nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
2-Anilinonicotinyl linked 2-aminobenzothiazoles and [1,2,4]triazolo[1,5-b] [1,2,4]benzothiadiazine conjugates as potential mitochondrial apoptotic inducers
|
Kamal, Ahmed |
|
2011 |
19 |
23 |
p. 7136-7150 15 p. |
artikel |
2 |
Benzenediol-berberine hybrids: Multifunctional agents for Alzheimer’s disease
|
Jiang, Huailei |
|
2011 |
19 |
23 |
p. 7228-7235 8 p. |
artikel |
3 |
Benzenepolycarboxylic acids with potential anti-hemorrhagic properties and structure–activity relationships
|
Aung, Hnin Thanda |
|
2011 |
19 |
23 |
p. 7000-7002 3 p. |
artikel |
4 |
1,2-Benzothiazine 1,1-dioxide carboxylate derivatives as novel potent inhibitors of aldose reductase
|
Chen, Xin |
|
2011 |
19 |
23 |
p. 7262-7269 8 p. |
artikel |
5 |
(2-Benzyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indol-8-yl)-acetic acid: An aldose reductase inhibitor and antioxidant of zwitterionic nature
|
Stefek, Milan |
|
2011 |
19 |
23 |
p. 7181-7185 5 p. |
artikel |
6 |
B-Ring-modified and/or 5-demethylated nobiletin congeners: Inhibitory activity against pro-MMP-9 production
|
Oshitari, Tetsuta |
|
2011 |
19 |
23 |
p. 7085-7092 8 p. |
artikel |
7 |
Design, synthesis and biological activity of original pyrazolo-pyrido-diazepine, -pyrazine and -oxazine dione derivatives as novel dual Nox4/Nox1 inhibitors
|
Gaggini, Francesca |
|
2011 |
19 |
23 |
p. 6989-6999 11 p. |
artikel |
8 |
Design, synthesis, and biological evaluation of a novel series of bisintercalating DNA-binding piperazine-linked bisanthrapyrazole compounds as anticancer agents
|
Zhang, Rui |
|
2011 |
19 |
23 |
p. 7023-7032 10 p. |
artikel |
9 |
Design, synthesis and biological evaluation of cycloalkyl arylpyrimidines (CAPYs) as HIV-1 NNRTIs
|
Gu, Shuang-Xi |
|
2011 |
19 |
23 |
p. 7093-7099 7 p. |
artikel |
10 |
Design, synthesis and biological evaluation of peptidyl-vinylaminophosphonates as novel cysteine protease inhibitors
|
Bhattacharya, Asish K. |
|
2011 |
19 |
23 |
p. 7129-7135 7 p. |
artikel |
11 |
13,13-Dimethyl-des-C,D analogues of (20S)-1α,25-dihydroxy-2-methylene-19-norvitamin D3 (2MD): Total synthesis, docking to the VDR, and biological evaluation
|
Plonska-Ocypa, Katarzyna |
|
2011 |
19 |
23 |
p. 7205-7220 16 p. |
artikel |
12 |
Discovery and pharmacological characterization of N-[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl}amino)-2-methylpropyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide hydrochloride (anagliptin hydrochloride salt) as a potent and selective DPP-IV inhibitor
|
Kato, Noriyasu |
|
2011 |
19 |
23 |
p. 7221-7227 7 p. |
artikel |
13 |
Editorial board
|
|
|
2011 |
19 |
23 |
p. IFC- 1 p. |
artikel |
14 |
Effect of 2′,6′-dimethyl-l-tyrosine (Dmt) on pharmacological activity of cyclic endomorphin-2 and morphiceptin analogs
|
Fichna, Jakub |
|
2011 |
19 |
23 |
p. 6977-6981 5 p. |
artikel |
15 |
Graphical contents list
|
|
|
2011 |
19 |
23 |
p. 6967-6976 10 p. |
artikel |
16 |
Identification of novel CYP2A6 inhibitors by virtual screening
|
Rahnasto, Minna K. |
|
2011 |
19 |
23 |
p. 7186-7193 8 p. |
artikel |
17 |
Inhibition of rat synaptic membrane Na+/K+-ATPase and ecto-nucleoside triphosphate diphosphohydrolases by 12-tungstosilicic and 12-tungstophosphoric acid
|
Čolović, Mirjana B. |
|
2011 |
19 |
23 |
p. 7063-7069 7 p. |
artikel |
18 |
In search of a cytostatic agent derived from the alkaloid lycorine: Synthesis and growth inhibitory properties of lycorine derivatives
|
Evdokimov, Nikolai M. |
|
2011 |
19 |
23 |
p. 7252-7261 10 p. |
artikel |
19 |
Metabolic and electrochemical mechanisms of dimeric naphthoquinones cytotoxicity in breast cancer cells
