nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors
|
Chimenti, Franco |
|
2010 |
18 |
3 |
p. 1273-1279 7 p. |
artikel |
2 |
4-Aryl-4-oxo-N-phenyl-2-aminylbutyramides as acetyl- and butyrylcholinesterase inhibitors. Preparation, anticholinesterase activity, docking study, and 3D structure–activity relationship based on molecular interaction fields
|
Vitorović-Todorović, Maja D. |
|
2010 |
18 |
3 |
p. 1181-1193 13 p. |
artikel |
3 |
Carbonic anhydrase activators: Activation of the β-carbonic anhydrases from the pathogenic fungi Candida albicans and Cryptococcus neoformans with amines and amino acids
|
Innocenti, Alessio |
|
2010 |
18 |
3 |
p. 1034-1037 4 p. |
artikel |
4 |
Cationic N-confused porphyrin derivative as a better molecule scaffold for G-quadruplex recognition
|
Du, Yuhao |
|
2010 |
18 |
3 |
p. 1111-1116 6 p. |
artikel |
5 |
Chemo-enzymatic synthesis of glycosylated insulin using a GlcNAc tag
|
Tomabechi, Yusuke |
|
2010 |
18 |
3 |
p. 1259-1264 6 p. |
artikel |
6 |
Comparative analysis of DNA alkylation by conjugates between pyrrole–imidazole hairpin polyamides and chlorambucil or seco-CBI
|
Minoshima, Masafumi |
|
2010 |
18 |
3 |
p. 1236-1243 8 p. |
artikel |
7 |
Design, synthesis and biological evaluation of chrysin long-chain derivatives as potential anticancer agents
|
Lv, Peng-Cheng |
|
2010 |
18 |
3 |
p. 1117-1123 7 p. |
artikel |
8 |
Design, synthesis and biological evaluation of new 2,3-diarylquinoline derivatives as selective cyclooxygenase-2 inhibitors
|
Ghodsi, Razieh |
|
2010 |
18 |
3 |
p. 1029-1033 5 p. |
artikel |
9 |
Design, synthesis, and biological evaluation of novel estradiol–bisphosphonate conjugates as bone-specific estrogens
|
Morioka, Masahiko |
|
2010 |
18 |
3 |
p. 1143-1148 6 p. |
artikel |
10 |
Design, synthesis and in vitro characterization of Glucagon-Like Peptide-1 derivatives for pancreatic beta cell imaging by SPECT
|
Behnam Azad, Babak |
|
2010 |
18 |
3 |
p. 1265-1272 8 p. |
artikel |
11 |
Design, synthesis and SAR analysis of novel selective σ1 ligands (Part 2)
|
Rossi, Daniela |
|
2010 |
18 |
3 |
p. 1204-1212 9 p. |
artikel |
12 |
Editorial board
|
|
|
2010 |
18 |
3 |
p. IFC- 1 p. |
artikel |
13 |
From anti-fouling to biofilm inhibition: New cytotoxic secondary metabolites from two Indonesian Agelas sponges
|
Hertiani, Triana |
|
2010 |
18 |
3 |
p. 1297-1311 15 p. |
artikel |
14 |
Ganodermasides A and B, two novel anti-aging ergosterols from spores of a medicinal mushroom Ganoderma lucidum on yeast via UTH1 gene
|
Weng, Yufang |
|
2010 |
18 |
3 |
p. 999-1002 4 p. |
artikel |
15 |
Graphical contents list
|
|
|
2010 |
18 |
3 |
p. 987-998 12 p. |
artikel |
16 |
Improved synthesis of a fluorogenic ceramidase substrate
|
Xia, Zuping |
|
2010 |
18 |
3 |
p. 1003-1009 7 p. |
artikel |
17 |
Inhibition of monoamine oxidase by 8-benzyloxycaffeine analogues
|
Strydom, Belinda |
|
2010 |
18 |
3 |
p. 1018-1028 11 p. |
artikel |
18 |
Inhibitory effect of novel tetrahydropyrimidine-2(1H)-thiones on melanogenesis
|
Thanigaimalai, P. |
|
2010 |
18 |
3 |
p. 1135-1142 8 p. |
artikel |
19 |
Isosorbide-based cholinesterase inhibitors; replacement of 5-ester groups leading to increased stability
|
Dillon, Gerald P. |
|
2010 |
18 |
3 |
p. 1045-1053 9 p. |
artikel |
20 |
Mevalonate analogues as substrates of enzymes in the isoprenoid biosynthetic pathway of Streptococcus pneumoniae
|
Kudoh, Takashi |
|
2010 |
18 |
3 |
p. 1124-1134 11 p. |
artikel |
21 |
β-Naphthoflavone analogs as potent and soluble aryl hydrocarbon receptor agonists: Improvement of solubility by disruption of molecular planarity
|
Fujita, Yuji |
|
2010 |
18 |
3 |
p. 1194-1203 10 p. |
artikel |
22 |
New benzoxanthone derivatives as topoisomerase inhibitors and DNA cross-linkers
|
Cho, Hee-Ju |
|
2010 |
18 |
3 |
p. 1010-1017 8 p. |
artikel |
23 |
Novel amidino substituted 2-phenylbenzothiazoles: Synthesis, antitumor evaluation in vitro and acute toxicity testing in vivo
|
Racané, Livio |
|
2010 |
18 |
3 |
p. 1038-1044 7 p. |
artikel |
24 |
Novel anilinophthalimide derivatives as potential probes for β-amyloid plaque in the brain
|
Duan, Xin-Hong |
|
2010 |
18 |
3 |
p. 1337-1343 7 p. |
