| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Abscinazole-E1, a novel chemical tool for exploring the role of ABA 8′-hydroxylase CYP707A
|
Okazaki, Mariko
|
|
2011
|
19 |
1 |
p. 406-413
8 p.
|
artikel
|
| 2 |
An efficient synthesis of γ-hydroxy-α,β-unsaturated aldehydic esters of 2-lysophosphatidylcholine
|
Choi, Jaewoo
|
|
2011
|
19 |
1 |
p. 580-587
8 p.
|
artikel
|
| 3 |
An on-bead assay for the identification of non-natural peptides targeting the Androgen Receptor–cofactor interaction
|
Göksel, Hülya
|
|
2011
|
19 |
1 |
p. 306-311
6 p.
|
artikel
|
| 4 |
A novel and efficient oxidative functionalization of lignin by layer-by-layer immobilised Horseradish peroxidase
|
Perazzini, Raffaella
|
|
2011
|
19 |
1 |
p. 440-447
8 p.
|
artikel
|
| 5 |
Antimalarials based on the dioxane scaffold of plakortin. A concise synthesis and SAR studies
|
Fattorusso, Caterina
|
|
2011
|
19 |
1 |
p. 312-320
9 p.
|
artikel
|
| 6 |
Antioxidant, anti-inflammatory and anti-hyperglycaemic activities of heterocyclic homoprostanoid derivatives
|
Manohara Reddy, S.A.
|
|
2011
|
19 |
1 |
p. 384-392
9 p.
|
artikel
|
| 7 |
Arylsulfanyl pyrazolones block mutant SOD1-G93A aggregation. Potential application for the treatment of amyotrophic lateral sclerosis
|
Chen, Tian
|
|
2011
|
19 |
1 |
p. 613-622
10 p.
|
artikel
|
| 8 |
A systematic protocol for the characterization of Hsp90 modulators
|
Matts, Robert L.
|
|
2011
|
19 |
1 |
p. 684-692
9 p.
|
artikel
|
| 9 |
Azido-iodo-N-benzyl derivatives of threo-methylphenidate (Ritalin, Concerta): Rational design, synthesis, pharmacological evaluation, and dopamine transporter photoaffinity labeling
|
Lapinsky, David J.
|
|
2011
|
19 |
1 |
p. 504-512
9 p.
|
artikel
|
| 10 |
Benzopyrazine derivatives: A novel class of growth factor receptor bound protein 7 antagonists
|
Ambaye, Nigus D.
|
|
2011
|
19 |
1 |
p. 693-701
9 p.
|
artikel
|
| 11 |
Benzothieno[3,2-b]quinolinium and 3-(phenylthio)quinolinium compounds: Synthesis and evaluation against opportunistic fungal pathogens
|
Boateng, Comfort A.
|
|
2011
|
19 |
1 |
p. 458-470
13 p.
|
artikel
|
| 12 |
Biologically active constituents from the fruiting body of Taiwanofungus camphoratus
|
Shi, Li-Shian
|
|
2011
|
19 |
1 |
p. 677-683
7 p.
|
artikel
|
| 13 |
Bioorganic & Medicinal Chemistry Reviews and Perspectives
|
|
|
2011
|
19 |
1 |
p. I-III
nvt p.
|
artikel
|
| 14 |
Cardenolides of Leptadenia madagascariensis from the Madagascar dry forest
|
Pan, Ende
|
|
2011
|
19 |
1 |
p. 422-428
7 p.
|
artikel
|
| 15 |
Cholinergic and neuroprotective drugs for the treatment of Alzheimer and neuronal vascular diseases. II. Synthesis, biological assessment, and molecular modelling of new tacrine analogues from highly substituted 2-aminopyridine-3-carbonitriles
|
Samadi, Abdelouahid
|
|
2011
|
19 |
1 |
p. 122-133
12 p.
