nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
5a-Carba-β-d-glucopyranose derivatives as novel sodium-dependent glucose cotransporter 2 (SGLT2) inhibitors for the treatment of type 2 diabetes
|
Ohtake, Yoshihito |
|
2011 |
19 |
18 |
p. 5334-5341 8 p. |
artikel |
2 |
A novel amino-benzosuberone derivative is a picomolar inhibitor of mammalian aminopeptidase N/CD13
|
Maiereanu, Carmen |
|
2011 |
19 |
18 |
p. 5716-5733 18 p. |
artikel |
3 |
A novel 3-arylethynyl-substituted pyrido[2,3,-b]pyrazine derivatives and pharmacophore model as Wnt2/β-catenin pathway inhibitors in non-small-cell lung cancer cell lines
|
Gong, Young-Dae |
|
2011 |
19 |
18 |
p. 5639-5647 9 p. |
artikel |
4 |
Anthraquinone derivatives induce G2/M cell cycle arrest and apoptosis in NTUB1 cells
|
Tu, Huang-Yao |
|
2011 |
19 |
18 |
p. 5670-5678 9 p. |
artikel |
5 |
Antifungal thiopeptide cyclothiazomycin B1 exhibits growth inhibition accompanying morphological changes via binding to fungal cell wall chitin
|
Mizuhara, Naoko |
|
2011 |
19 |
18 |
p. 5300-5310 11 p. |
artikel |
6 |
Assessment of dopamine D1 receptor affinity and efficacy of three tetracyclic conformationally-restricted analogs of SKF38393
|
Clark, Alia H. |
|
2011 |
19 |
18 |
p. 5420-5431 12 p. |
artikel |
7 |
Biochemical characterization of a novel type-II VEGFR2 kinase inhibitor: Comparison of binding to non-phosphorylated and phosphorylated VEGFR2
|
Iwata, Hidehisa |
|
2011 |
19 |
18 |
p. 5342-5351 10 p. |
artikel |
8 |
Chemical modifications of resveratrol for improved protein kinase C alpha activity
|
Das, Joydip |
|
2011 |
19 |
18 |
p. 5321-5333 13 p. |
artikel |
9 |
Corrigendum to “Discovery of potent, selective, and orally bioavailable quinoline-based dipeptidyl peptidase IV inhibitors targeting Lys554” [Bioorg. Med. Chem. 19 (2011) 4482–4498]
|
Maezaki, Hironobu |
|
2011 |
19 |
18 |
p. 5742- 1 p. |
artikel |
10 |
De novo design, synthesis and biological evaluation of 1,4-dihydroquinolin-4-ones and 1,2,3,4-tetrahydroquinazolin-4-ones as potent kinesin spindle protein (KSP) inhibitors
|
Jiang, Cheng |
|
2011 |
19 |
18 |
p. 5612-5627 16 p. |
artikel |
11 |
Design and synthesis of 1,3-biarylsulfanyl derivatives as new anti-breast cancer agents
|
Kumar, Atul |
|
2011 |
19 |
18 |
p. 5409-5419 11 p. |
artikel |
12 |
Design and synthesis of new prostaglandin D2 receptor antagonists
|
Iwahashi, Maki |
|
2011 |
19 |
18 |
p. 5361-5371 11 p. |
artikel |
13 |
Design, synthesis, and biological evaluation of curcumin analogues as multifunctional agents for the treatment of Alzheimer’s disease
|
Chen, Shang-Ying |
|
2011 |
19 |
18 |
p. 5596-5604 9 p. |
artikel |
14 |
Design, synthesis, and biological evaluation of imidazoline derivatives as p53–MDM2 binding inhibitors
|
Hu, Chunqi |
|
2011 |
19 |
18 |
p. 5454-5461 8 p. |
artikel |
15 |
6,7-Dihydro-5H-cyclopenta[d]pyrazolo[1,5-a]pyrimidines and their derivatives as novel corticotropin-releasing factor 1 receptor antagonists
|
Saito, Tetsuji |
|
2011 |
19 |
18 |
