| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A boronic acid chalcone analog of combretastatin A-4 as a potent anti-proliferation agent
|
Kong, Yali
|
|
2010
|
18 |
2 |
p. 971-977
7 p.
|
artikel
|
| 2 |
A diazirine-based photoaffinity etoposide probe for labeling topoisomerase II
|
Chee, Gaik-Lean
|
|
2010
|
18 |
2 |
p. 830-838
9 p.
|
artikel
|
| 3 |
Antifolate and antiproliferative activity of 6,8,10-triazaspiro[4.5]deca-6,8-dienes and 1,3,5-triazaspiro[5.5]undeca-1,3-dienes
|
Ma, Xiang
|
|
2010
|
18 |
2 |
p. 737-743
7 p.
|
artikel
|
| 4 |
Antitumor agents 270. Novel substituted 6-phenyl-4H-furo[3,2-c]pyran-4-one derivatives as potent and highly selective anti-breast cancer agents
|
Dong, Yizhou
|
|
2010
|
18 |
2 |
p. 803-808
6 p.
|
artikel
|
| 5 |
Apoptotic activities in closely related styryllactone stereoisomers toward human tumor cell lines: Investigation of synergism of styryllactone-induced apoptosis with TRAIL
|
Gupta, Shuchi
|
|
2010
|
18 |
2 |
p. 849-854
6 p.
|
artikel
|
| 6 |
Bisquaternary pyridinium oximes: Comparison of in vitro reactivation potency of compounds bearing aliphatic linkers and heteroaromatic linkers for paraoxon-inhibited electric eel and recombinant human acetylcholinesterase
|
Bharate, Sandip B.
|
|
2010
|
18 |
2 |
p. 787-794
8 p.
|
artikel
|
| 7 |
Cell permeability of Py–Im-polyamide-fluorescein conjugates: Influence of molecular size and Py/Im content
|
Nishijima, Shigeki
|
|
2010
|
18 |
2 |
p. 978-983
6 p.
|
artikel
|
| 8 |
Characterization of non-lipid autotaxin inhibitors
|
Hoeglund, Adrienne B.
|
|
2010
|
18 |
2 |
p. 769-776
8 p.
|
artikel
|
| 9 |
Click synthesis of estradiol–cyclodextrin conjugates as cell compartment selective estrogens
|
Kim, Hye-Yeong
|
|
2010
|
18 |
2 |
p. 809-821
13 p.
|
artikel
|
| 10 |
Comparative molecular field analysis of fenoterol derivatives: A platform towards highly selective and effective β2-adrenergic receptor agonists
|
Jozwiak, Krzysztof
|
|
2010
|
18 |
2 |
p. 728-736
9 p.
|
artikel
|
| 11 |
Corrigendum to “Design, synthesis and SAR studies of 4-allyoxyaniline amides as potent 15-lipoxygensae inhibitors” [Bioorg. Med. Chem. 17 (2009) 1614]
|
Seyedi, Seyed Mohammad
|
|
2010
|
18 |
2 |
p. 986-
1 p.
|
artikel
|
| 12 |
Corrigendum to “Evaluation of delocalized lipophilic cationic dyes as delivery vehicles for photosensitizers to mitochondria” [Bioorg. Med. Chem. 17 (2009) 6631]
|
Ngen, Ethel J.
|
|
2010
|
18 |
2 |
p. 984-
1 p.
|
artikel
|
| 13 |
Corrigendum to “SAR and biological evaluation of SEN12333/WAY-317538: Novel alpha 7 nicotinic acetylcholine receptor agonist” [Bioorg. Med. Chem. 17 (2009) 5247]
|
Haydar, Simon N.
|
|
2010
|
18 |
2 |
p. 985-
1 p.
|
artikel
|
| 14 |
Design and pharmacophore modeling of biaryl methyl eugenol analogs as breast cancer invasion inhibitors
|
Abdel Bar, Fatma M.
|
|
2010
|
18 |
2 |
p. 496-507
12 p.