|
artikel
|
| 16 |
Cytotoxicity and topoisomerase I/II inhibition of glycosylated 2-phenyl-indoles, 2-phenyl-benzo[b]thiophenes and 2-phenyl-benzo[b]furans
|
Shi, Wei
|
|
2011
|
19 |
1 |
p. 603-612
10 p.
|
artikel
|
| 17 |
Cytotoxicity of new polyfluorinated 1,4-naphtoquinones with diverse substituents in the quinone moiety
|
Zakharova, Ol’ga D.
|
|
2011
|
19 |
1 |
p. 256-260
5 p.
|
artikel
|
| 18 |
Cytotoxicity of δ-tocotrienols from Kielmeyera coriacea against cancer cell lines
|
de Mesquita, Mariana Laundry
|
|
2011
|
19 |
1 |
p. 623-630
8 p.
|
artikel
|
| 19 |
Design and synthesis of 3-pyridylacetamide derivatives as dipeptidyl peptidase IV (DPP-4) inhibitors targeting a bidentate interaction with Arg125
|
Miyamoto, Yasufumi
|
|
2011
|
19 |
1 |
p. 172-185
14 p.
|
artikel
|
| 20 |
Design, synthesis and antimycobacterial activities of 1-methyl-2-alkenyl-4(1H)-quinolones
|
Wube, Abraham A.
|
|
2011
|
19 |
1 |
p. 567-579
13 p.
|
artikel
|
| 21 |
Design, synthesis, and biological evaluation of N-acetyl-S-(p-chlorophenylcarbamoyl)cysteine and its analogs as a novel class of anticancer agents
|
Chen, Wei
|
|
2011
|
19 |
1 |
p. 287-294
8 p.
|
artikel
|
| 22 |
Design, synthesis, and biological evaluation of novel water-soluble N-mustards as potential anticancer agents
|
Kapuriya, Naval
|
|
2011
|
19 |
1 |
p. 471-485
15 p.
|
artikel
|
| 23 |
Design, synthesis and biological evaluation of small molecule inhibitors of CD4-gp120 binding based on virtual screening
|
LaLonde, Judith M.
|
|
2011
|
19 |
1 |
p. 91-101
11 p.
|
artikel
|
| 24 |
Design, synthesis, and testing of an 6-O-linked series of benzimidazole based inhibitors of CDK5/p25
|
Jain, Prashi
|
|
2011
|
19 |
1 |
p. 359-373
15 p.
|
artikel
|
| 25 |
DR396, an apoptotic DNase γ inhibitor, attenuates high mobility group box 1 release from apoptotic cells
|
Yamada, Yoichiro
|
|
2011
|
19 |
1 |
p. 168-171
4 p.
|
artikel
|
| 26 |
Editorial board
|
|
|
2011
|
19 |
1 |
p. IFC-
1 p.
|
artikel
|
| 27 |
Editor’s Note
|
|
|
2011
|
19 |
1 |
p. 20-
1 p.
|
artikel
|
| 28 |
Graphical contents list
|
|
|
2011
|
19 |
1 |
p. 1-19
19 p.
|
artikel
|
| 29 |
Herbal medicinal products target defined biochemical and molecular mediators of inflammatory autoimmune arthritis
|
Venkatesha, Shivaprasad H.
|
|
2011
|
19 |
1 |
p. 21-29
9 p.
|
artikel
|
| 30 |
Hypericins and thioredoxin reductase: Biochemical and docking studies disclose the molecular basis for effective inhibition by naphthodianthrones
|
Sorrentino, Francesca
|
|
2011
|
19 |
1 |
p. 631-641
11 p.
|
artikel
|
| 31 |
Identification of novel ASK1 inhibitors using virtual screening
|
Okamoto, Masako
|
|
2011
|
19 |
1 |
p. 486-489
4 p.
|
artikel
|
| 32 |
Identification of 3-phenylaminoquinolinium and 3-phenylaminopyridinium salts as new agents against opportunistic fungal pathogens
|
Mazu, Tryphon K.
