| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Antiproliferative activity of synthetic naphthoquinones related to lapachol. First synthesis of 5-hydroxylapachol
|
Bonifazi, Evelyn L.
|
|
2010
|
18 |
7 |
p. 2621-2630
10 p.
|
artikel
|
| 2 |
Application of the phosphoramidate ProTide approach to the antiviral drug ribavirin
|
Derudas, Marco
|
|
2010
|
18 |
7 |
p. 2748-2755
8 p.
|
artikel
|
| 3 |
Assessing the trypanocidal potential of natural and semi-synthetic diketopiperazines from two deep water marine-derived fungi
|
Watts, Katharine R.
|
|
2010
|
18 |
7 |
p. 2566-2574
9 p.
|
artikel
|
| 4 |
Bioconjugates of curcumin display improved protection against glutathione depletion mediated oxidative stress in a dopaminergic neuronal cell line: Implications for Parkinson’s disease
|
Harish, G.
|
|
2010
|
18 |
7 |
p. 2631-2638
8 p.
|
artikel
|
| 5 |
Chromene-3-carboxamide derivatives discovered from virtual screening as potent inhibitors of the tumour maker, AKR1B10
|
Endo, Satoshi
|
|
2010
|
18 |
7 |
p. 2485-2490
6 p.
|
artikel
|
| 6 |
‘Click chemistry’ synthesis of a library of 1,2,3-triazole-substituted galactose derivatives and their evaluation against Trypanosoma cruzi and its cell surface trans-sialidase
|
Carvalho, Ivone
|
|
2010
|
18 |
7 |
p. 2412-2427
16 p.
|
artikel
|
| 7 |
Conjugates of plumbagin and phenyl-2-amino-1-thioglucoside inhibit MshB, a deacetylase involved in the biosynthesis of mycothiol
|
Gammon, David W.
|
|
2010
|
18 |
7 |
p. 2501-2514
14 p.
|
artikel
|
| 8 |
Cu(II) cyclen cleavage agent for human islet amyloid peptide
|
Jeong, Keunhong
|
|
2010
|
18 |
7 |
p. 2598-2601
4 p.
|
artikel
|
| 9 |
Derivatives of schisandrin with increased inhibitory potential on prostaglandin E2 and leukotriene B4 formation in vitro
|
Blunder, Martina
|
|
2010
|
18 |
7 |
p. 2809-2815
7 p.
|
artikel
|
| 10 |
Design, synthesis and antimalarial/anticancer evaluation of spermidine linked artemisinin conjugates designed to exploit polyamine transporters in Plasmodium falciparum and HL-60 cancer cell lines
|
Chadwick, James
|
|
2010
|
18 |
7 |
p. 2586-2597
12 p.
|
artikel
|
| 11 |
Design, synthesis and evaluation of novel 2-thiophen-5-yl-3H-quinazolin-4-one analogues as inhibitors of transcription factors NF-кB and AP-1 mediated transcriptional activation: Their possible utilization as anti-inflammatory and anti-cancer agents
|
Giri, Rajan S.
|
|
2010
|
18 |
7 |
p. 2796-2808
13 p.
|
artikel
|
| 12 |
Discovery of inhibitors of brassinin oxidase based on the scaffolds of the phytoalexins brassilexin and wasalexin
|
Pedras, M. Soledade C.
|
|
2010
|
18 |
7 |
p. 2456-2463
8 p.
|
artikel
|
| 13 |
Editorial board
|
|
|
2010
|
18 |
7 |
p. IFC-
1 p.
|
artikel
|
| 14 |
Enhancement of antiproliferative activity by molecular simplification of catalpol
|
García, Celina
|
|
2010
|
18 |
7 |
p. 2515-2523
9 p.
|
artikel
|
| 15 |
Evaluation of retro-inverso modifications of HTLV-1 protease inhibitors containing a hydroxyethylamine isoster
|
Tatsumi, Tadashi
|
|
2010
|
18 |
7 |
p. 2720-2727
8 p.
|
artikel
|
| 16 |
18F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging
|
Zhang, Shuting
|
|
2010
|
18 |
7 |
p. 2394-2401
8 p.
|
artikel
|
| 17 |
Graphical contents list
|
|
|
2010
|
18 |
7 |
p. 2357-2369
13 p.
|
artikel
|
| 18 |
Inhibition of Escherichia coli glycosyltransferase MurG and Mycobacterium tuberculosis Gal transferase by uridine-linked transition state mimics
|
Trunkfield, Amy E.