|
artikel
|
| 15 |
Design and preliminary structure–activity relationship of redox-silent semisynthetic tocotrienol analogues as inhibitors for breast cancer proliferation and invasion
|
Elnagar, Ahmed Y.
|
|
2010
|
18 |
2 |
p. 755-768
14 p.
|
artikel
|
| 16 |
Design and synthesis of selective inhibitors of Placental Alkaline Phosphatase
|
Lanier, Marion
|
|
2010
|
18 |
2 |
p. 573-579
7 p.
|
artikel
|
| 17 |
Design, synthesis and biological evaluation of 6-(benzyloxy)-4-methylquinolin-2(1H)-one derivatives as PDE3 inhibitors
|
Nikpour, Mohsen
|
|
2010
|
18 |
2 |
p. 855-862
8 p.
|
artikel
|
| 18 |
Design, synthesis and primary activity assay of bi- or tri-peptide analogues with the scaffold l-arginine as amino-peptidase N/CD13 inhibitors
|
Mou, Jiajia
|
|
2010
|
18 |
2 |
p. 887-895
9 p.
|
artikel
|
| 19 |
Development of carbohydrate-derived inhibitors of acid sphingomyelinase
|
Roth, Anke G.
|
|
2010
|
18 |
2 |
p. 939-944
6 p.
|
artikel
|
| 20 |
2-Dialkynyl derivatives of (N)-methanocarba nucleosides: ‘Clickable’ A3 adenosine receptor-selective agonists
|
Tosh, Dilip K.
|
|
2010
|
18 |
2 |
p. 508-517
10 p.
|
artikel
|
| 21 |
2,4-Diamino-5-methyl-6-substituted arylthio-furo[2,3-d]pyrimidines as novel classical and nonclassical antifolates as potential dual thymidylate synthase and dihydrofolate reductase inhibitors
|
Gangjee, Aleem
|
|
2010
|
18 |
2 |
p. 953-961
9 p.
|
artikel
|
| 22 |
Discovery of 3-(4-bromophenyl)-6-nitrobenzo[1.3.2]dithiazolium ylide 1,1-dioxide as a novel dual cyclooxygenase/5-lipoxygenase inhibitor that also inhibits tumor necrosis factor-α production
|
Chen, Chien-Shu
|
|
2010
|
18 |
2 |
p. 597-604
8 p.
|
artikel
|
| 23 |
Di-substituted pyridinyl aminohydantoins as potent and highly selective human β-secretase (BACE1) inhibitors
|
Malamas, Michael S.
|
|
2010
|
18 |
2 |
p. 630-639
10 p.
|
artikel
|
| 24 |
Editorial board
|
|
|
2010
|
18 |
2 |
p. IFC-
1 p.
|
artikel
|
| 25 |
Enhancement of EGFR tyrosine kinase inhibition by C–C multiple bonds-containing anilinoquinazolines
|
Ban, Hyun Seung
|
|
2010
|
18 |
2 |
p. 870-879
10 p.
|
artikel
|
| 26 |
Fluoroalkene modification of mercaptoacetamide-based histone deacetylase inhibitors
|
Osada, Satoshi
|
|
2010
|
18 |
2 |
p. 605-611
7 p.
|
artikel
|
| 27 |
Graphical contents list
|
|
|
2010
|
18 |
2 |
p. 463-476
14 p.
|
artikel
|
| 28 |
Identification and characterisation of 2-aminopyridine inhibitors of checkpoint kinase 2
|
Hilton, Stephen
|
|
2010
|
18 |
2 |
p. 707-718
12 p.
|
artikel
|
| 29 |
Identification of novel allosteric nonpeptidergic inhibitors of the human cytomegalovirus-encoded chemokine receptor US28
|
Vischer, Henry F.
|
|
2010
|
18 |
2 |
p. 675-688
14 p.