|
|
2011
|
19 |
1 |
p. 524-533
10 p.
|
artikel
|
| 33 |
Identification of 3-sulfonylindazole derivatives as potent and selective 5-HT6 antagonists
|
Liu, Kevin G.
|
|
2011
|
19 |
1 |
p. 650-662
13 p.
|
artikel
|
| 34 |
3-[(Imidazolidin-2-yl)imino]indazole ligands with selectivity for the α2-adrenoceptor compared to the imidazoline I1 receptor
|
Sączewski, Franciszek
|
|
2011
|
19 |
1 |
p. 321-329
9 p.
|
artikel
|
| 35 |
Inhibition of monoamine oxidase by selected C5- and C6-substituted isatin analogues
|
Manley-King, Clarina I.
|
|
2011
|
19 |
1 |
p. 261-274
14 p.
|
artikel
|
| 36 |
Inhibition of the β-carbonic anhydrase from Streptococcus pneumoniae by inorganic anions and small molecules: Toward innovative drug design of antiinfectives?
|
Burghout, Peter
|
|
2011
|
19 |
1 |
p. 243-248
6 p.
|
artikel
|
| 37 |
Investigation of α-phenylnorstatine and α-benzylnorstatine as transition state isostere motifs in the search for new BACE-1 inhibitors
|
Wångsell, Fredrik
|
|
2011
|
19 |
1 |
p. 145-155
11 p.
|
artikel
|
| 38 |
Karavilagenin C derivatives as antimalarials
|
Ramalhete, Cátia
|
|
2011
|
19 |
1 |
p. 330-338
9 p.
|
artikel
|
| 39 |
Molecular modeling based approach, synthesis and in vitro assay to new indole inhibitors of hepatitis C NS3/4A serine protease
|
Ismail, Nasser S.M.
|
|
2011
|
19 |
1 |
p. 374-383
10 p.
|
artikel
|
| 40 |
New hydroxystilbenoid derivatives endowed with neuroprotective activity and devoid of interference with estrogen and aryl hydrocarbon receptor-mediated transcription
|
Villalonga-Barber, Carolina
|
|
2011
|
19 |
1 |
p. 339-351
13 p.
|
artikel
|
| 41 |
New imidazoline/α2-adrenoceptors affecting compounds—4(5)-(2-aminoethyl)imidazoline (dihydrohistamine) derivatives. Synthesis and receptor affinity studies
|
Treder, Adam P.
|
|
2011
|
19 |
1 |
p. 156-167
12 p.
|
artikel
|
| 42 |
NF kappa B inhibitors and antitrypanosomal metabolites from endophytic fungus Penicillium sp. isolated from Limonium tubiflorum
|
Aly, Amal H.
|
|
2011
|
19 |
1 |
p. 414-421
8 p.
|
artikel
|
| 43 |
Novel 9a,11-bridged azalides: One-pot synthesis of N′-substituted 2-imino-1,3-oxazolidines condensed to an azalide aglycone
|
Ištuk, Zorica Marušić
|
|
2011
|
19 |
1 |
p. 556-566
11 p.
|
artikel
|
| 44 |
Novel bifunctional alkylating agents, 5,10-dihydropyrrolo[1,2-b]isoquinoline derivatives, synthesis and biological activity
|
Chaniyara, Ravi
|
|
2011
|
19 |
1 |
p. 275-286
12 p.
|
artikel
|
| 45 |
Peripheral site ligand–oxime conjugates: A novel concept towards reactivation of nerve agent-inhibited human acetylcholinesterase
|
de Koning, M.C.
|
|
2011
|
19 |
1 |
p. 588-594
7 p.
|
artikel
|
| 46 |
Phosphoramidate pronucleotides of cytostatic 6-aryl-7-deazapurine ribonucleosides
|
Perlíková, Pavla
|
|
2011
|
19 |
1 |
p. 229-242
14 p.
