nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Avoidance of the Ames test liability for aryl–amines via computation
|
McCarren, Patrick |
|
2011 |
19 |
10 |
p. 3173-3182 10 p. |
artikel |
2 |
Biological evaluation of novel benzisoxazole derivatives as PPARδ agonists
|
Sakuma, Shogo |
|
2011 |
19 |
10 |
p. 3255-3264 10 p. |
artikel |
3 |
Cellular zwitterionic metabolite analogs simultaneously enhance reaction rate, thermostability, salt tolerance, and substrate specificity of α-glucosidase
|
Deguchi, Eisuke |
|
2011 |
19 |
10 |
p. 3128-3134 7 p. |
artikel |
4 |
Concise site-specific synthesis of DTPA–peptide conjugates: Application to imaging probes for the chemokine receptor CXCR4
|
Masuda, Ryo |
|
2011 |
19 |
10 |
p. 3216-3220 5 p. |
artikel |
5 |
Design of small molecule inhibitors of acetyl-CoA carboxylase 1 and 2 showing reduction of hepatic malonyl-CoA levels in vivo in obese Zucker rats
|
Bengtsson, Christoffer |
|
2011 |
19 |
10 |
p. 3039-3053 15 p. |
artikel |
6 |
Design, synthesis and inhibition activity of a novel cyclic enediyne amino acid conjugates against MPtpA
|
Chandra, Koushik |
|
2011 |
19 |
10 |
p. 3274-3279 6 p. |
artikel |
7 |
Design, synthesis and pharmacological evaluation of spirocyclic σ1 receptor ligands with exocyclic amino moiety (increased distance 1)
|
Rack, Elisabeth |
|
2011 |
19 |
10 |
p. 3141-3151 11 p. |
artikel |
8 |
Development of target protein-selective degradation inducer for protein knockdown
|
Itoh, Yukihiro |
|
2011 |
19 |
10 |
p. 3229-3241 13 p. |
artikel |
9 |
Editorial board
|
|
|
2011 |
19 |
10 |
p. IFC- 1 p. |
artikel |
10 |
Efficient synthesis and chiral separation of 11C-labeled ibuprofen assisted by DMSO for imaging of in vivo behavior of the individual isomers by positron emission tomography
|
Kikuchi, Tatsuya |
|
2011 |
19 |
10 |
p. 3265-3273 9 p. |
artikel |
11 |
Graphical contents list
|
|
|
2011 |
19 |
10 |
p. 3031-3038 8 p. |
artikel |
12 |
Inhibitory potential of chemical substitutions at bioinspired sites of β-d-galactopyranose on neoglycoprotein/cell surface binding of two classes of medically relevant lectins
|
Giguère, Denis |
|
2011 |
19 |
10 |
p. 3280-3287 8 p. |
artikel |
13 |
Molecular docking studies and in vitro screening of new dihydropyridine derivatives as human MRP1 inhibitors
|
Sirisha, Kalam |
|
2011 |
19 |
10 |
p. 3249-3254 6 p. |
artikel |
14 |
New 3-, 8-disubstituted pyrazolo[5,1-c][1,2,4]benzotriazines useful for studying the interaction with the HBp-3 area (hydrogen bond point area) in the benzodiazepine site on the γ-aminobutyric acid type A (GABAA) receptor
|
Guerrini, Gabriella |
|
2011 |
19 |
10 |
p. 3074-3085 12 p. |
artikel |
15 |
Peroxisome proliferator-activated receptor agonists with phenethylphenylphthalimide skeleton derived from thalidomide-related liver X receptor antagonists: Relationship between absolute configuration and subtype selectivity
|
Motoshima, Kazunori |
|
2011 |
19 |
10 |
p. 3156-3172 17 p. |
artikel |
16 |
Preparation of allosamidin and demethylallosamidin photoaffinity probes and analysis of allosamidin-binding proteins in asthmatic mice
|
Sato, Yosuke |
|
2011 |
19 |
10 |
p. 3054-3059 6 p. |
artikel |
17 |
Protective effect of ε-viniferin on β-amyloid peptide aggregation investigated by electrospray ionization mass spectrometry
|
Richard, Tristan |
|
2011 |
19 |
10 |
p. 3152-3155 4 p. |
artikel |
18 |
Structure-based design, synthesis, and nonalcoholic steatohepatitis (NASH)-preventive effect of phenylpropanoic acid peroxisome proliferator-activated receptor (PPAR) α-selective agonists
|
Ban, Shintaro |
|
2011 |
19 |
10 |
p. 3183-3191 9 p. |
artikel |
19 |
Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies
|
Carta, Fabrizio |
|
2011 |
19 |
10 |
p. 3105-3119 15 p. |
artikel |
20 |
Synthesis and antifungal activities of natural and synthetic biflavonoids
|
Sagrera, Gabriel |
|
2011 |
19 |
10 |
p. 3060-3073 14 p. |
artikel |
21 |
Synthesis and biological evaluation of new flavonoid fatty acid esters with anti-adipogenic and enhancing glucose consumption activities
|
Zhao, Wei |
|
2011 |
19 |
10 |
p. 3192-3203 12 p. |
artikel |
22 |
Synthesis and biological evaluation of unique stereodimers of sinomenine analogues as potential inhibitors of NO production
|
Teng, Peng |
|
2011 |
19 |
10 |
p. 3096-3104 9 p. |
artikel |
23 |
Synthesis and evaluation of carbaborane derivatives of indomethacin as cyclooxygenase inhibitors
|
Scholz, Matthias |
|
2011 |
19 |
10 |
p. 3242-3248 7 p. |
artikel |
24 |
Synthesis and evaluation of 1-(1H-indol-3-yl)ethanamine derivatives as new antibacterial agents
|
Burchak, Olga N. |
|
2011 |
19 |
10 |
p. 3204-3215 12 p. |
artikel |
25 |
Synthesis and evaluation of new carbonic anhydrase inhibitors
|
Xiao, Zhonghai |
|
2011 |
19 |
10 |
p. 3221-3228 8 p. |
artikel |
26 |
Thiazole-based chalcones as potent antimicrobial agents. Synthesis and biological evaluation
|
Liaras, K. |
|
2011 |
19 |
10 |
p. 3135-3140 6 p. |
artikel |
27 |
Tryptamine derivatives as novel non-nucleosidic inhibitors against hepatitis B virus
|
Qu, Shi-Jin |
|
2011 |
19 |
10 |
p. 3120-3127 8 p. |
artikel |
28 |
Virtual screening and further development of novel ALK inhibitors
|
Okamoto, Masako |
|
2011 |
19 |
10 |
p. 3086-3095 10 p. |
artikel |