|
artikel
|
| 30 |
Identification of triazinoindol-benzimidazolones as nanomolar inhibitors of the Mycobacterium tuberculosis enzyme TDP-6-deoxy-d-xylo-4-hexopyranosid-4-ulose 3,5-epimerase (RmlC)
|
Sivendran, Sharmila
|
|
2010
|
18 |
2 |
p. 896-908
13 p.
|
artikel
|
| 31 |
1-Indol-1-yl-propan-2-ones and related heterocyclic compounds as dual inhibitors of cytosolic phospholipase A2α and fatty acid amide hydrolase
|
Forster, Laura
|
|
2010
|
18 |
2 |
p. 945-952
8 p.
|
artikel
|
| 32 |
Isolation, structure, and bioactivities of abiesadines A–Y, 25 new diterpenes from Abies georgei Orr
|
Yang, Xian-Wen
|
|
2010
|
18 |
2 |
p. 744-754
11 p.
|
artikel
|
| 33 |
Labeled 3-aryl-4-indolylmaleimide derivatives and their potential as angiogenic PET biomarkers
|
Ilovich, Ohad
|
|
2010
|
18 |
2 |
p. 612-620
9 p.
|
artikel
|
| 34 |
Lobeline esters as novel ligands for neuronal nicotinic acetylcholine receptors and neurotransmitter transporters
|
Hojahmat, Marhaba
|
|
2010
|
18 |
2 |
p. 640-649
10 p.
|
artikel
|
| 35 |
Molecular design of N-linked tetravalent glycosides bearing N-acetylglucosamine, N,N′-diacetylchitobiose and N-acetyllactosamine: Analysis of cross-linking activities with WGA and ECA lectins
|
Masaka, Ryuichi
|
|
2010
|
18 |
2 |
p. 621-629
9 p.
|
artikel
|
| 36 |
New heteroaryl nitrones with spin trap properties: Identification of a 4-furoxanyl derivative with excellent properties to be used in biological systems
|
Barriga, Germán
|
|
2010
|
18 |
2 |
p. 795-802
8 p.
|
artikel
|
| 37 |
New thalidomide analogues derived through Sonogashira or Suzuki reactions and their TNF expression inhibition profiles
|
Stewart, Scott G.
|
|
2010
|
18 |
2 |
p. 650-662
13 p.
|
artikel
|
| 38 |
Novel and selective DNA methyltransferase inhibitors: Docking-based virtual screening and experimental evaluation
|
Kuck, Dirk
|
|
2010
|
18 |
2 |
p. 822-829
8 p.
|
artikel
|
| 39 |
Perchlorotrityl radical-fluorophore conjugates as dual fluorescence and EPR probes for superoxide radical anion
|
Wang, Jinhua
|
|
2010
|
18 |
2 |
p. 922-929
8 p.
|
artikel
|
| 40 |
Phenolics from Glycyrrhiza glabra roots and their PPAR-γ ligand-binding activity
|
Kuroda, Minpei
|
|
2010
|
18 |
2 |
p. 962-970
9 p.
|
artikel
|
| 41 |
Quinazolinone linked pyrrolo[2,1-c][1,4]benzodiazepine (PBD) conjugates: Design, synthesis and biological evaluation as potential anticancer agents
|
Kamal, Ahmed
|
|
2010
|
18 |
2 |
p. 526-542
17 p.
|
artikel
|
| 42 |
Quiquelignan A–H, eight new lignoids from the rattan palm Calamus quiquesetinervius and their antiradical, anti-inflammatory and antiplatelet aggregation activities
|
Chang, Chao-Lin
|
|
2010
|
18 |
2 |
p. 518-525
8 p.
|
artikel
|
| 43 |
Synthesis and anti-viral activity of azolo-adamantanes against influenza A virus
|
Zarubaev, Vladimir V.
|
|
2010
|
18 |
2 |
p. 839-848
10 p.