|
artikel
|
| 47 |
Rational design and synthesis of potent aminoglycoside antibiotics against resistant bacterial strains
|
Yan, Ri-Bai
|
|
2011
|
19 |
1 |
p. 30-40
11 p.
|
artikel
|
| 48 |
Reduction of vinyl groups in naturally occurring chlorophylls-a
|
Tamiaki, Hitoshi
|
|
2011
|
19 |
1 |
p. 52-57
6 p.
|
artikel
|
| 49 |
Stoichiometry-focused 18F-labeling of alkyne-substituted oligodeoxynucleotides using azido([18F]fluoromethyl)benzenes by Cu-catalyzed Huisgen reaction
|
Kuboyama, Takeshi
|
|
2011
|
19 |
1 |
p. 249-255
7 p.
|
artikel
|
| 50 |
Superoxide-dependent reduction of free Fe3+ and release of Fe2+ from ferritin by the physiologically-occurring Cu(I)–glutathione complex
|
Aliaga, Margarita E.
|
|
2011
|
19 |
1 |
p. 534-541
8 p.
|
artikel
|
| 51 |
Synthesis and antibacterial activity study of a novel class of cationic anthraquinone analogs
|
Zhang, Jianjun
|
|
2011
|
19 |
1 |
p. 498-503
6 p.
|
artikel
|
| 52 |
Synthesis and antitrypanosomal evaluation of derivatives of N-benzyl-1,2-dihydroquinolin-6-ols: Effect of core substitutions and salt formation
|
Reid, Carolyn S.
|
|
2011
|
19 |
1 |
p. 513-523
11 p.
|
artikel
|
| 53 |
Synthesis and biological evaluation of 7-substituted-1-(3-bromophenylamino)isoquinoline-4-carbonitriles as inhibitors of myosin light chain kinase and epidermal growth factor receptor
|
Rode, Haridas B.
|
|
2011
|
19 |
1 |
p. 429-439
11 p.
|
artikel
|
| 54 |
Synthesis and characterization of oligodeoxynucleotides containing a novel tetraazabenzo[cd]azulene:naphthyridine base pair
|
Hirama, Yasuyuki
|
|
2011
|
19 |
1 |
p. 352-358
7 p.
|
artikel
|
| 55 |
Synthesis and evaluation of β-carboline derivatives as potential monoamine oxidase inhibitors
|
Reniers, J.
|
|
2011
|
19 |
1 |
p. 134-144
11 p.
|
artikel
|
| 56 |
Synthesis and evaluation of 6-[1-(2-[18F]fluoro-3-pyridyl)-5-methyl-1H-1,2,3-triazol-4-yl]quinoline for positron emission tomography imaging of the metabotropic glutamate receptor type 1 in brain
|
Fujinaga, Masayuki
|
|
2011
|
19 |
1 |
p. 102-110
9 p.
|
artikel
|
| 57 |
Synthesis and in vitro anti-hepatitis B virus activity of six-membered azanucleoside analogues
|
Wang, Dan
|
|
2011
|
19 |
1 |
p. 41-51
11 p.
|
artikel
|
| 58 |
Synthesis and pharmacological evaluation of 4-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydronaphthalenyl amines as triple reuptake inhibitors
|
Shao, Liming
|
|
2011
|
19 |
1 |
p. 663-676
14 p.
|
artikel
|
| 59 |
Synthesis and SAR study of new phenylimidazole-pyrazolo[1,5-c]quinazolines as potent phosphodiesterase 10A inhibitors
|
Asproni, Battistina
|
|
2011
|
19 |
1 |
p. 642-649
8 p.
|
artikel
|
| 60 |
Synthesis and xanthine oxidase inhibitory activity of 7-methyl-2-(phenoxymethyl)-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one derivatives
|
Sathisha, K.R.
|
|
2011
|
19 |
1 |
p. 211-220
10 p.
