| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Aminomethyltetrazoles as potential inhibitors of the γ-aminobutyric acid transporters mGAT1–mGAT4: Synthesis and biological evaluation
|
Schaffert, Eva S.
|
|
2011
|
19 |
21 |
p. 6492-6504
13 p.
|
artikel
|
| 2 |
A sucrose-derived scaffold for multimerization of bioactive peptides
|
Rao, Venkataramanarao
|
|
2011
|
19 |
21 |
p. 6474-6482
9 p.
|
artikel
|
| 3 |
Binding of isoxazole and pyrazole derivatives of curcumin with the activator binding domain of novel protein kinase C
|
Das, Joydip
|
|
2011
|
19 |
21 |
p. 6196-6202
7 p.
|
artikel
|
| 4 |
Bioassay-guided identification of an anti-inflammatory prenylated acylphloroglucinol from Melicope ptelefolia and molecular insights into its interaction with 5-lipoxygenase
|
Shaari, Khozirah
|
|
2011
|
19 |
21 |
p. 6340-6347
8 p.
|
artikel
|
| 5 |
Chemical synthesis, biological evaluation and structure–activity relationship analysis of azaisoindolinones, a novel class of direct enoyl-ACP reductase inhibitors as potential antimycobacterial agents
|
Deraeve, Céline
|
|
2011
|
19 |
21 |
p. 6225-6232
8 p.
|
artikel
|
| 6 |
‘Click’ synthesis of dextran macrostructures for combinatorial-designed self-assembled nanoparticles encapsulating diverse anticancer therapeutics
|
Abeylath, Sampath C.
|
|
2011
|
19 |
21 |
p. 6167-6173
7 p.
|
artikel
|
| 7 |
Design, structure–activity relationship, and highly efficient asymmetric synthesis of 3-phenyl-4-benzylaminopiperidine derivatives as novel neurokinin-1 receptor antagonists
|
Shirai, Junya
|
|
2011
|
19 |
21 |
p. 6430-6446
17 p.
|
artikel
|
| 8 |
Design, synthesis and biological evaluation of benzo[1.3.2]dithiazolium ylide 1,1-dioxide derivatives as potential dual cyclooxygenase-2/5-lipoxygenase inhibitors
|
Tan, Chen-Ming
|
|
2011
|
19 |
21 |
p. 6316-6328
13 p.
|
artikel
|
| 9 |
Design, synthesis, and biological evaluation of callophycin A and analogues as potential chemopreventive and anticancer agents
|
Shen, Li
|
|
2011
|
19 |
21 |
p. 6182-6195
14 p.
|
artikel
|
| 10 |
Design, synthesis and biological evaluation of mannosyl triazoles as FimH antagonists
|
Schwardt, Oliver
|
|
2011
|
19 |
21 |
p. 6454-6473
20 p.
|
artikel
|
| 11 |
Design, synthesis, biophysical and biological studies of trisubstituted naphthalimides as G-quadruplex ligands
|
Peduto, Antonella
|
|
2011
|
19 |
21 |
p. 6419-6429
11 p.
|
artikel
|
| 12 |
1,1-Diarylalkenes as anticancer agents: Dual inhibitors of tubulin polymerization and phosphodiesterase 4
|
Ruchelman, Alexander L.
|
|
2011
|
19 |
21 |
p. 6356-6374
19 p.
|
artikel
|
| 13 |
Directed evolution of a pyruvate aldolase to recognize a long chain acyl substrate
|
Cheriyan, Manoj
|
|
2011
|
19 |
21 |
p. 6447-6453
7 p.
|
artikel
|
| 14 |
Discovery of orteronel (TAK-700), a naphthylmethylimidazole derivative, as a highly selective 17,20-lyase inhibitor with potential utility in the treatment of prostate cancer
|
Kaku, Tomohiro
|
|
2011
|
19 |
21 |
p. 6383-6399
17 p.
|
artikel
|
| 15 |
Discovery of pyridine-2-ones as novel class of multidrug resistance (MDR) modulators: First structure–activity relationships
|
Krawczyk, Sören
|
|
2011
|
19 |
21 |
p. 6309-6315
7 p.
|
artikel
|
| 16 |
3,4-Disubstituted oxazolidin-2-ones as constrained ceramide analogs with anticancer activities
|
Singh, Alok
|
|
2011
|
19 |
21 |
p. 6174-6181
8 p.
|
artikel
|
| 17 |
Editorial board
|
|
|
2011
|
19 |
21 |
p. IFC-
1 p.
|
artikel
|
| 18 |
Effect of different C3-aryl substituents on the antioxidant activity of 4-hydroxycoumarin derivatives
|
Rodríguez, Sergio A.
|
|
2011
|
19 |
21 |
p. 6233-6238
6 p.
|
artikel
|
| 19 |
Evaluation of apoptotic effect of cyclic imide derivatives on murine B16F10 melanoma cells
|
Machado, Karina Elisa
|
|
2011
|
19 |
21 |
p. 6285-6291
7 p.