p. 5432-5445 14 p. |
artikel |
16 |
Discovery, synthesis, and structure–activity relationship of 6-aminomethyl-7,8-dihydronaphthalenes as human melanin-concentrating hormone receptor 1 antagonists
|
Kamata, Makoto |
|
2011 |
19 |
18 |
p. 5539-5552 14 p. |
artikel |
17 |
Editorial board
|
|
|
2011 |
19 |
18 |
p. IFC- 1 p. |
artikel |
18 |
Extended targeting potential and improved synthesis of Microcin C analogs as antibacterials
|
Vondenhoff, Gaston H.M. |
|
2011 |
19 |
18 |
p. 5462-5467 6 p. |
artikel |
19 |
Fluorinated cannabinoid CB2 receptor ligands: Synthesis and in vitro binding characteristics of 2-oxoquinoline derivatives
|
Turkman, Nashaat |
|
2011 |
19 |
18 |
p. 5698-5707 10 p. |
artikel |
20 |
Graphical contents list
|
|
|
2011 |
19 |
18 |
p. 5279-5290 12 p. |
artikel |
21 |
Inhibition of LuxS by S-ribosylhomocysteine analogues containing a [4-aza]ribose ring
|
Malladi, Venkata L.A. |
|
2011 |
19 |
18 |
p. 5507-5519 13 p. |
artikel |
22 |
Inhibitory effects of chalcone glycosides isolated from Brassica rapa L. ‘hidabeni’ and their synthetic derivatives on LPS-induced NO production in microglia
|
Hara, Hirokazu |
|
2011 |
19 |
18 |
p. 5559-5568 10 p. |
artikel |
23 |
Isolation and structural identification of a direct-acting mutagen derived from N-nitroso-N-methylpentylamine and Fenton’s reagent with copper ion
|
Miura, Motofumi |
|
2011 |
19 |
18 |
p. 5693-5697 5 p. |
artikel |
24 |
Isolation, identification, and biological evaluation of HIF-1-modulating compounds from Brazilian green propolis
|
Hattori, Hisanori |
|
2011 |
19 |
18 |
p. 5392-5401 10 p. |
artikel |
25 |
N-(1,3-Diaryl-3-oxopropyl)amides as a new template for xanthine oxidase inhibitors
|
Nepali, Kunal |
|
2011 |
19 |
18 |
p. 5569-5576 8 p. |
artikel |
26 |
Norcantharimide analogues possessing terminal phosphate esters and their anti-cancer activity
|
Robertson, Mark J. |
|
2011 |
19 |
18 |
p. 5734-5741 8 p. |
artikel |
27 |
Novel macrocyclic C-aryl glucoside SGLT2 inhibitors as potential antidiabetic agents
|
Kim, Min Ju |
|
2011 |
19 |
18 |
p. 5468-5479 12 p. |
artikel |
28 |
Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C
|
Yoshimitsu, Yuji |
|
2011 |
19 |
18 |
p. 5402-5408 7 p. |
artikel |
29 |
2-({6-[(3R)-3-amino-3-methylpiperidine-1-yl]-1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-5H-pyrrolo[3,2-d]pyrimidine-5-yl}methyl)-4-fluorobenzonitrile (DSR-12727): A potent, orally active dipeptidyl peptidase IV inhibitor without mechanism-based inactivation of CYP3A
|
Nishio, Yukihiro |
|
2011 |
19 |
18 |
p. 5490-5499 10 p. |
artikel |
30 |
SAR studies of acidic dual γ-secretase/PPARγ modulators
|
Hieke, Martina |
|
2011 |
19 |
18 |
p. 5372-5382 11 p. |
artikel |
31 |
Substituted lactam and cyclic azahemiacetals modulate Pseudomonas aeruginosa quorum sensing
|
Malladi, Venkata L.A. |
|
2011 |
19 |
18 |
p. 5500-5506 7 p. |
artikel |
32 |
Synthesis and biological evaluation of 2′,4′- and 3′,4′-bridged nucleoside analogues
|
Nicolaou, K.C. |
|
2011 |