|
artikel
|
| 61 |
Synthesis, antiprotozoal, antimicrobial, β-hematin inhibition, cytotoxicity and methemoglobin (MetHb) formation activities of bis(8-aminoquinolines)
|
Kaur, Kirandeep
|
|
2011
|
19 |
1 |
p. 197-210
14 p.
|
artikel
|
| 62 |
Synthesis, in vitro and in vivo preliminary evaluation of anti-angiogenic properties of some pyrroloazaflavones
|
Ferlin, Maria Grazia
|
|
2011
|
19 |
1 |
p. 448-457
10 p.
|
artikel
|
| 63 |
Synthesis of a covalent gemcitabine-(carbamate)-[anti-HER2/neu] immunochemotherapeutic and its cytotoxic anti-neoplastic activity against chemotherapeutic-resistant SKBr-3 mammary carcinoma
|
Coyne, C.P.
|
|
2011
|
19 |
1 |
p. 67-76
10 p.
|
artikel
|
| 64 |
Synthesis of a-factor peptide from Saccharomyces cerevisiae and photoactive analogues via Fmoc solid phase methodology
|
Mullen, Daniel G.
|
|
2011
|
19 |
1 |
p. 490-497
8 p.
|
artikel
|
| 65 |
Synthesis of antiproliferative flavones from calycopterin, major flavonoid of Calycopteris floribunda Lamk.
|
Lewin, Guy
|
|
2011
|
19 |
1 |
p. 186-196
11 p.
|
artikel
|
| 66 |
Synthesis of novel 5-amino-thiazolo[4,5-d]pyrimidines as E. coli and S. aureus SecA inhibitors
|
Jang, Mi-Yeon
|
|
2011
|
19 |
1 |
p. 702-714
13 p.
|
artikel
|
| 67 |
Synthesis of sugar–amino acid–nucleosides as potential glycosyltransferase inhibitors
|
Vembaiyan, Kannan
|
|
2011
|
19 |
1 |
p. 58-66
9 p.
|
artikel
|
| 68 |
Synthesis of truncated analogues of the iNKT cell agonist, α-galactosyl ceramide (KRN7000), and their biological evaluation
|
Veerapen, Natacha
|
|
2011
|
19 |
1 |
p. 221-228
8 p.
|
artikel
|
| 69 |
Synthesis, pharmacological activity and structure affinity relationships of spirocyclic σ1 receptor ligands with a (2-fluoroethyl) residue in 3-position
|
Maestrup, Eva Große
|
|
2011
|
19 |
1 |
p. 393-405
13 p.
|
artikel
|
| 70 |
Synthetic biotinylated tetra β(1→5) galactofuranoside for in vitro aspergillosis diagnosis
|
Cattiaux, Laurent
|
|
2011
|
19 |
1 |
p. 547-555
9 p.
|
artikel
|
| 71 |
Synthetic conjugates of genistein affecting proliferation and mitosis of cancer cells
|
Rusin, Aleksandra
|
|
2011
|
19 |
1 |
p. 295-305
11 p.
|
artikel
|
| 72 |
Triazoloquinazolinediones as novel high affinity ligands for the benzodiazepine site of GABAA receptors
|
Nilsson, Jakob
|
|
2011
|
19 |
1 |
p. 111-121
11 p.
|
artikel
|
| 73 |
Tubulin photoaffinity labeling study with a plinabulin chemical probe possessing a biotin tag at the oxazole
|
Yamazaki, Yuri
|
|
2011
|
19 |
1 |
p. 595-602
8 p.
|
artikel
|
| 74 |
Vasorelaxant effect of flavonoids through calmodulin inhibition: Ex vivo, in vitro, and in silico approaches
|
Torres-Piedra, Mariana
|
|
2011
|
19 |
1 |
p. 542-546
5 p.
|
artikel
|
| 75 |
Virtual screening based identification of novel small-molecule inhibitors targeted to the HIV-1 capsid
|
Curreli, Francesca
|
|
2011
|
19 |
1 |
p. 77-90
14 p.
|
artikel
|
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