
|
2011
|
19 |
5 |
p. 1743-1750
8 p.
|
artikel
|
| 21 |
Synthesis and biological evaluation of 1,4-benzodiazepin-2-ones with antitrypanosomal activity
|
Spencer, John
|
|
2011
|
19 |
5 |
p. 1802-1815
14 p.
|
artikel
|
| 22 |
Synthesis and biological evaluation of imidazolo[2,1-b]benzothiazole derivatives, as potential p53 inhibitors
|
Christodoulou, Michael S.
|
|
2011
|
19 |
5 |
p. 1649-1657
9 p.
|
artikel
|
| 23 |
Synthesis and evaluation of cyclic RGD-boron cluster conjugates to develop tumor-selective boron carriers for boron neutron capture therapy
|
Kimura, Sadaaki
|
|
2011
|
19 |
5 |
p. 1721-1728
8 p.
|
artikel
|
| 24 |
Synthesis and hydrolytic evaluation of acid-labile imine-linked cytotoxic isatin model systems
|
Matesic, Lidia
|
|
2011
|
19 |
5 |
p. 1771-1778
8 p.
|
artikel
|
| 25 |
Synthesis, in vitro anti-inflammatory and cytotoxic evaluation, and mechanism of action studies of 1-benzoyl-β-carboline and 1-benzoyl-3-carboxy-β-carboline derivatives
|
Yang, Mei-Lin
|
|
2011
|
19 |
5 |
p. 1674-1682
9 p.
|
artikel
|
| 26 |
Synthesis, structure, molecular docking, and structure–activity relationship analysis of enamines: 3-Aryl-4-alkylaminofuran-2(5H)-ones as potential antibacterials
|
Xiao, Zhu-Ping
|
|
2011
|
19 |
5 |
p. 1571-1579
9 p.
|
artikel
|
| 27 |
Towards more specific O 6-methylguanine-DNA methyltransferase (MGMT) inactivators
|
Lopez, Sergio
|
|
2011
|
19 |
5 |
p. 1658-1665
8 p.
|
artikel
|
| 28 |
Unexpected stereochemical tolerance for the biological activity of tyroscherin
|
Tae, Hyun Seop
|
|
2011
|
19 |
5 |
p. 1708-1713
6 p.
|
artikel
|
| 29 |
X-ray and molecular modelling in fragment-based design of three small quinoline scaffolds for HIV integrase inhibitors
|
Majerz-Maniecka, Katarzyna
|
|
2011
|
19 |
5 |
p. 1606-1612
7 p.
|
artikel
|
Tijdschrift beschrijving