artikel |
25 |
Novel 4,4′-diether-2,2′-bipyridine cisplatin analogues are more effective than cisplatin at inducing apoptosis in cancer cell lines
|
Vo, Van |
|
2010 |
18 |
3 |
p. 1163-1170 8 p. |
artikel |
26 |
Preparation and biodistribution of [18F]FP2OP as myocardial perfusion imaging agent for positron emission tomography
|
Mou, Tiantian |
|
2010 |
18 |
3 |
p. 1312-1320 9 p. |
artikel |
27 |
Proteasome inhibition in human breast cancer cells with high catechol-O-methyltransferase activity by green tea polyphenol EGCG analogs
|
Huo, Congde |
|
2010 |
18 |
3 |
p. 1252-1258 7 p. |
artikel |
28 |
Salicylanilide carbamates: Antitubercular agents active against multidrug-resistant Mycobacterium tuberculosis strains
|
Férriz, Juana M. |
|
2010 |
18 |
3 |
p. 1054-1061 8 p. |
artikel |
29 |
Site-specific labeling of ‘second generation’ annexin V with 99mTc(CO)3 for improved imaging of apoptosis in vivo
|
De Saint-Hubert, Marijke |
|
2010 |
18 |
3 |
p. 1356-1363 8 p. |
artikel |
30 |
Square pyramidal copper(II) complexes with forth generation fluoroquinolone and neutral bidentate ligand: Structure, antibacterial, SOD mimic and DNA-interaction studies
|
Patel, Mohan N. |
|
2010 |
18 |
3 |
p. 1227-1235 9 p. |
artikel |
31 |
Structure–activity relationship of C5-curcuminoids and synthesis of their molecular probes thereof
|
Yamakoshi, Hiroyuki |
|
2010 |
18 |
3 |
p. 1083-1092 10 p. |
artikel |
32 |
Structure and in vitro antitumor activity evaluation of brominated diterpenes from the red alga Sphaerococcus coronopifolius
|
Smyrniotopoulos, Vangelis |
|
2010 |
18 |
3 |
p. 1321-1330 10 p. |
artikel |
33 |
Synthesis and biological evaluation of antitumour-active betulin derivatives
|
Csuk, René |
|
2010 |
18 |
3 |
p. 1344-1355 12 p. |
artikel |
34 |
Synthesis and biological evaluation of oxadiazole derivatives as inhibitors of soluble guanylyl cyclase
|
von Wantoch Rekowski, Margarete |
|
2010 |
18 |
3 |
p. 1288-1296 9 p. |
artikel |
35 |
Synthesis and biological evaluation of simple methoxylated chalcones as anticancer, anti-inflammatory and antioxidant agents
|
Bandgar, Babasaheb P. |
|
2010 |
18 |
3 |
p. 1364-1370 7 p. |
artikel |
36 |
Synthesis and disulfide bond connectivity–activity studies of a kalata B1-inspired cyclopeptide against dengue NS2B–NS3 protease
|
Gao, Yaojun |
|
2010 |
18 |
3 |
p. 1331-1336 6 p. |
artikel |
37 |
Synthesis and optimization of hyaluronic acid–methotrexate conjugates to maximize benefit in the treatment of osteoarthritis
|
Homma, Akie |
|
2010 |
18 |
3 |
p. 1062-1075 14 p. |
artikel |
38 |
Synthesis and structural and pharmacological properties of cyclopropane-based conformationally restricted analogs of 4-methylhistamine as histamine H3/H4 receptor ligands
|
Kobayashi, Takaaki |
|
2010 |
18 |
3 |
p. 1076-1082 7 p. |
artikel |
39 |
Synthesis and structure–activity relationship of 1,2,4-triazole-containing diarylpyrazolyl carboxamide as CB1 cannabinoid receptor–ligand
|
Seo, Hee Jeong |
|
2010 |
18 |
3 |
p. 1149-1162 14 p. |
artikel |
40 |
Synthesis and the biological evaluation of arylnaphthalene lignans as anti-hepatitis B virus agents
|
Janmanchi, Damodar |
|
2010 |
18 |
3 |
p. 1213-1226 14 p. |
artikel |
41 |
Synthesis, biological evaluation, and molecular modeling of berberine derivatives as potent acetylcholinesterase inhibitors
|
Huang, Ling |
|
2010 |
18 |
3 |
p. 1244-1251 8 p. |
artikel |
42 |
Synthesis of C-glycoside analogues of β-galactosamine-(1→4)-3-O-methyl-d-chiro-inositol and assay as activator of protein phosphatases PDHP and PP2Cα
|
Hans, Sunej K. |
|
2010 |
18 |
3 |
p. 1103-1110 8 p. |
artikel |
43 |
Synthesis of 1-(d-glucopyranosyl)-1,2,3-triazoles and their evaluation as glycogen phosphorylase inhibitors
|
Bokor, Éva |
|
2010 |
18 |
3 |
p. 1171-1180 10 p. |
artikel |
44 |
Toosendanin: Synthesis of the AB-ring and investigations of its anti-botulinum properties (Part II)
|
Nakai, Yuya |
|
2010 |
18 |
3 |
p. 1280-1287 8 p. |
artikel |
45 |
Utilization of the 1,2,3,5-thiatriazolidin-3-one 1,1-dioxide scaffold in the design of potential inhibitors of human neutrophil proteinase 3
|
Dou, Dengfeng |
|
2010 |
18 |
3 |
p. 1093-1102 10 p. |
artikel |