|
artikel
|
| 44 |
Synthesis and biological properties of iron chelators based on a bis-2-(2-hydroxy-phenyl)-thiazole-4-carboxamide or -thiocarboxamide (BHPTC) scaffold
|
Rodriguez-Lucena, David
|
|
2010
|
18 |
2 |
p. 689-695
7 p.
|
artikel
|
| 45 |
Synthesis and optimization of thiadiazole derivatives as a novel class of substrate competitive c-Jun N-terminal kinase inhibitors
|
De, Surya K.
|
|
2010
|
18 |
2 |
p. 590-596
7 p.
|
artikel
|
| 46 |
Synthesis, anti-HIV and anti-oxidant activities of caffeoyl 5,6-anhydroquinic acid derivatives
|
Ma, Chao-Mei
|
|
2010
|
18 |
2 |
p. 863-869
7 p.
|
artikel
|
| 47 |
Synthesis, biological evaluation and molecular docking studies of amide-coupled benzoic nitrogen mustard derivatives as potential antitumor agents
|
Zheng, Qing-Zhong
|
|
2010
|
18 |
2 |
p. 880-886
7 p.
|
artikel
|
| 48 |
Synthesis, characterization and antiglaucoma activity of a novel proton transfer compound and a mixed-ligand Zn(II) complex
|
Yenikaya, Cengiz
|
|
2010
|
18 |
2 |
p. 930-938
9 p.
|
artikel
|
| 49 |
Synthesis, DNA binding, fluorescence measurements and antiparasitic activity of DAPI related diamidines
|
Farahat, Abdelbasset A.
|
|
2010
|
18 |
2 |
p. 557-566
10 p.
|
artikel
|
| 50 |
Synthesis, in vitro structure–activity relationship, and in vivo studies of 2-arylthiazolidine-4-carboxylic acid amides as anticancer agents
|
Lu, Yan
|
|
2010
|
18 |
2 |
p. 477-495
19 p.
|
artikel
|
| 51 |
Synthesis of 6-N-(benzothiazol-2-yl)deoxyadenosine and its exciton-coupled circular dichroism
|
Masaki, Yoshiaki
|
|
2010
|
18 |
2 |
p. 567-572
6 p.
|
artikel
|
| 52 |
Synthesis of structurally simplified analogues of aplidinone A, a pro-apoptotic marine thiazinoquinone
|
Aiello, Anna
|
|
2010
|
18 |
2 |
p. 719-727
9 p.
|
artikel
|
| 53 |
Synthesis of α-tocohexaenol (α-T6) a fluorescent, oxidatively sensitive polyene analogue of α-tocopherol
|
Wang, Yongsheng
|
|
2010
|
18 |
2 |
p. 777-786
10 p.
|
artikel
|
| 54 |
Synthesis, pharmacological studies and molecular modeling of some tetracyclic 1,3-diazepinium chlorides
|
Grant, Julie-Ann A.
|
|
2010
|
18 |
2 |
p. 909-921
13 p.
|
artikel
|
| 55 |
The chemical synthesis and antibiotic activity of a diverse library of 2-aminobenzimidazole small molecules against MRSA and multidrug-resistant A. baumannii
|
Huigens III, Robert W.
|
|
2010
|
18 |
2 |
p. 663-674
12 p.
|
artikel
|
| 56 |
The effect of backbone cyclization on PK/PD properties of bioactive peptide-peptoid hybrids: The melanocortin agonist paradigm
|
Ovadia, Oded
|
|
2010
|
18 |
2 |
p. 580-589
10 p.
|
artikel
|
| 57 |
Towards the synthesis of bisubstrate inhibitors of protein farnesyltransferase: Synthesis and biological evaluation of new farnesylpyrophosphate analogues
|
Duez, Stéphanie
|
|
2010
|
18 |
2 |
p. 543-556
14 p.
|
artikel
|
| 58 |
Triazoloacridin-6-ones as novel inhibitors of the quinone oxidoreductases NQO1 and NQO2
|
Nolan, Karen A.
|
|
2010
|
18 |
2 |
p. 696-706
11 p.
|
artikel
|
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