|
artikel
|
| 20 |
Formulating a new basis for the treatment against botulinum neurotoxin intoxication: 3,4-Diaminopyridine prodrug design and characterization
|
Zakhari, Joseph S.
|
|
2011
|
19 |
21 |
p. 6203-6209
7 p.
|
artikel
|
| 21 |
Graphical contents list
|
|
|
2011
|
19 |
21 |
p. 6157-6166
10 p.
|
artikel
|
| 22 |
Identification of a potent and selective σ1 receptor agonist potentiating NGF-induced neurite outgrowth in PC12 cells
|
Rossi, Daniela
|
|
2011
|
19 |
21 |
p. 6210-6224
15 p.
|
artikel
|
| 23 |
Identification of new antimalarial leads by use of virtual screening against cytochrome bc 1
|
Rodrigues, Tiago
|
|
2011
|
19 |
21 |
p. 6302-6308
7 p.
|
artikel
|
| 24 |
Improvement in oral bioavailability of 2,4-diaminopyrimidine c-Met inhibitors by incorporation of a 3-amidobenzazepin-2-one group
|
Milkiewicz, Karen L.
|
|
2011
|
19 |
21 |
p. 6274-6284
11 p.
|
artikel
|
| 25 |
Melanin-concentrating hormone receptor 1 antagonists: Synthesis, structure–activity relationship, docking studies, and biological evaluation of 2,3,4,5-tetrahydro-1H-3-benzazepine derivatives
|
Kasai, Shizuo
|
|
2011
|
19 |
21 |
p. 6261-6273
13 p.
|
artikel
|
| 26 |
Multi-target drug discovery in anti-cancer therapy: Fragment-based approach toward the design of potent and versatile anti-prostate cancer agents
|
Speck-Planche, Alejandro
|
|
2011
|
19 |
21 |
p. 6239-6244
6 p.
|
artikel
|
| 27 |
New dammarane-type glucosides as potential activators of AMP-activated protein kinase (AMPK) from Gynostemma pentaphyllum
|
Nguyen, Phi Hung
|
|
2011
|
19 |
21 |
p. 6254-6260
7 p.
|
artikel
|
| 28 |
Novel biologically active nitro and amino substituted benzimidazo[1,2-a]quinolines
|
Perin, Nataša
|
|
2011
|
19 |
21 |
p. 6329-6339
11 p.
|
artikel
|
| 29 |
Sodium dl-α-tocopheryl-6-O-phosphate inhibits PGE2 production in keratinocytes induced by UVB, IL-1β and peroxidants
|
Kato, Eiko
|
|
2011
|
19 |
21 |
p. 6348-6355
8 p.
|
artikel
|
| 30 |
Synthesis and anticancer activity of 5′-chloromethylphosphonates of 3′-azido-3′-deoxythymidine (AZT)
|
Celewicz, Lech
|
|
2011
|
19 |
21 |
p. 6375-6382
8 p.
|
artikel
|
| 31 |
Synthesis and antitumor activity of β-carboline 3-(substituted-carbohydrazide) derivatives
|
Barbosa, Valéria Aquilino
|
|
2011
|
19 |
21 |
p. 6400-6408
9 p.
|
artikel
|
| 32 |
Synthesis and characterization of [125I]2-iodo N-[(S)-{(S)-1-methylpiperidin-2-yl}(phenyl)methyl]3-trifluoromethyl-benzamide as novel imaging probe for glycine transporter 1
|
Fuchigami, Takeshi
|
|
2011
|
19 |
21 |
p. 6245-6253
9 p.
|
artikel
|
| 33 |
Synthesis and evaluation of novel macrocyclic antifungal peptides
|
Mulder, Monique P.C.
|
|
2011
|
19 |
21 |
p. 6505-6517
13 p.
|
artikel
|
| 34 |
Synthesis, biological evaluation, and molecular docking studies of 1,3,4-oxadiazole derivatives possessing 1,4-benzodioxan moiety as potential anticancer agents
|
Zhang, Xiao-Min
|
|
2011
|
19 |
21 |
p. 6518-6524
7 p.
|
artikel
|
| 35 |
Synthesis, molecular modeling and preliminary biological evaluation of a set of 3-acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazole as potential antibacterial, anti-Trypanosoma cruzi and antifungal agents
|
Ishii, Marina
|
|
2011
|
19 |
21 |
p. 6292-6301
10 p.
|
artikel
|
| 36 |
The anti-malarial activity of bivalent imidazolium salts
|
Vlahakis, Jason Z.
|
|
2011
|
19 |
21 |
p. 6525-6542
18 p.
|
artikel
|
| 37 |
Three-dimensional quantitative structure–activity relationship analyses of substrates of the human proton-coupled amino acid transporter 1 (hPAT1)
|
Thondorf, Iris
|
|
2011
|
19 |
21 |
p. 6409-6418
10 p.
|
artikel
|
| 38 |
Tocotrienamines and tocopheramines: Reactions with radicals and metal ions
|
Galli, Francesco
|
|
2011
|
19 |
21 |
p. 6483-6491
9 p.
|
artikel
|
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