19 |
18 |
p. 5648-5669 22 p. |
artikel |
33 |
Synthesis and biological evaluation of a peptide–paclitaxel conjugate which targets the integrin αvβ6
|
Li, Shunzi |
|
2011 |
19 |
18 |
p. 5480-5489 10 p. |
artikel |
34 |
Synthesis and biological evaluation of HQCAs with aryl or benzyl substituents on N-1 position as potential HIV-1 integrase inhibitors
|
He, Qiu-Qin |
|
2011 |
19 |
18 |
p. 5553-5558 6 p. |
artikel |
35 |
Synthesis and biological evaluation of Matijing-Su derivatives as potent anti-HBV agents
|
Qiu, Jingying |
|
2011 |
19 |
18 |
p. 5352-5360 9 p. |
artikel |
36 |
Synthesis and characterization of tritylthioethanamine derivatives with potent KSP inhibitory activity
|
Rodriguez, Delany |
|
2011 |
19 |
18 |
p. 5446-5453 8 p. |
artikel |
37 |
Synthesis and glycosidase inhibitory profiles of functionalised morpholines and oxazepanes
|
Burland, Peter A. |
|
2011 |
19 |
18 |
p. 5679-5692 14 p. |
artikel |
38 |
Synthesis and pharmacological evaluation of 1-alkyl-N-[2-ethyl-2-(4-fluorophenyl)butyl]piperidine-4-carboxamide derivatives as novel antihypertensive agents
|
Watanuki, Susumu |
|
2011 |
19 |
18 |
p. 5628-5638 11 p. |
artikel |
39 |
Synthesis and photobiological study of a novel chlorin photosensitizer BCPD-18MA for photodynamic therapy
|
Zhang, Jialiang |
|
2011 |
19 |
18 |
p. 5520-5528 9 p. |
artikel |
40 |
Synthesis and protective effects of aralkyl alcoholic 2-acetamido-2-deoxy-β-d-pyranosides on hypoglycemia and serum limitation induced apoptosis in PC12 cell
|
Meng, Ying |
|
2011 |
19 |
18 |
p. 5577-5584 8 p. |
artikel |
41 |
Synthesis and SAR requirements of adamantane–colchicine conjugates with both microtubule depolymerizing and tubulin clustering activities
|
Zefirova, Olga N. |
|
2011 |
19 |
18 |
p. 5529-5538 10 p. |
artikel |
42 |
Synthesis, antibacterial activities and molecular docking studies of Schiff bases derived from N-(2/4-benzaldehyde-amino) phenyl-N′-phenyl-thiourea
|
Zhang, Hong-Jia |
|
2011 |
19 |
18 |
p. 5708-5715 8 p. |
artikel |
43 |
Synthesis, antitubercular activity, and SAR study of N-substituted-phenylamino-5-methyl-1H-1,2,3-triazole-4-carbohydrazides
|
Jordão, Alessandro K. |
|
2011 |
19 |
18 |
p. 5605-5611 7 p. |
artikel |
44 |
Synthesis of benzo[3,4]azepino[1,2-b]isoquinolin-9-ones from 3-arylisoquinolines via ring closing metathesis and evaluation of topoisomerase I inhibitory activity, cytotoxicity and docking study
|
Van, Hue Thi My |
|
2011 |
19 |
18 |
p. 5311-5320 10 p. |
artikel |
45 |
Synthesis of pheophorbide-a conjugates with anticancer drugs as potential cancer diagnostic and therapeutic agents
|
You, Hyun |
|
2011 |
19 |
18 |
p. 5383-5391 9 p. |
artikel |
46 |
Synthesis, structural, and biological evaluation of bis-heteroarylmaleimides and bis-heterofused imides
|
Ferri, Nicola |
|
2011 |
19 |
18 |
p. 5291-5299 9 p. |
artikel |
47 |
The structure–activity relationship of urea derivatives as anti-tuberculosis agents
|
Brown, Joshua R. |
|
2011 |
19 |
18 |
p. 5585-5595 11 p. |
artikel |