|
|
2010
|
18 |
7 |
p. 2651-2663
13 p.
|
artikel
|
| 19 |
Investigating the anti-proliferative activity of styrylazanaphthalenes and azanaphthalenediones
|
Mrozek-Wilczkiewicz, Anna
|
|
2010
|
18 |
7 |
p. 2664-2671
8 p.
|
artikel
|
| 20 |
Isolation, structure and biological activities of platencin A2–A4 from Streptomyces platensis
|
Zhang, Chaowei
|
|
2010
|
18 |
7 |
p. 2602-2610
9 p.
|
artikel
|
| 21 |
New 3-methylquinoxaline-2-carboxamide 1,4-di-N-oxide derivatives as anti-Mycobacterium tuberculosis agents
|
Ancizu, Saioa
|
|
2010
|
18 |
7 |
p. 2713-2719
7 p.
|
artikel
|
| 22 |
Novel acyl coenzyme A (CoA): Diacylglycerol acyltransferase-1 inhibitors: Synthesis and biological activities of diacylethylenediamine derivatives
|
Nakada, Yoshihisa
|
|
2010
|
18 |
7 |
p. 2785-2795
11 p.
|
artikel
|
| 23 |
Novel azalides derived from 16-membered macrolides. III. Azalides modified at the C-15 and 4″ positions: Improved antibacterial activities
|
Miura, Tomoaki
|
|
2010
|
18 |
7 |
p. 2735-2747
13 p.
|
artikel
|
| 24 |
Novel DNA–peptide interaction networks
|
Huang, Jonathan T.B.
|
|
2010
|
18 |
7 |
p. 2575-2585
11 p.
|
artikel
|
| 25 |
Novel 8-(furan-2-yl)-3-substituted thiazolo [5,4-e][1,2,4] triazolo[1,5-c] pyrimidine-2(3H)-thione derivatives as potential adenosine A2A receptor antagonists
|
Mishra, Chandra Bhushan
|
|
2010
|
18 |
7 |
p. 2491-2500
10 p.
|
artikel
|
| 26 |
Phosphoramidates of 2′-β-d-arabinouridine (AraU) as phosphate prodrugs; design, synthesis, in vitro activity and metabolism
|
Mehellou, Youcef
|
|
2010
|
18 |
7 |
p. 2439-2446
8 p.
|
artikel
|
| 27 |
Polysubstituted pyrazoles, part 6. Synthesis of some 1-(4-chlorophenyl)-4-hydroxy-1H-pyrazol-3-carbonyl derivatives linked to nitrogenous heterocyclic ring systems as potential antitumor agents
|
Rostom, Sherif A.F.
|
|
2010
|
18 |
7 |
p. 2767-2776
10 p.
|
artikel
|
| 28 |
Preparation and in vitro photodynamic activity of amphiphilic zinc(II) phthalocyanines substituted with 2-(dimethylamino)ethylthio moieties and their N-alkylated derivatives
|
Duan, Wubiao
|
|
2010
|
18 |
7 |
p. 2672-2677
6 p.
|
artikel
|
| 29 |
Pyrazolone-fused combretastatins and their precursors: synthesis, cytotoxicity, antitubulin activity and molecular modeling studies
|
Burja, Bojan
|
|
2010
|
18 |
7 |
p. 2375-2387
13 p.
|
artikel
|
| 30 |
Regioselective one-pot synthesis and anti-proliferative and apoptotic effects of some novel tetrazolo[1,5-a]pyrimidine derivatives
|
Hussein, Ahmed M.
|
|
2010
|
18 |
7 |
p. 2639-2644
6 p.
|
artikel
|
| 31 |
Statistical molecular design of a focused salicylidene acylhydrazide library and multivariate QSAR of inhibition of type III secretion in the Gram-negative bacterium Yersinia
|
Dahlgren, Markus K.
|
|
2010
|
18 |
7 |
p. 2686-2703
18 p.
|
artikel
|
| 32 |
Structural development studies of anti-hepatitis C virus agents with a phenanthridinone skeleton
|
Nakamura, Masahiko
|
|
2010
|
18 |
7 |
p. 2402-2411
10 p.
|
artikel
|
| 33 |
Structure–activity relationship of novel DAPK inhibitors identified by structure-based virtual screening
|
Okamoto, Masako
|
|
2010
|
18 |
7 |
p. 2728-2734
7 p.
