| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
3-(2-Aminocarbonylphenyl)propanoic acid analogs as potent and selective EP3 receptor antagonists. Part 3: Synthesis, metabolic stability, and biological evaluation of optically active analogs
|
Asada, Masaki
|
|
2010
|
18 |
9 |
p. 3212-3223
12 p.
|
artikel
|
| 2 |
A novel kavalactone derivative protects against H2O2-induced PC12 cell death via Nrf2/ARE activation
|
Tanaka, Arisa
|
|
2010
|
18 |
9 |
p. 3133-3139
7 p.
|
artikel
|
| 3 |
Antagonism of 4-substituted 1,4-dihydropyridine-3,5-dicarboxylates toward voltage-dependent L-type Ca2+ channels CaV1.3 and CaV1.2
|
Chang, Che-Chien
|
|
2010
|
18 |
9 |
p. 3147-3158
12 p.
|
artikel
|
| 4 |
Anti-microtubule ‘plinabulin’ chemical probe KPU-244-B3 labeled both α- and β-tubulin
|
Yamazaki, Yuri
|
|
2010
|
18 |
9 |
p. 3169-3174
6 p.
|
artikel
|
| 5 |
Antitumor activity and COMPARE analysis of bis-indole derivatives
|
Andreani, Aldo
|
|
2010
|
18 |
9 |
p. 3004-3011
8 p.
|
artikel
|
| 6 |
Azetidinone-isothiazolidinones: Stereoselective synthesis and antibacterial evaluation of new monocyclic beta-lactams
|
Cerić, Helena
|
|
2010
|
18 |
9 |
p. 3053-3058
6 p.
|
artikel
|
| 7 |
Design and synthesis of biotin-tagged photoaffinity probes of jasmonates
|
Gu, Min
|
|
2010
|
18 |
9 |
p. 3012-3019
8 p.
|
artikel
|
| 8 |
Design of pentapeptidic BACE1 inhibitors with carboxylic acid bioisosteres at P 1 ′ and P4 positions
|
Tagad, Harichandra D.
|
|
2010
|
18 |
9 |
p. 3175-3186
12 p.
|
artikel
|
| 9 |
Design of potential reverse transcriptase inhibitor containing Isatin nucleus using molecular modeling studies
|
Pawar, Vidya
|
|
2010
|
18 |
9 |
p. 3198-3211
14 p.
|
artikel
|
| 10 |
Design, synthesis, biological evaluation and computational investigation of novel inhibitors of dihydrofolate reductase of opportunistic pathogens
|
Bag, Seema
|
|
2010
|
18 |
9 |
p. 3187-3197
11 p.
|
artikel
|
| 11 |
3,5-Diaryl-1H-pyrazole as a molecular scaffold for the synthesis of apoptosis-inducing agents
|
Shaw, Arthur Y.
|
|
2010
|
18 |
9 |
p. 3270-3278
9 p.
|
artikel
|
| 12 |
DNA strand cleaving properties and hypoxia-selective cytotoxicity of 7-chloro-2-thienylcarbonyl-3-trifluoromethylquinoxaline 1,4-dioxide
|
Junnotula, Venkatraman
|
|
2010
|
18 |
9 |
p. 3125-3132
8 p.
|
artikel
|
| 13 |
Dodecaborate lipid liposomes as new vehicles for boron delivery system of neutron capture therapy
|
Ueno, Manabu
|
|
2010
|
18 |
9 |
p. 3059-3065
7 p.
|
artikel
|
| 14 |
Editorial board
|
|
|
2010
|
18 |
9 |
p. IFC-
1 p.
|
artikel
|
| 15 |
Elaborate ligand-based pharmacophore exploration and QSAR analysis guide the synthesis of novel pyridinium-based potent β-secretase inhibitory leads
|
Al-Nadaf, Afaf
|
|
2010
|
18 |
9 |
p. 3088-3115
28 p.
|
artikel
|
| 16 |
Graphical contents list
|
|
|
2010
|
18 |
9 |
p. 2987-2996
10 p.
|
artikel
|
| 17 |
Identification of serotonin 5-HT1A receptor partial agonists in ginger
|
Nievergelt, Andreas
|
|
2010
|
18 |
9 |
p. 3345-3351
7 p.
|
artikel
|
| 18 |
In silico directed chemical probing of the adenosine receptor family
|
Areias, Filipe M.
|
|
2010
|
18 |
9 |
p. 3043-3052
10 p.
|
artikel
|
| 19 |
In vitro TRPV1 activity of piperine derived amides
|
Correa, Edwin Andrés
|
|
2010
|
18 |
9 |
p. 3299-3306
8 p.
|
artikel
|
| 20 |
Novel 2-[(benzylamino)methyl]pyrrolidine-3,4-diol derivatives as α-mannosidase inhibitors and with antitumor activities against hematological and solid malignancies
|
Bello, Claudia
|
|
2010
|
18 |
9 |
p. 3320-3334
15 p.