|
Emadi, Ashkan |
|
2011 |
19 |
23 |
p. 7057-7062 6 p. |
artikel |
20 |
Molecular modeling studies, synthesis, configurational stability and biological activity of 8-chloro-2,3,5,6-tetrahydro-3,6-dimethyl-pyrrolo[1,2,3-de]-1,2,4-benzothiadiazine 1,1-dioxide
|
Battisti, Umberto M. |
|
2011 |
19 |
23 |
p. 7111-7119 9 p. |
artikel |
21 |
Novel pyridopyrazine and pyrimidothiazine derivatives as FtsZ inhibitors
|
Mathew, Bini |
|
2011 |
19 |
23 |
p. 7120-7128 9 p. |
artikel |
22 |
N9-Substituted N 6-[(3-methylbut-2-en-1-yl)amino]purine derivatives and their biological activity in selected cytokinin bioassays
|
Mik, Václav |
|
2011 |
19 |
23 |
p. 7244-7251 8 p. |
artikel |
23 |
Pharmacophore-based discovery of FXR agonists. Part I: Model development and experimental validation
|
Schuster, Daniela |
|
2011 |
19 |
23 |
p. 7168-7180 13 p. |
artikel |
24 |
Quinoline tricyclic derivatives. Design, synthesis and evaluation of the antiviral activity of three new classes of RNA-dependent RNA polymerase inhibitors
|
Carta, Antonio |
|
2011 |
19 |
23 |
p. 7070-7084 15 p. |
artikel |
25 |
Screening of a library of T7 phage-displayed peptides identifies alphaC helix in 14-3-3 protein as a CBP501-binding site
|
Matsumoto, Yuki |
|
2011 |
19 |
23 |
p. 7049-7056 8 p. |
artikel |
26 |
Searching for the Multi-Target-Directed Ligands against Alzheimer’s disease: Discovery of quinoxaline-based hybrid compounds with AChE, H3R and BACE 1 inhibitory activities
|
Huang, Wenhai |
|
2011 |
19 |
23 |
p. 7158-7167 10 p. |
artikel |
27 |
Synthesis and activity of new macrolones: Conjugates between 6(7)-(2′-aminoethyl)-amino-1-cyclopropyl-3-carboxylic acid (2′-hydroxyethyl) amides and 4″-propenoyl-azithromycin
|
Kapić, Samra |
|
2011 |
19 |
23 |
p. 7270-7280 11 p. |
artikel |
28 |
Synthesis and biological profile of new 1,2,3,4-tetrahydroisoquinolines as selective carbonic anhydrase inhibitors
|
Gitto, Rosaria |
|
2011 |
19 |
23 |
p. 7003-7007 5 p. |
artikel |
29 |
Synthesis and in vitro evaluation of analogues of avocado-produced toxin (+)-(R)-persin in human breast cancer cells
|
Brooke, Darby G. |
|
2011 |
19 |
23 |
p. 7033-7043 11 p. |
artikel |
30 |
Synthesis, molecular modeling studies and biological evaluation of fluorine substituted analogs of GW 501516
|
Ciocoiu, Calin C. |
|
2011 |
19 |
23 |
p. 6982-6988 7 p. |
artikel |
31 |
Synthesis of 6-(het) ary Xylocydine analogues and evaluating their inhibitory activities of CDK1 and CDK2 in vitro
|
Xiao, Chuan |
|
2011 |
19 |
23 |
p. 7100-7110 11 p. |
artikel |
32 |
Synthesis of macrolones with central piperazine ring in the linker and its influence on antibacterial activity
|
Kapić, Samra |
|
2011 |
19 |
23 |
p. 7281-7298 18 p. |
artikel |
33 |
Targeting pancreatic cancer with a G-quadruplex ligand
|
Gunaratnam, Mekala |
|
2011 |
19 |
23 |
p. 7151-7157 7 p. |
artikel |
34 |
The arginine mimicking β-amino acid β 3hPhe(3-H2N-CH2) as S1 ligand in cyclotheonamide-based β-tryptase inhibitors
|
Janke, Dennis |
|
2011 |
19 |
23 |
p. 7236-7243 8 p. |
artikel |
35 |
The effect of the placement and total charge of the basic amino acid clusters on antibacterial organism selectivity and potency
|
Russell, Amanda L. |
|
2011 |
19 |
23 |
p. 7008-7022 15 p. |
artikel |
36 |
Trace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine class
|
Lewin, Anita H. |
|
2011 |
19 |
23 |
p. 7044-7048 5 p. |
artikel |
37 |
Tyrphostin-like compounds with ubiquitin modulatory activity as possible therapeutic agents for multiple myeloma
|
Peng, Zhenghong |
|
2011 |
19 |
23 |
p. 7194-7204 11 p. |
artikel |