|
artikel
|
| 34 |
Synthesis and antibacterial studies of binaphthyl-based tripeptoids. Part 1
|
Bremner, John B.
|
|
2010
|
18 |
7 |
p. 2611-2620
10 p.
|
artikel
|
| 35 |
Synthesis and anticancer activity evaluation of 2(4-alkoxyphenyl)cyclopropyl hydrazides and triazolo phthalazines
|
De, Prithwiraj
|
|
2010
|
18 |
7 |
p. 2537-2548
12 p.
|
artikel
|
| 36 |
Synthesis and biological evaluation of antitumor-active γ-butyrolactone substituted betulin derivatives
|
Csuk, René
|
|
2010
|
18 |
7 |
p. 2549-2558
10 p.
|
artikel
|
| 37 |
Synthesis and biological evaluation of 4-(hydroxyimino)arylmethyl diarylpyrimidine analogues as potential non-nucleoside reverse transcriptase inhibitors against HIV
|
Feng, Xiao-Qing
|
|
2010
|
18 |
7 |
p. 2370-2374
5 p.
|
artikel
|
| 38 |
Synthesis and evaluation of novel benzothiazole derivatives based on the bithiophene structure as potential radiotracers for β-amyloid plaques in Alzheimer’s disease
|
Cui, Meng-Chao
|
|
2010
|
18 |
7 |
p. 2777-2784
8 p.
|
artikel
|
| 39 |
Synthesis and pharmacological characterization of a new series of 5,7-disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazine derivatives as adenosine receptor antagonists: A preliminary inspection of ligand–receptor recognition process
|
Pastorin, Giorgia
|
|
2010
|
18 |
7 |
p. 2524-2536
13 p.
|
artikel
|
| 40 |
Synthesis and preliminary pharmacological characterisation of a new class of nitrogen-containing bisphosphonates (N-BPs)
|
Lolli, Marco L.
|
|
2010
|
18 |
7 |
p. 2428-2438
11 p.
|
artikel
|
| 41 |
Synthesis and structure–activity relationships of antimalarial 4-oxo-3-carboxyl quinolones
|
Zhang, Yiqun
|
|
2010
|
18 |
7 |
p. 2756-2766
11 p.
|
artikel
|
| 42 |
Synthesis, molecular modeling and biological evaluation of PSB as targeted antibiotics
|
Cheng, Kui
|
|
2010
|
18 |
7 |
p. 2447-2455
9 p.
|
artikel
|
| 43 |
Synthesis of 26-hydroxy-22-oxocholestanic frameworks from diosgenin and hecogenin and their in vitro antiproliferative and apoptotic activity on human cervical cancer CaSki cells
|
Fernández-Herrera, María A.
|
|
2010
|
18 |
7 |
p. 2474-2484
11 p.
|
artikel
|
| 44 |
Synthesis of mono-carbonyl analogues of curcumin and their effects on inhibition of cytokine release in LPS-stimulated RAW 264.7 macrophages
|
Zhao, Chengguang
|
|
2010
|
18 |
7 |
p. 2388-2393
6 p.
|
artikel
|
| 45 |
Synthesis of new β-1-C-alkylated imino-l-iditols: A comparative study of their activity as β-glucocerebrosidase inhibitors
|
Schönemann, Wojciech
|
|
2010
|
18 |
7 |
p. 2645-2650
6 p.
|
artikel
|
| 46 |
Synthesis, X-ray crystal structure study and antitumoral evaluations of 5,6-disubstituted pyrimidine derivatives
|
Kraljević, Tatjana Gazivoda
|
|
2010
|
18 |
7 |
p. 2704-2712
9 p.
|
artikel
|
| 47 |
Total synthesis, antiprotozoal and cytotoxicity activities of rhuschalcone VI and analogs
|
Mihigo, Shetonde O.
|
|
2010
|
18 |
7 |
p. 2464-2473
10 p.
|
artikel
|
| 48 |
Water-soluble polymer–drug conjugates for combination chemotherapy against visceral leishmaniasis
|
Nicoletti, Salvatore
|
|
2010
|
18 |
7 |
p. 2559-2565
7 p.
|
artikel
|
| 49 |
Zinc(II) complexes of the second-generation quinolone antibacterial drug enrofloxacin: Structure and DNA or albumin interaction
|
Tarushi, Alketa
|
|
2010
|
18 |
7 |
p. 2678-2685
8 p.
|
artikel
|
Tijdschrift beschrijving