| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
3-(2-Aminocarbonylphenyl)propanoic acid analogs as potent and selective EP3 receptor antagonists. Part 2: Optimization of the side chains to improve in vitro and in vivo potencies
|
Asada, Masaki
|
|
2010
|
18 |
4 |
p. 1641-1658
18 p.
|
artikel
|
| 2 |
Antimalarial and antitubercular nostocarboline and eudistomin derivatives: Synthesis, in vitro and in vivo biological evaluation
|
Bonazzi, Simone
|
|
2010
|
18 |
4 |
p. 1464-1476
13 p.
|
artikel
|
| 3 |
2-Arylthiomorpholine derivatives as potent and selective monoamine oxidase B inhibitors
|
Lühr, Susan
|
|
2010
|
18 |
4 |
p. 1388-1395
8 p.
|
artikel
|
| 4 |
Binding of curcumin and its long chain derivatives to the activator binding domain of novel protein kinase C
|
Majhi, Anjoy
|
|
2010
|
18 |
4 |
p. 1591-1598
8 p.
|
artikel
|
| 5 |
Bioorganic & Medicinal Chemistry Reviews and Perspectives
|
|
|
2010
|
18 |
4 |
p. 1736-1738
3 p.
|
artikel
|
| 6 |
CoMFA analysis of tgDHFR and rlDHFR based on antifolates with 6–5 fused ring system using the all-orientation search (AOS) routine and a modified cross-validated r2-guided region selection (q2-GRS) routine and its initial application
|
Gangjee, Aleem
|
|
2010
|
18 |
4 |
p. 1684-1701
18 p.
|
artikel
|
| 7 |
Design and synthesis of anti-breast cancer agents from 4-piperazinylquinoline: A hybrid pharmacophore approach
|
Solomon, V. Raja
|
|
2010
|
18 |
4 |
p. 1563-1572
10 p.
|
artikel
|
| 8 |
Design of novel nicotinamides as potent and selective monoamine oxidase a inhibitors
|
Shi, Lei
|
|
2010
|
18 |
4 |
p. 1659-1664
6 p.
|
artikel
|
| 9 |
Developing a complete pharmacology for AMPA receptors: A perspective on subtype-selective ligands
|
Fleming, James J.
|
|
2010
|
18 |
4 |
p. 1381-1387
7 p.
|
artikel
|
| 10 |
Diamination by N-coupling using a commercial laccase
|
Wellington, Kevin W.
|
|
2010
|
18 |
4 |
p. 1406-1414
9 p.
|
artikel
|
| 11 |
2,3-Diamino acid modifying 3S-tetrahydroisoquinoline-3-carboxylic acids: Leading to a class of novel agents with highly unfolded conformation, selective in vitro anti-platelet aggregation and potent in vivo anti-thrombotic activity
|
Zhang, Xiaoyi
|
|
2010
|
18 |
4 |
p. 1536-1554
19 p.
|
artikel
|
| 12 |
Discovery of potent BACE-1 inhibitors containing a new hydroxyethylene (HE) Scaffold: Exploration of P1′ alkoxy residues and an aminoethylene (AE) central core
|
Björklund, Catarina
|
|
2010
|
18 |
4 |
p. 1711-1723
13 p.
|
artikel
|
| 13 |
Editorial board
|
|
|
2010
|
18 |
4 |
p. IFC-
1 p.
|
artikel
|
| 14 |
Evaluation of 3,4-dihydroquinazoline-2(1H)-thiones as inhibitors of α-MSH-induced melanin production in melanoma B16 cells
|
Thanigaimalai, P.
|
|
2010
|
18 |
4 |
p. 1555-1562
8 p.
|
artikel
|
| 15 |
Graphical contents list
|
|
|
2010
|
18 |
4 |
p. 1371-1380
10 p.
|
artikel
|
| 16 |
11β-Hydroxysteroid dehydrogenase 1 inhibiting constituents from Eriobotrya japonica revealed by bioactivity-guided isolation and computational approaches
|
Rollinger, Judith M.
|
|
2010
|
18 |
4 |
p. 1507-1515
9 p.
|
artikel
|
| 17 |
Interaction between double helix DNA fragments and the new antitumor agent sabarubicin, Men10755
|
Mazzini, Stefania
|
|
2010
|
18 |
4 |
p. 1497-1506
10 p.
|
artikel
|
| 18 |
Interaction between ghrelin and the ghrelin receptor (GHS-R1a), a NMR study using living cells
|
Martín-Pastor, Manuel
|
|
2010
|
18 |
4 |
p. 1583-1590
8 p.
|
artikel
|
| 19 |
Mitochondrial biotransformation of ω-(phenoxy)alkanoic acids, 3-(phenoxy)acrylic acids, and ω-(1-methyl-1H-imidazol-2-ylthio)alkanoic acids: A prodrug strategy for targeting cytoprotective antioxidants to mitochondria
|
Roser, Kurt S.
|
|
2010
|
18 |
4 |
p. 1441-1448
8 p.
|
artikel
|
| 20 |
New pterocarpanquinones: Synthesis, antineoplasic activity on cultured human malignant cell lines and TNF-α modulation in human PBMC cells
|
Netto, Chaquip D.