|
artikel
|
| 21 |
Novel DNA intercalators without basic side chains as efficient antitumor agents: Design, synthesis and evaluation of benzo-[c,d]-indol-malononitrile derivatives
|
Li, Xiaolian
|
|
2010
|
18 |
9 |
p. 3279-3284
6 p.
|
artikel
|
| 22 |
Phosphate ester derivatives of homocamptothecin: Synthesis, solution stabilities and antitumor activities
|
Miao, Zhenyuan
|
|
2010
|
18 |
9 |
p. 3140-3146
7 p.
|
artikel
|
| 23 |
Prenylated pterocarpans as bacterial neuraminidase inhibitors
|
Nguyen, Phi Hung
|
|
2010
|
18 |
9 |
p. 3335-3344
10 p.
|
artikel
|
| 24 |
Publisher’s Note
|
|
|
2010
|
18 |
9 |
p. 2997-
1 p.
|
artikel
|
| 25 |
Structure–activity relationships in a novel series of 7-substituted-aryl quinolines and 5-substituted-aryl benzothiazoles at the metabotropic glutamate receptor subtype 5
|
Zhang, Peng
|
|
2010
|
18 |
9 |
p. 3026-3035
10 p.
|
artikel
|
| 26 |
Structure–activity relationships in the conversion of vitamin K analogues into menaquinone-4. Substrates essential to the synthesis of menaquinone-4 in cultured human cell lines
|
Suhara, Yoshitomo
|
|
2010
|
18 |
9 |
p. 3116-3124
9 p.
|
artikel
|
| 27 |
Structure–activity relationships of bioisosteric replacement of the carboxylic acid in novel androgen receptor pure antagonists
|
Yoshino, Hitoshi
|
|
2010
|
18 |
9 |
p. 3159-3168
10 p.
|
artikel
|
| 28 |
Sugar-based peptidomimetics as potential inhibitors of the vascular endothelium growth factor binding to neuropilin-1
|
Novoa, Alexandre
|
|
2010
|
18 |
9 |
p. 3285-3298
14 p.
|
artikel
|
| 29 |
Synthesis and biological activity of cyclotetrapeptide analogues of the natural HDAC inhibitor FR235222
|
Terracciano, Stefania
|
|
2010
|
18 |
9 |
p. 3252-3260
9 p.
|
artikel
|
| 30 |
Synthesis and biological evaluation of isoflavone fatty acid esters with potential weight loss and hypolipidemic activities
|
Xiang, Hua
|
|
2010
|
18 |
9 |
p. 3036-3042
7 p.
|
artikel
|
| 31 |
Synthesis and biological evaluation of novel C5 halogen-functionalized S-DABO as potent HIV-1 non-nucleoside reverse transcriptase inhibitors
|
Qin, Hua
|
|
2010
|
18 |
9 |
p. 3231-3237
7 p.
|
artikel
|
| 32 |
Synthesis and evaluation of new N 6-substituted adenosine-5′-N-methylcarboxamides as A3 adenosine receptor agonists
|
Devine, Shane M.
|
|
2010
|
18 |
9 |
p. 3078-3087
10 p.
|
artikel
|
| 33 |
Synthesis, characterization and vasculoprotective effects of nitric oxide-donating derivatives of chrysin
|
Zou, Xiao-Qing
|
|
2010
|
18 |
9 |
p. 3020-3025
6 p.
|
artikel
|
| 34 |
Synthesis, topoisomerase I and II inhibitory activity, cytotoxicity, and structure–activity relationship study of hydroxylated 2,4-diphenyl-6-aryl pyridines
|
Karki, Radha
|
|
2010
|
18 |
9 |
p. 3066-3077
12 p.
|
artikel
|
| 35 |
The anti-cancer, anti-inflammatory and tuberculostatic activities of a series of 6,7-substituted-5,8-quinolinequinones
|
Mulchin, Benjamin J.
|
|
2010
|
18 |
9 |
p. 3238-3251
14 p.
|
artikel
|
| 36 |
The bisnaphthalimides as new active lead compounds against Plasmodium falciparum
|
Tischer, Maximilian
|
|
2010
|
18 |
9 |
p. 2998-3003
6 p.
|
artikel
|
| 37 |
The evaluation of quinonoid compounds against Trypanosoma cruzi: Synthesis of imidazolic anthraquinones, nor-β-lapachone derivatives and β-lapachone-based 1,2,3-triazoles
|
da Silva Júnior, Eufrânio N.
|
|
2010
|
18 |
9 |
p. 3224-3230
7 p.
|
artikel
|
| 38 |
Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: Structure-based drug design, synthesis, and biological evaluation
|
Vernier, William
|
|
2010
|
18 |
9 |
p. 3307-3319
13 p.
|
artikel
|
| 39 |
3′-(1,2,3-Triazol-1-yl)-3′-deoxythymidine analogs as substrates for human and Ureaplasma parvum thymidine kinase for structure–activity investigations
|
Lin, Jay
|
|
2010
|
18 |
9 |
p. 3261-3269
9 p.
|
artikel
|
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