|
|
2010
|
18 |
4 |
p. 1610-1616
7 p.
|
artikel
|
| 21 |
Novel 1,3-dihydro-benzimidazol-2-ones and their analogues as potent non-nucleoside HIV-1 reverse transcriptase inhibitors
|
Monforte, Anna-Maria
|
|
2010
|
18 |
4 |
p. 1702-1710
9 p.
|
artikel
|
| 22 |
Novel matrix metalloproteinase inhibitors derived from quinoxalinone scaffold (Part I)
|
Li, Yonggang
|
|
2010
|
18 |
4 |
p. 1516-1525
10 p.
|
artikel
|
| 23 |
Potent inhibitor scaffold against Trypanosoma cruzi trans-sialidase
|
Arioka, Shingo
|
|
2010
|
18 |
4 |
p. 1633-1640
8 p.
|
artikel
|
| 24 |
Quinolinotriazole-β-cyclodextrin and its adamantanecarboxylic acid complex as efficient water-soluble fluorescent Cd2+ sensors
|
Zhang, Ying-Ming
|
|
2010
|
18 |
4 |
p. 1415-1420
6 p.
|
artikel
|
| 25 |
RETRACTED: Carboxylated calixarenes bind strongly to CD69 and protect CD69+ killer cells from suicidal cell death induced by tumor cell surface ligands
|
Bezouška, Karel
|
|
2010
|
18 |
4 |
p. 1434-1440
7 p.
|
artikel
|
| 26 |
Stereoselective synthesis of desloratadine derivatives as antagonist of histamine
|
Liu, Gai-Zhi
|
|
2010
|
18 |
4 |
p. 1626-1632
7 p.
|
artikel
|
| 27 |
Structural analogues of schweinfurthin F: Probing the steric, electronic, and hydrophobic properties of the D-ring substructure
|
Ulrich, Natalie C.
|
|
2010
|
18 |
4 |
p. 1676-1683
8 p.
|
artikel
|
| 28 |
Structural basis for selective inhibition of purine nucleoside phosphorylase from Schistosoma mansoni: Kinetic and structural studies
|
Castilho, Marcelo S.
|
|
2010
|
18 |
4 |
p. 1421-1427
7 p.
|
artikel
|
| 29 |
Synthesis and anti-influenza virus activity of dihydrofuran-fused perhydrophenanthrenes with a benzyloxy-type side-chain
|
Matsuya, Yuji
|
|
2010
|
18 |
4 |
p. 1477-1481
5 p.
|
artikel
|
| 30 |
Synthesis and anti-leishmanial activity of heterocyclic betulin derivatives
|
Alakurtti, Sami
|
|
2010
|
18 |
4 |
p. 1573-1582
10 p.
|
artikel
|
| 31 |
Synthesis and biological evaluation of (phenylpiperazinyl-propyl)arylsulfonamides as selective 5-HT2A receptor antagonists
|
Yoo, Euna
|
|
2010
|
18 |
4 |
p. 1665-1675
11 p.
|
artikel
|
| 32 |
Synthesis and cancer cell cytotoxicity of substituted xanthenes
|
Giri, Rajan
|
|
2010
|
18 |
4 |
p. 1456-1463
8 p.
|
artikel
|
| 33 |
Synthesis and carbohydrate binding studies of fluorescent α-amidoboronic acids and the corresponding bisboronic acids
|
Jin, Shan
|
|
2010
|
18 |
4 |
p. 1449-1455
7 p.
|
artikel
|
| 34 |
Synthesis and induction of apoptosis signaling pathway of ent-kaurane derivatives
|
Hueso-Falcón, Idaira
|
|
2010
|
18 |
4 |
p. 1724-1735
12 p.
|
artikel
|
| 35 |
Synthesis and SAR of thiazolidinedione derivatives as 15-PGDH inhibitors
|
Wu, Ying
|
|
2010
|
18 |
4 |
p. 1428-1433
6 p.
|
artikel
|
| 36 |
Synthesis, characterization, and in vitro and in vivo evaluation of a novel pectin–adriamycin conjugate
|
Tang, Xiao-Hai
|
|
2010
|
18 |
4 |
p. 1599-1609
11 p.
|
artikel
|
| 37 |
Synthesis of novel aminoglycosides via allylic azide rearrangement for investigating the significance of 2′-amino group
|
Zhang, Jianjun
|
|
2010
|
18 |
4 |
p. 1396-1405
10 p.
|
artikel
|
| 38 |
Synthesis, photophysical properties and photocytotoxicity of mono-, di-, tri- and tetra-glucosylated fluorophenylporphyrins
|
Hirohara, Shiho
|
|
2010
|
18 |
4 |
p. 1526-1535
10 p.
|
artikel
|
| 39 |
Synthesis, structure–activity relationship and crystallographic studies of 3-substituted indolin-2-one RET inhibitors
|
Mologni, Luca
|
|
2010
|
18 |
4 |
p. 1482-1496
15 p.
|
artikel
|
| 40 |
The first low μM SecA inhibitors
|
Chen, Weixuan
|
|
2010
|
18 |
4 |
p. 1617-1625
9 p.
|
artikel
|
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